Patents
Patents for C07D 413 - Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms (64,687)
02/2005
02/24/2005US20050043357 Mitotic kinesin inhibitors
02/24/2005US20050043337 Selective beta3 adrenergic agonists
02/24/2005US20050043336 Quinazoline derivatives as antitumor agents
02/24/2005US20050043335 Heterocyclic derivatives of glycinamide and their medical use
02/24/2005US20050043334 Such as N6-(4,5-dihydrooxazol-2-yl)-N4-[3-methyl-4-(6-methylpyridin-3-yloxy)-phenyl]-quinazoline-4,6-diamine; for treatment of hyperproliferative disorders such as cancer
02/24/2005US20050043331 Substituted 3-(2,5-disubstituted)pyridyl-4-aryl pyrroles for treating inflammatory diseases
02/24/2005US20050043330 Antiinflammation agents
02/24/2005US20050043326 Compounds
02/24/2005US20050043317 Biaryl heterocyclic compounds and methods of making and using the same
02/24/2005US20050043313 1-(phenylaminocarbonylmethyl)-3-alkylamino-5,6-disubstituted-2-pyazinones; serine protease inhibitors; anticoagulants; coronary artery and cerebrovascular diseases
02/24/2005US20050043310 Such as (R)-4-bromo-N-[1-(2,4-dichlorophenyl)-ethyl]-2-(quinoxaline-5-quinoxaline-sulfonylamino)-benzamide via sulfonylation; cholecystokinin receptor modulators
02/24/2005US20050043308 Process for total synthesis of ecteinascidins and intermediates therefor
02/24/2005US20050043305 Aryl substituted pyridines, pyrimidines, pyrazines and triazines and the use thereof
02/24/2005US20050043302 New indole derivatives as factor Xa inhibitors
02/24/2005US20050043295 Pharmaceutically effective compounds
02/24/2005US20050043292 eg S)-[5-amino-6-oxo-6-(3,3,4,4-tetrafluoro-pyrrolidin-1-yl)-hexyl-carbamic acid benzylester; Type 2 diabetes, metabolic syndrome (syndrome X or insulin resistance syndrome), hyperglycemia, impaired glucose tolerance, glucosuria, metabolic acidosis, arthritis, cataracts, diabetic neuropathy
02/24/2005US20050043290 for treating neurodegenerative disease such as Alzheimer's disease
02/24/2005DE102004010545A1 Pyrazoline Pyrazolines
02/24/2005CA2536470A1 Pyrrole compositions useful as inhibitors of c-met
02/24/2005CA2535665A1 Substituted arylalkanoic acid derivative and use thereof
02/24/2005CA2534950A1 Cyclic amine bace-1 inhibitors having a benzamide substituent
02/24/2005CA2534887A1 Process for the preparation of 2- (quinoxalin-5-ylsulfonylamino) -benzamide compounds
02/24/2005CA2534300A1 Aminopyrones and their use as atm inhibitors
02/24/2005CA2534047A1 Oxazoles derivatives, their manufacture and their use as tyrosine kinase inhibitors
02/24/2005CA2518774A1 Heterocyclic n-aryl carboxamides as cytokine inhibitors
02/24/2005CA2500358A1 Probes for diseases in which amyloid accumulates, agents for staining amyloid, drugs for treatment and prophylaxis of diseases with accumulated amyloid, and probes for diagnosis of neurofibrillary tangles and agents for staining neurofibrillary tangles
02/23/2005EP1507764A1 Novel enantiomers of tetrahydroisoquinoline derivatives and their pharmaceutically acceptable salts, their preparations and pharmaceutical compositions
02/23/2005EP1507762A1 Pesticidal pyridinecarboxamide derivatives
02/23/2005EP1507761A1 Pyridine carboxamide derivatives and their use as pesticides
02/23/2005EP1507756A1 Ccr9 inhibitors and methods of use thereof
02/23/2005EP1507549A2 Drug therapy for celiac sprue
02/23/2005EP1507528A2 Methods for using jnk inhibitors for treating or preventing disease-related wasting
