Patents
Patents for C07D 417 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group (62,773)
05/2004
05/27/2004CA2505797A1 Process for converting a cis-trans mixture of substituted benzylidene amines into the pure cis isomer
05/27/2004CA2505127A1 Ophthalmic compositions for treating ocular hypertension
05/27/2004CA2504737A1 Aromatic sulfone hydroxamic acids and their use as protease inhibitors
05/27/2004CA2502190A1 Pyrimidine compounds
05/26/2004EP1422553A1 Improved base precursors for use in a photothermographic element
05/26/2004EP1422224A1 Dithiazole compounds, matrix metalloprotease inhibitors and external preparations for the skin
05/26/2004EP1422218A1 Antiviral agent
05/26/2004EP1421389A2 Neurofibrillary labels
05/26/2004EP1421082A1 New piperidinyl-morpholinyl derivatives as modulators of chemokine receptor activity
05/26/2004EP1421078A1 Beta-3 adrenergic agonists
05/26/2004EP1421074A1 Novel compounds
05/26/2004EP1421070A1 New piperidinyl derivates as modulators of chemokine receptor activity
05/26/2004EP1421063A1 Disulfide and thiosulfonate ligands and libraries comprising these ligands
05/26/2004EP1420784A1 Compounds effecting glucokinase
05/26/2004EP1420780A2 Cyclopropyl and cyclobutyl epothilone analogs
05/26/2004EP1216245B1 Pharmaceutically active sulfonyl hydrazide derivatives
05/26/2004EP1173176B1 Utilization of polycyclic 2-amino-thiazole systems in the production of medicaments for prophylaxis or treatment of obesity
05/26/2004EP1117661B1 Propanolamine derivatives substituted with heterocyclic compounds, methods for their production, pharmaceutical compositions containing said compounds and the use thereof
05/26/2004EP1117642B1 Substituted 1,3-diaryl-2-pyridine-2-yl-3-(pyridine-2-ylamino)-propanol derivatives, methods for their production, pharmaceutical compositions containing the same and their use
05/26/2004EP1027332B1 Novel lactam metalloprotease inhibitors
05/26/2004EP1022272B1 Substituted fused heterocyclic compounds
05/26/2004EP0968194B1 Atropisomers of 3-aryl-4(3h)-quinazolinones and their use as ampa-receptor antagonists
05/26/2004CN1500086A Aminopiperidine derivatives
05/26/2004CN1500082A Cyano-5ubstituted dihydropyrimidine compounds and their use to treat diseases
05/26/2004CN1500080A 稠合杂环化合物 Fused heterocyclic compounds
05/26/2004CN1499970A Use of GAL3 receptor antagonists for treatment of. depression and/or anxiety and compounds useful in such methods
05/26/2004CN1151161C Medicine nitrate salts
05/26/2004CN1151147C Indole derivatives as 5-HT receptor antagonist
05/26/2004CN1151133C Anthranilic acid amides and use thereof as medicaments
05/26/2004CN1151131C Piperidine derivatives useful as CCR5 antagonists
05/25/2004US6740760 Such as 1-((s)-3-mercapto-2-methyl-propionyl)-(r)-pyrrol-idine-2-carboxylic acid for treating diseases associated with amyloidosis (alzheimer's disease, diabetes, and familial amyloid polyneuropathy)
05/25/2004US6740682 Treatment of thrombotic diseases, asthma, emphysema, cirrhosis, arthritis, carcinoma, melanoma, restenois, atheroma, trauma, shock and reperfusion injury.
05/25/2004US6740666 Substituted 8-arylquinoline phosphodiesterase-4 inhibitors
05/25/2004US6740655 3',5'-cyclic nucleotide phosphodiesterase 4-specific inhibitors reduce eosinophil influx to the lungs; side effect reduction; antiinflammatory agent; antiallergens; respiratory system disorders, especially asthma
05/25/2004US6740649 Cyclic hydroxamic acids as inhibitors of matrix metalloproteinases and/or TNF- α converting enzyme (TACE)
05/25/2004CA2302058C A process for preparing 5-methoxy-4-methyl-2,4-dihydro-3h-1,2,4-triazol-3-one
05/21/2004WO2004041818A1 Anti-infective agents
05/21/2004WO2004041816A1 Azacyclic compounds as orexin receptor antagonist
05/21/2004WO2004041815A1 Indole derivative with 5ht1a affinity
05/21/2004WO2004041813A1 Compositions useful as inhibitors of rock and other protein kinases
05/21/2004WO2004041809A2 Substituted imidazolylmethyl pyridine and pyrazine derivatives and their use as gabaa receptor ligands
05/21/2004WO2004041808A1 4-imidazol-1-ylmethyl-pyrimidine derivatives_as ligands for gabaa receptors
05/21/2004WO2004041799A1 5- (substituted phenyl) -thiadiazolidine-3-ones and their use as ptp1b
05/21/2004WO2004041795A1 Novel inhibitors of dipeptidyl peptidase iv
05/21/2004WO2004041794A1 Antiinflammatory 3-arylthio-3-thiazolyl-alkylamines
05/21/2004WO2004041793A1 Phenylalkyl and pyridylalkyl piperazine derivatives
05/21/2004WO2004041782A1 Indoles useful in the treatment of androgen-receptor related diseases
05/21/2004WO2004041777A2 Heteroarylpiperidine modulators of chemokine receptor activity
05/21/2004WO2004041776A2 SULFONYLAMINOVALEROLAC TAMS AND DERIVATIVES THEREOF AS FACTOR Xa INHIBITORS
05/21/2004WO2004041282A1 Receptor regulator
