Patents
Patents for C07D 417 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group (62,773)
03/2004
03/11/2004US20040048843 And aza- and diaza-derivatives thereof; especially treating allergy or nasal congestion
03/11/2004US20040048797 Regulation of TNF-alpha
03/11/2004US20040048774 Inhibitors of IMPDH enzyme
03/11/2004CA2496580A1 3-(sulfonamidoethyl)-indole derivaties for use as glucocorticoid mimetics in the treatment of inflammatory, allergic and proliferative diseases
03/11/2004CA2495917A1 Oxazolidin-2-one and thiazolidin-2-one derivatives for use as ep4 receptor agonists in the treatment of glaucoma
03/11/2004CA2495914A1 N-biarylmethyl aminocycloalkanecarboxamide derivatives
03/11/2004CA2495248A1 Anabaseine derivatives useful in the treatment of neurodegenerative diseases
03/11/2004CA2494931A1 Hetereoaryl nitrile derivatives
03/11/2004CA2488739A1 Nitrogen-containing aromatic derivatives
03/10/2004EP1396487A1 Phenylpyridine carbonyl piperazine derivative
03/10/2004EP1395606A1 Pyrrolidin-2-one derivatives as inhibitors of factor xa
03/10/2004EP1395578A1 Carbazole derivatives and their use for the preparation of pharmaceutical compositions for the treatment of npy related diseases
03/10/2004EP1395576A1 4-(phenyl-piperidin-4-ylidene-methyl)-benzamide derivatives and their use for the treatment of pain, anxiety or gastrointestinal disorders
03/10/2004EP1395575A1 4-(penyl-piperidin-4-ylidene-methyl)-benzamide derivatives and their use for the treatment of pain, anxiety or gastrointestinal disorders
03/10/2004EP1395574A1 4-(phenyl-piperidin-4-ylidene-methyl)-benzamide derivatives and their use for the treatment of pain, anxiety or gastrointestinal disorders
03/10/2004EP1395571A1 Compounds and methods for the treatment or prevention of flavivirus infections
03/10/2004EP1395565A1 Herbicidal substituted benzoylpyrazoles
03/10/2004EP1395559A1 4-(phenyl-piperidin-4-ylidene-methyl)-benzamide derivatives and their use for the treatment of pain anxiety or gastrointestinal disorders
03/10/2004EP1395558A1 4-(phenyl-(piperidin-4-yl)-amino)-benzamide derivatives and their use for the treatment of pain, anxiety or gastrointestinal disorders
03/10/2004EP1395557A1 4-(phenyl-(piperidin-4-yl)-amino)-benzamide derivatives and their use for the treatment of pain, anxiety or gastrointestinal disorders
03/10/2004EP1395556A1 4-(phenyl-(piperidin-4-yl)-amino)-benzamide derivatives and their use for the treatment of pain, anxiety or gastrointestinal disorders
03/10/2004EP1395555A1 4-(phenyl-(piperidin-4-yl)-amino)-benzamide derativatives and their use for the treatment of pain, anxiety or gastrointestinal disorders
03/10/2004EP1395553A1 Pyrrolidine derivatives as factor xa inhibitors
03/10/2004EP1395251A2 Aminediols as agents for the treatment of alzheimer's disease
03/10/2004CN1481382A Isoindolin-1-one glucokinase activators
03/10/2004CN1481380A Novel benzazepines and related heterocyclic derivatives which are useful as orexin receptor antagonists
03/10/2004CN1481377A Cyclic Beta-amino acid derivatives as inhibitors of matrix metalloproteases and TNF alhpa
03/10/2004CN1481376A Oxybenzamides derivatives as factor xa inhibitors
03/10/2004CN1481373A 1,5-benzothiazepines compounds and its use as antilipemic agent
03/10/2004CN1481372A 1,1-dioxo-2H-1,2-benzothiazine-3-carboxamide derivatives, method for preparing same and pharmaceutical compsns comprising same
