Patents
Patents for C07D 491 - Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups , , or (29,726)
05/2006
05/03/2006CN1254243C Pharmaceutical compositions comprising chelidonine or derivatives thereof
05/02/2006US7038052 Process for the synthesis of derivatives of 2, 3-dihydro-1, 4-dioxino- [2, 3-f] quinoline
05/02/2006US7037926 Anticarcinogenic, antiallergen, and antiinflammatory agents; autoimmuned diseases
05/02/2006US7037925 for treating or preventing organ transplant rejection, lupus, multiple sclerosis, rheumatoid arthritis, psoriasis, Type I diabetes, asthma, rhinitis, atopic dermatitis, autoimmune disorders, Alzheimer's disease, leukemia
05/02/2006US7037920 Substituted tricyclic himbacine derivatives that are useful as thrombin receptor antagonists
05/02/2006US7037919 novel nonsteroidal compounds and salts; have a specific and strong binding affinity for androgen receptors and exhibit AR agonism or antagonism; therapeutic effect on AR-mediated diseases such as male hypogonadism, male sexual dysfunction, anemia, aids, breast, prostate cancer
05/02/2006US7037915 fused thienopyrimidine compounds useful as phosphatidylinositol 3-kinase inhibitors and carcinostatic agents
04/2006
04/27/2006WO2006043490A1 Pyrimidine derivative fused with nonaromatic ring
04/27/2006WO2006029146A3 6H-[1]BENZOPYRANO[4,3-b]QUINOLINES AND THEIR USE AS ESTROGENIC AGENTS
04/27/2006US20060089397 Synthetic diazonamides
04/27/2006US20060089379 Tetrahydropyranyl cyclopentyl tetrahydroisoquinoline modulators of chemokine receptor activity
04/27/2006US20060089354 ligands for receptor localization studies; for inhibiting binding of vanilloid ligand to a capsaicin receptor; Phosphoric acid dibenzyl ester 4-(4-tert-butyl-phenylamino)-7-(3-trifluoromethyl-pyridin-2-yl)-quinazolin-2-ylmethyl ester; to treat neuropathic pain, itch, urinary incontinence, cough, obesity
04/27/2006US20060089344 E.g., 2-(Methylamino)-2-oxoethyl 3-[1-(1-isoquinolyl)-4-piperidyl]propylcarbamate hydrochloride and 3{2-[1-(2-quinolyl)-4-piperidyl]-ethyl}-1,3-oxazolidine-2,4-dione; preventing or treating a pathology in which endogenous cannabinoids and/or any other substrate metabolized by the enzyme FA; analgesics
04/27/2006US20060089262 Substituted (thioxo)carbonylamino phenyl uraciles
04/27/2006CA2584507A1 Flavanoids and isoflavanoids for the prevention and treatment of cardiovascular diseases
04/26/2006EP1650235A1 Vinyl monomer, polymer derived from such monomer, and a light-emitting device using such polymer
04/26/2006EP1648923A1 Spatially-defined macrocycles incorporating peptide bond surrogates
04/26/2006EP1648905A1 Thienopyridine and furopyridine kinase inhibitors
04/26/2006EP1648904A1 N-sulfonylheterocyclopyrrolylalkylamine compounds as 5-hydroxytryptamine-6 ligands
04/26/2006EP1648871A1 Piperidine or 8-aza-bicyclo 3.2.1 oct-3-yl derivatives useful as modulators of chemokine receptor activity
04/26/2006EP1648870A2 Sulfonic acid derivatives of polycyclic dyes used for analytical applications
04/26/2006EP1409485B1 Immunomodulating compounds
04/26/2006CN1764663A Method for preparing topotecan from 10-hydroxy-4-(S)-camptothecine
04/26/2006CN1764662A Cyclic benzimidazoles.
