Patents for C07D 471 - Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups (64,559) |
---|
03/03/1993 | EP0529636A1 Novel isatinoxime derivatives, their preparation and use |
03/03/1993 | EP0529452A2 1,7-Condensed 2-(piperazinoalkyl)indol derivatives, process and intermediates for their preparation and pharmaceutical compositions containing them |
03/03/1993 | EP0529253A1 Phenylalkylderivatives, compounds containing them and process for their fabrication |
03/03/1993 | EP0528922A1 New sulfonyl compounds |
03/03/1993 | CN1019973C Piperidine derivative and pharmaceutical composition containing the same |
03/02/1993 | US5190953 Heterocyclic carboxylic acid amides and esters of azabicyclic compounds as gastric prokinetic, antiemetic, anxiolytic and antiarrhythmic agents |
03/02/1993 | US5190951 Quinoline derivatives |
03/02/1993 | US5190862 Peptide modified compound |
03/02/1993 | CA1314044C Imidazopyridine derivatives |
02/25/1993 | DE4227791A1 New psychotherapeutic pyrrolo-2,3-c pyridine deriv. - useful as benzodiazepine antagonists, inverse agonists and agonists |
02/24/1993 | EP0528026A1 New meso-azacyclic aromatic acid amides and esters as novel serotonergic agents |
02/24/1993 | EP0527889A1 Quinolizinone type compounds |
02/24/1993 | EP0527817A1 Gamma-butyrolactol ether derivatives |
02/24/1993 | CN1069270A Heteraryloxy-beta-carboline, processes for its production and use in pharmaceutical agents |
02/24/1993 | CA2076553A1 1,7-fused 2-(piperazinoalkyl) indole derivatives, processes and intermediates for their preparation, and pharmaceutical compositions containing them |
02/23/1993 | US5189168 1'-amino-2[(benzothiazolyl)methyl]spiro-[isoquinoline-4(1H),3'-pyrrolidine]-1,2'3,5'(2H)-tetrones and analogs thereof useful as aldose reductase inhibitors |
02/23/1993 | US5189167 Useful for prevention or treatment of diabetes mellitus associated complications |
02/23/1993 | US5189158 Acid mediated ring closure |
02/23/1993 | US5189055 Phenylpyrrolic compounds used as drugs, their preparation and application |
02/23/1993 | US5189045 Antiserotonine agent |
02/23/1993 | CA2076556A1 A method and intermediates for the preparation of 6-fluorobenzisothiazoles |
02/23/1993 | CA2076281A1 Oxidation process for preparing quinacridone pigments |
02/18/1993 | WO1993003034A1 Quinazoline derivatives as acetylcholinesterase inhibitors |
02/18/1993 | WO1993003030A1 Quinoline derivatives as immunostimulants |
02/18/1993 | WO1993003026A1 Novel quinolone carboxylic acid derivatives |
02/18/1993 | WO1993002711A1 Use of persistent free-radicals in magnetic resonance imaging |
02/18/1993 | WO1993002710A2 Use of persistent free radicals in magnetic resonance imaging |
02/18/1993 | WO1993002678A1 Use of quinozilinederivatives as orexigenics |
02/18/1993 | WO1993002677A1 5-ht4 receptor antagonists |
02/18/1993 | WO1993000095A3 Bicyclic fibrinogen antagonists |
02/18/1993 | CA2115260A1 Use of persistent free-radicals in magnetic resonance imaging |
02/18/1993 | CA2113115A1 Quinazoline derivatives as acetylcholinesterase inhibitors |
02/17/1993 | EP0527534A1 Quinoline and azaquinoline angiotensin II antagonists |
02/17/1993 | EP0527494A1 Compositon containing rhodacyanine dyes for treating cancer |
02/17/1993 | EP0527186A1 Photodynamic plant defoliants and chlorophyll biosynthesis modulators |
02/17/1993 | EP0527181A1 Heterocyclicethenediyl compounds which inhibit egf receptor tyrosine kinase |
02/17/1993 | EP0527131A1 Chelants |
02/17/1993 | CN1069025A Aryl, amide, imide, and carbamate pyridine antagonists of platelet activating factor |
02/16/1993 | US5187279 Synthesis of (-) swainsonine and intermediate compounds employed in such synthesis |
02/16/1993 | US5187180 (quinolin-2-ylmethoxy)heterotetrahydrocarbazoles as inhibitors of the biosynthesis of leukotrienes |
02/16/1993 | US5187166 Azabicyclo derivatives and their use as antiemetics |
02/16/1993 | US5187164 Psychological disorders, antiemetics |
02/16/1993 | US5187159 Angiotensin II antagonists incorporating a substituted 1,3-benzodioxole or 1,3-benzodithiole |
02/14/1993 | CA2075652A1 Quinoline and azaquinoline angiotensin ii antagonists incorporating a substituted benzyl element |
02/10/1993 | WO1993003025A1 Thiophene compound |
02/10/1993 | EP0526840A1 Condensed naphthyridine derivatives |
02/10/1993 | EP0526545A1 Isoquinoline amides and esters as 5 ht3 receptor antagonists |
02/10/1993 | CN1068822A Substituted benzothiazol derivatives, their preparation and use as herbicides |
02/10/1993 | CN1068814A Tetracyclic antibiotic and process for preparing same |
