Patents
Patents for C07D 417 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group (62,773)
12/2004
12/09/2004WO2004105750A1 3-aminomethyl-pyrrolidines as n-type calcium channel blockers
12/09/2004WO2004094388A3 Indazole derivatives as jnk inhibitors
12/09/2004WO2004087699A3 Thiazoles useful as inhibitors of protein kinases
12/09/2004WO2004087698A3 Thiazoles useful as inhibitors of protein kinases
12/09/2004WO2004071440A3 Thiazolyl-based compounds useful as kinase inhibitors
12/09/2004WO2004061084A8 Modulation of protein functionalities
12/09/2004WO2004018478A3 Synthesis of epothilones, intermediates thereto, analogues and uses thereof
12/09/2004WO2003080582A3 Fredericamycin derivatives
12/09/2004US20040249150 Positive allosteric modulators of the nicotinic acetylcholine receptor
12/09/2004US20040248950 Apo ai expression accelerating agent
12/09/2004US20040248945 Thiazolidinedione derivative and its use as antidiabetic
12/09/2004US20040248936 such as (R)-1-{4-[4-(4-Phenoxy-2-propyl-phenoxy)-butoxy]-benzenesulfonyl}-azetidine-2-carboxylic acid, used as peroxisome proliferator-activated receptor agonists; hypoglycemic agents
12/09/2004US20040248934 peroxisome proliferator activator receptor agonists; anticholesterol, antidiabetic agents; 2-Methyl-2-{2-[4-methyl-2-(4-trifluoromethyl-phenyl)-thiazole-5-carbonyl]-1,2,3,4-tetrahydro-isoquinolin-7-yloxy}-propionic acid
12/09/2004US20040248923 Novel 4-anilinoquinoline-3-carboxamides
12/09/2004US20040248899 Fused bicyclic-substituted amines as histamine-3 receptor ligands
12/09/2004US20040248890 Voltage gated sodium and calcium channel inhibitors
12/09/2004US20040248885 Use of thiazole derivatives for preparing a medicine for protecting mitochondria
12/09/2004US20040248851 Substituted diphenyloxazoles, the synthesis thereof, and the use thereof as fluorescence probes
12/09/2004US20040248740 for controlling undesirable plants
12/09/2004US20040248225 Luciferin hydrazides
12/09/2004CA2527731A1 Substituted pyrrole derivatives as hmg-coa reductase inhibitors
12/09/2004CA2527174A1 Benzothiazole derivatives and use thereof in the treatment of diseases related to the adenosine a2a receptor
12/09/2004CA2527159A1 3-aminomethyl-pyrrolidines as n-type calcium channel blockers
12/09/2004CA2526749A1 3-[2-(3-amino-2-oxo-2h-pyridin-1-yl)-acetylamino]-4-oxo-pentanoic acid derivatives and their use as caspase inhibitors
12/08/2004EP1484328A1 Derivatives of quinolyl-propyl-piperidine and their use as antimicrobial agents
12/08/2004EP1484327A1 Nitrogenous heterocyclic compound and medicine thereof
12/08/2004EP1483263A1 Thiazolyl urea compounds for the treatment of cancer
12/08/2004EP1483262A1 Coumarines useful as biomarkers
12/08/2004EP1483260A1 Cdk inhibiting 2-heteroaryl pyrimidine, the production thereof, and use thereof as a medicament
12/08/2004EP1483259A1 Pyrimidines as novel openers of potassium ion channels
12/08/2004EP1483251A1 C3-cyano epothilone derivatives
12/08/2004EP1482940A2 Prodrugs of substituted polycyclic compounds useful for selective inhibition of the coagulation cascade
12/08/2004EP1482935A1 Thiazole and oxazole derivatives which modulate ppar activity
12/08/2004EP1482932A1 N3 alkylated benzimidazole derivatives as mek inhibitors
12/08/2004EP1482924A2 Cathepsin cysteine protease inhibitors
12/08/2004EP1363898A4 Compounds useful as modulators of melanocortin receptors and pharmaceutical compositions comprising same
