Patents for C07D 471 - Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups (64,559) |
---|
08/25/1993 | EP0556319A1 Sampangine and derivatives useful as antifungal agents |
08/25/1993 | EP0556225A1 SUBSTITUTED PYRIDO 2,3-d]PYRIMIDIN-2,4(1H,3H)-DIONES |
08/24/1993 | US5239070 Alkyl esters of 5-heterocyclic-pyridine-2,3-dicarboxylic acids |
08/24/1993 | US5238932 Mercaptoacetylamide tricyclic derivatives useful as inhibitors of enkephalinase |
08/24/1993 | CA1321586C Bicyclic compounds, their use as pharmaceuticals, their preparation, and intermediates useful in their preparation |
08/20/1993 | CA2089689A1 Substituted biphenylyl derivatives, pharmaceutical compositions containing these compounds and processes for preparing them |
08/19/1993 | WO1993016103A1 Aminoacetylmercaptoacetylamide derivatives useful as inhibitors of enkephalinase and ace |
08/19/1993 | WO1993016078A1 PROCESS FOR PREPARING CHIRAL ETHYL (5-AMINO-1,2-DIHYDRO-2-METHYL-3-PHENYLPYRIDO[3,4-b]PYRAZIN-7-YL)CARBAMATE |
08/19/1993 | WO1993016077A1 7-substituted quinolones and naphthyridones as antibacterial agents |
08/19/1993 | WO1993016076A1 3-(1h^_-tetrazol-5-yl)-4h^_-pyrido[1,2-a^_]pyrimidine-4-ones, pharmaceutical compositions containing the same and the preparation thereof |
08/19/1993 | WO1993016075A1 4-(1H-2-METHYLIMIDAZO[4,5-c]PYRIDINYLMETHYL)PHENYLSULPHONAMIDE DERIVATIVES AS ANTAGONISTS OF PAF |
08/19/1993 | WO1993016074A1 Novel isoindolinone derivative, preparation thereof, and pharmaceutical compositions containing same |
08/19/1993 | WO1993016073A1 Piperazine and piperidine derivatives, and their use as antipsychotics |
08/19/1993 | WO1993016071A1 Heterocyclic derivatives as angiotensin ii antagonists |
08/19/1993 | WO1993016070A1 3-(pyridylamino)-2-(1h^_-tetrazol-5-yl)-acrylnitriles and a process for the preparation thereof |
08/19/1993 | WO1993016050A1 Antipsychotic nitrogen-containing bicyclic compounds |
08/19/1993 | WO1993016047A1 Hydroisoindolines and hydroisoquinolines as psychotropic drugs |
08/19/1993 | WO1993015734A1 Method of treating abnormal tissue proliferation by administering an angiotensin ii antagonist |
08/19/1993 | CA2130123A1 Hydroisoindolines and hydroisoquinolines as psychotropic |
08/19/1993 | CA2130110A1 Antipsychotic-nitrogen-containing bicyclic compounds |
08/19/1993 | CA2129898A1 4-(1h-2-methylimidazo¬4,5-c|pyridinylmethyl)phenylsulphonamide derivatives as antagonists of paf |
08/19/1993 | CA2127456A1 Process for preparing chiral ethyl (5-amino-1,2-dihydro-2-methyl-3-phenylpyrido[3,4-b]pyrazin-7-yl) carbamate |
08/19/1993 | CA2117434A1 Piperazine and piperidine derivatives, and their use as antipsychotics |
08/18/1993 | EP0556080A1 Bicyclic pyridine derivatives, process for their preparation, intermediates, their use as medicaments and pharmaceutical compositions containing them |
08/18/1993 | EP0556060A1 Biphenyl-substituted quinoline and naphthyridines derivatives as angiotensine II antagonists |
08/18/1993 | EP0556008A1 Condensed imidazopyridine derivatives with psychotropic activity |
08/18/1993 | EP0555957A1 Pyrido 2,3-d pyridazine derivatives as herbicides |
08/18/1993 | EP0555825A1 Imidazo(1,2-a)pyridines as angiotensin-II-antagonists |
