Patents
Patents for C07D 417 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group (62,773)
01/2004
01/15/2004US20040009990 Especially piperidinylcarbonyl- and piperazinylcarbonyl-derivatives of indoles having oxalyl groups
01/15/2004US20040009987 4-phenylpiperidinyl- or 4-phenylpiperazinyl-; including N-oxides
01/15/2004US20040009981 Oxazole, thiazole, 1,3,4-oxadiazole and 1,3,4-thiadiazole derivatives of pyrimidines, 1,2,4- and 1,3,5-triazines
01/15/2004US20040009977 For use in the prophylaxis and the treatment of Picornavirus and human rotavirus infections.
01/15/2004US20040009974 Pyrimidylamino- or triazinylamino- substituted pyrazoles or 1,2,3-triazoles
01/15/2004US20040009969 Diazacycloalkanes containing a 2,5-dioxo-1H-pyrrolyl- or 4-oxo-2-thioxoimidazolidinyl- groups; treating prostate cancer, benign prostate hyperplasia, androgenetic alopecia, hirsutism and androgen-dependent acne.
01/15/2004US20040009968 Indazole compounds useful as protein kinase inhibitors
01/15/2004US20040009967 May contain further anticancer or immunosuppressive agents
01/15/2004US20040009966 Interleukin converting enzyme inhibitors
01/15/2004US20040009877 Hetaryl-substituted heterocycles
01/15/2004US20040009527 4-(2-imino-4-oxo-thiazolidin-5-ylidenemethyl)-benzoic acid, having at least two binding sites, selectivity binding to a receptor protein or oxidoreductase enzyme; drug design
01/15/2004US20040009526 Common ligand mimics: thiazolidinediones and rhodanines
01/15/2004DE10229370A1 2,1,3-Benzothiadiazole 2,1,3-benzothiadiazoles
01/15/2004DE10229070A1 Phenylderivate 5 Phenyl derivatives 5
01/15/2004CA2492121A1 3,6-disubstituted azabicyclo [3.1.0]hexane derivatives useful as muscarinic receptor antagonists
01/15/2004CA2491998A1 Azabicyclo derivatives as muscarinic receptor antagonists
01/15/2004CA2490463A1 1-amido-4-phenyl-4-benzyloxymethyl-piperidine derivatives and related compounds as neurokinin-1(nk-1) antagonists for the treatment of emesis, depression, anxiety and cough
01/15/2004CA2490097A1 Di-aryl-substituted-ethane pyridone pde4 inhibitors
01/15/2004CA2489166A1 Substituted anthranilic amide derivatives and methods of use
01/14/2004EP1380577A1 Thiazoline acid derivatives
01/14/2004EP1380575A1 1,2-disubstituted 1,4-dihydro-4-oxoquinoline compounds
01/14/2004EP1380562A1 Carboxylic acid derivative and salt thereof
01/14/2004EP1379525A2 Heteropolycyclic compounds and their use as metabotropic glutamate receptor antagonists
01/14/2004EP1379522A1 DIHYDRO-BENZO(b)(1,4)DIAZEPIN-2-ONE DERIVATIVES AS MGLUR2 ANTAGONISTS I
01/14/2004EP1379520A1 N-substituted nonaryl-heterocyclic nmda/nr2b antagonists
01/14/2004EP1379514A2 5-membered heterocycles, preparation and application thereof as medicaments
01/14/2004EP1379511A1 DIHYDRO-BENZO (b) (1, 4) DIAZEPIN-2-ONE DERIVATIVES AS MGLUR2 ANTAGONISTS II
01/14/2004EP1379508A2 N-(aryl)-2-arylethenesulfonamides and therapeutic uses thereof
01/14/2004EP1379504A1 Bipiperidinyl-derivatives and their use as chemokine receptors inhibitors
01/14/2004EP1379493A2 Non-imidazole aryl alkylamines compounds as histamine h3 receptor antagonists, preparation and therapeutic uses
01/14/2004EP1379252A2 Nociceptin analogs
01/14/2004EP1379249A1 Fused cyclic succinimide compounds and analogs thereof, modulators of nuclear hormone receptor function
01/14/2004EP1379243A1 Methods for treating metabolic diseases using malonyl-coa decarboxylase inhibitors
01/14/2004EP1379239A2 N-(2-arylethyl) benzylamines as antagonists of the 5-ht6 receptor
01/14/2004EP1379138A1 Liquid formulations for dermal application in treatment of parasitic insects in animals
01/14/2004EP1019385B1 Aminoaryl oxazolidinone n-oxides
01/14/2004EP0900088B1 Inclusion complexes of aryl-heterocyclic salts
01/14/2004CN1468243A Polymorphs of an epothilone analog
01/14/2004CN1468235A Aminoheterocyclylamides as pesticides and antiparasitic agents
01/14/2004CN1468233A Novel aminotriazolone compounds, method for preparing same and pharmaceutical compositions containing same
01/14/2004CN1468232A Heterocyclic sodium/proton exchange inhibitors and method
01/14/2004CN1468226A Biphenyl derivatives and their use as ppar-gamma receptor activators
01/14/2004CN1468220A New piperidine derivatives
01/14/2004CN1468217A Aliphatic nitrogenous five-membered ring compounds
01/14/2004CN1468216A Nitrogenous five-membered ring compounds
01/14/2004CN1468211A Nitroso diphenylamine derivatives
01/14/2004CN1467207A Method for preparing solid optical pure neutral S- (-) - and (R) - (+) -Omeprazole
01/14/2004CN1134444C Epothilone analog and medicine combination
01/14/2004CN1134438C Bicyclic heteroaromatic compounds, method for prepearing the same and uses
01/14/2004CN1134434C Novel 2-heterocyclically substituted dihydropyrimidines
01/14/2004CN1134421C Antifungal and its preparation method and intermediate
01/14/2004CN1134414C Substituted oximes, hydrazones and olefins as neurokinin antagonists
01/14/2004CN1134256C Application of substituted aminomethyl chromans in order to prevent neural degeneration and to promote neural regeneration.