12/08/2004EP1339403B1 Repinotan kit
12/08/2004EP1218370B1 Quinolyl propyl piperidine derivatives and their use as antibacterial agents
12/08/2004EP1119548B1 3-(3-chloro-4-hydroxyphenylamino)-4-(2-nitrophenyl)-1h-pyrrole-2,5-dione as glycogen synthase kinase-3 inhibitor (gsk-3)
12/08/2004EP0915868B1 Carbanilides used as pesticides
12/08/2004CN1553910A Heterocyclylindazole and -azaindazole compounds as 5-hydroxytryptamine-6 ligands
12/08/2004CN1553909A Benzimidazole and pyridylimidazole derivatives as ligands for GABA receptors
12/08/2004CN1553907A Tetrazoyl oxime derivative and agrochemical containing the same as active ingredient
12/08/2004CN1178937C Preparation of intermediate for thiazolylisopseudoindole dyes
12/08/2004CN1178935C 1,3-disubstituted pyrrolidines as alpha-2-adrenoceptor antagonists
12/08/2004CN1178932C Amide derivatives
12/08/2004CN1178922C Substituted 1-aminoalkyl-lactams compound and their use as muscarinic receptor antagonists
12/08/2004CN1178917C N-oxides as NK1 receptor antagonist prodrugs of 4-phenyl-pyridine derivatives
12/08/2004CN1178912C Small molecule inhibitors of rotamase enzyme activity
12/08/2004CN1178665C Water soluble prodrugs of azole compounds
12/08/2004CN1178663C Use of 1,4-benzothiazepine derivatives as drugs overcoming carcinostatic tolerance
12/08/2004CN1178657C Treatment and prophylaxis of pancreatitis
12/07/2004US6828427 Oligomeric aminodiol-containing compounds, libraries thereof, and process of preparing the same
12/07/2004US6828344 Direct inhibition of the activity of phospholipase A2 has been suggested as a useful mechanism for a therapeutic agent for inflammation
12/07/2004US6828341 Brain disorders; anticonvulsants; central nervous system disorders; psychological disorders
12/07/2004US6828340 Especially for cancer which has developed a multidrug-resistant phenotype.
12/07/2004US6828335 Oxazole or thiazole-ethyl-oxy-indane acetic acid derivatives; useful for the treatment of diseases such as diabetes, obesity, hyperlipidemia and atherosclerosis
12/07/2004US6828333 Ether derivatives useful as inhibitors of PDE4 isozymes
12/07/2004US6828317 Bactericides; gramnegative, grampositive bacteria
12/07/2004US6828116 Energy transfer assay method and reagent
12/07/2004CA2272136C Pyrazole derivatives having crf antagonist activity
12/07/2004CA2150123C Aminomethylene substituted non-aromatic heterocycles
12/07/2004CA2112331C Novel naphthalene derivatives
12/07/2004CA2108817C Arylidene-1-azacycloalkanes and arylalkyl-1-azacycloalkanes, their salts, medicaments containing these compounds and their use, and processes for their preparation
12/02/2004WO2004103999A1 AZTREONAM β POLYMORPH WITH VERY LOW RESIDUAL SOLVENT CONTENT
12/02/2004WO2004103998A1 Quinoline derivatives as phosphodiesterase inhibitors
12/02/2004WO2004103997A1 TETRAHYDROISOQUINOLINE DERIVATIVES AS PPAR-α ACTIVATORS
12/02/2004WO2004103995A1 N-acyl nitrogen heterocycles as ligands of peroxisome proliferator-activated receptors
12/02/2004WO2004103981A1 Process for preparing a 4,7-bis(5-halothien-2-yl)-2,1,3-benzothiadiazole and a precursor therefor
12/02/2004WO2004103980A1 Inhibitors of 11-beta-hydroxy steroid dehydrogenase type i
12/02/2004WO2004103367A1 Benzothiazole derivatives and use thereof in the treatment of diseases relates to the adenosine a2a receptor
12/02/2004WO2004076413A3 Phenyl- and pyridylpiperidine-derivatives as modulators of glucose metabolism
