Patents
Patents for C07D 401 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom (107,979)
04/2002
04/09/2002US6369074 Aminomethylene substituted non-aromatic heterocycles and use as substance P antagonists
04/09/2002US6369069 Cardiovascular disorders
04/09/2002US6369068 Amino substituted pyrimidine containing compounds
04/09/2002US6369061 4-bromo-6-(3-(4-chlorophenyl)propoxy)-5-(3-pyridylmethylamino) -3(2h)-pyridazinone
04/09/2002US6369060 Central nervous system disorders such as anxiety; 5-methyl-6-trifluoromethyl-1-(6-(2-methylpyridin-3-yloxy)-pyridin-3-yl carbamoyl)indoline and 5-methyl-1-(6-(2-methylpyridin-3-yloxy) -pyridazin-3-ylcarbamoyl)-6-trifluoromethylindoline
04/09/2002US6369057 Quinoxalines, processes for their preparation and their use
04/09/2002US6369053 2-Aminoquinolinecarboxamides: neurokinin receptor ligands
04/09/2002US6369002 Hetero is pyrimidine or pyridazine; 1-(3-fluoro-5-chloro pyridin-2-yl)-3-methyl-4-trifluoromethylpyrimidin-2,6-dione
04/09/2002US6368520 Synergistic stabilizer mixture
04/09/2002CA2229000C 1-biphenylimidazole derivatives, their preparation and their therapeutic use
04/09/2002CA2215732C Quinazoline derivatives
04/09/2002CA2095338C Individual stereoisomers of 7-¬3-(aminoalkyl)-1-pyrrolidinyl|-quinolonesand naphthyridones as antibacterial agents
04/09/2002CA2048842C Substituted pyrimidine derivatives, a process for the preparation thereof and the use thereof as reagents
04/04/2002WO2002026734A1 PIPERAZIN-2-ONE AMIDES AS INHIBITORS OF FACTOR Xa
04/04/2002WO2002026731A2 Quaternary amidino based inhibitors of factor xa
04/04/2002WO2002026720A2 PIPERAZINE BASED INHIBITORS OF FACTOR Xa
04/04/2002WO2002026718A2 Bicyclic pyrimidin-4-one based inhibitors of factor xa
04/04/2002WO2002026714A1 Spiro compounds
04/04/2002WO2002026708A1 Nitrogen-containing compounds and ccr3 inhibitors containing the same as the active ingredient
04/04/2002WO2002014281A8 Pyridine derivatives as inhibitors of p38
04/04/2002WO2002008195A8 Pyrazolyl biphenyl carboxamides and the use thereof for controlling undesired microorganisms
04/04/2002WO2002004421A3 Pyridoxine and pyridoxal analogues: cardiovascular therapeutics
04/04/2002WO2002002521A3 Aroyl aminoacyl pyrrole compounds and their pharmaceutical use
04/04/2002WO2001090079A3 Novel carbamates and carbamides, production and use thereof as endothelin receptor antagonists
04/04/2002WO2001089451A3 Protease inhibitors
04/04/2002WO2001087376A8 Drug/drug delivery systems for the prevention and treatment of vascular disease
04/04/2002WO2001087263A3 Delivery systems for treatment of vascular disease
04/04/2002WO2001081308A3 Aminopiperidines for use as glyt-1 inhibitors
04/04/2002WO2001074815A3 Phenyl-substituted imidazopyridines
04/04/2002WO2001074810A3 Method for using 2-aryloxyalkylaminobenzoxazoles and 2-aryloxyalkylaminobenzothiazoles as h3 antagonists
04/04/2002WO2001074773A3 Phenyl-substituted indoles as histamine h3-receptor antagonists
04/04/2002WO2001066098A3 Therapeutic uses of ppar mediators
04/04/2002WO2001064643A3 Benzamides and related inhibitors of factor xa
04/04/2002WO2001047898A3 Substituted piperazine derivatives and their use as inhibitors of the microsomal triglyceride transfer protein (mtp)
04/04/2002WO2001047507A3 Combinations of receptor tyrosine kinase inhibitor with an a1-acidic glycoprotein binding compound
04/04/2002US20020040148 Diphenyl heterocyclic thioamide derivatives
