Patents
Patents for C07D 417 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group (62,773)
01/2005
01/19/2005CN1566099A Isoquinoline-1, 3, 4-trione compounds, preparation method and uses thereof
01/19/2005CN1566096A Prostaglandin agonists and their use to treat bonedisorders
01/19/2005CN1185230C N-substituted carbamoyloxyalkyl-azolium derivs.
01/19/2005CN1185228C Hydroxyphenyl-piperidin-4-ylidene-methyl-benzamide derivatives for treatment of pain
01/19/2005CN1185220C Para-amino substituted phenylamide glucokinase activators
01/19/2005CN1185217C Propanolamine derivatives, processes for their preparation, pharmaceuticals comprising these compounds, and their use
01/19/2005CN1185216C Fungicides
01/18/2005US6844357 Anticarcinogenic agents
01/18/2005US6844347 Substituted 4-amino-2aryl-pyrimidines, their production and use and pharmaceutical preparations containing same
01/18/2005US6844344 Depression, anxiety; tobacco or nicotine withdrawal; such as 1-(benzofuran-4-yl)oxy-3-(4-(6-methoxybenzo(b)thiophen-2-yl)piperidinyl)-2 -propanol oxalate
01/18/2005US6844342 Heterocyclic substituted 2-methyl-benzimidazole antiviral agents
01/18/2005US6844338 Piperidyindoles as serotonin receptor ligands
01/18/2005US6844295 2-Pyridin-2-yl derivatives
01/13/2005WO2005003128A1 Thiazolylpiperidine derivatives as mtp inhibitors
01/13/2005WO2005003127A1 Bicyclic heteroaromatic derivatives as modulators of cxcr3 function
01/13/2005WO2005003118A1 Amide-substituted 1,2,4-triazin-5(2h)-ones for the treatment of chronically inflammatory diseases
01/13/2005WO2005003103A2 2, 4, 6-tri-substituted 6-membered heterocycles and their use in the treatment of neurodegenerative diseases
01/13/2005WO2005003102A1 Methods of preparation of dehydro-diketopiperazines in liquid phase or of solid supported phase
01/13/2005WO2005003097A1 Cis-2,4,5-triaryl-imidazolines
01/13/2005WO2005003087A2 Oxazole derivatives as antibacterial agents
01/13/2005WO2005003071A1 Method for producing c1-c15 fragments of epothilones and the derivatives thereof
01/13/2005WO2005002577A1 Dual nk1/nk3 antagonists for treating schizophrenia
01/13/2005WO2004099192A3 Heterocycle substituted carboxylic acids as inhibitors of protein tyrosine phosphatase-1b
01/13/2005WO2004099134A3 Glutaminyl based dp iv-inhibitors
01/13/2005WO2004092130A3 N-containing heteroaromatic compounds as modulators of ppars and methods of treating metabolic disorders
01/13/2005WO2004064764A3 Substituted alkyl amido piperidines
01/13/2005WO2004050035A3 Benzimidazoles and analogs thereof as antivirals
01/13/2005US20050009892 Phenyloxazole derivatives lower blood triglyceride, glucose, insulin; hyperlipidemia, arteriosclerosis, diabetes mellitus, hypertension, obesity; 2-methyl-2-[6-(5-methyl-2-phenyloxazol-4-yl)-(E)-4-hexenyloxy]propionic acid
01/13/2005US20050009890 E.g., 1) (2R)-N-(4-phenoxybenzyl)-3-cyclohexylmethylthio-2-((4R)-3-methoxymethylcarbonylthiazolidin-4-ylcarbonylamino)propanamide; treatment of cerebral infarct, transient ischemic attack, encephalomyelopathy, spinal angiopathy, hypertension with stress, neurosis, epilepsy, asthma, pollakiuria, and pain
01/13/2005US20050009876 Indazole compounds, compositions thereof and methods of treatment therewith
01/13/2005US20050009874 Tetrahydropyridin or piperidino heterocyclic derivatives
01/13/2005US20050009873 1-Acyl-2,4-dicarbonyldihydropyrrole derivatives, e.g., rel-(2S,5R)-1-(4-tert-butylbenzoyl)-2-isobutyl-5-(1,3-thiazol-2-yl)-2,5-dihydro-1H-pyyrole-2,4-dicarboxylic acid; properation by acylating the corresponding dihydropyrrole derivative