04/26/2006CN1764655A Aromatic sulfone hydroxamates and their use as protease inhibitors
04/26/2006CN1764648A hydroxamid acid derivatives as histone deacetylase (HDAC) inhibitors
04/26/2006CN1763042A Preparation method of indole-containing heterocycle pyridinedihydrofuranketone
04/26/2006CN1253455C 2-3-methylen-dioxy dibenzo [a,g] quinolizine onium hydrochloride and its uses in treatment of diabete
04/26/2006CN1253441C Protease inhibitors
04/25/2006US7034163 From alkoxycyclopropane with nitrile in presence of Lewis acid catalyst
04/25/2006US7034153 Antidepressants; anxiolytic agents; eating disorders; antiulcer agents; drug abuse; Alzheimer's disease
04/25/2006US7034041 Substituted 4-phenyl-1-(1-phenylcyclohexyl)-1,2,3,6-tetrahydropyridine
04/25/2006US7034021 Dihydro-1,3,5-triazine amine derivatives and their therapeutic uses
04/25/2006CA2189525C 2-(aminomethyl)-3,4,7,9-tetrahydro-2h-pyrano-[2,3e]indol-8-ones and derivatives
04/20/2006WO2006041872A2 Thrombin receptor antagonists
04/20/2006WO2006040351A1 Indazoles, benzisoxazoles and benzisothiazoles and their use as estrogenic agents
04/20/2006WO2006040338A1 Difluoro-substituted imidazopyridines
04/20/2006WO2005115398A3 Hiv integrase inhibitors
04/20/2006WO2005111039A3 Compounds and methods for inhibiting mitotic progression by inhibition of aurora kinase
04/20/2006WO2005016913A8 Tetrahydroisoquinoline or isochroman compounds as orl-1 receptor ligands for the treatment of pain and cns disorders
04/20/2006US20060084803 Bicyclic pyridine and pyrimidine P38 kinase inhibitors
04/20/2006US20060084576 Hetaryl substituted homotetramic and homotetronic acids and their use thereof as pesticides
04/20/2006US20060083676 For marking and identifying metabotropic glutamate receptor sites and for imaging an organ; in particular non-competitive mGlu1 receptor ligands
04/20/2006CA2583253A1 Difluoro-substituted imidazopyridines
04/20/2006CA2582639A1 Thrombin receptor antagonists
04/20/2006CA2582180A1 Indazoles, benzisoxazoles and benzisothiazoles, process for preparing them, pharmaceutical compositions and use as estrogenic agents
04/19/2006EP1647549A1 Indazoles, benzisoxazoles and benzisothiazoles as estrogenic agents
04/19/2006EP1646661A2 Living radical polymerization initiator comprising a functional group capable of reacting with polypeptides or the like, comb polymer obtained therewith, polypeptide conjugates and drung obtained therefrom
04/19/2006EP1646615A1 Pyrimidine derivatives as modulators of atp-binding cassette transporters
04/19/2006EP1646388A2 Cytotoxic indeno and isoindoloisoquinolones
04/19/2006EP1646380A2 Indolocarbazole anticancer agents and methods of using same
04/19/2006EP1537112B1 Condensed pyridines and pyrimidines with tie2 (tek) activity
04/19/2006EP1363883B1 Hydroxy-substituted n-alkoxy hindered amines and compositions stabilized therewith
04/19/2006EP1080726B1 Agents for relieving side effects
04/19/2006EP1044197B1 Piperidinyl-substituted pyridylalkane, alkene and alkyne carboxamides as cytostatic agents and immunosuppressants
04/19/2006EP0885215B1 Novel benzo-1,3-dioxolyl- and benzofuranyl substituted pyrrolidine derivatives as endothelin antagonists
04/19/2006CN1761668A 7-imino derivatives of camptothecin having antitumor activity
04/19/2006CN1761667A 3-phenyl substituted 3-substituted-4ketolactams and ketolactones
04/19/2006CN1761660A Indeno-fused photochromic naphthopyrans, naphthols and photochromic articles
04/19/2006CN1761651A 2,4-dihalogen-6-(c2-c3-alkyl)-phenyl substituted tetramic acid derivatives
04/19/2006CN1760195A Method for separating and purifying 9-nitro camptothecin
04/18/2006US7030245 A chemical intermediate, toluene-4-sulfonic acid 7,8-dihydro-6H-5-oxa-1-aza-phenanthren-6-ylmethyl ester for preparing antidepressant, 6-[4-(5-fluoro-1H-indol-3-yl)-3,6-dihydro-2H-pyridin-1-ylmethyl]-7,8-dihydro-6H-5-oxa-1aza-phenanthrene; treating psychological disorders