04/04/2002US20020040147 Novel catechols as antimicrobial agents
04/04/2002US20020040146 Useful as inhibitors of metalloproteases, e.g. zinc proteases, and which are effective in therapy of disease states associated with vasoconstriction
04/04/2002US20020040144 For therapy of thrombotic disease, asthma, emphysema, cirrhosis, arthritis, carcinoma, melanoma, restenois, atheroma, trauma, shock and reperfusion injury
04/04/2002US20020040140 Crystalline therapeutic agent
04/04/2002US20020040136 Vitronectin receptor antagonist
04/04/2002US20020040048 (2S,4R)-4-Mercapto-1-(naphthalene-2-sulfonyl)-pyrrolidine-2 -carboxylic acid N'-isobutyl-N'-(4-methyl-benzenesulfonyl)-hydrazide, for example; inhibitors of metalloproteases, e.g. zinc proteases; vasodilators
04/04/2002US20020040040 N-(3,5-bis-trifluoromethyl-benzyl)-6-(4-hydroxyacetyl-piperazin-1 -yl)-N-methyl-4-o-tolyl-nicotinamide, for example
04/04/2002US20020040028 2-amine substituted quinoline or quinozoline derivatives useful for treating benign prostatic hyperplasia
04/04/2002US20020040026 Phenyloxy-and phenylthiosubstituted pyrimidines and triazines and derivatives useful for treating anxiety, depression, effective disorders, post-traumatic stress disorders etc.
04/04/2002US20020040024 A phenoxy substituted piperidine derivative, useful for treating or preventing histamine H3 receptor activity
04/04/2002US20020040016 Derivatives of azetidine and pyrrolidine
04/04/2002US20020039998 Administering to human therapeutically effective amount of a combination of drug which is metabolized by cytochrome p450 monooxygenase or pharmaceutically acceptable salt thereof and ritonavir
04/04/2002US20020039598 Stabilized pharmaceutical composition and its production
04/04/2002DE10044792A1 Substituierte Phenylcyclohexancarbonsäureamide und ihre Verwendung Substituted Phenylcyclohexancarbonsäureamide and their use
04/04/2002CA2422873A1 Piperazin-2-one amides as inhibitors of factor xa
04/03/2002EP1193266A1 Quinolinecarboxylic acid derivative or salts thereof
04/03/2002EP1193265A2 A process for the preparation of 4-[2-(aryl or heterocyclo)-1H-imidazol-1-yl]benzenesulfonamides
04/03/2002EP1193259A1 Dihydropyrimidine derivatives
04/03/2002EP1192189A2 Catalysts containing n-pyrrolyl substituted nitrogen donors
04/03/2002EP1192139A1 Preparation of quinoline-substituted carbonate and carbamate derivatives
04/03/2002EP1192137A1 COMPOUNDS FOR THE MODULATION OF PPAR$g(g) ACTIVITY
04/03/2002EP1192135A2 Serine protease inhibitors
04/03/2002EP1192133A1 N-cyclopentyl modulators of chemokine receptor activity
04/03/2002EP1192132A2 Serine protease inhibitors
04/03/2002EP1192131A1 Method of inhibiting amyloid protein aggregation and imaging amyloid deposits using isoindoline derivatives
04/03/2002EP1192129A2 Pharmaceutical compounds
04/03/2002EP1162201A9 Farnesyl protein transferase inhibiting (imidazol-5-yl)methyl-2-quinolinone derivatives
04/03/2002EP1161240A4 N-ureidoalkyl-piperidines as modulators of chemokine receptor activity
04/03/2002EP1158980A4 N-ureidoalkyl-piperidines as modulators of chemokine receptor activity
04/03/2002EP1156807A4 N-ureidoalkyl-piperidines as modulators of chemokine receptor activity
04/03/2002EP1140087A4 N-ureidoalkyl-piperidines as modulators of chemokine receptor activity
04/03/2002EP1007512B1 Branched alkoxy-subsituted 2-aminopyridines as nos inhibitors
04/03/2002EP0865440B1 Farnesyl protein transferase inhibiting (imidazol-5-yl)methyl-2-quinolinone derivatives
