Patents
Patents for C07D 471 - Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups (64,559)
08/2004
08/12/2004US20040156788 Delivery of erectile dysfunction drugs through an inhalation route
08/12/2004CA2514656A1 5ht7 antagonists and inverse agonists
08/12/2004CA2514612A1 2,4-diaminopyrimidine derivatives useful as inhibitors of pkc-theta
08/12/2004CA2513141A1 Hiv-integrase inhibitors, pharmaceutical compositions, and methods for their use
08/11/2004EP1445252A1 Sulphonamide derivatives, the preparation thereof and the application of same as medicaments
08/11/2004EP1444232A1 Phenyl substituted triazoles and their use as selective inhibors of akl5 kinase
08/11/2004EP1444231A1 Amine salts of an integrin receptor antagonist
08/11/2004EP1444228A2 Substituted heteroarylalkanoic acids and their use as aldose reductase inhibitors
08/11/2004EP1444227A1 Thiazolyl substituted triazoles as alk5 inhibitors
08/11/2004EP1444210A1 Qunazoline derivatives as antitumor agents
08/11/2004EP1444209A2 Mitotic kinesin inhibitors
08/11/2004EP1444207A2 Substituted pyrazolyl-compounds for the treatment of inflammation
08/11/2004EP1443927A2 Carboline derivatives as inhibitors of ikb in the treatment of multiple myeloma and other cancers
08/11/2004EP1443925A1 Naphthyridine derivatives, their preparation and their use as phosphodiesterase isoenzyme 4 (pde4) inhibitors
08/11/2004EP1443916A1 Pharmaceutical composition comprising an adenosine a1/a2 agonist and a sodium hydrogen exchanger inhibitor
08/11/2004EP1334092A4 Process for preparation of bicyclic and polycyclic molecules
08/11/2004EP1109813B1 Pyrroloindoles, pyridoindoles and azepinoindoles as 5-ht2c agonists
08/11/2004EP1042294B1 Heterocyclic cytotoxic agents
08/11/2004CN1520414A Novel compound, its prepn. and application
08/11/2004CN1520413A Technical synthesis method for producing tropenol
08/11/2004CN1520412A New derivatives of oxazolidinones as antibacterial agents
08/11/2004CN1520409A Piperazine oxime derivatives having Nk-1 receptor antagonistic activity
08/11/2004CN1520295A Indole, azaindole and related heterocyclic amidopiperazine derivatives
08/11/2004CN1520293A 3-flworo-pyrrolidines as antidiabetic agents
08/11/2004CN1519240A Substituted nitrogen contg. heterocycles as inhibitors of P38 progein kinase
08/11/2004CN1519239A Ramification of a compound of medication as well as preparation method and application
08/11/2004CN1161355C New compounds
08/11/2004CN1161341C Fused pydiopyridazine inhibitors of cGMP phosphodiesterase
08/11/2004CN1161334C Nitrogen-containing tegracyclic compounds
08/10/2004US6774237 Vascular endothelial growth factor receptor tyrosine kinases inhibitors; angiogenesis inhibitors, anticarcinogenic agents
08/10/2004US6774236 Process for the preparation of enantiomerically pure cycloalkano-indol -and azaindol -and pyrimido [1,2A]indolcarbocyclic acids and their activated derivatives
08/10/2004US6774230 Such as 1-(3-carboxypyridyl-2)-4-methyl-2- phenylpiperazine dihydrate; antidepressants
08/10/2004US6774229 Coupling condensation synthesis of heterocycles
08/10/2004US6774134 For therapy of respiratory syncytial virus infection
08/10/2004US6774133 Substituted spiroheterocyclic 1H-3-aryl-pyrrolidine-2,4-dione derivatives, processes for their preparation, and their use as pesticides
08/10/2004US6774132 Spirooxindole derivatives that act as analgesics
08/10/2004CA2134566C 1-piperazino-1,2-dihydroindene derivatives
08/10/2004CA2124999C Loracarbef isopropanolate and a process for converting loracarbef isopropanolate to loracarbef monohydrate
08/05/2004WO2004065520A1 Light-emitting device, condensed polycyclic compound used therein and method for producing same
08/05/2004WO2004064778A2 3-amino-4-phenylbutanoic acid derivatives as dipeptidyl peptidase inhibitors for the treatment or prevention of diabetes
08/05/2004WO2004064764A2 Substituted alkyl amido piperidines
08/05/2004WO2004064741A2 Compounds, compositions, and methods
08/05/2004WO2004043925A3 3-substituted-6-aryl pyridined as ligands of c5a receptors
08/05/2004WO2004043389A3 Methods of treating cancer and related methods
08/05/2004WO2004032861A3 Hexahydro-benzimidazolone compounds useful as anti-inflammatory agents
08/05/2004WO2004026867A3 Imidazopyridines as cyclin dependent kinase inhibitors
08/05/2004WO2003103590A3 (halo-benzo carbonyl)heterobicyclic p38 kinase inhibiting agents
08/05/2004WO2003101953A3 Triazaspiro compounds useful for treating or preventing pain
08/05/2004WO2003086319A3 Pharmaceutical compositions containing an hiv integrase inhibitor and a nonionic surfactant
08/05/2004WO2003059289A3 Melanin concentrating hormone receptor ligands: substituted benzoimidazole analogues
08/05/2004WO2002102976A3 Mutations in the bcr-abl tyrosine kinase associated with resistance to sti-571
08/05/2004WO2002066435B1 Metal complexes and therapeutic uses thereof
08/05/2004US20040152897 Synthesis of indolizines