02/23/2005EP1507504A1 Cycloalkyl inhibitors of potassium channel function
02/23/2005EP1395583B1 New phenylpiperazines
02/23/2005EP1317421B1 2-amino-2-alkyl-5 heptenoic and heptynoic acid derivatives useful as nitric oxide synthase inhibitors
02/23/2005EP1261606B1 Substituted oxazolidinones and their use in the field of blood coagulation
02/23/2005EP1177177B1 Substituted 4-oxo-quinoline-3-carboxamides: gaba brain receptor ligands
02/23/2005EP1133482B1 Il-5 inhibiting 6-azauracil derivatives
02/23/2005EP1041980B1 Acyl guanidine sodium/proton exchange inhibitors and method
02/23/2005CN1585768A Pyrazole derivatives as psychopharmaceuticals
02/23/2005CN1585763A Piperidine derivatives and their use as modulators of chemokine receptor activity especially CCR5
02/23/2005CN1585756A Substituted diphenyl heterocycles useful for treating HCV infection
02/23/2005CN1585754A Quinazoline derivatives as antitumor agents
02/23/2005CN1585749A Cannabinoid receptor ligands
02/23/2005CN1585742A Aryl aniline beta-2 adrenergic receptor agonists
02/23/2005CN1585643A Benzotriazepines as gastrin and cholecystokinin receptor ligands
02/23/2005CN1585633A Phenethanolamine derivatives for treatment of respiratory diseases
02/23/2005CN1585152A Current carrier transmtiting material with high-effect and balancing electronic cavity transmitting performance
02/23/2005CN1190434C Novel heterocyclic compounds and process for its preparation, and pharmaceutical compositions containing them and their use in treatment of diabetes and related diseases
02/23/2005CN1190433C Phenylpiperazine
02/23/2005CN1190432C Piperazing derivatives as 5-HTIB antagonists
02/23/2005CN1190424C Quinoline-containing Alpha-ketoamide cysteine and serine protease inhibitors
02/23/2005CN1190423C Heteroycle derivatives and drugs
02/22/2005US6858740 2-oxo-1-pyrrolidine derivatives, process for preparing them and their uses
02/22/2005US6858727 Intermediate of carbapenem antibiotics and process for the preparation thereof
02/22/2005US6858642 For use in pharmaceutical, skin-protective and cosmetic formulations
02/22/2005US6858638 Substituted indazoles, compositions containing them, method of production and use
02/22/2005US6858635 Photoreceptive detectors such as 2-(4-(4-((5S)-5-((Acetylamino )methyl)-2-oxo-3-oxazolidinyl)-2-fluorophenyl)-1-piperazinyl)-2-oxoethyl-4 -azido-2-hydroxy-5-iodobenzoate, used for analyzing binding in grampositive and negative bacteria
02/22/2005US6858628 Substituted cyclic amine metalloprotease inhibitors
02/22/2005US6858623 Amidino and guanidino peptidyl compounds
02/22/2005CA2218493C Benzimidazole compounds and their use as modulators of the gabaa receptor complex
02/22/2005CA2129039C Tri-substituted phenyl derivatives as phosphodiesterase inhibitors
02/17/2005WO2005014578A1 Phenylsulfonyl compounds as antipsychotic agents
02/17/2005WO2005014571A1 Substituted piperidines as histamine h3 receptor ligands
02/17/2005WO2005014559A1 Amide derivatives
02/17/2005WO2005014558A1 Condensed pyramidine compounds as inhibitors of voltage-gated ion channels
02/17/2005WO2005014554A1 1h-indazole-3-carboxamide compounds as mapkap kinase modulators
02/17/2005WO2005014552A1 Quinoline and quinazoline derivatives having affinity for 5ht1-type receptors
02/17/2005WO2005014540A1 Cyclic amine base-1 inhibitors having a heterocyclic substituent
02/17/2005WO2005014539A2 Pyrrole-based hmg-coa reductase inhibitors
