Patents for C07D 471 - Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups (64,559) |
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12/23/1993 | WO1993025546A1 Bicyclic(azaaromatic)indoles as inhibitors of leukotriene biosynthesis |
12/23/1993 | WO1993025545A1 Novel quinoline derivatives and processes for preparing the same |
12/23/1993 | WO1993025206A1 ORALLY ADMINISTRABLE COMPOSITION OF PYRIDO[1,2-a]PYRIMIDINE DERIVATIVE |
12/23/1993 | WO1993025205A1 Pyrazolopyridine compounds for the treatment of anemia |
12/23/1993 | DE4243287A1 N-Substituierte Azabicycloheptan-Derivate, ihre Herstellung und Verwendung N-substituted Azabicycloheptan derivatives, their preparation and use |
12/23/1993 | DE4220384A1 Use of 9-amino-pyridazino (4',5'3,4)pyrrolo-(2,1-a)isoquinoline derivs. - are inhibitors of non-selective cation channels and useful for treating chromic inflammations |
12/23/1993 | DE4220380A1 Treatment of ulcerative colitis and Crohn's disease - by admin. of 9-amino-pyridazino:pyrrolo:isoquinoline derivs. which act as vaso-spasmolytic endothelin antagonists |
12/23/1993 | DE4220373A1 New fused ring di:hydro-pyridine-acetic acid derivs. - useful as cardio-protective and cerebro-protective agents, antiinflammatory agents and anticoagulants |
12/23/1993 | DE4220369A1 New fused-ring di:hydro-pyridine-acetic acid derivs. - useful as cardio-protective and cerebro-protective agents, antiinflammatory agents and anticoagulants |
12/23/1993 | DE4220368A1 New fused-ring di:hydro-pyridine-acetic acid derivs. - useful as cardio-protective and cerebro-protective agents, antiinflammatory agents and anticoagulants or platelet aggregation inhibitors |
12/23/1993 | DE4220361A1 Pyridazino:pyrrolo:isoquinoline deriv. anti:proliferative agents - used as non-selective cation channel blockers for inhibiting calcium flow into cells, and as antitumour agents |
12/23/1993 | DE4220355A1 New fused di:hydro-pyridine cpds. - useful in treatment of stroke, asthma, arthritis, etc. |
12/23/1993 | DE4220353A1 Use of fused di:hydro-pyridinyl phenyl acetic acid derivs. - as anti-proliferative agents in treatment of tumours |
12/23/1993 | DE4220345A1 New fused di:hydro:pyridine cpds. - exhibit cardio- and cerebro-protective activity useful in treatment of Crohn's disease, asthma, arthritis, etc. |
12/23/1993 | DE4220319A1 New use of fused di:hydro-pyridine(s) - in treatment of ulcerative colitis and Crohn's disease |
12/23/1993 | DE4220312A1 New fused ring di:hydro-pyridine derivs. - used e.g. as cardio-protective or cerebral-protective agents, antiinflammatories and blood platelet aggregation inhibitors |
12/23/1993 | CA2136547A1 Novel biologically active eburnamenine derivatives, pharmaceutical compositions containing them and process for preparing same |
12/23/1993 | CA2136240A1 Bicyclic(azaaromatic)indoles as inhibitors of leukotriene biosynthesis |
12/23/1993 | CA2112360A1 Bicyclic fibrinogen antagonists |
12/22/1993 | EP0574846A2 Imidazopyridines as angiotensin II antagonistes |
12/22/1993 | EP0574787A2 Benzimidazole derivatives as angiotensin II antagonists |
12/22/1993 | EP0574783A2 Asymmetric hydrogenation |
12/22/1993 | CN1023226C Prepn. method of medical compounds |
12/21/1993 | US5272269 Disubstituted polycyclic systems and preparative methods therefor |
12/21/1993 | US5272167 Pharmaceutically active compounds |
12/21/1993 | US5272154 3,7 substituted indole and indazole compounds and pharmaceutical compositions containing them |
12/21/1993 | US5272150 Hydroxyalkylfuranyl derivatives |