01/13/2004US6677457 Halogenation
01/13/2004US6677368 4-aryl substituted indolinones
01/13/2004US6677365 Antagonists of MCP-1 function and methods of use thereof
01/13/2004US6677360 Biphenyl and biphenyl-analogous compounds as integrin antagonists
01/13/2004US6677354 Treating sleep, brain, sexual, cardiovascular, nervous system, psychological, glandular, and gastrointestinal disorders
01/13/2004US6677349 Sulfonamide and sulfamide substituted imidazoquinolines
01/13/2004US6677340 Gonadotropin-releasing hormone receptor antagonists and methods relating thereto
01/13/2004US6677337 1,2-dihydropyrazol-3-ones which controls inflammatory cytokines
01/13/2004US6677333 2H-phthalazin-1-one derivatives and drug containing its derivatives as active ingredient
01/13/2004US6676909 Method for recovery of metals from metal-containing materials using medium temperature pressure leaching
01/13/2004CA2139731C 2-heterocyclic-5-hydroxy-1,3-pyrimidines useful as antiinflammatory agents
01/13/2004CA2053359C Heteroaroyl derivatives of monocyclic beta-lactam antibiotics
01/08/2004WO2004003108A1 Luminescent compositions
01/08/2004WO2004002992A1 Compounds
01/08/2004WO2004002970A1 2,1,3-benzothiadiazoles for use as electronic active components
01/08/2004WO2004002967A1 Difluorothioacetamides of oxazolidinones as antibacterial agents
01/08/2004WO2004002965A1 Arylcarbonylpiperazines and heteroarylcarbonylpiperazines and the use thereof for treating benign and malignant tumour diseases
01/08/2004WO2004002964A1 Diaminopyrimidinecarboxa mide derivative
01/08/2004WO2004002960A1 Substituted quinoline ccr5 receptor antagonists
01/08/2004WO2004002948A1 Amide compound and medicinal use thereof
01/08/2004WO2004002481A1 Aryl carbonyl derivatives as therapeutic agents
01/08/2004WO2004002477A1 2-(phenyl)-2h-pyrazole-3-carboxylic acid-n-4-(thioxo-heterocyclyl)-phenyl-amide derivatives and corresponding imino-heterocyclyl derivatives and relates compounds for use as inhibitors of the coagulation factors xa and/or viia for treating thromboses
01/08/2004WO2004002470A1 Compounds useful for the inhibition of aldh
01/08/2004WO2003087088A3 (condensed) pyrimidone and (condensed) pyridone compounds, processes for their preparation, and pharmaceutical compositions containing them
01/08/2004WO2003077828A3 Novel florfenicol-type antibiotics
01/08/2004US20040006230 Substituted polycyclic aryl and heteroaryl pyrazinones useful for selective inhibition of the coagulation cascade
01/08/2004US20040006229 Indole derivatives for the treatment of depression and anxiety
01/08/2004US20040006123 Interleukin-4 gene expression inhibitors
01/08/2004US20040006112 Benzylidene thiazolidinediones and their use as antimycotic agents
01/08/2004US20040006110 1,4-dihydropyridine and pyridine compounds as calcium channel blockers
01/08/2004US20040006107 For prophylaxis of asthma and other allergic diseases
01/08/2004US20040006105 Thrombin receptor antagonists
01/08/2004US20040006101 Quinolinone derivatives
01/08/2004US20040006099 Amidine compounds
01/08/2004US20040006091 Therapeutic agents useful for treating or preventing pain
01/08/2004US20040006089 For therapy of acromegalia, hypophyseal adenomas or endocrine gastroenteropancreatic tumors including carcinoid syndrome
01/08/2004US20040006088 Substituted N-(indole-2-carbonyl) -amides and derivatives as glycogen phosphorylase inhibitors
01/08/2004US20040006086 For therapy of metabolic and eating disorders such as obesity and hyperphagia, diabetes
01/08/2004US20040006081 Pharmaceutically active piperidine derivatives, in particular as modulators of chemokine receptor activity
01/08/2004US20040006080 Chemical compounds
01/08/2004US20040006078 For therapy of autoimmune diseases, asthma, osteoporosis, atherosclerosis, Alzheimer's disease
01/08/2004US20040006076 Thiazolyl amide derivatives
01/08/2004US20040006069 For therapy inflammatory and immune system disorders such as stroke, myocardial infarction, atherosclerosis, ischemic heart disease, ischemia-reperfusion injury
01/08/2004US20040006067 Substituted piperidines and methods of use
01/08/2004US20040006062 For use as anticoagulant agents for therapy of thromboembolic disorders
01/08/2004US20040006058 As inhibitors of cyclin-dependent kinase 4 (Cdk4); antiproliferative agents; for therapy of cancer, tumors
01/08/2004US20040005986 Pyridazin-3-one derivatives, their use, and intermediates for their production