Patents
Patents for C07D 417 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group (62,773)
01/2000
01/11/2000US6013651 Meta-azacyclic amino benzoic acid compounds and derivatives thereof
01/11/2000CA2195027C Hiv protease inhibitors useful for the treatment of aids
01/06/2000WO2000000487A1 5-ht1f agonists
01/06/2000WO2000000485A1 Epothilon derivatives, their preparation process, intermediate products and their pharmaceutical use
01/06/2000WO2000000477A1 Non-peptidyl inhibitors of vla-4 dependent cell binding useful in treating inflammatory, autoimmune, and respiratory diseases
01/06/2000WO2000000470A1 Amino acid derivatives and drugs containing the same as the active ingredient
01/06/2000WO2000000465A1 Hydrazine derivatives
01/06/2000WO2000000197A1 4-benzyl piperidine alkylsulfoxide heterocycles and their use as subtype-selective nmda receptor antagonists
01/06/2000WO1999043661A3 Substituted cycloalkyl-4-oxonicotinic carboxamides; gaba brain receptor ligands
01/06/2000CA2336625A1 Non-peptidyl inhibitors of vla-4 dependent cell binding useful in treating inflammatory, autoimmune, and respiratory diseases
01/06/2000CA2336254A1 5-ht1f agonists
01/06/2000CA2336162A1 Amino acid derivatives and pharmaceutical composition comprising, as active ingredients, them
01/06/2000CA2335245A1 Hydrazine derivatives
01/06/2000CA2327888A1 4-benzyl piperidine alkylsulfoxide heterocycles and their use as subtype-selective nmda receptor antagonists
01/05/2000EP0969003A2 Process for the preparation of benzo[f]quinolinone derivatives and intermediates
01/05/2000EP0968209A1 THIAZOLE BENZENESULFONAMIDES AS $g(b) 3? AGONISTS FOR THE TREATMENT OF DIABETES AND OBESITY
01/05/2000EP0968206A1 N-heterocyclic derivatives as nos inhibitors
01/05/2000EP0968194A1 Atropisomers of 3-aryl-4(3h)-quinazolinones and their use as ampa-receptor antagonists
01/05/2000EP0968193A1 Phenylsulphonyl ureas, processes for their preparation and their use as herbicides and plant-growth regulators
01/05/2000EP0968190A1 Substituted isoquinoline derivatives and their use as anticonvulsants
01/05/2000EP0968175A1 Spiro compounds and the use thereof
01/05/2000EP0967980A2 Use of aminothiazoles for treating wounds and skin
01/05/2000EP0666856B1 4-arylmethyloxymethyl piperidines as tachykinin antagonists
01/05/2000EP0539420B1 substituted thiazolyl and substituted pyridinyl derivatives
01/05/2000CN1240446A Insoluble s-triazine derivatives and their use as UV filters
01/05/2000CN1240212A Process for reducing prochiral ketone to produce optically active alcohol of high optical purity
01/04/2000US6011154 Substituted heterocyclic compounds, method of preparing them and pharmaceutical compositions in which they are present
01/04/2000US6011150 Synthetic intermediate of a 1 beta-methylcarbapenem derivative
01/04/2000US6011048 Thiazole benzenesulfonamides as β3 agonists for treatment of diabetes and obesity
01/04/2000US6011039 Aminopyridine derivatives
01/04/2000US6011037 Thiazole derivatives with phosphodiesterase-inhibiting action
01/04/2000US6011036 Heterocyclic compounds having antidiabetic hypolipidemic antihypertensive properties process for their preparation and pharmaceutical compositions containing them
01/04/2000US6011033 Phenylene derivatives
01/04/2000US6011032 Heterocyclic compounds for treating myocardial ischemia
01/04/2000US6011031 Azolidinediones useful for the treatment of diabetes, dyslipidemia and hypertension: process for their preparation and pharmaceutical compositions containing them
01/04/2000US6011029 Benzodiazepine compounds
01/04/2000US6011028 Cyclic amidino agents useful as nitric oxide synthase inhibitors
12/1999
12/29/1999WO1999067253A2 Desmethyl epothilones
12/29/1999WO1999067252A2 Epothilone derivatives and their synthesis and use
12/29/1999WO1999067230A1 INHIBITORS OF α4β1 MEDIATED CELL ADHESION
12/29/1999WO1999067221A1 Compounds for inhibiting beta-amyloid peptide release and/or its synthesis
12/29/1999WO1999067220A1 Compounds for inhibiting beta-amyloid peptide release and/or its synthesis
12/29/1999WO1999067219A1 Compounds for inhibiting beta-amyloid peptide release and/or its synthesis
12/29/1999WO1999066944A1 Methods for identifying novel multimeric agents that modulate receptors
12/29/1999WO1999066934A1 CYCLIC AMINO ACID COMPOUNDS, PHARMACEUTICAL COMPOSITIONS COMPRISING SAME, AND METHODS FOR INHIBITING β-AMYLOID PEPTIDE RELEASE AND/OR ITS SYNTHESIS BY USE OF SUCH COMPOUNDS
12/29/1999WO1999066925A1 Protease inhibitors
12/29/1999WO1999054326A8 Dihydropyrimidines
12/29/1999EP0967207A1 Nitrone derivatives, process for their preparation and pharmaceutical compositions containing them
12/29/1999EP0966465A1 Inhibitors of impdh enzyme
12/29/1999EP0966454A1 Disubstituted bicyclic heterocycles, their production and use as medicaments
12/29/1999EP0966452A1 Process for preparing sulphurous 2-chloro-3-(4,5-dihydroisoxazol-3-yl)-benzoic acids
12/29/1999EP0966443A1 Heteroaryl-hexanoic acid amide derivatives, their preparation and their use as selective inhibitors of mip-1-alpha binding to its ccr1 receptor
12/29/1999EP0612314B1 2-pyrazinylethylamine derivatives and their use as pharmaceuticals
12/29/1999CN1239952A 6-phenylpyridyl-2-amine derivatives useful as NOS inhibitors
12/29/1999CN1239941A Aryl or heteroaryl substd. 3, 4-dihydroanthracene and benzo [1,2-g]-chrom-3-ene, benzo [1,2-g]-thiochrom-3-ene and benzo [1,2-g]-1,2-dihydroquinoline derivs.