08/18/1993 | EP0555657A1 4-Cinnolinyl- and 4-naphthyridinyl-dihydropyridines, process for their preparation and their use in drugs |
08/18/1993 | EP0555347A1 SUBSTITUTED INDOLIZINO 1,2-b]QUINOLINONES |
08/18/1993 | EP0555327A1 Alkylidene analogs of 1'-aminospiro-[isoquinoline- 4(1h),3'-pyrrolidine]-1,2',3,5'(2h)-tetrones useful as aldose reductase inhibitors in vivo |
08/18/1993 | CN1075318A Benzopyran and related LTB4 antagonists |
08/18/1993 | CN1021825C Prepn. for aromatic w-alkylimide-tetrahydro-6h-1,3-thiazine-6-one derivatives |
08/18/1993 | CN1021824C Substituted benzofurans herbicide active compound |
08/18/1993 | CN1021820C Process for n-substituted adenine and n'-substituted cytimidine |
08/17/1993 | US5237060 Cyclization; amination |
08/17/1993 | US5236952 Catechol derivatives |
08/17/1993 | US5236937 Pyridinyl compounds which are useful as angiotensin ii antagonists |
08/17/1993 | US5236917 Respiratory system disorders, antiarthritic agents |
08/15/1993 | CA2089470A1 Azaindoles, preparation processes and medicinal products containing them |
08/15/1993 | CA2089185A1 Biphenyl-substituted quinoline derivatives |
08/12/1993 | CA2089141A1 Imidazo[1,2-a]pyridines, pharmaceutical compositions containing these compounds and processes for preparing them |
08/11/1993 | EP0554434A1 Imaging of infections |
08/11/1993 | EP0554247A1 Neuroprotective indolone and related derivatives |
08/10/1993 | US5235056 Discoloration inhibitors |
08/10/1993 | US5235054 3-carboxaldehyde substituted quinolines and naphthyridines |
08/10/1993 | US5234930 Pyrazolopyridine compounds which have useful pharmaceutical utility |
08/10/1993 | US5234923 Hypotensive agents |
08/10/1993 | US5234818 3-aminopyrazolo heterocyclic derivatives, and use for colorimetric determinations |
08/10/1993 | CA1321145C Pharmaceutical preparations |
08/10/1993 | CA1321144C Pharmaceutical preparations |
08/05/1993 | WO1993015091A1 Diphosphine ligands |
08/05/1993 | WO1993015090A1 Diphosphine ligands |
08/05/1993 | WO1993015080A1 Azabicyclo compounds as calcium channel antagonists |
08/05/1993 | WO1993015079A1 Pyrroloimidazolyl and imidazopyridinyl substituted 1h-benzimidazole derivatives as aromatase inhibitors |
08/05/1993 | WO1993015074A1 Substituted phenylheterocyclic herbicides |
08/05/1993 | WO1993015073A1 Azabricyclic compounds as calcium channel antagonists |
08/05/1993 | WO1993015067A1 Benzopyran and related ltb4 antagonists |
08/05/1993 | WO1993015051A1 N-sulphonyl-2-oxoindole derivatives having affinity for vasopressin and/or ocytocin receptors |
08/05/1993 | WO1993015046A1 Carbamates and plant-protecting agents containing them |
08/05/1993 | CA2128736A1 Substituted phenylheterocyclic herbicides |
08/05/1993 | CA2128536A1 Azabicyclo compounds as calcium channel antagonists |
08/05/1993 | CA2127689A1 Pyrroloimidazolyl and imidazopyridinyl substituted 1h-benzimidazole derivatives as aromatase inhibitors |
08/05/1993 | CA2107348A1 N-sulfonyl-2-oxoindole derivatives having affinity for vasopressin and/or ocytocin receptors |
08/04/1993 | EP0554098A2 Process for the preparation of imidazo 4,5-b pyridine derivatives |
08/04/1993 | EP0553682A1 Imidazo 4,5-b pyridine derivatives as Angiotensin II antagonists |