04/18/2006US7030243 Process for making camptothecin derivatives
04/18/2006US7030196 Process for reducing the molecular weight of polypropylene
04/18/2006US7030135 A sulfonylamino-tetrahydro(1,3)thiazolo(5,4-c)pyridinyl or benzothiazole derivatives, for treating diabetes, syndrome X, obesity, glaucoma, hyperlipidemia, hyperglycemia, hyperinsulinemia, osteoporosis, tuberculosis, dementia
04/18/2006CA2247513C Camptothecin derivatives and the use thereof as antitumor agents
04/18/2006CA2241852C Fused pyrrolo(2,3-c)carbazole-6-ones which potentiate activity of gamma interferon
04/18/2006CA2207443C Tricyclic compounds
04/13/2006WO2006038596A1 Pharmaceutical composition for xerophthalmia and xerostomia treatment
04/13/2006WO2006038526A1 Acid addition salt of irinotecan
04/13/2006US20060079567 Tricyclic heteroaryl piperazines, pyrrolidines and azetidines as serotonin receptor modulators
04/13/2006US20060079563 Cyclic protein tyrosine kinase inhibitors
04/13/2006US20060078518 Cosmetic compositions containing fluorescent colorants for natural skin appearance
04/13/2006CA2582615A1 Pharmaceutical composition for treatment of tear and salivary fluid drying
04/13/2006CA2582294A1 Condensed tricyclic benzimidazoles for the treatment of gastrointestinal disorders
04/12/2006EP1644372A2 Substituted quinolin-4-ylamine analogues
04/12/2006EP1644363A1 Triheterocyclic compounds, compositions, and methods for treating cancer or viral diseases
04/12/2006EP1644343A1 5-substituted quinazolinone derivatives
04/12/2006EP1644012A1 Quaternary chelidonine and alkaloid derivatives, process for their preparation and their use in manufacture of medicaments
04/12/2006EP1644001A2 Pancratistatin cyclic phosphate prodrugs an phenpanstatin cyclic phosphate prodrugs
04/12/2006EP1643998A1 Dual nk1/nk3 antagonists for treating schizophrenia
04/12/2006EP1643984A2 Use of parthenolide derivatives as antileukemic and cytotoxic agents
04/12/2006EP1546151B1 Antidepressant cycloalkylamine derivatives of heterocycle-fused benzodioxans
04/12/2006EP1349854B1 Hetaryl substituted homotetramic and homotetronic acids and the use thereof as pesticides
04/12/2006EP1054887B1 Bicyclic pyridine and pyrimidine derivatives as neuropeptide y receptor antagonists
04/12/2006CN1759110A Pyrazole derivative
04/12/2006CN1250553C Antidepressant azaheterocyclylmethyl derivatives of 2, 3-dihydro-1,4-dioxino [2,3-f] quinoxaline
04/12/2006CN1250551C Spirocyclic-6,7-dihydro-5h-pyrazolo[1,2-a]pyrazol-1-ones which control inflammatory cytokines
04/12/2006CN1250550C Process for preparation of amidine derivatives
04/12/2006CN1250544C Pyridoarylphenyl oxazolidinone antibacterials and related compositions and methods
04/12/2006CN1250542C 2-(1H-indol-3-yl)-2-oxo-acetamides with antitumor activity
04/12/2006CN1250528C Cyclic nitrones and pharmaceutical compositions containing them
04/12/2006CN1250293C Drug composites
04/11/2006US7026489 e.g., (9R)-1-{(2'S,8'S,10'S,11'R)-2',8'-dihydroxy-7'-oxo-11'-[(Z)-2-pentenyl]-9'-oxa-4'-azatricyclo[6.3.1.01.5]dodec-5'-en-10'-yl}-9-hydroxy-10-oxoundecanoic acid and N-[9-hydroxy-10-oxo-12(Z),15(Z)-octadecadienoyl]-L-isoleucine.
04/11/2006US7026484 For therapy of cancer
04/11/2006US7026472 for example 1-(methylthio)-3-methoxy-4-(2-fluorophenyl)azetidin-2-one; induce neoplastic cell apoptosis or inhibit neoplastic cell proliferation
04/11/2006US7026341 Hetaryl substituted homotetramic and homotetronic acids and their use thereof as pesticides
04/11/2006US7025900 Perylenetetracarboxylic acid dibenzimidazole sulfoderivatives containing oxo-groups in the perylene core which form part of a para-quinoid system of bonds, lyotropic liquid crystal systems and anisotropic films containing the same, and methods for making the same
04/06/2006WO2006036527A1 Substituted dipiperdine ccr2 antagonists
04/06/2006US20060074248 Process for the stereoselective synthesis of lactones