Patents
Patents for C07D 401 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom (107,979)
05/2002
05/15/2002CN1349503A Renin ihibitors
05/15/2002CN1349500A 3,3-substituted indoline derivatives
05/15/2002CN1349416A Contraceptive compositions contaiing indoline derivatives and progestational agents
05/15/2002CN1348956A Substituted diazacycloheptane compound, medicine composite contg. same and the use thereof
05/15/2002CN1084751C Palladium catalyzed indolization
05/15/2002CN1084744C N-substituted azaheterocyclic compounds
05/15/2002CN1084743C 毒蕈碱拮抗剂 Muscarinic antagonist
05/15/2002CN1084620C Medicine for prophylaxis and treatment of thromboxane A2-mediated diseases
05/15/2002CN1084619C Process for preparing medicine composition
05/14/2002US6388094 Method for making intermediates useful in synthesis of retroviral protease inhibitors
05/14/2002US6388092 Antitumor agent
05/14/2002US6388088 Antidiabetic agents
05/14/2002US6388081 4-substituted-quinoline derivatives and 4-substituted-quinoline combinatorial libraries
05/14/2002US6388080 Polymorphic forms of 6-[4-(1-cyclohexyl-1H-tetrazol-5-yl)butoxy]-3,4-dihydro-2(1H)-quinolinone
05/14/2002US6388071 Alkynyl phenyl heteroaromatic glucokinase activators
05/14/2002US6387992 Heat, oxidation and light resistance
05/14/2002US6387940 Heterocyclylmethyl-substituted pyrazole derivatives
05/14/2002US6387932 Somatostatin agonists
05/14/2002US6387930 Antiarthritic agents; antiallergens; skin disorders; inflammatory bowel disorders
05/14/2002US6387929 4-heteroaryl-tetrahydroquinolines and their use as inhibitors of the cholesterin-ester transfer protein
05/14/2002US6387928 Antimicrobial quinolones, their compositions and uses
05/14/2002US6387926 Inhibitors of farnesyl protein transferase
05/14/2002US6387919 Substituted oxindole derivatives as protein tyrosine kinase and as protein serine/threonine kinase inhibitors
05/14/2002US6387915 Isoxazole-sulfonamide endothelin antagonists
05/14/2002US6387911 Pyrazinone thrombin inhibitors
05/14/2002US6387905 Compounds useful for inhibition of farnesyl protein transferase
05/14/2002US6387898 Treatment for CNS injuries
05/14/2002US6387897 Preferentially substituted calcium channel blockers
05/14/2002US6387893 Adrenergic blocking agent; benign prosatatic hyperplasia
05/14/2002CA2267186C Method of using cyclooxygenase-2 inhibitors in the treatment and prevention of neoplasia
05/14/2002CA2247105C Novel substituted n-methyl-n-(4-(4-(1h-benzimidazol-2-yl-amino)piperidin-1-yl)-2-(aryl)butyl)benzamides useful for the treatment of allergic di seases
05/14/2002CA2150162C New n-pyridyl carboxamides and derivatives thereof, preparation processes thereof and pharmaceutical compositions containing thereof
05/14/2002CA2105071C Use of nicotinic analogs for treatment of degenerative diseases of the nervous system
05/10/2002WO2002036734A2 Aza-and polyaza-naphthalenyl ketones useful as hiv integrase inhibitors
05/10/2002WO2002036589A1 Indolylpiperidine derivatives as antihistaminic and antiallergic agents
05/10/2002WO2002036586A1 N-type calcium channel antagonists for the treatment of pain
05/10/2002WO2002036577A1 Quinazoline derivatives and drugs
05/10/2002WO2002036576A1 Phthalazinone derivatives
05/10/2002WO2002036575A1 Tagging compounds and process for use in aida libraries
05/10/2002WO2002036573A2 8- substituted-2, 6-methano-3-benzazocines and 3-substituted morphinanes as opioid receptor binding agents
05/10/2002WO2002036570A1 4-substituted quinolines as antitumor agents
05/10/2002WO2002036567A1 N-type calcium channel antagonists for the treatment of pain
05/10/2002WO2002036564A1 Sulfonylamino substituted 3-(aminomethylide)-2-indolinones as cell proliferation inhibitors
05/10/2002WO2002036560A1 Aminoalkylpyrrolidine serotonin receptor ligands and compositions, their pharmaceutical uses, and methods for their synthesis
05/10/2002WO2002036173A2 Simultaneous dual isotope imaging of cardiac perfusion and cardiac inflammation
05/10/2002WO2002036119A1 Δ2,-1,2,3-triazoline anticonvulsants and their active metabolite analogues, the aminoalkylpyridines, are excitatory amino acid antagonists and antiischemic agents, useful in the treatment of cerebral ischemia resulting from stroke
05/10/2002WO2002036116A2 Tripeptidyl peptidase inhibitors
05/10/2002WO2002022600A3 Chemokine receptor binding heterocyclic compounds
05/10/2002WO2002020437A3 Basic compounds containing tertiary amides with activity on tachykinin receptors, and pharmaceutical compositions containing them
05/10/2002WO2002016338A8 Aminoalkenylbenzoyl-benzofuran or benzothiophene derivatives, method for preparing same and compositions containing same
05/10/2002WO2002008200A3 Arylethene-sulfonamides, their preparation and their use as endothelin antagonists