02/10/1993 | CN1019890C Process for preparation of 4-heterocyclic sulfonyl (or thio-) propyl-oxy-2-hydroxy-3-propyl-hypnone derivatives |
02/10/1993 | CA2093516A1 Thiophene compound |
02/09/1993 | US5185449 Process and intermediate for certain bis-aza-bicyclic anxiolytic agents |
02/09/1993 | US5185447 Treating polycyclic nitro compounds with aqueous base; cognition activators |
02/09/1993 | US5185337 Pyrroloquinoline derivatives and pharmaceutical compositions for antimicrobial use |
02/04/1993 | WO1993003714A2 Method for treatment of metabolic disorders |
02/04/1993 | WO1993002090A1 Manganese complexes of nitrogen-containing macrocyclic ligands effective as catalysts for dismutating superoxide |
02/04/1993 | WO1993002080A1 Imidazo (4,5-c) pyridine derivatives as paf antagonists |
02/04/1993 | WO1992018475A3 Substituted phenylazacycloalkanes as cns agents |
02/04/1993 | CA2113817A1 A method for treatment of metabolic disorders |
02/03/1993 | EP0525538A2 Process for the continuous preparation of perylenetetracarboxylic diimides |
02/03/1993 | EP0525057A1 Antimicrobial quinolonyl lactams |
02/02/1993 | US5183822 Substituted 3,4-annelated benzimidazol-2(1h)-ones |
02/02/1993 | US5183820 Lactam derivatives |
02/02/1993 | CA2075010A1 Aryl, amide, imide, and carbamate pyridine antagonists of platelet activating factor |
01/28/1993 | DE4223164A1 New 9-carbamoyl-beta-carboline derivs. - used as benzodiazepine antagonists, inverse agonists and agonists for treating neuro:degenerative and psychiatric disorders |
01/26/1993 | US5182391 Process and intermediates for the preparation of oxophthalazinyl acetic acids and analogs thereof |
01/26/1993 | US5182291 Pyrozala-pyridyl aminoabkoxyphenol compounds |
01/26/1993 | US5182289 Pyrrolo 2,3-b!Pyridin-2-one Derivatives |
01/26/1993 | US5182287 Antitumor agents, fungicides |
01/26/1993 | US5182283 Alzheimer's disease |
01/21/1993 | WO1993001195A1 DIBENZ[b,e]AZEPINE DERIVATIVES AND DRUGS CONTAINING THEM |
01/21/1993 | WO1993001191A1 Cyclic ether acetal paf antagonists |
01/21/1993 | WO1993001190A1 Novel 2-amino naphthyridine derivative, its preparation and use |
01/21/1993 | WO1993001189A1 Method for preparating optical isomers of a 2-amino naphthyridine derivative |
01/21/1993 | WO1993001188A1 Method for preparing optical isomers of a 2-amino naphthyridine derivative |
01/21/1993 | WO1993001187A1 Process for the preparation of a dextrogyral isomer of an isoindolinone derivative |
01/21/1993 | WO1993001186A1 Hydroisoquinoline derivatives |
01/21/1993 | WO1993001178A1 Diaminic compounds, preparation, use and intermediates |
01/21/1993 | WO1993000906A1 Muscarinic antagonists |
01/21/1993 | WO1993000897A1 Cholecystokinin antagonists useful in the treatment of panic attacks |
01/21/1993 | CA2112744A1 Hydroisoquinoline derivatives |
01/21/1993 | CA2111710A1 Dibenz[b,e]azepin derivatives and medicaments containing these |
01/21/1993 | CA2110986A1 Cholecystokinin antagonists useful in the treatment of panic attacks |
01/20/1993 | EP0524161A1 Manganese complexes of nitrogen containing macrocyclic ligands effective as catalysts for dismutating superoxide |
01/20/1993 | EP0524004A1 Decahydro-8H-isoquino[2,1-g][1,6]naphthyridine and decahydrobenzo[a]pyrrolo[2,3-e]quinolizine derivatives |
01/20/1993 | EP0523845A2 New benzodiazepine analogs |
01/20/1993 | EP0523533A1 Substituted pyrimidin derivatives and their use for combatting the growth of undesirable plants |
01/20/1993 | EP0523512A1 8-vinyl- and 8-ethinyl-quinolone carboxylic acids |
01/20/1993 | CN1068115A 7-isoindolinyl-quinolone-and-naphthyridone carboxylic acid herivatives |
01/20/1993 | CN1068114A 7-azaisoindolinyl-quinolone-and-naphthyridonecarboxylic acid derivatives |
01/20/1993 | CN1068113A Preparation of tetrahydropalmatinum by using guaiacol as material |
01/20/1993 | CA2073993A1 8-vinyl- and 8-ethinyl-quinolone-carboxylic acids |
01/19/1993 | US5180823 Intramolecular Cyclization |
01/19/1993 | US5180744 Renin inhibitors; hypotensive agents |
01/19/1993 | US5180725 Quinoxalinyl/quinoxaliy; alkyl-N-terminal amino hydroxy |
01/19/1993 | US5180724 Platelet activating factor |
01/19/1993 | US5180723 Certain sulfonamide heterobicyclic platelet activating factor antagonists |
01/19/1993 | US5180722 10,11-methylenedioxy-20(RS)-camptothecin and 10,11-methylenedioxy-20(S)-camptothecin analogs |
01/19/1993 | US5180418 Herbicidally active thiadiazabicyclononanes and nonenes |
01/18/1993 | CA2074038A1 Decahydro-8h-isoquino[2,1-g][1,6]naphthyridine and decahydrobenzo[a] pyrrol[2,3-e]quinolizine derivatives |