08/05/2004US20040152739 Bone disorders; cardiovascular disorders; gastrointestinal disorders; angiogenesis inhibitors; metabolism disorders; central nervous system disorders; traumas; skin disorders; inflammatory bowel disorders; anticancer agents
08/05/2004US20040152738 Wound healing agents; antiarthritic agents; osteoporosis; congestive heart failure; antiulcer agents; Alzheimer's disease; anticholesterol agents; antiarthritic agents
08/05/2004US20040152730 Novel compounds
08/05/2004US20040152726 Quinoline-4-carboxamide derivatives as nk-3 and nk-2 receptor antagonists
08/05/2004US20040152724 Analgesics; anticholinergic agents; Alzheimer's and Parkinson's disease; attention deficit hydroactivity; antidepressants; schizophrenia
08/05/2004US20040152707 Analgesics; anxiolytic agents; antihistamines; antitussive agents; antidepressants; alcoholism
08/05/2004US20040152705 Pyrazino 1',2':1,6 pyrido 3,4-b indole1,4-dione derivatives
08/05/2004US20040152704 Bicyclic-substituted amines as histamine-3 receptor ligands
08/05/2004US20040152697 Pyrrolidin-2-one derivatives as inhibitors of factor xa
08/05/2004US20040152690 Analgesics; neuropathic pain; antiinflamamtory agents; oral diseases; headaches; antiarthritic agents; vision disorders; skin disorders; inflammatory bowel disorders; benzimidazole compounds
08/05/2004US20040152686 Metal complexes and therapeutic uses thereof
08/05/2004US20040152659 For therapy and prophylaxis of Parkinson's disease and symptoms associating therewith such as anxiety, depression and/or memory disorder which contain as the active ingredient an adenosine A1A2a receptor dual antagonist or salts thereof
08/05/2004US20040151945 Binaphthol based chromophores for the fabrication of blue organic light emitting diodes
08/05/2004CA2512546A1 3-amino-4-phenylbutanoic acid derivatives as dipeptidyl peptidase inhibitors for the treatment or prevention of diabetes
08/05/2004CA2509456A1 Substituted alkyl amido piperidines
08/04/2004EP1442137A2 Universal nucleotides for nucleic acid analysis
08/04/2004EP1442133A2 Methods for improving the treatment of major depression by genotyping for the gene for apolipoproteine e4
08/04/2004EP1442041A1 Azabicyclic-substituted-heteroaryl compounds for the treatment of disease
08/04/2004EP1442040A1 Bridged bicycle (1,4) benzodiazepine vasopressin receptor antagonists
08/04/2004EP1442015A1 Use of 2-acylindoles in the treatment of tumors
08/04/2004EP1441734A1 Dihydroxypyrimidine carboxamide inhibitors of hiv integrase
08/04/2004EP1441728A2 Modulators of the cholesterol biosynthetic pathway
08/04/2004EP1441725A1 Benzimidazoles and analogues and their use as protein kinases inhibitors
08/04/2004EP1441719A1 N-substituted pyrrolidin derivatives as dipeptidyl peptidase iv inhibitors
08/04/2004EP1317455B1 Process for preparing a substituted imidazopyridine compound
08/04/2004EP1077957B1 Oxyiminoalkanoic acid derivatives with hypoglycemic and hypolipidemic activity
08/04/2004EP1064256B1 Bicyclo [2.2.1] heptanes and related compounds
08/04/2004EP0912571B1 Naphthyridines which affect il-4 and g-csf
08/04/2004EP0842933B1 Novel naphthyridine derivatives
08/04/2004CN1518551A Triazaspiro [5,5] undecane derivatrives and drugs containing the same as active ingredient
08/04/2004CN1518550A Imidazo [1,2-A] pyridine derivatives for prophylaxis and treatment of herpes viral infections
08/04/2004CN1518541A Phenyl derivatives
08/04/2004CN1518534A Copper-catalyzed formation of carbon-heteroatom and carbon-carbon bonds
08/04/2004CN1518447A Synthesis and evaluation of novel phthalimide mimics as anti-angiogenic agents
08/04/2004CN1160353C Prepn. of 8-cyclopentyl-6-ethyl-3-[substituted]-5,8-dihydro-4H-1,2,3A,7,8-pentaaza-asymmetric indacene
08/04/2004CN1160352C Three-site substituted beta-carboline novel compound having anti-HIV and anti-cancer activity, preparation method and its composition and use
08/04/2004CN1160074C Aqueous suspensions of submicron 9-hydroxyrisperidone fatty acid esters
08/03/2004US6770666 Fused-ring compounds and use thereof as drugs
08/03/2004US6770664 Bicyclic heterocyclic substituted phenyl oxazolidinone antibacterials, and related compositions and methods
08/03/2004US6770655 2-imidazomethyl- pyrido(4,3-b)indol-1-one or -carbazol-1-one derivatives containing an ester group; especially for treating irritable bowel syndrome.
08/03/2004US6770647 Osteoporosis; rheumatic diseases
08/03/2004US6770643 Inhibit protein kinases
08/03/2004US6770642 For use in treatment of cns disorders such as anxiety, depression, epilepsy, obsessive compulsive disorder, attention deficit disorder, migraine, cognitive memory enhancement, alzheimer's disease
08/03/2004US6770641 Fused heteroaryl derivatives
08/03/2004US6770639 Cell proliferative; autoimmune diseases; antiallergens; antiinflammatory agents; anticancer agents
08/03/2004CA2136836C Piperidinyl-terminated n-(dihydroxy alkyl)-ethynyl-alanine amides for treatment of hypertension
07/2004
07/29/2004WO2004063330A2 (2-carboxamido) (3-amino) thiophene compounds