Patents
Patents for C07D 401 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom (107,979)
08/2002
08/20/2002US6437123 Triazine compounds and their use
08/20/2002US6437120 Chemical intermediate for mirtazepine, antidepressants
08/20/2002US6436985 Disubstituted pyrazolines and triazolines as factor Xa inhibitors
08/20/2002US6436981 Dihydrotriazolone derivatives as pesticides
08/20/2002US6436967 Process for preparing prodrugs of benzenesulfonamide-containing cox-2 inhibitors
08/20/2002US6436965 Inhibition of phosphodiesterase; 3-carbocyclic(alkyl)oxy-2-aryl(alkyl)aminocarbonyl-1-aryl(alkyl)indole or azaindole derivatives
08/20/2002US6436964 Piperidine derivatives having effects on serotonin related systems
08/20/2002US6436962 Alpha 1a adrenergic receptor antagonists; relief from benign prostatic hyperplasia by less hindered urine flow by relaxing smooth muscle tissue; with a testosterone 5-alpha reductase inhibitor, finasteride; acute and chronic relief
08/20/2002US6436961 Substance p receptor antagonist; 2-phenyl-3-benzylaminopiperidines
08/20/2002US6436960 Farnesyl transferase inhibitors having a piperidine structure and process for preparation thereof
08/20/2002US6436949 Heterocyclically substituted benzamides and their use
08/20/2002US6436943 Use of dihydropyrimidines as medicaments, and novel substances
08/20/2002US6436941 Treating schizophrenia, depression, and parkinson's disease; side effect reduction
08/20/2002US6436939 Treatment of central nervous system disorders including sleep/wake disorders, dementia, alzheimer's disease, epilepsy, narcolepsy, eating disorders, motion sickness, vertigo
08/20/2002US6436928 Selective neurokinin antagonists
08/20/2002US6436923 Compounds and methods for modulation of estrogen receptors
08/20/2002US6436915 Antiproliferative and antitumor agents and angiogenesis inhibitors
08/20/2002US6436904 Treatment of inflammatory diseases in mammals
08/20/2002CA2240138C Quinazolin-4-one ampa antagonists
08/15/2002WO2002062789A1 Pyrazole compounds useful as protein kinase inhibitors
08/15/2002WO2002062788A1 Sulfonamide compounds, their preparation and use
08/15/2002WO2002062787A1 Pyrazoles as tgf inhibitors
08/15/2002WO2002062786A1 Processes for the production of substituted 2-(2-pyridylmethyl) sulfinyl-1h-benzimidazoles
08/15/2002WO2002062785A1 Benzimidazole derivatives, method for their production and use thereof as tryptase inhibitors
08/15/2002WO2002062784A1 Piperidinee derivatives as neurokinin 1 antagonists
08/15/2002WO2002062764A1 Fused heterocyclic compounds
08/15/2002WO2002062763A2 Inhibition of raf kinase using quinolyl isoquinolyl or pyridyl ureas
08/15/2002WO2002062762A2 Potassium channel openers
08/15/2002WO2002062755A2 Polyamide analogs as dna minor groove binders
08/15/2002WO2002062423A1 Composition and antiviral activity of substituted azaindoleoxoacetic piperazine derivatives
08/15/2002WO2002062295A2 Pyridine-substituted benzanilides as potassium ion channel openers
08/15/2002WO2002062290A2 Heterocyclic substituted 2-methyl-benzimidazole antiviral agents
08/15/2002WO2002040465A3 Aryloxy piperidinyl indoles for treating depression
08/15/2002WO2002032861A3 Orally active salts with tyrosine kinase activity
08/15/2002WO2002011724A3 Neuroprotective 2-pyridinamine compositions and related methods
08/15/2002WO2001030768A9 Methods and compositions utilizing quinazolinones
08/15/2002US20020111495 Nicotinamide acids, amides, and their mimetics active as inhibitors of PDE4 isozymes
08/15/2002US20020111494 N-type calcium channel blockers, antiischemic agents
08/15/2002US20020111492 Bactericides
08/15/2002US20020111461 Peptidomimetic compound for us ein the treatment of diabetes
08/15/2002US20020111374 Estrogen receptor modulators
08/15/2002US20020111371 Delta2-1,2,3-triazoline anticonvulsants and their active metabolite analogues, the aminoalkylpyridines, are excitatory amino acid antagonists and antiischemic agents, useful in the treatment of cerebral ischemia resulting from stroke
08/15/2002US20020111370 Compounds useful as antibacterial agents
08/15/2002US20020111367 Phenyl substituted pyridine and benzene derivatives
08/15/2002US20020111364 ABCA-1 elevating compounds
08/15/2002US20020111358 Phenoxypropylamine compounds
08/15/2002US20020111353 Antiinflammatory agents; central nervous system disorders;antidiabgetic agents; rheumatic disorders
