Patents
Patents for C07D 409 - Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms (52,226)
02/2001
02/27/2001US6194574 Selectively bind to corticotropin-releasing factor (crf1) receptors; for treating stress related disorders such as post traumatic stress disorder (ptsd) as well as depression, headache and anxiety
02/27/2001US6194450 Polyaromatic heterocyclic compounds and pharmaceutical compositions comprised thereof
02/27/2001US6194448 N, N-disubstituted amides that inhibit the binding of integrins to their receptors
02/27/2001US6194438 Derivatives of 2-(2-oxo-ethylidene)-imidazolidin-4-one, and compositions and methods for inhibiting abnormal cell growth comprising said derivatives
02/27/2001US6194427 Brain disorders; psychological disorders; sleep disorders; anticonvulsants
02/27/2001US6194418 Bactericides, pesticides
02/27/2001US6194406 Histamine receptor antagonists; tachykinin receptor antagonists; asthma; bronchitis; inflammatory bowel diseases, including crohn's disease and ulcerative colitis; seasonal rhinitis; sinusitis; antiallergens; emetic agents
02/27/2001CA2317053A1 New pyridine derivatives, the process for preparing them and the pharmaceutical compositions that contain them
02/22/2001WO2001012609A1 Pyrazoloanthrone and derivatives thereof as jnk inhibitors and their compositions
02/22/2001WO2001012604A1 Fungicides
02/22/2001WO2001012600A1 INHIBITORS OF FACTOR Xa
02/22/2001WO2001012575A1 Methods for preparing perfluorinated [18f]-radiolabelled nitroimidazole derivatives for cellular hypoxia detection
02/22/2001WO2001012189A1 3(5)-amino-pyrazole derivatives, process for their preparation and their use as antitumor agents
02/22/2001WO2001012187A2 Benzoic acid derivatives and their use as ppar receptor agonists
02/22/2001WO2001012186A1 Cell adhesion inhibitors
02/22/2001WO2001011966A1 Fungicides
02/22/2001WO2001011965A1 Fungicides
02/22/2001WO2000055126A3 N-cyanomethylamides as protease inhibitors
02/22/2001WO2000039716A3 Arylpropenylimidazoles as farnesyl-protein transferase inhibitors
02/22/2001WO2000032588A3 Carboxylic acids and carboxylic acid isosteres of n-heterocyclic compounds
02/22/2001DE19939756A1 New 1-(1-ethyl-piperidin-4-yl)-1-(phenyl or heterocyclyl)-alkanol derivatives, are 5-HT(2A) receptor antagonists useful e.g. for treating schizophrenia, depression, memory disorders or eating disorders
02/22/2001DE19939463A1 Tryptase inhibitors useful e.g. for treating inflammatory or allergic disease, arteriosclerosis or neoplasia, comprising new or known 2-phenethyl-benzimidazole-5-carboxamides
02/22/2001DE10025830A1 New 4-acyl-2,3-dihydro-benzofuran or -benzothiophene derivatives, useful as pre- or post-emergence, total or selective herbicides or as plant growth inhibitors
02/22/2001CA2383268A1 Pyrazoloanthrone and derivatives thereof as jnk inhibitors and their compositions
02/22/2001CA2380817A1 Cell adhesion inhibitors
02/22/2001CA2380775A1 Benzoic acid derivatives and their use as ppar receptor agonists
02/22/2001CA2378712A1 Methods for preparing perfluorinated [18f]-radiolabelled nitroimidazole derivatives for cellular hypoxia detection
02/21/2001EP1077213A2 Inhibition of serotonin reuptake
02/21/2001EP1076557A1 Ccr-3 receptor antagonists
02/21/2001CN1284947A Carboxyl acid substituted heterocycles as metalloproteinase inhibitors
02/21/2001CN1284946A Substituted isoquinoline derivatives and their use as anticonvulsants
02/21/2001CN1284945A Substituted pyriding and pyridazine compounds and their pharmaceutical use
02/21/2001CN1062270C Amino-acid derrivatives having benzothiophene ring, prep. thereof and use as fungus-killing agent
02/21/2001CN1062269C Novel (R)-5-carbamyl-8-fluoro-3-N, N-disubstituted amino-3, 4-dihydro-2H-1-benzopyranes
02/21/2001CN1062265C Method for producing triazine derivatives
02/21/2001CN1062264C Amino-acid indole or quinoline derivatives, prep. thereof and use as fungus-killing agent
02/20/2001US6191266 Sugar modified nucleosides
02/20/2001US6191149 Heterocyclic derivative and medicine
02/20/2001US6191134 Stroke therapy, antiischemic agents, brain disorders
02/15/2001WO2001010863A2 Substituted thienyl(amino)sulfonylureas
02/15/2001WO2001010847A2 Novel integrin receptor antagonists
02/15/2001WO2001010842A2 Melanocortin-4 receptor binding compounds and methods of use thereof
02/15/2001WO2001010799A1 Methods for preparing n-[(aliphatic or aromatic)carbonyl)]-2-aminoacetamide compounds and for cyclizing such compounds
02/15/2001WO2001010381A2 Methods for treating or preventing pain and anxiety
02/15/2001WO2001010380A2 Benzanilides as potassium channel openers
02/15/2001WO2000064874A3 Heterosubstituted pyridine derivatives as pde 4 inhibitors
