Patents
Patents for C07D 409 - Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms (52,226)
09/2000
09/21/2000CA2368122A1 Novel compounds and compositions as protease inhibitors
09/21/2000CA2367595A1 Lxr modulators
09/21/2000CA2367461A1 Heterocyclic aromatic compounds useful as growth hormone secretagogues
09/20/2000EP1036793A2 A process for preparing 2-alkyl-3-aminothiophene derivative and 3-aminothiophene derivative
09/20/2000EP1036072A1 Thrombin receptor antagonists
09/20/2000EP1036067A2 Pdgf receptor kinase inhibitory compounds, their preparation and compositions
09/20/2000EP1036065A1 Substituted imidazole derivatives having agonist-like activity at alpha 2b or 2b/2c adrenergic receptors
09/20/2000EP1036063A1 Heteroaryl aminoguanidines and alkoxyguanidines and their use as protease inhibitors
09/20/2000CN1267300A Benzo (5,6) cyclohepta (1,2-b) pyridine derivs useful for inhibition of farnesyl protein transferase
09/20/2000CN1267299A Aminooxyamide tricyclic inhibitors of farnesylprotein transferase
09/20/2000CN1267293A Benzo (5,6) cyclohepta (1,2-b) pyridine derivs. useful for inhibition of farnesyl-protein transferase
09/19/2000US6121309 Fused-ring carboxylic acid derivatives
09/19/2000US6121308 Indole and benzimidazole antithrombotic compounds, such as 1-methyl-2-(n-(4-amidinophenyl)-aminomethyl)-5-(n-(hydroxycarbonylmethyl) -quinoline-8-sulphonylamino)-indole
09/19/2000US6121293 Benzothiophene compounds, compositions, and methods
09/19/2000US6121283 N-substituted-6-(2-(4-trifluoromethylphenyl)phenylcarbonyl-amino) -1,2,3,4-tetrahydroisoquinolines; treating disorders including obesity, hyperlipidemia, and diabetes; microsomal triglyceride transfer protein (mtp); apolipoprotein b (apo-b)
09/19/2000US6121271 Antidiabetic agents
09/19/2000US6121267 Substituted piperazines and piperidines as central nervous system agents
09/19/2000US6121260 Appetite stimulation with dosage of neuropeptide y (npy) receptor agonist
09/19/2000US6121258 For treatment of arthritis, cancer, cardiovascular disorders, skin disorders, ocular disorders, inflammation, gum disease
09/19/2000US6121204 Selective control of monocotyledonous and dicotyledonous weeds in monocotyledonous and dicotyledonous crops, both pre-emergence and post-emergence
09/19/2000US6121202 2-((thienyl or furyl) (oxy or thio))-pyridine and 6-((thienyl or furyl) (oxy or thio))-pyrimidine compounds
09/19/2000US6120696 Proton conductors in liquid form
09/14/2000WO2000053580A2 N-protected synthesis method for use in making porphyrins
09/14/2000WO2000053573A1 Medicinal compositions with [2.2.1] and [3.1.1] bicycloskeleton antagonistic to both of pgd2/txa2 receptors
09/14/2000WO2000053282A1 Crystallization process for producing fine crystal products
09/14/2000WO2000037469A3 Process for preparing n6-substituted deaza-adenosine derivatives
09/14/2000WO2000037422A3 Ion channel modulating agents
09/14/2000WO2000022129A9 Non-endogenous, constitutively activated human g protein-coupled receptors
09/13/2000EP1035121A1 Pyrrole derivatives, film-forming material and method of preparing the derivatives
09/13/2000EP1035113A2 Process for the preparation of 2-aryl-5-(perfluoroalkyl)pyrrole compounds from N-[1-chloro-1-(perfluoroalkyl)methyl]arylimidoyl chloride compounds
09/13/2000EP1034167A1 Alpha-alkylthio substituted pyrimidine ethers and thioethers as viral reverse transcriptase inhibitors
