Patents
Patents for C07D 401 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom (107,979)
07/2002
07/18/2002CA2434152A1 Therapeutic heterocyclic compounds
07/18/2002CA2434044A1 1,2-disubstituted cyclic inhibitors of matrix metallorproteases and tnf-alpha
07/18/2002CA2434015A1 Therapeutic chroman compounds
07/18/2002CA2433950A1 Therapeutic chromone compounds
07/18/2002CA2433723A1 Chemical derivatives and their use as anti-telomerase agent
07/18/2002CA2432114A1 4-(hetero)aryl substituted indolinones
07/17/2002EP1223170A1 Pyrimidine-5-carboxamide compounds, process for producing the same and use thereof
07/17/2002EP1223166A1 Linked cyclic polyamines with activity against hiv.
07/17/2002EP1222922A1 Method for stabilizing benzimidazole compounds
07/17/2002EP1222305A2 Enzymatic process for the resolution of enantiomeric mixtures of beta-lactams
07/17/2002EP1222185A1 Tetrahydrobenzindolone derivatives, their preparation and their use as 5-ht7 receptor antagonists
07/17/2002EP1222176A1 AMINO LACTAM SULFONAMIDES AS INHIBITORS OF A$g(b) PROTEIN PRODUCTION
07/17/2002EP1222175A1 4,5-disubstituted-2-aminopyrimidines
07/17/2002EP1222173A1 Process for preparing 4-trifluoromethylsulphinylpyrazole derivative
07/17/2002EP1222171A1 Pyridinium derivatives for the management of aging-related and diabetic vascular complications, process for their preparation and therapeutic uses thereof
07/17/2002EP1222170A1 Novel nicotinonitrile compounds
07/17/2002EP1221953A1 Treating sleep disorders using desloratadine
07/17/2002EP1049670B1 Azetidinecarboxamide derivatives for treating cns disorders
07/17/2002EP0939629A4 Thiol sulfonamide metalloprotease inhibitors
07/17/2002EP0888340B1 4-(benzo-1,3-dioxolyl)-pyrrolidine-3-carboxylic acid derivatives as endothelin antagonists
07/17/2002EP0882044B1 1,4-dihydropyridine compounds as bradykinin antagonists
07/17/2002CN1359377A Dihydrobenzodiazepins and their use for treating dyslipidemia
07/17/2002CN1359289A Selective iGLuR5 receptor antagonists for the treatment of migraine
07/17/2002CN1087741C New indole and inidazole compounds, process for their preparation and pharmaceutical compositions containing them
07/17/2002CN1087740C New benzimidzole, benzoxazole and benzothiazole compounds, process for their preparation and pharmaceutical compositions containing them
07/17/2002CN1087739C Inclusion and resolution preparation process of optical purity benzimidazoles medicines resisting peptic ulcer
07/17/2002CN1087737C Dihygropyridine derivatives as bradykinin ant agonists
07/17/2002CN1087736C Novel amidinonaphthyl derivative or salt thereof
07/17/2002CN1087735C Process for preparation of pesticidal 1-(haloaryl) heteroyclic compounds
07/16/2002US6420975 Interior rearview mirror sound processing system
07/16/2002US6420563 Inverse antagonist
07/16/2002US6420560 H1—histamine receptor antagonists
07/16/2002US6420559 1-(4-arylpiperazin-1-yl)-ω-[N-(α,ω-dicarboximido)]-alkanes useful as uro-selective α1-adrenoceptor blockers
07/16/2002US6420558 Aminopiperidine derivates as integrin αvβ3 antagonists
07/16/2002US6420557 For therapy of male erectile dysfunction
07/16/2002US6420555 Imidazolyl derivatives
07/16/2002US6420462 Oxidation resistance, heat resistant and actinic degradationheterocyclic amine oxides
07/16/2002US6420438 1-amino-7-isoquinoline derivatives as serine protease inhibitors
07/16/2002US6420415 Thiol compounds, their production and use
07/16/2002US6420414 Amino derivatives of EM-138 and methods of treating angiogenesis with same
07/16/2002US6420409 Benzimidazole derivatives
07/16/2002US6420406 Triazolyl disulphides
07/16/2002US6420396 Biphenyl and biphenyl-analogous compounds as integrin antagonists
07/16/2002US6420395 Disorders or diseases involving the cholinergic system of the central nervous system, pain, inflammatory diseases, diseases caused by smooth muscle contractions and as assistance in the cessation of chemical substance abuse.
