Patents
Patents for C07D 471 - Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups (64,559)
06/2004
06/24/2004CA2507607A1 Heterocyclic compounds, preparation method thereof and use of same as medicaments, such as anti-bacterial medicaments and beta-lactamaseinhibitors
06/24/2004CA2505887A1 Pyrazole and imidazole compounds and uses thereof
06/23/2004EP1430058A1 Sodium salt of an hiv integrase inhibitor
06/23/2004EP1430053A1 Chemical compounds
06/23/2004EP1430052A2 Substituted imidazo 1, 2-a]-5, 6, 7,8-tetrahydropyridine-8-ones, method for their production and the use thereof for producing imidazo 1, 2-a]pyridines
06/23/2004EP1430050A1 Piperidine derivatives and their use as modulators of chemokine (especially ccr3) activity
06/23/2004EP1429763A2 NOVEL LIGANDS FOR THE HisB10 Zn2+ SITES OF THE R-STATE INSULIN HEXAMER
06/23/2004EP1429759A2 Compounds useful for treating hepatitus c virus
06/23/2004CN1507447A Substituted pyrazolopyrimidines and thiazolopyrimidines used as analgesics
06/23/2004CN1154648C Stable crystal salt of 5-methyl tetrahydrofolic acid
06/23/2004CN1154647C Imidazonephthyridines and their use in inducing cytokine biosynthesis
06/23/2004CN1154646C Benzisozazoles and phenones as alpha antagonist
06/22/2004US6753430 Optically active quinoline carboxylic acid derivatives with 7-pyrrolidine substituents causing optical activity and a process for the preparation thereof
06/22/2004US6753429 1,4-disubstituted benzenes as insecticides
06/22/2004US6753427 2,6-disubstituted 7-oxopyrido(2,3-d)pyrimidines; inhibitors of protein kinases; treating diseases mediated by the pro-inflammatory cytokines, e.g., tumor necrosis factor, inter-leukins, cycloxygenase; chronic obstructive pulmonary disease
06/22/2004US6753333 Arginine salt forms of s-(-)-9- fluoro-6,7-dihydro 8-(4-hydroxypiperidin-1-yl)-5-methyl-1-oxo-1h,5h-benzo(i,j)quinolizine-2 -carboxylic acid, a process for their preparation and pharmaceutical formulations which are
06/22/2004US6753331 Heterocyclic derivatives which inhibit factor Xa
06/17/2004WO2004050681A2 Kinase modulators
06/17/2004WO2004050658A1 Novel substituted imidazo-pyridinones and imidazo-pyridazeiones, the production and use thereof as medicaments
06/17/2004WO2004050656A1 1,3-dihydroimidazole fused-ring compound
06/17/2004WO2004050651A1 Anilinopyrazole derivatives useful for the treatment of diabetes
06/17/2004WO2004050650A1 Anilinopyrazole derivatives useful for the treatment of diabetes
06/17/2004WO2004050629A2 The use of 4-phenyl substituted tetrahydroisoquinolines in the treatment of pain, migraine and urinary incontinence
06/17/2004WO2004050623A1 Methods for preparing phenylalkyne derivatives
06/17/2004WO2004050610A2 Modulators of melanocortin receptor
06/17/2004WO2004050036A2 Quinolines and nitrogenated derivatives thereof and their use as antibacterial agents
06/17/2004WO2004050035A2 Benzimidazoles and analogs thereof as antivirals
06/17/2004WO2004018414A3 Antibacterial agents
06/17/2004WO2004014869A3 5,6-fused 3,4-dihydropyrimidine-2-one derivatives as matrix metalloproteinase inhibitors
06/17/2004US20040116706 Therapeutic ureas
06/17/2004US20040116698 6-Substituted pyrido-pyrimidines
06/17/2004US20040116697 Novel compounds
06/17/2004US20040116509 Antiviral agent; reducing the activity of viral polymerase; 3-(4-Chloro-2,5-dimethyl-benzenesulfonylamino)-5-(4-chloro-phenyl)-thiophene-2-carboxylic acid for example
06/17/2004US20040116499 treatment of inflammatory or proliferative diseases of the skin and other organ systems; from yeast of the genus Malassezia; for example, 2,3-dihydro-4,5-bis(indol-3-yl)furan-2,3-dione; against multiresistent staphylococci
06/17/2004US20040116493 Anti-helicobacterial agents
06/17/2004US20040116474 Novel pyrazole compounds as transforming growth factor (TGF) inhibitors
06/17/2004US20040116473 useful in the treatment of TGF- beta related disease states including, for example, cancer and fibrotic diseases
06/17/2004US20040116467 Hexahydro-benzimidazolone compounds useful as anti-inflammatory agents
06/17/2004US20040116466 Phenyl-aza-benzimidazole compounds for modulating IgE and inhibiting cellular proliferation
06/17/2004US20040116465 Novel compounds
06/17/2004US20040116463 excellent in stability than amorphous one and are more preferable for treatment of hyperlipidemia and atherosclerosis
06/17/2004US20040116462 Antiinflammatory agents
06/17/2004US20040116461 Immunomodulatory compounds
06/17/2004US20040116458 Chemical compounds
06/17/2004US20040116457 Agents for improving excretory potency of urinary bladder
06/17/2004US20040116454 Pyrazole compounds useful as protein kinase inhibitors
06/17/2004US20040116443 Dopamine D4 ligands for the treatment of novelty-seeking disorders
06/17/2004US20040116438 Compositions for treatment of cell proliferation disorders
06/17/2004US20040116429 5-Phenylpyrimidines, methods and intermediate products for the production thereof and use of the same for controlling pathogenic fungi
