Patents
Patents for C07D 417 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group (62,773)
02/2005
02/17/2005WO2005014553A1 Novel gamma-secretase inhibitors
02/17/2005WO2005014552A1 Quinoline and quinazoline derivatives having affinity for 5ht1-type receptors
02/17/2005WO2005014540A1 Cyclic amine base-1 inhibitors having a heterocyclic substituent
02/17/2005WO2005013977A1 Indol-5-yl sulfonamide derivatives, their preparation and their use 5-ht-6 as modulators
02/17/2005WO2005013914A2 Heteroarylaminosulfonylphenyl derivatives for use as sodium or calcium channel blockers in the treatment of pain
02/17/2005WO2004110993A3 N-ureidoalkyl-piperidines as modulators of chemokine receptor activity
02/17/2005WO2004110344A3 New azetidine compounds
02/17/2005WO2004092115A3 Hydroxamates as therapeutic agents
02/17/2005WO2004084813A3 Chemical compounds
02/17/2005US20050038247 topoisomerase inhibitors such as [5-(4-Cyclopropylcarbamoyl-imidazol-1-yl)-7-pyrimidin-2-yl-1H-benzoimidazol-2-yl]-carbamic acid ethyl ester, used for prophylaxis of bacterial infections in mammals
02/17/2005US20050038243 2, 4-pyrimidinediamine compounds and their uses
02/17/2005US20050038101 Substituted 2 5-diamidoindoles as ece inhibitors for the treatment of cardiovascular diseases
02/17/2005US20050038100 Eating disorders; anticholesterol agents; hypotensive agents; sleep disorders; hyperphagia
02/17/2005US20050038099 3-Amido-5-substituted pyrazole derivatives and related compounds useful as bradykinin B1 receptor antagonists to relieve adverse symptoms in mammals mediated, at least in part, by bradykinin B1 receptor including pain, inflammation, septic shock, scarring process
02/17/2005US20050038092 effective against aerobic and anerobic pathogens such as multi-resistant staphylococci, streptococci and enterococci, Bacteroides spp., Clostridia spp. species; side effect reductions
02/17/2005US20050038089 Thiazole derivatives
02/17/2005US20050038087 Derivatives of heterocycles with 5 members, their preparation and their use as medicaments
02/17/2005US20050038086 Epothilone derivatives and methods for making and using the same
02/17/2005US20050038078 Antimetastasis agents e.g. 6-[4-Amino-5-(2,6-difluoro-benzoyl)-thiazol-2-ylamino]-N-pyridin-2-ylmethyl-nicotinamide; protein kinase inhibitor
02/17/2005US20050038075 Intermediates for N-substituted carbamoyloxyalkyl-azolium derivatives
02/17/2005US20050038074 Kinesin spindle protein (KSP) inhibitors, e.g., 4-(2,5-Difluorophenyl)-N-[(3S,4S)-3-fluoropiperidin-4-yl]-2-hydroxymethyl)-N-methyl-2-phenyl-2,5-dihydro-1N-pyrrole-1-carboxamide; antiproliferative and -carcinogenic agents
02/17/2005US20050038073 Thiazole derivatives
02/17/2005US20050038072 Nitrogeneous cyclic ketone derivative, process for producing the same, and use
02/17/2005US20050038069 Tumor necrosis factor antagonist; antiinflammatory agents; such as 2-Cyclopropyl-4-(3,5-dimethyl-4-pyridylmethoxy)-7-methoxy-3H-benzimidazole
02/17/2005US20050038060 Spiropoperidine compounds as ligands for orl-1 receptor
02/17/2005US20050038059 N-{4-[2-(1-Dimethylamino-ethylimino)-4-phenyl-thiazol-5-yl]-pyrimidin-2-yl}-N-phenyl-amine; fungicides against infestation by phytopathogenic organisms, nematodes, insects, fungi, bacteria, viruses
02/17/2005US20050038040 Corticotropin releasing factor antagonist; antiinflammatory agents; drug abuse; analgesics; antihistamines; skin disorders; neurodegenerative disease; eating disorders;eating disorders; antiepileptic agents; cardiovascular disorders
02/17/2005US20050038038 N-phenyl substituted carbamoyloxyalkyl-azolium derivatives