12/29/1999CN1239889A Novel compounds useful as neuro-protective agents
12/29/1999CA2342778A1 Inhibitors of .alpha.4.beta.1 mediated cell adhesion
12/29/1999CA2335876A1 Protease inhibitors
12/29/1999CA2325389A1 Compounds for inhibiting beta-amyloid peptide release and/or its synthesis
12/29/1999CA2325388A1 Compounds for inhibiting beta-amyloid peptide release and/or its synthesis
12/29/1999CA2324475A1 Cyclic amino acid compounds, pharmaceutical compositions comprising same, and methods for inhibiting .beta.-amyloid peptide release and/or its synthesis by use of such compounds
12/29/1999CA2324474A1 Compounds for inhibiting beta-amyloid peptide release and/or its synthesis
12/29/1999CA2319650A1 Methods for identifying novel multimeric agents that modulate receptors
12/28/1999US6008370 Fungicidal imidazolinone and imidazolinethione compounds for use in plant protection
12/28/1999US6008365 Adrenoreceptor agonists and dopamine da2-receptor agonists, useful in the treatment of obstructive airway diseases
12/28/1999US6008257 Pesticidal composition containing the hydroxamic acid derivatives of given formula; applying to control pests
12/28/1999US6008245 Treatment of prophylaxis and cardiovascular disorders, in particular arrhythmias, for the treatment of ulcers of the gastrointestinal disorders, diarrheal diseases
12/28/1999US6008237 Potent agonists of peroxidsome proliferator activated receptor; for controlling or preventing of diabetes, hyperglycemia, hyperlipidemia, hypercholesterolemia, atherosclerosis, obesity, vascular restenosis
12/28/1999US6008234 Treating a human having a disease-state characterized by thrombotic activity, inhibiting human blood coagulation factor xa
12/28/1999US6008230 Treating bone diseases caused by abnormal bone metabolism in human being or animals as the inhibitors of bone resorption or the inhibitors of bone metastasis
12/26/1999CA2273545A1 Processed lumber material
12/23/1999WO1999065922A2 Prenyl transferase inhibitors
12/23/1999WO1999065913A2 Epothilone minor constituents
12/23/1999WO1999065901A1 1,3-oxazoline and 1,3-thiazoline derivatives, method for producing the same and their use as pesticides
12/23/1999WO1999065898A1 Imidazolyl derivatives
12/23/1999WO1999065897A1 Inhibitors of glycogen synthase kinase 3
12/23/1999WO1999065896A1 Preparation of heteroaryl compounds
12/23/1999WO1999065893A1 Novel benzopyran or thiobenzopyran derivatives
12/23/1999WO1999065884A1 Carbon substituted aminothiazole inhibitors of cyclin dependent kinases
12/23/1999WO1999065882A1 2,4-diamino-1,3,5-triazine, method for the production and use of the same as herbicides and plant growth regulators
12/23/1999WO1999065878A1 Synthesis of benzo[f]quinolinones
12/23/1999WO1999065871A2 Thiolesters and uses thereof
12/23/1999WO1999065870A2 Sulfonamide inhibitors of aspartyl protease
12/23/1999WO1999065867A1 Cyclic hydroxamic acids as metalloproteinase inhibitors
12/23/1999WO1999065487A1 Inhibitors of serotonin reuptake
12/23/1999WO1999055156A3 The use of derivatives of iminotriazole as crop protection agents and novel iminotriazoles
12/23/1999DE19925329A1 New triazine derivatives useful as selective herbicides and plant growth regulators
12/23/1999DE19826988A1 Epothilon-Nebenkomponenten Epothilone secondary components
12/23/1999DE19826671A1 1,3-Oxazolin- und 1,3-Thiazolin-Derivate, Verfahren zu ihrer Herstellung und ihre Verwendung als Schädlingsbekämpfungsmittel 1,3-oxazoline and 1,3-thiazoline derivatives, processes for their preparation and their use as pesticides
12/23/1999CA2337603A1 Prenyl transferase inhibitors
12/23/1999CA2336189A1 Epothilone minor constituents
12/23/1999CA2335464A1 Novel thiolesters and uses thereof
12/23/1999CA2335435A1 Imidazolyl derivatives
12/23/1999CA2335352A1 1,3-oxazoline and 1,3-thiazoline derivatives, their preparation, and their use as pesticides
12/23/1999CA2335327A1 2,4-diamino-1,3,5-triazines, their preparation, and their use as herbicides and plant growth regulators
12/23/1999CA2335322A1 Inhibitors of serotonin reuptake
12/23/1999CA2334701A1 Synthesis of benzo¬f|quinolinones
12/23/1999CA2334677A1 Preparation of heteroaryl compounds
12/23/1999CA2334634A1 Novel benzopyran or thiobenzopyran derivatives
12/23/1999CA2333554A1 Cyclic hydroxamic acids as metalloproteinase inhibitors