08/15/2002US20020111351 New hydroxyindoles, their use as inhibitors of phosphodiesterase 4 and processes for their preparation
08/15/2002US20020111348 Substituted oximes and hydrazones as neurokinin antagonists
08/15/2002US20020111347 Nervous system disorders
08/15/2002CA2437492A1 Fused heterocyclic compounds
08/15/2002CA2437405A1 Potassium channel openers
08/15/2002CA2436467A1 Processes for the production of substituted 2-(2-pyridylmethyl) sulfinyl-1h-benzimidazoles
08/15/2002CA2436461A1 Pyridine-substituted benzanilides as potassium ion channel openers
08/14/2002EP1230249A1 Transition metal complexes with bidentate ligand having an imidazole ring
08/14/2002EP1230248A2 Transition metal complexes attached to a polymer via a flexible chain
08/14/2002EP1230244A2 Pyrazolecarboxylic acid tricyclic derivatives, preparation and pharmaceutical compositions containing same
08/14/2002EP1230237A1 Magnesium omeprazole
08/14/2002EP1230236A1 Compound with growth hormone releasing properties
08/14/2002EP1230235A1 Compounds with antibacterial and antiparasitic properties
08/14/2002EP1230224A1 Substituted 5-benzyl-2,4-diaminopyrimidines
08/14/2002EP1230219A1 Aromatic sulfons hydroxamic acid metalloprotease inhibitor
08/14/2002EP1229915A1 Protease inhibitors
08/14/2002EP1229914A1 Protease inhibitors
08/14/2002EP1229907A1 Prevention of plaque rupture by acat inhibitors
08/14/2002EP1087961B1 Phenoxylpropanolamines, method for the production thereof and pharmaceutical compositions containing the same
08/14/2002EP0988038B1 (imidazol-5-yl)methyl-2-quinolinone derivatives as inhibitors of smooth muscle cell proliferation
08/14/2002EP0807111B1 Substituted heterocyclic compounds, preparation method therefor and pharmaceutical compositions containing same
08/14/2002EP0763024B1 Processes and intermediates for the preparation of piperazine derivatives
08/14/2002EP0754683B1 Ether compound, use thereof, and intermediate for producing the compound
08/14/2002EP0722439B1 Hiv protease inhibitors
08/14/2002DE10106457A1 DELTA·1·-Pyrroline DELTA · 1 · -Pyrrolines
08/14/2002CN1364167A Endogenous constitutively activated G protein-coupled orphan receptors
08/14/2002CN1364155A N-Cyanomethyl amides as protease inhibitors
08/13/2002US6433187 Certain polycyclic compounds useful as tubulin-binding agents
08/13/2002US6433186 Treatment of conditions where inhibition of thrombin is required (e.g. thrombosis) or as anticoagulants.
08/13/2002US6433182 Nitrosated and nitrosylated α-adrenergic receptor antagonist compounds, compositions and their uses
08/13/2002US6433178 3-alkyl-3-phenyl-piperidines
08/13/2002US6433177 Reacting n-carboxyanhydride and butylamine
08/13/2002US6433165 Chemokine receptor antagonists and methods of use therefor
08/13/2002US6432995 Inhibit the release of inflammatory cytokines such as interleukin-1 and tumor necrosis factor from cells
08/13/2002US6432988 2-arylalkylthio -imidazoles, 2-arylalkenyl -thio -imidazoles and 2-arylalkinyl -thio -imidazoles as anti -inflammatory substances and substances inhibiting the release of cytokine
08/13/2002US6432987 Substituted N-benzylindol-3-ylglyoxylic acid derivatives having antitumor action
08/13/2002US6432981 Cyclopentyl modulators of chemokine receptor activity
08/13/2002US6432980 Aliphatic amine substituted piperidyl diaryl pyrrole derivatives as antiprotozoal agents
08/13/2002US6432978 4-hydroxy-1-methyl-1,2-dihydroquinolin-2-one derivatives; cardiovascular, atopic, and rheumatic disorders; antiallergens, antiinflammatory agents, antiasthmatics, and hypotensive agents
08/13/2002US6432972 Desloratadine as non-sedating antihistamine, decongestant
08/13/2002US6432969 Non-insulin dependent diabetes, obesity, arthritis, and osteoporosis treatment
08/13/2002US6432963 Antiinflammatory agents; tyrosine kinase inhibitor
08/13/2002US6432959 Antitumor agents
08/13/2002US6432957 Piperazine derivative
08/13/2002US6432955 Heterocyclic derivatives and their use as antithrombotic agents
08/13/2002US6432949 Amide derivatives useful as inhibitors of the production of cytokines
08/13/2002US6432947 N-heterocyclic derivatives as NOS inhibitors
08/13/2002US6432921 Oligopeptides
08/13/2002US6432900 Antisoilants
08/13/2002US6432879 Substituted phenyl uracils
08/13/2002CA2216633C Synthesis of bis-indolylmaleimides
08/08/2002WO2002060894A2 Sulfonamide lactam inhibitors of factor xa
08/08/2002WO2002060893A1 Method for carbamoylating alcohols