03/10/2004CN1481361A Piperidine MCH antagonists and their use in treatment of obesity
03/10/2004CN1481358A Carboxylic acid amide derivatives and their use in treatment of thromboembolic diseases and tumours
03/10/2004CN1480451A Photoactive compound used as intermediate for preparing photoactive 2-imidazoline-5-ketone or 2-imdazoline-5-thio-ketone derivative
03/10/2004CN1141300C Acrylonitrile compounds
03/09/2004US6703503 Pyridazin-3-one derivatives, their use, and intermediates for their production
03/09/2004US6703403 Method for improving pharmacokinetics
03/09/2004US6703388 Dibenzodiazepine derivatives; antihistamines, leukotriene inhibitors, antiallergens, antiasthmatics; hay fever, atopic dermatitis, and urticaria treatment
03/09/2004US6703387 Inhibitors of HPV E1 helicase enzyme
03/09/2004US6703347 Insecticides, fungicides, nematocides, molluscicides, and miticides for plants
03/04/2004WO2004018478A2 Synthesis of epothilones, intermediates thereto, analogues and uses thereof
03/04/2004WO2004018463A2 Pyridyl substituted heterocycles useful for treating or preventing hcv infection
03/04/2004WO2004018461A2 Antibacterial benzoic acid derivatives
03/04/2004WO2004018458A1 2-thio-substituted imidazole derivatives and their use in pharmaceutics
03/04/2004WO2004018448A1 Novel thiophene derivatives, preparation method thereof and pharmaceutical compositions containing same
03/04/2004WO2004018438A2 Microbiocidal (e.g. fungicidal) 1,2,3-triazole derivatives
03/04/2004WO2004018435A1 Pyrimidine derivatives as modulators of chemokine receptor activity
03/04/2004WO2004018428A1 Antibacterial benzoic acid derivatives
03/04/2004WO2004017995A1 Preventive and/or therapeutic drugs for itch
03/04/2004WO2004017973A1 Remedy for integration dysfunction syndrome
03/04/2004WO2004017966A1 Five-membered heterocyclic compounds in the treatment of chronic and acute pain
03/04/2004WO2004017965A1 1,3-thiazolin-4-ones as therapeutic compounds in the treatment of pain
03/04/2004WO2004017961A2 Derivatives of 3-hydroxy-4-(cyclyl-alkylaminoalkyl)-5-phenyl-1h-pyrazole as antagonists of the gonadotropin releasing hormone (gnrh) for use in the treatment of sex hormone related conditions, such as prostatic of uterine cancer
03/04/2004WO2004017911A2 Protease inhibitors
03/04/2004WO2004001059A3 Heterocyclic inhibitors of kinases
03/04/2004WO2003106448A3 Nicotinoyl derivatives as herbicidal compounds
03/04/2004WO2003088917A3 Regulation of tnf-alpha
03/04/2004WO2003082350A3 Radiolabelled quinoline and quinolinone derivatives and their use as metabotropic glutamate receptor ligands
03/04/2004WO2003032916A3 Organosulfur inhibitors of tyrosine phosphatases
03/04/2004WO2003022844A3 Synthesis of epothilones intermediates thereto and analogues thereof
03/04/2004WO2002098856A3 Piperazine oxyquinoline (naphthaline) platelet adenosine diphosphate receptor antagonists
03/04/2004WO2002070469A3 Selective pde3b inhibitors and use of the same in therapy
03/04/2004US20040044221 Anticancer ganets; drug resistance
03/04/2004US20040044211 Substituted 4-phenyltetrahydroisoquinolinium, process for their preparation, their use as a medicament, and medicament containing them
03/04/2004US20040044203 Anticancer agents
03/04/2004US20040044057 5- substituted tetralones as inhibitors of ras farnesyl trransferase
03/04/2004US20040044052 N-Aryl-2-oxazolidinone-5-carboxamides and their derivatives
03/04/2004US20040044047 Alpha and beta-amino acid hydroxyethylamino sulfonamides useful as retroviral protease inhibitors