05/21/2004WO2004041279A1 Gamma-aminoamide modulators of chemokine receptor activity
05/21/2004WO2004041277A1 Carbonylamino-benzimidazole derivatives as androgen receptor modulators
05/21/2004WO2004041258A2 Cyclic nucleotide phosphodiesterase inhibitors, preparation and uses
05/21/2004WO2004041201A2 Benzofuran compounds, compositions and methods for treatment and prophylaxis of hepatitis c viral infections and associated diseases
05/21/2004WO2004041164A2 Kinase inhibitors
05/21/2004WO2004041163A2 Piperidinyl cyclopentyl aryl benzylamide modulators of chemokine receptor activity
05/21/2004WO2004041161A2 Tetrahydropyranyl cyclopentyl benzylamide modulators of chemokine receptor activity
05/21/2004WO2004026226A8 Compounds, compositions and methods
05/21/2004WO2004014860A3 Fused heterocyclic compounds as peptidase inhibitors
05/21/2004WO2004004629A3 3,6-disubstituted azabicyclo [3.1.0]hexane derivatives useful as muscarinic receptor antagonists
05/21/2004WO2004000817A3 Benzimidazole compounds and their use as estrogen agonists/antagonists
05/21/2004CA2505397A1 Phenylalkyl and pyridylalkyl piperazine derivatives
05/21/2004CA2504805A1 Receptor regulator
05/21/2004CA2504344A1 Benzofuran compounds, compositions and methods for treatment and prophylaxis of hepatitis c viral infections and associated diseases
05/21/2004CA2504320A1 Compositions useful as inhibitors of rock and other protein kinases
05/21/2004CA2504044A1 Carbonylamino-benzimidazole derivatives as androgen receptor modulators
05/21/2004CA2503720A1 Gamma-aminoamide modulators of chemokine receptor activity
05/21/2004CA2503716A1 Cyclic nucleotide phosphodiesterase inhibitors, preparation and uses
05/21/2004CA2503715A1 Kinase inhibitors
05/21/2004CA2503713A1 Piperidinyl cyclopentyl aryl benzylamide modulators of chemokine receptor activity
05/21/2004CA2502178A1 Heteroarylpiperidine modulators of chemokine receptor activity
05/21/2004CA2502174A1 Tetrahydropyranyl cyclopentyl benzylamide modulators of chemokine receptor activity
05/21/2004CA2495708A1 4-imidazol-1-ylmethyl-pyrimidine derivatives as ligands for gabaa receptors
05/21/2004CA2484936A1 Substituted imidazolylmethyl pyridine and pyrazine derivatives and their use as gabaa receptor ligands
05/20/2004US20040097734 Aryl- and heteroarylcarbonylpiperazines and their use for the treatment of benign and malignant oncoses
05/20/2004US20040097732 Peptide deformylase inhibitors
05/20/2004US20040097730 Amide containing a pyridinone or pyrazinone compound as serine protease enzyme inhibitors
05/20/2004US20040097729 Substituted pyridine herbicides
05/20/2004US20040097728 Method for producing anellated tetrahydro-{1h}-triazoles
05/20/2004US20040097594 Sulfonamide inhibitors of aspartyl protease
05/20/2004US20040097579 Taxane formulations
05/20/2004US20040097574 For therapy of inflammatory, allergic, or proliferative processes
05/20/2004US20040097571 Imidazole compounds and their use as adenosine deaminase inhibitors
05/20/2004US20040097566 For therapy of diseases related to uncontrolled cellular proliferation, useful for modulating lipid and/or carbohydrate metabolism, for therapy of Type II diabetes, hyperglycemia or obesity, inflammatory diseases such as arthritis
05/20/2004US20040097564 Method and compounds for treating glaucoma VI
05/20/2004US20040097560 N-alkyl-4-methyleneamino-3-hydroxy-2-pyridones
05/20/2004US20040097559 N-sulfonyl-4-methyleneamino-3-hydroxy-2-pyridones
05/20/2004US20040097558 Hetaryl substituted homotetramic and homtetronic acids and the use thereof as pesticides
05/20/2004US20040097555 Useful as a prophylactic or therapeutic agent of the diseases such as rheumatism, arthritis and the like, and other diseases
05/20/2004US20040097553 Hydrate of 5-[4-[2-(N-methyl-N-(2-pyridil)amino)ethoxy]benzyl]thiazolidine-2,4-dione maleic acid salt
05/20/2004US20040097545 Quinolinone derivatives
05/20/2004US20040097531 For therapy of inflammatory disease, autoimmune disease, destructive bone disorder, proliferative disorder, infectious disease, neurodegenerative disease, allergy, reperfusion/ischemia in stroke, heart attack, hypoxia
05/20/2004US20040097513 Novel non-imidazole compounds
05/20/2004US20040097503 Substituted 2-aryl-4-arylaminopyrimidines and analogs as activators of caspases and inducers of apoptosis and the use thereof
05/20/2004US20040097501 Triazole compounds useful as protein kinase inhibitors
05/20/2004US20040097497 4-heteroaryl-3-heteroarylidenyl-2-indolinones and their use as protein kinase inhibitors
05/20/2004US20040097496 Novel thiazine derivatives
05/20/2004US20040097494 For use as nitric oxide synthase inhibitors
05/20/2004US20040097492 For inhibiting hepatitis C virus (HCV) polymerase; therapy and prophylaxis of HCV infection
05/20/2004US20040097487 To inhibits matrix metalloprotease activity