02/17/2005US20050038037 N-(naphth-2-ylaminocarbonylacetyl)- or N-(naphth-2-ylcarbonylamino- acetyl)- piperazine derivatives, e.g., 2-[((4-(ethoxycarbonyl)piperazin-1-yl)carbonylmethyl)carbonyl]aminonaphthalene; useful as antithrombotic agents
02/17/2005US20050038035 Heterocyclic amide compounds as apolipoprotein b inhibitors
02/17/2005US20050038031 Novel bicyclic urea derivatives useful in the treatment of cancer and other disorders
02/17/2005US20050038029 Transferring, releasing nitric oxide; side effect reduction; using a compound containing nitrosos group
02/17/2005US20050038023 Inhibitors of glycogen synthase kinase-3 (gsk-3) and aurora-2, both serine/threonine protein kinases; for treating diseases such as cancer, diabetes and alzheimer's disease
02/17/2005US20050038021 2,4,5,-trisubstituted phenylketo-enols for use as pesticides and herbicides
02/17/2005US20050038016 Arylamine-substituted quinazolinone compounds useful as alpha 1A/B adrenergic receptor antagonists
02/17/2005US20050038009 1,1-dioxo-3,3-dibutyl-5-phenyl-7-methylthio-8-(N-{(R)- alpha -[N-((S)-1-carboxypropyl) carbamoyl]-4-hydroxybenzyl}carbamoylmethoxy)-2,3,4,5-tetrahydro-1,2,5-benzothiadiazepine
02/17/2005US20050037997 Detoxification; hydrolases or esterases; short half-life; non-insulin dependent diabetes; side effect reduction
02/17/2005US20050037925 Mixture with other herbicides
02/17/2005CA2539227A1 Heteroarylaminosulfonylphenyl derivatives for use as sodium or calcium channel blockers in the treatment of pain
02/17/2005CA2534405A1 Halogenated quinazolinyl nitrofurans as antibacterial agents
02/17/2005CA2534057A1 Novel gamma-secretase inhibitors
02/17/2005CA2533976A1 Indol-5-yl sulfonamide derivatives, their preparation and their use 5-ht-6 as modulators
02/17/2005CA2533464A1 Thiazole derivatives as npy antagonists
02/17/2005CA2533463A1 2-amino-5-benzoylthiazole npy antagonists
02/17/2005CA2532452A1 Quinoline and quinazoline derivatives having affinity for 5ht1-type receptors
02/16/2005EP1506967A1 Dipeptidyl peptidase inhibitors
02/16/2005EP1506962A2 Nitrogen-containing aromatic heterocycles
02/16/2005EP1506203A2 Synthesis of epothilones, intermediates thereto, analogues and uses thereof
02/16/2005EP1506197A1 Acyl bicyclic derivatives of pyrrol
02/16/2005EP1506189A1 Pyrrole derivatives as inhibitors of erk2 and uses thereof
02/16/2005EP1506179A1 Benzoxazine derivatives as 5-ht6 modulators and uses thereof
02/16/2005EP1506176A1 Aminoindazole derivatives active as kinase inhibitors, process for their preparation and pharmaceutical compositions comprising them
02/16/2005EP1505977A2 Administration of a partial fatty acid inhibitor such as ranolazine for the treatment of diabetes
02/16/2005EP1505968A1 Multicyclic compounds for use as melanin concentrating hormone antagonists in the treatment of obesity and diabetes
02/16/2005EP1505963A1 Hepatitis c virus inhibitors
02/16/2005EP1395553B1 Pyrrolidine derivatives as factor xa inhibitors
02/16/2005EP1240166B1 N-[5-[[[5-alkyl-2-oxazolyl]methyl]thio]-2-thiazolyl carboxamide inhibitors of cyclin dependent kinases
02/16/2005CN1582287A Thiophenylthiopyrane dioxides as MMP or TNF-alpha inhibitors
02/16/2005CN1582285A Heteroaryl amines as glycogen synthase kinase 3beta inhibitors (GSK3 inhibitors)
02/16/2005CN1582284A Aminopyrimidines and pyridines
02/16/2005CN1582281A Mch受体拮抗剂 Mch receptor antagonist
02/16/2005CN1582280A 3, 4-di-substituted pyridazinediones as CXC chemokine receptor antagonists
02/16/2005CN1582277A Amide derivatives as glycogen synthase kinase 3-beta inhibitors
02/16/2005CN1582151A Benzothiazepine and benzothiazepine derivatives with ileal bile acid transport (IBAT) inhibitory activity for the treatment hyperlipidaemia