12/21/1993 | US5272146 1,2-dihydroellipticines with activity against CNS specific cancer cell lines |
12/18/1993 | CA2098473A1 Imidazopyridines |
12/15/1993 | EP0574231A1 Quinolone and naphthyridine derivatives having at the 3-position a group other than a carboxy group, as antibacterials |
12/15/1993 | EP0574195A1 Antitumoral aza- and diazaanthracenes |
12/15/1993 | EP0574174A2 Angiotensin II antagonists |
12/15/1993 | EP0573464A1 Process for preparing trans-piperidine-2,5-dicarboxylates. |
12/15/1993 | CN1023054C Oxo-1, 2-dihydroindene and tetrahydronaphthalene herbicide |
12/14/1993 | US5270322 Imidazo[1,2-a]pyridines, pharmaceutical compositions containing these compounds and processes for preparing them |
12/14/1993 | US5270317 N-substituted heterocyclic derivatives, their preparation and the pharmaceutical compositions in which they are present |
12/14/1993 | US5270316 Condensed purine derivatives |
12/14/1993 | CA2098243A1 Benzimidazole derivatives |
12/14/1993 | CA1325205C Substituted flavanoid compounds, their salts, their manufacture and medicines containing these materials |
12/09/1993 | WO1993024487A1 Nitrogen containing heterocyclic compounds as angiotensin-ii-antagonists |
12/09/1993 | WO1993024482A1 Heterocyclically bisubstituted sulphonyl amino(thio)carbonyl compounds |
12/09/1993 | WO1993024481A1 7-substituted-6-fluoro-1,4-dihydro-4-oxo-quinoline-3-carboxylic acid compounds and related compounds as antibacterial agents |
12/09/1993 | WO1993024480A1 Pyridine compound and medicinal use thereof |
12/09/1993 | CA2136993A1 Pyridine compound and pharmaceutical use thereof |
12/08/1993 | EP0572455A1 Substituted pyridinones and pyrimidinones as angiotensin ii antagonists |
12/08/1993 | CN1079222A Pharmaceutical composition containing quinoline and quinazoline derivatives and novel compounds therefor |
12/07/1993 | US5268481 3-7-diheterabicyclo (3.3.1)nonanes and derivatives as antiarrhythmic agents |
12/07/1993 | US5268470 Reacting a spiro quaternary amine with a secondary amine |
12/07/1993 | US5268377 Imidazoindolizine derivatives process for preparation thereof and use thereof to treat hypertension |
12/07/1993 | US5268376 Containing alkoxy substitution |
12/06/1993 | CA2097731A1 Antitumoral compounds |
12/04/1993 | CA2097460A1 Angiotensin ii antagonists |
12/02/1993 | DE4217719A1 Zweifach heterocyclisch substituierte Sulfonylamino(thio)carbonylverbindungen Dual heterocyclic-substituted sulfonyl amino (thio) carbonyl compounds |
12/01/1993 | EP0572259A1 Aminoquinolone derivatives as anti-HIV agents |
12/01/1993 | EP0572235A2 Beta-carboline derivatives with anticholecystoquinine activity |
12/01/1993 | EP0422154B1 Therapeutic use of 5-ht3 receptor antagonists |
12/01/1993 | CN1078969A Condensed heterocyclic ketone derivatives, their production and use |
11/30/1993 | US5266699 Near infrared radiation absorbers; optical recording media |
11/30/1993 | US5266698 Certain aryl and cycloalkyl fused imidazopyrazinediones; a new class of GABA brain receptor ligands |
11/30/1993 | US5266576 N-myristoyl transferase inhibitors |
11/30/1993 | US5266575 2-ethyl 1H-imidazo[4,5-ciquinolin-4-amines |
11/30/1993 | US5266569 Azatricyclo carboxylic acids useful as anti-bacterial agents |
11/30/1993 | CA1324793C 17-aza derivatives of 20, 21-dinoreburnamenine, process for their preparation and their intermediates, their application as medecines and compositions containing them |
11/29/1993 | CA2097112A1 .beta.-carboline derivative |
11/28/1993 | CA2096998A1 Aryl group- or aromatic heterocyclic group-substituted aminoquinolone derivatives and anti-hiv agent |