09/12/2000US6117987 Alkyl or aryl substituted dihydronaphthalene derivatives having retinoid and/or retinoid antagonist like biological activity
09/12/2000US6117898 Bicyclic amidine derivatives as inhibitors of nitric oxide synthetase
09/12/2000US6117874 Benzopyran and benzo-fused compounds, their preparation and their use as leukotriene B4 (LTB4 ) antagonists
09/12/2000US6117869 Compounds for and methods of inhibiting matrix metalloproteinases
09/12/2000US6117866 For inhibiting platelet aggregation or clot formation and reocclusion of an artery or vein in a mammal following fibrinolytic therapy or angioplasty; for treating stroke, transient ischemia attacks, or myocardial infarction
09/12/2000CA2105384C Treatment of addiction to drugs and substances of abuse
09/12/2000CA2047773C Derivatives of benzofuran, benzothiophene, indole and indolizine, process for their preparation as well as the compositions containing them
09/09/2000CA2300412A1 Process for the preparation of 2-aryl-5-(perfluoro-alkyl) pyrrole compounds from n-[1-chloro-1-(perfluoroalkyl) methyl] arylimidoyl chloride compounds
09/08/2000WO2000051986A1 Cyclopentanone dihydropyridine compounds useful as potassium channel openers
09/08/2000WO2000051610A1 Pyrrolidine modulators of chemokine receptor activity
09/08/2000WO2000051609A1 3-alkyl substituted pyrrolidine modulators of chemokine receptor activity
09/08/2000WO2000051608A1 3-thienyl and 3-furanyl pyrrolidine modulators of chemokine receptor activity
09/08/2000WO2000051607A1 3-cyclopropyl and 3-cyclobutyl pyrrolidine modulators of chemokine receptor activity
09/08/2000CA2330541A1 Cyclopentanone dihydropyridine compounds useful as potassium channel openers
09/06/2000EP1032559A1 Aminoalkylphenol derivatives and related compounds
09/06/2000EP1032556A1 Pharmaceutically active compounds and methods of use
09/06/2000EP1032393A1 QUINOLINE-CONTAINING $g(a)-KETOAMIDE CYSTEINE AND SERINE PROTEASE INHIBITORS
09/06/2000CN1265658A 5-naphthalen-1-yl-1,3-dioxane derivatives, preparation and therapeutic application
09/06/2000CN1265656A O-substituted hydroxycumaranone derivatives as anttumor and antimetastatic agents
09/06/2000CN1265654A 1-(N-phenylaminoalkyl)-piperazine derivatives substituted at position 2 of phenyl ring
09/06/2000CN1265649A Indole derivatives as MCP-1 receptor antagonists
09/06/2000CN1265591A Coumpound
09/06/2000CN1265394A Compound as intermediates for use in preparation of optically active 2-imidazoline-5-one or 2-imidazoline-5-thionone derivatives
09/06/2000CN1056144C New use of 6-heterocyclic-4-amino-3,4,5-tetrahydrobenz (CD) indoles compound
09/06/2000CN1056143C Piperidine derivatives and its use
09/05/2000US6114374 2-and 2,5-substituted phenylketoenols
09/05/2000US6114371 3-(cyclohexanoheteroarylidenyl)-2-indolinone protein tyrosine kinase inhibitors
09/05/2000US6114360 Pyrrole compounds
09/05/2000US6114359 Endothelin receptor antagonists
09/05/2000US6114354 N-substituted azaheterocyclic compounds
09/05/2000US6114335 Benzoylguanidine derivatives, process for their preparation their use in the preparation of medicines
09/05/2000US6114334 Piperazine derivatives as therapeutic agents
09/05/2000US6114330 Substituted 2,4-diaminopyrimidines
09/05/2000US6113937 Sustained release sufentanil compositions
09/05/2000CA2001160C Pyridine derivatives
08/2000
08/31/2000WO2000050470A2 Catalysts containing n-pyrrolyl substituted nitrogen donors
08/31/2000WO2000050419A1 Substituted bicyclic heterocycles and the use thereof as thrombin inhibitors