01/13/2005US20050009870 3-(amino)sulfonylamino-substituted, e.g., N-(1,6-Dibenzyl-2-oxo-1,2,3,4-tetrahydroquinolin-3-yl)-benzenesulfonamide and N-(1-Benzyl-2-oxo-6-(thiophen-3-yl)-1,2,3,4-tetrahydroquinolin-3-yl)benzenesulfonamide; eating, metabolic, obesity, cognitive, neurological, pain, inflammatory and psychiatric disorders
01/13/2005US20050009867 Quinoline derivatives and their use as tyrosine kinase inhibitors
01/13/2005US20050009864 Substituted 4-phenyltetrahydroisoquinolinium, process for their preparation, their use as a medicament, and medicament containing them
01/13/2005US20050009855 1-(hydroxy, oxo, or epoxy)-3-oxo-3'-benzaminocarbonyl-4'-(carboxy or carboxylate)-1,2,3-trihydroindene-2-spiro-2'-tetrahydrofuran derivatives; these compounds interfere with the E1-E2-DNA complex during initiation of DNA replication
01/13/2005US20050009853 Pyrimidine derivatives for the treatment of abnormal cell growth
01/13/2005US20050009843 Thiazole derivatives of pyrido-1,2-a-pyrimidines, quinolones, pyridopyridazinoness, cinnolinones and naphthyridones; identifying a drug efflux pump expressed in a microorganism
01/13/2005US20050009840 2-amino- pyridines and pyrazines additionally substituted witn one or more carbocyclic or heterocyclic groups, e.g., 4-[6-amino-5-(2,6-dichloro-benzyloxy)-pyridin-3-yl]-phenol, for treating many kinds of cancer
01/13/2005US20050009839 Novel azoles having an insecticidal action
01/13/2005US20050009838 Piperidinyl-and piperazinyl-sulfonylmethyl hydroxamic acids and their use as protease inhibitors
01/13/2005US20050009834 E.g., 3-(2-chloro-6-fluorophenyl)-1-[4-(3,5-dichloropyridin-2-yloxymethyl)phenyl]-5-methyl-1H-1,2,4-triazole and 3-(3-chloropyridin-2-yl)-1-[4-(3-chloro-5-trifluoromethylpyridin-2-yloxymethyl)phenyl]-5-methyl-1H-1,2,4-triazole; for use as pesticides, especially insecticides and acaricides
01/13/2005US20050009829 1-Substituted 2-carboxamide derivatives of fused ring imidazoles, e.g., -[5-(5-Chloro-thiophen-2-yl)-isoxazol-3-ylmethyl]-1H-benzoimidazole-2-carboxylic acid (1-isopropyl-piperidin-4-yl)-amide
01/13/2005US20050009821 Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1
01/13/2005US20050009820 Thiochromenones used to combat painful conditions and neurodegenerative diseases
01/13/2005US20050009818 Therapeutic heterocyclic compounds
01/13/2005US20050009817 Substituted heteroaryls
01/13/2005US20050009816 Potassium channel modulators
01/13/2005US20050009785 Heterocyclic compounds
01/13/2005US20050009756 Polymorph of a pharmaceutical
01/13/2005US20050009058 Nitro-substituted non-fluorescent asymmetric cyanine dye compounds
01/13/2005DE10327472A1 New thia-epothilone derivatives useful in the preparation of medicaments for the treatment of cancer
01/13/2005CA2531078A1 Method for producing c1-c15 fragments of epothilones and the derivatives thereof
01/13/2005CA2530886A1 Dual nk1/nk3 antagonists for treating schizophrenia
01/13/2005CA2530816A1 Amide-substituted 1,2,4-triazin-5(2h)-ones for the treatment of chronic inflammatory diseases
01/13/2005CA2528119A1 Cis-2,4,5-triaryl-imidazolines
01/12/2005EP1496053A1 Kappa-opioid receptor agonist comprising 2-phenylbenzothiazoline derivative
01/12/2005EP1496052A1 Novel aminobenzamide derivative
01/12/2005EP1495018A1 Tricyclic thrombin receptor antagonists
01/12/2005EP1495005A1 Pyrazole compounds as anti-inflammatory and analgesic agents