06/17/2004US20040116425 Prenylation inhibitors and methods of their synthesis and use
06/17/2004US20040116410 Diazepinones as antiviral agents
06/17/2004US20040116399 for preventing or treating coagulation disorders
06/17/2004US20040116388 triazine compoound inhibitors of enzymes that catalyze phosphoryl transfer and/or that bind ATP/GTP nucleotides
06/17/2004US20040116328 Condensed imidazole derivatives
06/17/2004DE10256405A1 New 4-substituted quinoline derivatives, useful for treating bacterial infections, optionally including additional ring nitrogens
06/17/2004DE10247233A1 New 4-substituted quinoline derivatives, useful for treating bacterial infections, optionally including additional ring nitrogens
06/17/2004CA2508914A1 Modulators of melanocortin receptor
06/17/2004CA2508311A1 The use of 4-phenyl substituted tetrahydroisoquinolines in the treatment of pain, migraine and urinary incontinence
06/17/2004CA2507875A1 Methods for preparing phenylalkyne derivatives
06/17/2004CA2507763A1 Fused 1,3-dihydro-imidazole ring compounds
06/17/2004CA2507186A1 Anilinopyrazole derivatives useful for the treatment of diabetes
06/17/2004CA2506546A1 Kinase modulators
06/16/2004EP1428531A1 Oxyiminoalkanoic acid derivatives with hypoglycemic and hypolipidemic activity
06/16/2004EP1427729A1 Carbazole derivatives and their use as npy5 receptor antagonists
06/16/2004EP1427726A1 Process for preparing 5-sulfonamido-8-hydroxy-1, 6-naphthyridine-7-carboxamides
06/16/2004EP1427707A1 Substituted indazole compounds for the treatment of inflammation
06/16/2004EP1427706A1 Substituted pyrazolo compounds for the treatment of inflammation
06/16/2004EP1427421A1 2,4-disubstituted pyrimidinyl derivatives for use as anticancer agents
06/16/2004EP1427415A1 Lactam-containing compounds and derivatives thereof as factor xa inhibitors
06/16/2004EP1427414A1 Inhalation compositions comprising tricyclic 5,6-dihydro-9h-pyrazolo (3,4-c)-1,2,4-triazolo (4,3-alpha) pyridines
06/16/2004EP1427413A2 2-aroylimidazole compounds for treating cancer
06/16/2004EP1427411A2 (-)-1-(3,4-dichlorophenyl)-3-azabicyclo 3.1.0]hexane, compositions thereof, and uses as a dopamine-reuptake inhibitor
06/16/2004EP1427408A2 CYCLIC HYDROXAMIC ACIDS AS INHIBITORS OF MATRIX METALLOPROTEINASES AND/OR TNF-$g(a) CONVERTING ENZYME (TACE)
06/16/2004EP1427287A1 Pesticidal and parasitical di-and trifluorosubstituted alkene compounds
06/16/2004EP1196418B1 METHOD FOR PREPARING SUBSTITUTED 1,4]DIAZEPINO 6,7,1- i hi /i ]INDOL-4-ONES
06/16/2004EP1147083B1 Arylpiperazinyl-cyclohexyl indole derivatives for the treatment of depression
06/16/2004EP1109810B1 Benzonaphthyridine-n-oxides comprising a pde3 and pde4 inhibiting activity
06/16/2004EP0807105B1 Pyridopyrimidones, quinolines and fused n-heretocycles as bradykinin antagonists
06/16/2004CN1505630A Pyrazolo[1,5-a]pyridines and medicaments containing thereof
06/16/2004CN1505607A Peptide-deformylase inhibitors
06/16/2004CN1505514A Combinations of aldose reductase inhibitors and cyclooxygenase-2 inhibitors
06/16/2004CN1505511A Use of pyridoindolone derivatives for preparing medicines
06/16/2004CN1505510A Medicine combinations using pyridoindolone derivatives and anticancer agent as base
06/16/2004CN1505509A Method for treating allergies using substituted pyrazoles
06/16/2004CN1153770C Substitued nitrogen heterocyclic ring as inhibitors of P38 protein kinase
06/15/2004US6750348 Protective effects against infection by hiv through binding to chemokine receptors, including cxcr4 and ccr5;n-(2-pyridinylmethyl)-n'-(2-(phenylureido)ethyl)-n'-(5,6,7,8-tetrahydro-8-quinolinyl)-1,4-benzenedimethanamine
06/15/2004US6750341 Preparation of risperidone
06/15/2004US6750241 Two or more ligand moieties covalently linked together by one or more linking groups enabling binding to multiple binding sites; increased efficacy, selectivity and duration; anti-proliferative and anticarcinogenic
06/15/2004US6750228 Uncontrolled breakdown of connective tissue by metalloproteases is a feature of many pathological conditions
06/15/2004US6750225 Anticoagulants
06/15/2004US6750220 Amine salt of an integrin receptor antagonist
06/15/2004US6750214 Quinoline and quinazoline compounds useful in therapy
06/15/2004US6750005 Reagent system and method for increasing the luminescence of lanthanide(III) macrocyclic complexes
06/15/2004US6749978 Electrophotographic organophotoreceptors with novel charge transport compounds
06/15/2004CA2183735C Hetero-annulated indazoles
06/10/2004WO2004048378A1 Pyrazoloquinolines with immunomodulating activity
06/10/2004WO2004048377A2 Method of preparing inhibitors of phosphodiesterase-4
06/10/2004WO2004048376A1 Bicyclic naphthylidine nucleosides
06/10/2004WO2004048375A1 Novel vitronectin receptor antagonist derivatives, method for preparing same, use thereof as medicines and pharmaceutical compositions containing same
06/10/2004WO2004048374A1 4-oxo-1-(3-substituted phenyl-1,4-dihydro-1,8-naphthyridine-3-carboxamide phosphodiesterase-4 inhibitors