11/25/1993 | WO1993023400A1 Pentacyclic antihistamines |
11/25/1993 | WO1993023399A1 6-AMINO SUBSTITUTED IMIDAZO[4,5-b]PYRIDINES AS ANGIOTENSIN II ANTAGONISTS |
11/25/1993 | WO1993023398A1 Substituted pyrido[1,2-a]pyrimidinone derivatives as fungicides |
11/25/1993 | WO1993023397A1 4-mercaptoacetylamino-[2] benzazepinone(3) derivatives, and use as enkephalinase inhibitors |
11/25/1993 | WO1993023396A1 Fused imidazole and triazole derivatives as 5-ht1 receptor agonists |
11/25/1993 | WO1993023391A1 Substituted indoles and azaindoles as angiotensin ii antagonists |
11/25/1993 | WO1993023036A1 Optically active condensed pyrazole compound for use in treating thrombocytopenia and erythropenia |
11/25/1993 | CA2136228A1 Use for treating thrombocytopenia, use for treating erythropenia and optically active fused pyrazole compound |
11/25/1993 | CA2135605A1 Substituted indoles and azaindoles as angiotensin ii antagonists |
11/25/1993 | CA2135188A1 6-amino substituted imidazo(4,5-b)pyridines as angiotensin ii antagonists |
11/25/1993 | CA2134986A1 Fused imidazole and triazole derivatives as 5-htl receptor agonists |
11/24/1993 | EP0570575A1 Bicycloazamacrocyclophosphonic acid, conjugates, contrast agents and preparation |
11/23/1993 | US5264576 Pyrazolo[4,3-c]pyridines which are intermediates |
11/23/1993 | US5264575 Reacting 1,3-benzodiazocine-8-ol derivative with lutidine/2,6-/, triisoproylsilyltrifluoro methane, formed intermediate reacted with lithium chloride, tetrabutylammonium fluoride and isocyanate |
11/23/1993 | US5264439 Quinazolinone, triazolinone and pyrimidinone angiotensin II antagonists incorporating a substituted benzyl element |
11/23/1993 | US5264437 Antiinflammatory agents, immunosuppressants or antiallergens |
11/18/1993 | EP0569794A1 Biphenylmethyl-substituted pyridones useful as angiotensin II receptor antagonists. |
11/18/1993 | EP0569387A1 Resolution of trans-2-(2-pyrimidinyl)-7-(hydroxymethyl)octahydro-2h-pyrido 1,2-a]pyrazine. |
11/17/1993 | CN1078471A Pharmaceuticals |
11/17/1993 | CN1078470A Optionally substituted pyrido |2,3-d¨ pyrimidine-2,4(1H,3H)-diones and pyrido |2,3-d¨ pyrimidine-2(1H,3H)-ones |
11/17/1993 | CN1078469A Substituted indole, azaindole and tetrahydro-1H-pyrrol pyrrolo |2,3-c¨ pyridin-7-one derivatives |
11/16/1993 | US5262537 Treatment of nausea and vomiting |
11/16/1993 | US5262526 Fluorescent compound, complex, reagent, and specific binding assay employing said reagent |
11/16/1993 | US5262426 Treatment of cardiovascular disorders, antiinflammatory agents |
11/16/1993 | US5262417 Antibacterial quinolone compounds |
11/16/1993 | US5262387 Pyridine derivatives and their use for controlling undesirable plant growth |
11/16/1993 | US5262384 Pyridine derivatives and their use for controlling undesirable plant growth |
11/16/1993 | CA1324382C Isoxazole-.beta.-carboline derivatives |
11/16/1993 | CA1324381C Aryl-substituted naphthyridine and pyridopyrazine derivatives |
11/16/1993 | CA1324378C Perhydroazacycloalka [1,2-a] imidazole derivatives and use thereof as nootropic agents |
11/13/1993 | CA2095802A1 Biphenylmethyl-substituted pyridones |
11/11/1993 | WO1993023405A1 Use of tricyclic pyrimidine derivatives as anti-viral medicaments |
11/11/1993 | WO1993022316A1 Process for preparing 10-deazaaminopterins and 5,10- and 8,10-dideazaaminopterins from pteroic dicarboxylic acid diesters |
11/11/1993 | WO1993022314A1 Certain aryl and cycloalkyl fused imidazopyrazinediones; a new class of gaba brain receptor ligands |
11/11/1993 | WO1993022313A1 Tricyclic compound having antiallergic effect |