02/16/2005CN1582148A Derivatives of phenoxy-n-'4-(isothiazolidin-1, 1-dioxid-2yl)pheny!-valerian- acid amide and other compounds as inhibitors of the coagulation factor Xa in the treatment of thromboembolic diseases and tu
02/16/2005CN1580179A White electroluminescent polymer material and its preparing method
02/16/2005CN1580056A Heterocyclic derivatives their preparing methods and uses
02/16/2005CN1189469C 3-(heteroaryl acetamido)-2-oxo-azeridine-1-sulfonic acid derivatives as anti-bacterial agents
02/16/2005CN1189468C Preparation method of 5-[4-[2-(5-ethyl-2-pyridine)ethoxy]benzylidene]-2, 4thiazolidine diketone
02/16/2005CN1189467C Pharmaceutically active sulfonamide derivatives
02/16/2005CN1189466C New direct chain or cyclic urea, its preparing method and medicinal composition containing them
02/15/2005US6855726 Heterocyclic amides such as 3-(1-5-((2R,6S)-2,6-dimethyltetra-hydro-1(2H)-pyridinyl)pentyl-2-oxo-1,2 -dihydro-3-quinolinyl) benzenecarboximidamide, administered as anticoagulants or for prophylaxis of cardiovascular disorders
02/15/2005US6855715 Drugs such as 1-(3-Amino-4-chlorobenzoyl-D-phenylglycinyl)-4-(4-fluoro-2 -methylsulphonylphenyl)piperazine, used as anticoagulants
02/10/2005WO2005012298A1 Pyridinylamino-pyrimidine derivatives as protein kinase inhibitors
02/10/2005WO2005012297A1 Benzimidazole, benzthiazole and benzoxazole derivatives and their use as lta4h modulators
02/10/2005WO2005012296A1 Benzimidazole, benzthiazole and benzoxazole derivatives and their use as lta4h modulators
02/10/2005WO2005012295A1 Substituted thiazole-benzoisothiazole dioxide derivatives, method for the production thereof and use of the same
02/10/2005WO2005012294A1 2,4-pyrimidinediamine compounds for use in the treatment or prevention of autoimmune diseases
02/10/2005WO2005012292A1 Gyrase inhibitors and uses thereof
02/10/2005WO2005012288A1 Bicyclic imidazol derivatives against flaviviridae
02/10/2005WO2005012281A1 Neuroprotective benzo[1,3]oxathol-2-ones
02/10/2005WO2005012275A2 Benzo [1, 2, 5] thiadiazole compounds as cck2 modulators
02/10/2005WO2005012272A1 Benzoxazepine compound
02/10/2005WO2005012271A2 Process for the synthesis of biaryl oxazolidinones
02/10/2005WO2005012263A1 5-ht2b receptor antagonists
02/10/2005WO2005012252A1 Novel 6-phenylphenantridines
02/10/2005WO2005011812A1 Cyanoamide compounds useful as malonyl-coa decarboxylase inhibithors
02/10/2005WO2005011693A1 Piperidine compounds useful as malonyl-coa decarboxylase inhibitors
02/10/2005WO2005011686A1 2-imino-4-(thio) oxo-5-poly cyclovinylazolines for use as p13 kinase ihibitors
02/10/2005WO2005011681A1 Chemical compounds
02/10/2005WO2005011611A2 Bicyclic compounds and compositions as pdf inhibitors
02/10/2005WO2005011601A2 6-menbered heteroaryl compounds for the treatment of neurodegenerative disorders
02/10/2005WO2004060305A3 Anti-cancer medicaments
02/10/2005WO2003099793A9 1,2-azole derivatives with hypoglycemic and hypolipidemic activity
02/10/2005US20050033059 Synthesis of epothilones, intermediates thereto, analogues and uses thereof
02/10/2005US20050032874 Indole derivatives
02/10/2005US20050032868 Selected substituted pyrazole derivatives and related compounds as bradykinin B1 receptor antagonists
02/10/2005US20050032864 Azolidinedione derivatives such as 5-[4-[[3-methyl-4-oxo-3,4-dihydro-2-quinazolinyl]methoxy]phenylmethyl]thiazolidine-2,4-dione potassium salt; dyslipidaemia; eating, cardiovascular and kidney disorders; atherosclerosis, obesity, psoriasis, polycystic ovarian syndrome; hypotensive agents
02/10/2005US20050032861 Antibiotic (vancomycin) resistant Grampositive and Gramnegative bacteria; cycloadditon, reduction, coupling, salt formation, deprotecting, amination, oxidation
02/10/2005US20050032858 Novel heterocyclic compound and anti-inflamatory agent