08/04/1993 | EP0553263A1 1'-aminospiro-[isoquinoline-4(1h),3'-pyrrolidine]- 1,2',3,5'(2h)-tetrones and analogs thereof useful as aldose reductase inhibitors in vivo |
08/04/1993 | CN1074907A Pyrroloimidazolyl and imidazopyridinyl substituted 1H-benzimidizole derivatives |
08/04/1993 | CN1074906A New 4-cinnolinyl- and 4-naphthyridinyl-dihydropyridines, processes for their preparation and their use in medicaments |
08/03/1993 | US5232924 Cardiovascular disorders |
08/03/1993 | CA1320952C Antitumor alkaloids |
08/01/1993 | CA2088464A1 A new pyridine bicyclic derivatives, process for preparing the same, new intermediates obtained, apllication of the same as drugs, and pharmac eutical compositions containing thesame |
07/31/1993 | CA2088209A1 4-cinnolinyl- and 4-naphthyridinyl-dihydropyridines, processes for their preparation and their use in medicaments |
07/29/1993 | CA2088220A1 Heterocyclic derivatives |
07/29/1993 | CA2086647A1 Chemical process |
07/28/1993 | EP0552552A2 5-Deazafolic acid derivatives and their use as antineoplastics agents |
07/28/1993 | EP0552237A1 Certain cycloalkyl and azacycloalkyl pyrrolopyrimidines; a new class of gaba brain receptor ligands |
07/28/1993 | CN1074683A Benzofuran derivatives |
07/28/1993 | CN1074682A Pyridylthiozolidine carboxylic amide derivative preparation thereof and its application in medical treatment |
07/28/1993 | CN1074606A Method of using M1-selective antimuscarinic pyridobenzodiazepinones in axial myopia therapy |
07/27/1993 | US5231182 Platelet activating factor inhibitor |
07/27/1993 | US5231181 Crystallization and resolution |
07/27/1993 | US5231111 Imidazolyl/imidazolylalkyl-N-terminal cycloalkoxy-C-terminal amino hydroxy β-amino acid derivatives |
07/27/1993 | US5231100 Antineoplastic modified imidazoacridines |
07/27/1993 | US5231098 Insecticidal nitro-substituted heterocyclic compounds |
07/24/1993 | WO1993014636A1 Insect control with substituted oxadiazole and thiadiazole compounds |
07/24/1993 | CA2105556A1 Insect control with substituted oxadiazole and thiadiazole compounds |
07/22/1993 | WO1993014092A1 Disubstituted polycyclic systems as cognition enhancers |
07/22/1993 | WO1993014091A1 Alkyl derivatives of trazodone with cns activity |
07/22/1993 | WO1993014090A1 Heterocyclic compounds and their preparation and use |
07/22/1993 | WO1993014089A1 Heterocyclic compounds and their preparation and use |
07/22/1993 | WO1993014088A1 Antihistaminic piperazinyl derivatives |
07/22/1993 | WO1993014083A1 Pharmaceutically active substituted benzimidazole derivatives |
07/22/1993 | WO1993014072A1 Amino acid derivatives as paf-receptor antagonists |
07/22/1993 | WO1993014069A1 Heterocyclic sulfonamide derivatives as antagonists of paf and angiotensin ii |
07/22/1993 | WO1993013777A1 Method of using m1-selective antimuscarinic pyridobenzodiazepinones in axial myopia therapy |
07/22/1993 | CA2128234A1 Disubstituted polycyclic systems as cognition enhancers |
07/22/1993 | CA2127367A1 Heterocyclic sulfonamide derivatives as antagonists of paf and angiotensin ii |
07/22/1993 | CA2127365A1 Amino acid derivatives as paf-receptor antagonists |
07/22/1993 | CA2127251A1 Heterocyclic compounds and their preparation and use |