02/17/2005WO2005014517A2 Novel dibenzo[b,f]oxepine-10-carboxamides and pharmaceutical uses thereof
02/17/2005WO2005013995A1 4-substituted 7-alkoxy-2-aminosulfonyl-1,2-dihydro-phtalazin derivatives as phosphodiesterase 4 inhibitors for the treatment of allergies and inflammations
02/17/2005WO2005013914A2 Heteroarylaminosulfonylphenyl derivatives for use as sodium or calcium channel blockers in the treatment of pain
02/17/2005WO2005013909A2 Novel cathepsin k inhibitors
02/17/2005WO2005013907A2 Pyrrolo[1,2-b]pyridazine derivatives
02/17/2005WO2004110993A3 N-ureidoalkyl-piperidines as modulators of chemokine receptor activity
02/17/2005WO2004110344A3 New azetidine compounds
02/17/2005WO2004108068A3 4-[4-(4-morpholino)anilino]pyrimidine derivatives, method for preparing thereof and antiviral pharmaceutical composition comprising the same
02/17/2005WO2004094386A8 Isoquinoline-5-sulfonic acid amides as inhibitors of akt (protein kinase b)
02/17/2005WO2004092115A3 Hydroxamates as therapeutic agents
02/17/2005WO2004084813A3 Chemical compounds
02/17/2005WO2004078114A3 Pyridine, pyrimidine, quinoline, quinazoline, and naphthalene urotensin-ii receptor antagonists.
02/17/2005WO2004069790A3 Crystalline modifications of triazinylaminostilbenes
02/17/2005WO2004002491A8 Morpholine and tetrahydropyran drivatives and their use as cathepsin inhibitors
02/17/2005WO2003097059A8 Polymorphic forms of phenyl oxazolidinone derivatives
02/17/2005US20050038247 topoisomerase inhibitors such as [5-(4-Cyclopropylcarbamoyl-imidazol-1-yl)-7-pyrimidin-2-yl-1H-benzoimidazol-2-yl]-carbamic acid ethyl ester, used for prophylaxis of bacterial infections in mammals
02/17/2005US20050038243 2, 4-pyrimidinediamine compounds and their uses
02/17/2005US20050038107 Substituted 2-phenyl benzofurans as estrogenic agents
02/17/2005US20050038099 3-Amido-5-substituted pyrazole derivatives and related compounds useful as bradykinin B1 receptor antagonists to relieve adverse symptoms in mammals mediated, at least in part, by bradykinin B1 receptor including pain, inflammation, septic shock, scarring process
02/17/2005US20050038092 effective against aerobic and anerobic pathogens such as multi-resistant staphylococci, streptococci and enterococci, Bacteroides spp., Clostridia spp. species; side effect reductions
02/17/2005US20050038091 Novel oxazoles, their manufacture and use as pharmaceutical agents
02/17/2005US20050038090 cytotoxic agents; made by fermentation of Streptomyces sparsogenes
02/17/2005US20050038087 Derivatives of heterocycles with 5 members, their preparation and their use as medicaments
02/17/2005US20050038086 Epothilone derivatives and methods for making and using the same
02/17/2005US20050038084 Phenylalanine enamide derivatives
02/17/2005US20050038074 Kinesin spindle protein (KSP) inhibitors, e.g., 4-(2,5-Difluorophenyl)-N-[(3S,4S)-3-fluoropiperidin-4-yl]-2-hydroxymethyl)-N-methyl-2-phenyl-2,5-dihydro-1N-pyrrole-1-carboxamide; antiproliferative and -carcinogenic agents
02/17/2005US20050038072 Nitrogeneous cyclic ketone derivative, process for producing the same, and use
02/17/2005US20050038069 Tumor necrosis factor antagonist; antiinflammatory agents; such as 2-Cyclopropyl-4-(3,5-dimethyl-4-pyridylmethoxy)-7-methoxy-3H-benzimidazole
02/17/2005US20050038067 A compound with azo containing mono and a bicyclic rings attached with an aryl or heteroaryl ring; both therapeutic and diagnostic
02/17/2005US20050038060 Spiropoperidine compounds as ligands for orl-1 receptor