04/03/2002EP0865281B1 Naphthyl-substituted benzimidazole derivatives as anticoagulants
04/03/2002CN1343201A Bicyclic heterocycles, pharmaceutical compositions containing these compounds, and processes for preparing them
04/02/2002US6365621 Remedies or preventives for intractable epilepsy
04/02/2002US6365603 Aromatic compounds and pharmaceutical compositions containing them
04/02/2002US6365602 For therapy of depression, anxiety, asthma, pain, inflammation, urinary incontinence and other disease conditions
04/02/2002US6365600 For therapy of condition associated with smooth muscle cell proliferation in a warm-blooded animal which comprises administering imidazol-5-yl-methyl-2-quinolinone derivatives
04/02/2002US6365599 For therapy of benign prostatic hyperplasia
04/02/2002US6365588 Tricyclic amide and urea compounds useful for inhibition of G-protein function and for treatment of proliferative diseases
04/02/2002US6365587 Substituted aryl hydroxamic acids as metalloproteinase inhibitors
04/02/2002US6365584 For prophylaxis and therapy of inflammatory and/or allergic diseases, lung fibrosis, fibrosing alveolitis and scarring, collagenoses such as lupus erythematodes and sclerodermia as well as arteriosclerosis, psoriasis and neoplasm
04/02/2002US6365583 Methods to enhance white blood cell count
04/02/2002US6365552 Substituted 3-phenylpyrazoles
04/02/2002US6365184 Multiple unit tableted dosage forms containing acid susceptible proton pump inhibitor in combination with one or more nsaids and wherein at least proton pump inhibitor is protected by enteric coated layer
04/02/2002CA2253906C Process for preparation of pyrimidine derivatives
04/02/2002CA2223574C Biphenyl-2-carboxylic acid-tetrahydro-isoquinolin-6-yl amide derivatives, their preparation and their use as inhibitors of microsomal triglyceride transfer protein and/or apolipoprotein b (apo b) secretion
04/02/2002CA2178130C Method of producing 2-naphthamide derivative, and compounds for producing 2-naphthamide derivative
04/02/2002CA2099868C Substituted 4,6-di-tertiary-butyl-5-hydroxy-pyrimidines
04/02/2002CA2097928C Uracil derivatives
03/2002
03/28/2002WO2002024693A1 A process for producing 3,4-dihydro naphthyridinone analogs
03/28/2002WO2002024687A1 Farnesyl transferase inhibiting 6-heterocyclylmethyl quinolinone derivatives
03/28/2002WO2002024686A2 Farnesyl transferase inhibiting 6-heterocyclylmethyl quinoline and quinazoline derivatives
03/28/2002WO2002024684A1 Quinoline derivatives as antibacterials
03/28/2002WO2002024683A1 Farnesyl transferase inhibiting 6-[(substituted phenyl)methyl]-quinoline and quinazoline derivatives
03/28/2002WO2002024682A1 Farnesyl transferase inhibiting quinoline and quinazoline derivatives as farnesyl transferase inhibitors
03/28/2002WO2002024681A2 Pyrazine derivatives as modulators of tyrosine kinases
03/28/2002WO2002024680A1 Imidazole derivatives as raf kinase inhibitors
03/28/2002WO2002024679A1 PYRIDINE DERIVATIVES WITH IKB-KINASE (IKK-β) INHIBITING ACTIVITY
03/28/2002WO2002024667A1 4-amino-quinazolines
03/28/2002WO2002024665A1 Arylalkane-sulfonamides having endothelin-antagonist activity
03/28/2002WO2002024662A1 New benzimidazolone derivatives displaying affinity at the serotonin and dopamine receptors
03/28/2002WO2002024661A2 New n, n'-disubstituted benzimidazolone derivatives with affinity at the serotonin and dopamine receptors