02/15/2001WO2000054759A3 Lxr modulators
02/15/2001DE19936780A1 Neue Antagonisten von Integrinrezeptoren New antagonists of integrin
02/15/2001CA2381008A1 Melanocortin-4 receptor binding compounds and methods of use thereof
02/15/2001CA2379977A1 Novel integrin receptor antagonists
02/15/2001CA2378241A1 Benzanilides as potassium channel openers
02/14/2001EP1075475A1 Heterocyclic carboxamide derivatives as inhibitors of nitric oxide production
02/14/2001EP1075470A1 Novel analgesic and immunomodulatory cannabinoids
02/14/2001EP1075467A1 Pyrazole derivatives as p-38 map kinase inhibitors
02/14/2001EP1075466A1 Cyclopentanone dihydropyridine compounds useful as potassium channel openers
02/14/2001EP0836593B1 5-pyrazolylbenzoic acid derivatives as herbicides
02/14/2001EP0773964B1 Gas phase production of polydienes
02/14/2001EP0714897B1 Fused heteroaromatic cyclopentene derivative having endothelin-antagonist activity
02/14/2001EP0708767B1 Haptens, tracers, immunogens and antibodies for carbazole and dibenzofuran derivatives
02/14/2001CN1284069A Substituted 2,4-diamino-1,3,5-triazines
02/14/2001CN1284068A Substituted phenyl uracils
02/14/2001CN1284066A Substituted inidazole derivatives having agonist-like activity at alpha 2B or 2B/2C adrenergic receptors
02/14/2001CN1284064A 2,3-substituted indole compounds as cox-2 inhibitors
02/14/2001CN1283622A 6-hydroxy-3(4-[2-(piperidine-1-group)oxyethyl group]phenoxy)-2-(4-methoxy phenyl) benzo[b] thiophene hydrochloride salt
02/14/2001CN1061977C Aryl substituted heterocycles
02/13/2001US6187944 A phenyl acrylonitrile compounds useful as active ingredients of an insecticide, a miticide, a nematicide, a soil pesticide, a fungicide and a marine antifouling agent
02/13/2001US6187933 Bind to retinoid receptors; treating skin disorders
02/13/2001US6187805 Indole and indoline derivatives as 5-HT6 selective ligands
02/13/2001US6187799 Inhibition of raf kinase activity using aryl ureas
02/13/2001US6187792 Compounds with analgesic effect
02/13/2001US6187781 Corticotropin releasing factor receptor antagonists; alzheimer*s, huntington, and parkinson disease; antidepressants, anxiolytic agents
02/08/2001WO2001055118A1 Benzene-fused heterocycle derivatives and drugs containing the same as the active ingredient
02/08/2001WO2001009138A2 Chemokine receptor antagonists and methods of use therefor
02/08/2001WO2001009126A1 Serotonergic benzothiophenes
02/08/2001WO2001009121A2 2-pyrazolin-5-ones_as tyrosine kinase inhibitors
02/08/2001WO2001009120A1 Amine and amide derivatives as ligands for the neuropeptide y y5 receptor useful in the treatment of obesity and other disorders
02/08/2001WO2001009119A2 Chemokine receptor antagonists
02/08/2001WO2001009116A2 A NOVEL CRYSTALLINE FORM OF 6-HYDROXY-3- (4-[2-(PIPERIDIN-1-YL) ETHOXY]PHENOXY)- 2-(4-METHOXYPHENYL)BENZO[b]THIOPHENE HYDROCHLORIDE
02/08/2001WO2001009115A2 A NOVEL CRYSTALLINE FORM OF 6-HYDROXY-3- (4-[2-(PIPERIDIN-1- YL)ETHOXY] PHENOXY)-2- (4-METHOXYPHENYL) BENZO[b]THIOPHENE HYDROCHLORIDE
02/08/2001WO2001009110A1 Novel succinate derivative compounds useful as cysteine protease inhibitors
02/08/2001WO2001009106A1 Diamino-1,2,4-triazole-carboxylic and derivatives as gsk-3 inhibitors
02/08/2001WO2001009094A2 Chemokine receptor antagonists and methods of use therefor
02/08/2001WO2001009090A2 Hydantoin, thiohydantoin, pyrimidinedione and thioxopyrimidinone derivatives, preparation method and use as medicines
02/08/2001WO2001008685A1 Acyclic and cyclic amine derivatives
02/08/2001WO2001008673A1 Calcilytic compounds
02/08/2001WO2000076984A3 Novel compounds, their use and preparation
02/08/2001WO2000069855A3 Furanone derivatives as inhibitors of cathepsin s
02/08/2001WO2000059898A3 Process for the dehalogenation of thiochroman and dihydrobenzothiophene derivatives
02/08/2001DE19937118A1 Substituierte Thienyl(amino)sulfonylharnstoffe Substituted thienyl (amino) sulfonylureas
02/08/2001CA2391267A1 Chemokine receptor antagonists and methods of use therefor
02/08/2001CA2380644A1 2-pyrazolin-5-ones
02/08/2001CA2380081A1 Calcilytic compounds
02/08/2001CA2380032A1 Amine and amide derivatives as ligands for the neuropeptide y y5 receptor useful in the treatment of obesity and other disorders
02/08/2001CA2379993A1 Acyclic and cyclic amine derivatives
02/08/2001CA2378879A1 Serotonergic benzothiophenes
02/07/2001EP1074551A2 Phenylpyrazoles with a herbicidal activity
02/07/2001EP1074542A1 Sulfonamide-containing indole compounds
02/07/2001EP1073650A1 Guanidine derivatives
02/07/2001EP1073642A1 The use of dihydropyrimidines as medicaments, and novel substances
02/07/2001EP1073637A1 3-(amino- or aminoalkyl)pyridinone derivatives and their use for the treatment of hiv related diseases