03/04/2004US20040044044 Thiazolyl urea compounds and methods of uses
03/04/2004US20040044043 Hyperglycemic agents; antilipemic agents
03/04/2004US20040044031 Controlling appetite; dietetics; sleep disorders
03/04/2004US20040044029 Azabicyclic compounds are central nervous system active agents
03/04/2004US20040044015 Quinazoline derivatives
03/04/2004US20040044003 Therapeutic agents useful for treating pain
03/04/2004US20040044000 Cardiovascular disorders; antiarthritic agents; inflammatory bowel disorders; vision defects; respiratory system disorders
03/04/2004US20040043988 Cycloalkyl alkanoic acids as intergrin receptor antagonists
03/04/2004US20040043987 Novel compounds and their use as positive AMPA receptor modulators
03/04/2004US20040043984 3,4-Dihydroquinolin-2-one, 5,6-fused oxazin-3-one, and 5,6-fused thiazin-3-one derivatives as matrix metalloproteinase inhibitors
03/04/2004US20040043903 2-Aryl-5-trifluoromethylpyridines
03/04/2004DE10238742A1 New N-(maleimidyl- or thiohydantoinyl-alkyl)-piperazine derivatives, are androgen receptor destabilizers and/or inhibitors useful e.g. for treating prostate carcinoma or hyperplasia
03/04/2004DE10238725A1 New heterocyclyl-substituted 2-(difluorobutenyl-sulfanyl)-pyrimidine derivatives, useful as pesticides, e.g. insecticides, acaricides, nematocides, ectoparasiticides or antifouling agents
03/04/2004DE10238045A1 2-Thio-substituierte Imidazolderivate und ihre Verwendung in der Pharmazie 2-thio-substituted imidazole derivatives and their use in the pharmaceutical
03/04/2004CA2501849A1 2-thio-substituted imidazole derivatives and their use in treating diseases associated with a disorder of the immune system
03/04/2004CA2497632A1 Novel thiophene derivatives, preparation method thereof and pharmaceutical compositions containing same
03/04/2004CA2496464A1 Agent for prevention and/or treatment of itching
03/04/2004CA2494263A1 Microbiocidal (e.g. fungicidal) 1,2,3-triazole derivatives
03/04/2004CA2494164A1 Pyridyl substituted heterocycles useful for treating or preventing hcv infection
03/03/2004EP1394162A1 Intermediates of azole antifungal agents and processes for the preparation thereof
03/03/2004EP1394159A1 New thiophene derivatives, process for their preparation and pharmaceutical compositions containing them
03/03/2004EP1394154A1 Five-membered heterocyclic alkanoic acid derivative
03/03/2004EP1394152A1 2-iminoimidazole derivatives (1)
03/03/2004EP1394147A1 Carboxylic acid derivative and medicine comprising salt or ester of the same
03/03/2004EP1394142A1 Carboxylic acid intermediates of antifungal agents and processes for the preparation thereof
03/03/2004EP1392684A1 Thiazole compounds useful as inhibitors of protein kinases
03/03/2004EP1392665A1 Thiazole or oxazole derivatives which are useful in the treatment of cardiovascular and related diseases
03/03/2004EP1392664A1 Epothilone derivatives
03/03/2004EP1392662A1 Cdk inhibiting pyrimidines, production thereof and their use as medicaments
03/03/2004EP1392661A1 Diarylurea derivatives useful as anti-inflammatory agents
03/03/2004EP1392656A2 Process for preparing chiral diol sulfones and dihydroxy acid hmg coa reductase inhibitors
03/03/2004EP1392317A2 Substituted 1-benzazepines and derivatives thereof
03/03/2004EP1392300A1 2,5-disubstituted pyridine, pyrimidine, pyridazine and 1, 2, 4-triazine derivatives for use as p38 inhibitors