05/10/2002WO2001081342A3 Novel epothilone derivatives, method for the preparation thereof and their pharmaceutical use
05/10/2002WO2001038324A3 Imidazole derivatives and their use as raf kinase inhibitors
05/10/2002WO2001034600A9 Protease inhibitors
05/10/2002WO2001034599A9 Protease inhibitors
05/10/2002WO2001032650A3 Alkaline salts of n-(6-alkyl-2,4-dioxo-1,2,3,4-tetrahydro-5-pyrimidinesulfone)-n'-isonicotinoylhydrazide, possess for their preparation, and pharmaceutical composition based on these salts
05/10/2002WO2001024827A3 INHIBITORS OF THE ENDOTHELIN SIGNALLING PATHWAY AND αVβ3 INTEGRIN RECEPTOR ANTAGONISTS FOR COMBINATION THERAPY
05/10/2002CA2427911A1 Simultaneous dual isotope imaging of cardiac perfusion and cardiac inflammation
05/10/2002CA2427589A1 Indolylpiperidine derivatives as antihistaminic and antiallergic agents
05/10/2002CA2425286A1 Aminoalkylpyrrolidine serotonin receptor ligands and compositions, their pharmaceutical uses, and methods for their synthesis
05/10/2002CA2425067A1 Aza-and polyaza-naphthalenyl ketones useful as hiv integrase inhibitors
05/09/2002US20020055639 Pyrazole derivatives as herbicides
05/09/2002US20020055632 Such as (3R,5S)-1-pyrimidin-2-yl-5-(2,4,5-trifluoro-benzyloxymethyl)-pyrrolidine-3 -thiol trifluoro-acetate useful as inhibitors of metalloproteases for treating diseases associated with vasoconstriction
05/09/2002US20020055631 N-acylsulfonamide apoptosis promoters
05/09/2002US20020055524 Novel aryl substituted tetrahydroindazoles as ligands of the GABA receptor
05/09/2002US20020055522 Treatment of thrombotic diseases, asthma, emphysema, cirrhosis, arthritis, carcinoma, melanoma, restenois, atheroma, trauma, shock and reperfusion injury.
05/09/2002US20020055516 Nitrogen-containing heterocyclic compounds and medicaments containing the compounds
05/09/2002US20020055507 Ureas and thioureas inhibit production of cytokines
05/09/2002US20020055501 Treatment of neurological disorders related to beta -amyloid production such as Alzheimer's disease and Down's Syndrome.
05/09/2002US20020055499 Integrin receptor antagonists
05/09/2002US20020055469 Anticoagulants
05/09/2002US20020055437 Stability of liquid formulations of various pesticides can be enhanced by utilizing quaternary ammoniuim salts
05/09/2002US20020054926 Administering tobacco extract, Yerbamate extract, and extract of chewing gum and lozenges for increasing levels of norepinephrine, dopamine, and serotonin to treat psychological disorders and aid in smoking cessation
05/09/2002US20020054899 Methods and compositions for the prevention and treatment of atherosclerosis, restenosis and related disorders
05/08/2002EP1203767A1 Heterocyclic-substituted alkylamide acat inhibitors
05/08/2002EP1203766A2 Carboxylic acid derivatives that inhibit the binding of integrins to their receptors
05/08/2002EP1202990A2 Neurotrophic pyrrolidines and piperidines, and related compositions containing them
05/08/2002EP1202988A2 Novel integrin receptor antagonists
05/08/2002EP1202987A2 Quinoline derivatives and their use as antibacterial agents
05/08/2002EP1202986A1 Amine and amide derivatives as ligands for the neuropeptide y y5 receptor useful in the treatment of obesity and other disorders
05/08/2002EP1202985A2 Chemokine receptor antagonists
05/08/2002EP1202984A1 Novel diphenyl-piperidine derivate
05/08/2002EP1202976A1 Pyrazinones, compositions containing such compounds
05/08/2002EP1202975A1 Substituted polycyclic aryl and heteroaryl pyrazinones useful for selective inhibition of the coagulation cascade
05/08/2002EP1202971A2 Pharmaceutical compositions comprising 4-quinolones
05/08/2002EP1202969A2 Biphenyl derivatives, production thereof and use as medicines
05/08/2002EP1202968A2 Antibacterial agents
05/08/2002EP1202966A1 Piperidine alcohols
05/08/2002EP1202738A1 Dihydropyrazine derivatives as npy antagonists
05/08/2002EP1202736A1 Nicotine in therapeutic angiogenesis and vasculogenesis
05/08/2002EP1202733A1 3(5)-amino-pyrazole derivatives, process for their preparation and their use as antitumor agents
05/08/2002EP1202729A1 Phosphate transport inhibitors
05/08/2002EP0914332B1 Isoquinolines useful as analgesics
05/08/2002EP0804464B1 Aromatic heterocyclic derivatives as enzyme inhibitors
05/08/2002EP0790994B1 Heterocycle substituted propenoic acid derivatives as nmda antagonists
05/08/2002CN1348450A Tetrahydroisoquinolinyl-indole derivatives for the treatment of depression
05/08/2002CN1348449A Heteroaryl diazacycloalkanes, their preparation and use
05/08/2002CN1348444A 丝氨酸蛋白酶抑制剂 Serine protease inhibitors
05/08/2002CN1348363A Novel pharmaceutical salt form
05/08/2002CN1347881A 法呢基蛋白转移酶抑制剂 Farnesyl protein transferase inhibitor