Patents
Patents for C07D 471 - Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups (64,559)
09/2004
09/21/2004US6794391 Inhibitors of phosphodiesterase (pde) isoenzymes; useful for treatment of respiratory disorders such as asthma.
09/21/2004US6794388 Succinic acid salts of 5,7,14-triazatetracyclo[10.3.1.02,11.04,9] -hexadeca-1(11),3,5,7,9-pentaene and pharmaceutical compositions thereof
09/21/2004US6794382 Benzimidazole derivatives, preparation and therapeutic use thereof
09/21/2004US6794379 Antiinflammatory agents; autoimmune disease; skin disorders
09/21/2004US6793839 Forming methylene bridges between glycoluril units; attaining oligimers with up to twelve units at high yield
09/21/2004CA2280587C Growth hormone secretagogues
09/21/2004CA2155843C Novel urea derivatives, their preparation and use
09/21/2004CA2114017C Amide tetrazole acat inhibitors
09/21/2004CA2033143C Alkyl esters of 5-heterocyclic-pyridine-2,3-dicarboxylate acids, 5-heterocyclic 2-(2-imidazoline-2-yl)pyridines, useful as herbicidal agents and methods for the preparation thereof
09/16/2004WO2004078943A2 Alternative heterocycles for dna recognition
09/16/2004WO2004078759A1 Substituted 2-(diaza-bicyclo-alkyl)-pyrimidone derivatives
09/16/2004WO2004078758A1 Novel fused heterocycles and uses thereof
09/16/2004WO2004078757A2 Synthesis of 5-substituted 7-azaindoles and 7-azaidonines
09/16/2004WO2004078756A2 Jnk inhibitors
09/16/2004WO2004078755A1 Substituted pyrido(1,2-a)pyrimidines and their use as nos inhibitors
09/16/2004WO2004078733A1 Quinazolines useful as modulators of ion channels
09/16/2004WO2004078731A1 Quinoline-carboxylic acids and the derivatives thereof, a focused library
09/16/2004WO2004078717A1 Acylated piperazine derivatives as melanocortin-4 receptor agonists
09/16/2004WO2004078716A1 Acylated piperazine derivatives as melanocortin-4 receptor agonists
09/16/2004WO2004078712A2 Isoquinoline derivatives and methods of use thereof
09/16/2004WO2004078682A2 Cyclic compounds and compositions as protein kinase inhibitors
09/16/2004WO2004078116A2 P38 inhibitors and methods of use thereof
09/16/2004WO2004078110A2 Fused imizadoles as transforming growth factor (tgf) inhibitors
09/16/2004WO2004078109A2 PROCESS FOR SYNTHESISING USEFUL INTERMEDIATES FOR THE PREPARATION OF ανβ3 RECEPTOR ANTAGONISTS
09/16/2004WO2004071445A3 2-(aminomethyl)arylamide analgesics
09/16/2004WO2004069782A3 2-aryl-acetic acids, their derivatives and pharmaceutical compositions containing them
09/16/2004WO2004058176A3 Acyclic pyrazole compounds
09/16/2004WO2004043389B1 Methods of treating cancer and related methods
09/16/2004WO2004039803A3 Hiv-integrase inhibitors, pharmaceutical compositions, and methods for their use
09/16/2004WO2004028459A3 Piperidine derivatives
09/16/2004WO2003092586A3 Tetrahydropyranyl cyclopentyl tetrahydropyridopyridine modulators of chemokine receptor activity
09/16/2004WO2003072553A8 N-aryl-2-oxazolidinone-5-carboxamides and their derivates and their use as antibacterials
09/16/2004WO2003028729A3 Prodrugs of substituted polycyclic compounds useful for selective inhibition of the coagulation cascade
09/16/2004US20040181075 Process of making chalcone derivatives
09/16/2004US20040181064 Bicyclic modulators of androgen receptor function
09/16/2004US20040181059 Aryl or heteroaryl fused imidazole compounds as anti-inflammatory and analgesic agents
09/16/2004US20040180947 Sulfonamide compounds and pharmaceutical use thereof
09/16/2004US20040180934 Dihydropyrrolo[1,2-a]indole and tetrahydropyrido[1,2-a]-indole derivatives as prostaglandin d2 receptor antagonists
09/16/2004US20040180923 obesity, diabetes, male sexual dysfunction, and female sexual dysfunction
09/16/2004US20040180921 Nitrogen compounds such as 2-benzofuran-2-yl-imidazo(1,2-a) pyridine administered as g protein coupled receptor antagonists for prophylaxis of psychological and neurodegenerative disorders, and as analgesics
09/16/2004US20040180920 Pyrano[2,3-C]imidazo[-1,2-A]pyridine derivatives for the treatment of gastrointestinal disorders
09/16/2004US20040180917 Novel tricyclic dihydro-quinoline derivatives, method for preparing same and pharmaceutical compositions containing the same
09/16/2004US20040180910 Heterocycle carboxamides as antiviral agents
09/16/2004US20040180897 anticarcinogenic agents
09/16/2004US20040180896 P38 inhibitors and methods of use thereof
09/16/2004US20040180887 N-aroyl cyclic amine derivatives as orexin receptor antagonists
09/16/2004US20040180877 Nicotinic acetylcholine receptor cholinergic ligands, monoamine receptor and transporter modulators; such as 1-(2-Benzo[b]thiophenyl-1,1-dioxide)-imidazolidine
09/16/2004US20040180875 Obesity, anorexia, bulemia, depression, anxiety, psychosis, schizophrenia, migraine, addictive behavior, obsessive-compulsive disorder, sexual disorders