08/31/2000WO2000050405A1 Quinoline derivatives as tyrosine kinase inhibitors
08/31/2000WO2000050396A1 Aromatic sulfone hydroxamic acid metalloprotease inhibitor
08/31/2000WO2000050395A1 Sulfonamide-containing indole compounds
08/31/2000WO2000050390A1 N-substituted arylsulfonylamino hydroxamic acids useful as inhibitors of c-proteinase and for treating or preventing disorders related to unregulated collagen production
08/31/2000WO2000012074A3 Use of piperidines and/or piperazines as inhibitors of p38-alpha kinase
08/31/2000WO2000007996A3 Pyrazoles as estrogen receptor modulators
08/31/2000DE19907813A1 Substituierte bicyclische Heterocyclen, deren Herstellung und deren Verwendung als Arzneimittel Substituted bicyclic heterocycles, their preparation and their use as medicaments
08/31/2000CA2371876A1 Aromatic sulfone hydroxamic acid metalloprotease inhibitor
08/31/2000CA2364804A1 N-substituted arylsulfonylamino hydroxamic acids useful as inhibitors of c-proteinase and for treating or preventing disorders related to unregulated collagen production
08/31/2000CA2363628A1 Catalysts containing n-pyrrolyl substituted nitrogen donors
08/30/2000EP1031572A1 Pyridylpyrrole derivatives
08/30/2000EP1031563A1 Sulfonyl derivatives
08/30/2000EP1030844A1 Compounds which inhibit tryptase activity
08/30/2000EP1030843A1 Substituted benzene compounds, process for their preparation, and herbicidal and defoliant compositions containing them
08/30/2000EP1030840A1 Cyclic amine derivatives and their use as drugs
08/30/2000EP1030835A2 Urea derivatives and their use as integrin inhibitors
08/30/2000EP0821680B1 Novel taxoids, preparation thereof, and pharmaceutical compositions containing same
08/30/2000EP0710367B1 Photochromic substituted naphthopyran compounds
08/30/2000EP0690843B1 Formyl- or cyano- substituted indole derivatives having dopaminergic activity
08/30/2000CN1265107A Indole and 2,3-dihydronindole derivatives, their prepn. and use
08/30/2000CN1265106A Compounds derived from thophene and benzothiophene, and related utilisation and compsn.
08/30/2000CN1265033A Certain diarylimidaozle derivatives, new class of NPY speific ligands
08/29/2000US6110959 Carboxylic acid derivatives having fused rings
08/29/2000US6110953 A therapeutic drug mixture comprising a 1h-1,2,4-triazole with a chemotherapeutic agents can both reduce and suppress the growth of cancers, tumors and leukemia; synergistic effect
08/29/2000US6110947 An analgesic agent for treating stroke, abdominal pain; as antiinflammatory, diuretic, anesthetic or neuroprotective agents
08/29/2000US6110943 An antipsychotic agent, antidepressant and anxiolytic agent
08/29/2000US6110939 As a substance p antagonists treating tachykinin-mediated disease, asthma, central nervous system disorder
08/29/2000US6110936 A bactericide treating a bacterial infection in a warm blooded animal
08/29/2000US6110924 Barbituric acid derivatives, processes for their production and pharmaceutical agents containing these compounds
08/29/2000US6110910 Antiinflammatory agents, antiarthritic agents, antirheumatic agents, anticarcinogenic agents
08/29/2000US6110872 2,4,5-trisubstituted phenylketo-enols for use as pesticides and herbicides
08/29/2000US6110871 2-((phenyl, pyridyl or pyrazolyl)(oxy or thio)), 6-((substituted)phenyl)-cyanopyridines; herbicidal activity with the necessary selectivity and enhanced soil degradation