07/16/2002US6420390 Heteroarylpiperidines and their use as antipsychotics
07/16/2002US6420387 Antitumor
07/16/2002US6420385 Substituted pyrimidinone and pyridone compounds and methods of use
07/16/2002US6420376 Amido spiropiperidines promote the release of growth hormone
07/16/2002US6420372 Tropical malarial antiprotozoan
07/16/2002US6420371 Angiogenesis inhibitor
07/16/2002US6420366 1-(4-arylpiperazin-1-yl)-ω-[N-(αω-dicarboximido)]-alkanes useful as uro-selective α1-adrenoceptor blockers
07/16/2002US6420364 Treating autoimmune diseases,alzheimer's disease, atherosclerosis, osteoporosis,
07/16/2002US6420315 5-thien-3-yl-2-oxy- or -2-thio-pyridines; high selectivity for broadleaf and grassy weeds in crops, such as maize and rice; pre- and post-emergence
07/16/2002CA2240846C Tricyclic amides useful for inhibition of g-protein function and for treatment of proliferative diseases
07/16/2002CA2205998C Certain 4-aminomethyl-2-substituted imidazole derivatives and 2-aminomethyl-4-substituted imidazole derivatives; new classes of dopamine receptor subtype specific ligands
07/16/2002CA2119511C Benzimidazole compounds, their use and preparation
07/16/2002CA2063594C 5-(1-aminocyclohexyl)-2(1h)-pyridinone and related compounds
07/16/2002CA2050875C 3-(1h-indazol-3-yl)-4-pyridinamines, a process and intermediates for their preparation and their use as medicaments
07/11/2002WO2002053561A1 Excitatory amino acid receptor antagonists
07/11/2002WO2002053560A1 Microbiocidal n-phenyl-n-[4-(4-pyridyl-2-pyrimidin-2-yl]-amine derivatives
07/11/2002WO2002053559A1 Sodium channel modulators derived from 2-piperidylimidazoles
07/11/2002WO2002053558A1 Quinazolone derivatives as alpha 1a/b adrenergic receptor antagonists
07/11/2002WO2002053557A1 Novel sulfamides and their use as endothelin receptor antagonists
07/11/2002WO2002053556A2 Pyrrolidinylmethyl substituted decahydroisoquinolines as excitatory amino acid receptor antagonists
07/11/2002WO2002053555A2 Pyrrolidinylmethyl- and piperidinyl substituted decahydroisoquinolines as excitatory amino acid receptor antagonists
07/11/2002WO2002053546A1 Heterocycle derivatives as ppar-gamma agonists
07/11/2002WO2002053543A1 Pyridone derivative having affinity for cannabinoid 2-type receptor
07/11/2002WO2002053535A2 Process for making amlodipine, derivatives thereof, and precursors therefor
07/11/2002WO2002053534A1 Vla-4 inhibitors
07/11/2002WO2002053533A2 Kappa opioid receptor ligands
07/11/2002WO2002053528A1 Method for the regioselective preparation of substituted benzo[g]quinoline-3-carbonitriles and benzo[g]quinazolines
07/11/2002WO2002053516A2 N(phenylsulphonyl)glycine derivatives and their therapeutic use
07/11/2002WO2002053155A1 Telomerase inhibitor
07/11/2002WO2002053135A1 Amlodipine free base
07/11/2002WO2002053097A2 Pharmaceutical compositions of a non-enteric coated proton pump inhibitor with a carbonate salt and bicarbonate salt combination
07/11/2002WO2002036734A3 Aza-and polyaza-naphthalenyl ketones useful as hiv integrase inhibitors
07/11/2002WO2002024658A3 Substituted imidazoles as dual histamine h1 and h3 agonists or antagonists
07/11/2002WO2002024657A3 Substituted imidazoles as dual histamine h1 and h3 agonists or antagonists
07/11/2002WO2002018348A3 Quinazoline derivatives as alpha-1 adrenergic antagonists
07/11/2002WO2002008221A3 Capsaicin receptor ligands
07/11/2002WO2001040187A3 Compound having effect of promoting neuron differentiation
07/11/2002WO2001022919A3 Spiro[bicyclic -azacycloalkyl and -cycloalkyl] derivatives and uses thereof
07/11/2002WO2001017568A3 Bioconjugation in vivo to pulmonary or blood components
07/11/2002WO2000072834A3 Agent for expression of long-term potentiation of synaptic transmission comprising compound having brain somatostatin activation property
07/11/2002US20020091273 Method for the regioselective preparation of substituted benzo[g]quinoline3-carbonitriles and benzo[g]quinazolines
07/11/2002US20020091265 4-phenyl-pyridine derivatives
07/11/2002US20020091262 Armoatic or heteroarmoatic compound containing substituted amides or thioamides
07/11/2002US20020091261 Phthalazines with angiogenesis inhibiting activity
07/11/2002US20020091148 3-substituted indole antiproliferative angiogenesis inhibitors
07/11/2002US20020091143 Use of 4-substituted tetrahydropyridines for the manufacture of medicament s acting upon TGF-beta 1
07/11/2002US20020091141 Treating serotonin-related central nervous system disorders
07/11/2002US20020091138 Treating vascular proliferative disorders
07/11/2002US20020091127 Semicarbazides and their uses
07/11/2002US20020091124 Also used as an antimitotic and for direct and/or indirect inhibition of tubulin polymerization in mammalian
07/11/2002US20020091122 Voltage-dependent
07/11/2002US20020091120 2-substituted heterocyclic compounds for treating multidrug resistance
07/11/2002US20020091116 Show selectivity for factor Xa versus other proteases of coagulation or the fibrinolytic cascades
07/11/2002US20020091090 Somatostatin antagonists and agonists
07/11/2002US20020091089 (Substituted)acyl dipeptidyl inhibitors of the ICE/ced-3 family of cysteine proteases
07/11/2002US20020091078 Treating diabetes, especially Type II diabetes