01/12/2005EP1495002A1 Benzamide derivatives useful as histone deacetylase inhibitors
01/12/2005EP1495001A1 Antibacterial agents
01/12/2005EP1494671A1 1-(4-piperidinyl)benzimidazolones as histamine h3 antagonists
01/12/2005EP1494668A2 Use of benzimidazole analogs in the treatment of cell proliferation
01/12/2005EP1494667A1 Imidazole compounds as anti-inflammatory and analgesic agents
01/12/2005EP1494663A1 Derivatives of 1-(oxoaminoacetyl) pentylcarbamate as cathepsin k inhibitors for the treatment of bone loss
01/12/2005EP1434773A4 Heteroaryl substituted tetrazole modulators of metabotropic glutamate receptor-5
01/12/2005EP1353918B1 Morpholine derivatives as antagonists of orexin receptors
01/12/2005CN1564820A Heterocyclic compounds for use in the treatment of disorders of the urinary tract
01/12/2005CN1564817A Novel benzothiazine derivatives, their preparation and use
01/12/2005CN1564816A Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1
01/12/2005CN1564811A Acylsulfonamides as inhibitors of steroid sulfatase
01/12/2005CN1563003A Suitable industrialized method of preparing Lamivudine
01/12/2005CN1184215C Substd. oxazoles and thiazoles derivs. as HPPAR alpha activators
01/12/2005CN1184214C Alpha-acyl and alpha-heteroatom-bustituted benzene acetamide glucokinase activators
01/12/2005CN1184204C Piperidine compounds for use as CCR-3 inhibitors
01/12/2005CN1183989C Reaction crystallizing method for improving grain size
01/11/2005US6841682 Prevent binding of adrenergenic receptors
01/11/2005US6841674 N-heterocyclic derivatives as NOS inhibitors
01/11/2005US6841673 Enzyme inhibitors; antiinflammatory agents; rheumatic diseases; antidiabetic agents
01/11/2005US6841566 Viral polymerase inhibitors
01/11/2005US6841564 Tri-aryl-substituted-ethane PDE4 inhibitors
01/11/2005US6841560 Substituted isoquinoline derivatives and their use as anticonvulsants
01/11/2005CA2269128C Piperazino derivatives as neurokinin antagonists
01/11/2005CA2104909C Decahydroisoquinolines as excitatory amino acid receptor antagonists
01/11/2005CA2100924C Oxadiazine derivatives
01/06/2005WO2005000852A2 Product containing at least one phosphatase cdc25 inhibitor combined with at least one other anticancer agent
01/06/2005WO2005000844A1 Process for the preparation of insulin sensitizer and intermediate compound thereof
01/06/2005WO2005000843A2 Benzothiazole-4,7-diones and benzoxazole-4,7-diones with substituents in position 5 or 6 and method for production thereof
01/06/2005WO2005000842A1 Benzothiazole derivatives as adenosine receptor ligands
01/06/2005WO2005000826A1 Urea derivatives of piperazines and piperidines as fatty acid oxidation inhibitors
01/06/2005WO2005000821A1 Tachykinin receptor antagonists
01/06/2005WO2005000309A2 Chemical compounds
01/06/2005WO2005000298A2 5-membered heterocycle-based p-38 inhibitors
01/06/2005WO2005000249A2 Preparation of chemical compounds
01/06/2005WO2004101528A3 Isoquinoline derivatives and their use as gfat inhibitors
01/06/2005WO2004087646A3 Pyrrolidino-1,2-dicarboxy-1-(phenylamide)-2-(4-(3-oxo-morpholino-4-yl)-phenylamide) derivatives and related compounds for use as inhibitors of coagulation factor xa in the treatment of thrombo-embolic diseases
01/06/2005WO2004060281A3 2-aryl thiazole derivatives as kcnq modulators
01/06/2005WO2003042177A8 Piperidine derivatives and their use as modulators of chemokine receptor activity (especially ccr5)
01/06/2005US20050004360 Compounds and methods for modulation of estrogen receptors