12/02/2004WO2004072031A3 Phenylacetamides and their use as glucokinase modulators
12/02/2004WO2004066952A3 Benzoxazole, benzothiazole, and benzimidazole derivatives for the treatment of cancer and other diseases
12/02/2004WO2004058174A3 Indane acetic acid derivatives and their use as pharmaceutical agents, intermediates, and method of preparation
12/02/2004US20040242928 Reverse hydroxamic acid derivatives
12/02/2004US20040242871 Nitric oxide synthease inhibitors; antiinflamamtory agents; analgesics; inflamamtory bowel disorders; antiarthritic agents;
12/02/2004US20040242868 Controlling cytokines; antiinflammatory agents; rheumatic disoreders; skin disorders; respiratory system disorders; Alzheimer's disease; Parkinson's disease; Huntington"s disease ; amyotrophic lateral sclerosis
12/02/2004US20040242672 Pyrrolidine derivatives
12/02/2004US20040242668 Capable of increasing lipolysis and energy expenditure in cells and therefore is useful for treating Type 2 diabetes and/or obesity
12/02/2004US20040242666 Isoxazole and isothiazole compounds for the treatment of neurodegenerative disorders
12/02/2004US20040242664 Pyrazolyl-substituted heterocycles and their use as phytosanitary products
12/02/2004US20040242660 Combinations of oxazolidinones with other active ingredients for the prophylaxis and/or treatment of thromboembolic disorders
12/02/2004US20040242658 Recrystallizing rosiglitazone maleate from solvent; for treatment or prophylaxis of diabetes mellitus, conditions associated with diabetes mellitus and complication thereof in a mammal
12/02/2004US20040242656 N-heterocyclicamide compounds; useful in the treatment of cardiovascular disorders, in particular, as an anticoagulant
12/02/2004US20040242637 drugs used for signal transduction modulation, and for prophylaxis of angiogenesis, cancers, tumors, atherosclerosis, vision disorders and inflammatory diseases in mammals
12/02/2004US20040242633 Compound used to lower cholesterol, reduce weight for dietetics, antidepressants and antidiabetic agents
12/02/2004US20040242628 administering N-(1H-Indol-7-yl)-4-nitrobenzenesulfonamide; treating cachexia during cancer therapy
12/02/2004US20040242627 2-Iminoimidazole derivatives (1)
12/02/2004US20040242615 enhancing the expression of apoAI; prevention or therapy of dislipidemia
12/02/2004US20040242609 Therapy for eating disorders, sexual disorders, psychological disorders
12/02/2004US20040242602 Novel thiazolidine compounds as calcium sensing receptor modulators
12/02/2004US20040242593 Cannabinoid derivatives, methods of making, and use thereof
12/02/2004US20040242580 can be applied as sprays by methods commonly employed in crops such as vegetables, fruits, ornamentals, seeds, turf, cereal and vines among other plants
12/02/2004US20040242577 N-methyl 2-morpholine-4-carbonyl or sulfonyl substituted; for example: 2-{[4-(3,4-dichlorophenoxy)piperidin-1-yl]methyl}morpholine; useful for treating asthma and/or rhinitis
12/02/2004US20040242576 Urea substituted benzothiazoles
12/02/2004US20040242575 for use with various disorders including sleep disorders; depression; cardiovascular disorders; pain; neurodegenerative disorders; psychiatric disorders etc.
12/02/2004US20040242574 Anticancer agents; antiarthritic agents
12/02/2004US20040242573 Novel compounds
12/02/2004US20040242571 Novel benzothiazine derivatives, their preparation and use