09/16/2004US20040180234 Electroluminescent devices
09/16/2004DE10310106A1 Substituierte Pyridot [1,2-a]pyrimidin-Verbindungen Substituted Pyridot [1,2-a] pyrimidine compounds
09/16/2004DE10309927A1 New trisubstituted dihydro-imidazo-pyridazinone or imidazo-pyridinone derivatives, useful as dipeptidylpeptidase-IV inhibitors for e.g. treating diabetes mellitus type I or II, arthritis or obesity
09/16/2004CA2517844A1 Quinazolines useful as modulators of ion channels
09/16/2004CA2517358A1 Isoquinoline derivatives and methods of use thereof
09/15/2004EP1457490A1 5-membered N-heterocyclic compounds with hypoglycemic and hypolipidemic activity
09/15/2004EP1457488A1 Intermediates for use in the preparation of urea compounds having muscarinic receptor antagonist activity
09/15/2004EP1457199A1 Coupling agents having a 2,3,5-triaminopyridine structure and their use for dyeing keratinic fibres
09/15/2004EP1456208A1 Pyridoquinoxaline antivirals
09/15/2004EP1456207A2 Heterocyclic acridone inhibitors of impdh enzyme
09/15/2004EP1456206A1 Azaindolylalkylamine derivatives as 5-hydroxytryptamine-6 ligands
09/15/2004EP1456205A1 Imidazoquinoline derivatives
09/15/2004EP1456204A1 Triazolo-quinolin derivatives useful as adenosine receptor ligands
09/15/2004EP1455792A1 Ureas of 2-aminobenzothiazoles as adenosine modulators
09/15/2004EP1455779A1 Indolylalkylamine derivatives as 5-hydroxytryptamine-6 ligands
09/15/2004EP1455700A2 Methods and compositions related to irm compounds and toll-like receptor pathways
09/15/2004EP1202992B1 Ascididemin derivatives and their therapeutic applications
09/15/2004EP1196408B1 Respiratory syncytial virus replication inhibitors
09/15/2004EP1173440B1 Tetracyclic azepinoindole compounds as 5-ht receptor ligands
09/15/2004EP0986384A4 Inhibitors of protein isoprenyl transferases
09/15/2004CN1529705A Tri-and tetraaza-acenaphthylen derivatives as CRF receptor antagonists
09/15/2004CN1529704A 3-(4-amidopyrrol-2-2ylmethlidene)-2-indolinone derivatives as protein kinase inhibitors
09/15/2004CN1529597A Imidazo (1,2-A)_pyridine derivatives as mGLUR5 antagonists
09/15/2004CN1166668C Method for preparing substituted [1,4] diazepino (6,7,1-hi) indol-4-ones
09/15/2004CN1166666C Fused imiazole compounds and remedies for diabetes mellitus
09/15/2004CN1166640C Substituted 1,2,3,4,5,6-hyxahydro-2,6-methano-3-benzazocine-10-oles, method for production and use thereof as medicaments
09/15/2004CN1166636C Arylpiperazinyl-cyclohexyl indole derivatives for the treatment of depression
09/14/2004US6790961 Reacting a 3-amino-4-(substituted)amino-2-chloroquinoline with an alkylcarbonyl chloride to form the 2-alkylcarboxamide intermediate
09/14/2004US6790960 Compounds
09/14/2004US6790844 Muscle relaxants; antiserotonine agent
09/10/2004WO2004076463A1 Inhibitors
09/10/2004WO2004076457A1 Solvent-free process for the preparation of pyrrolo (3,4c) pyrrole compounds
09/10/2004WO2004076456A1 Solvent-free process for the preparation of diketopyrrolopyrrole derivatives
09/10/2004WO2004076453A1 Novel diazabicyclic aryl derivatives
09/10/2004WO2004076452A1 5,8-DIFLUOROIMIDAZO[1,2-a]PYRIDINES AS GABA-A α2/α3 LIGANDS FOR TREATING ANXIETY AND/OR DEPRESSION
09/10/2004WO2004076451A1 Imidazo[4,5-b]quinoline-derivatives and their use as no-synthase inhibitors
09/10/2004WO2004076450A1 Pyrazolopyridine derivates
09/10/2004WO2004076449A2 3-substituted-2(arylalkyl)-1-azabicycloalkanes and methods of use thereof
09/10/2004WO2004076418A1 Ligands that modulate lxr-type receptors
09/10/2004WO2004076411A2 Aminocyclopentyl fused heterotricylicamide modulators of chemokine receptor activity
09/10/2004WO2004075891A1 1,3-substituted cycloalkyl derivatives containing acidic, mainly heterocyclic groups, corresponding production method and use of said derivatives as medicaments
09/10/2004WO2004075863A2 Cxcr3 antagonists
09/10/2004WO2004056727A8 Process of making chalcone derivatives
09/10/2004WO2004052847A3 Tricyclic steroid hormone nuclear receptor modulators
09/10/2004WO2004047769A3 Benzimidazoles and analogs thereof as antibacterials
09/10/2004WO2004022523A3 1, 3-diamino-2-hydroxypropane prodrug derivatives
09/10/2004WO2004014352A3 Methods for treating carbonic anhydrase mediated disorders
09/10/2004WO2003087092A3 Inhibitors of serine proteases, particularly hepatitis c virus ns3 - ns4 protease
09/10/2004CA2518675A1 Novel diazabicyclic aryl derivatives
09/10/2004CA2517307A1 1,3-substituted cycloalkyl derivatives containing acidic, mainly heterocyclic groups, corresponding production method and use of said derivatives as medicaments
09/10/2004CA2516705A1 Aminocyclopentyl fused heterotricylicamide modulators of chemokine receptor activity
09/10/2004CA2516522A1 Imidazo[4,5-b]quinoline-derivatives and their use as no-synthase inhibitors