Patents
Patents for C07D 401 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom (107,979)
10/2002
10/17/2002US20020151555 Pyrimidine matrix metalloproteinase inhibitors
10/17/2002US20020151553 Such as 4-(4-chlorophenyl)1-(3-(5-cyano-5H-dibenzo(a,d) cycloheptene-5-yl)propyl)piperidin-4-ol for treatment of diseases associated with aberrant leukocyte recruitment and/or activation
10/17/2002US20020151547 Substituted phenyl-piperidine methanone compounds
10/17/2002US20020151545 Anticoagulants in treating and preventing cardiovascular diseases, as anti-inflammatory agents, and metastasis inhibitors in treating cancer
10/17/2002US20020150947 Detecting preferential biopolymer in sample; obtain sample, incubate with ligand, allow complex to form, detect complex
10/17/2002CA2444024A1 Thiohydantoins and use thereof for treating diabetes
10/17/2002CA2443108A1 N-substituted nonaryl-heterocyclo amidyl nmda/nr2b antagonists
10/17/2002CA2442904A1 Benzamidine derivative
10/17/2002CA2442695A1 Indolinones substituted in the 6-position, the preparation thereof and their use as medicaments
10/16/2002EP1248782A1 Anticancer compound and enantiomer separation method useful for synthesizing said compound
10/16/2002EP1248781A1 Pyrazole cyclic amp-specific pde inhibitors
10/16/2002EP1248777A2 Tricyclic compounds with antiviral activity
10/16/2002EP1248771A1 Method for preparing hydroxypicolinic acid derivatives
10/16/2002EP1248770A1 1,3,4-substituted piperidine analogs and uses thereof in treating addictions
10/16/2002EP1248624A1 3,4-DIHYDRO-(1H)-QUINAZOLIN-2-ONES AND THEIR USE AS CSBP/p38 KINASE INHIBITORS
10/16/2002EP1248622A1 Anxiety method
10/16/2002EP0934316B1 Azabicyclic carbamoyloxy mutilin derivatives for antibacterial use
10/16/2002EP0927161B1 Substituted cyclic amine metalloprotease inhibitors
10/16/2002EP0831826B1 Pharmaceutical composition comprising a proteinase inhibitor and a monoglyceride
10/16/2002EP0763033B1 Imidazole derivatives and processes for the preparation thereof
10/16/2002EP0641203B1 Pharmaceutical compositions of an imidazolyl-akenoic acid salt and their use as angiotensin ii antagonists
10/16/2002EP0542136B1 1-[(1,4-benzodioxanyl)alkyl]-4-(heteroaryl) piperidines, piperazines and pyrrolidines as antipsychotic agents
10/16/2002CN1374995A Fluorescent maleimides and uses thereof
10/16/2002CN1374960A Novel integrain receptor antagonists
10/16/2002CN1374959A Piperidine quinolyl propyl derivatives, preparation method and compositions containing same
10/16/2002CN1374953A Aromatic nitrogenous six-membered ring compounds
10/16/2002CN1374952A Benzimidazolone derivatives and their use as phosphodiesterase inhibibors
10/16/2002CN1374950A Indazole compounds and pharmaceutical compositions for inhibiting protein kinases, and methods for their use
10/16/2002CN1374949A 毒蕈碱拮抗剂 Muscarinic antagonist
10/16/2002CN1374948A 4-amino-1-aryl-1,5-dihydro-pyrrole-2-one with anti-convulsive and anxiolytic properties and a method for producing the same
10/16/2002CN1374865A Nociceptin receptor ORL-1 agonists for use in treating cough
10/16/2002CN1374306A Prepn of improved pesticide intermediate
10/16/2002CN1374082A Use of glycogen sulphofoenzyme inhibitor
10/16/2002CN1092651C Pyridyl methylene process for producing amino triazineone compound
10/16/2002CN1092643C Certain aminomethyl phenylidazole derivatives, for intensifying memory
10/16/2002CN1092642C Quinoline derivatives as tachykinin NK 3 receptor antagonists
10/15/2002USRE37886 4-(1-(3,5bis(trifluoromethyl) benzoyl)-2-(phenylmethyl)-4-piperidinyl)-n-(2,6dimethylphenyl)-1-piperazine acetamide, having tachykinin and substance p antagonistic activity; analgesic and antiinflammatory agents
10/15/2002US6465693 Metal-catalyzed arylations of hydrazines, hydrazones, and related substrates
10/15/2002US6465661 Methods of making HIV-protease inhibitors and intermediates for making HIV-protease inhibitors
10/15/2002US6465645 Containing triazine groups and n-alkyloxypiperidine groups; candle wax which is effectively stabilized against discoloration and fading
10/15/2002US6465504 Such as 4-(3,5-bis(2-hydroxyphenyl)-(1,2,4)triazol-1-yl)-benzoic acid; treatment of iron overload by mobilizing and eliminating iron deposits; preventing organ damage, in particular of liver, heart and endocrine organs
10/15/2002US6465493 Such as 4-(4-(4-fluorophenyl)-5-(2-pyridyl)-1-hydroxy-1h-imidazol-2-yl)benzonitrile; alk5 mediated diseases such as arthritis, osteoporosis, kidney and renal diseases, conges-tive heart failure, ulcers, diabetic nephropathy
10/15/2002US6465492 Heterocyclic compounds
10/15/2002US6465491 6-phenylpyridyl-2-amine derivatives
10/15/2002US6465489 Such as 1-benzoyl-3-(3,4-dichlorophenyl)-3-(3-(4-(n',n'-dimethylureido)-4 -phenylpiperidin-1-)propyl)piperidine; psychiatric and psychosomatic illnesses, hypertension, central or peripheral pathology
10/15/2002US6465486 Alpha2 adrenoceptor modulators; hypertension, glaucoma, sexual dysfunction, depression, attention deficit hyperactivity disorder, parkinsonism, need for anesthesia, cardiac arrythmia
10/15/2002US6465485 Tetrahydroisoquinoline derivatives as modulators of dopamine D3 receptors
10/15/2002US6465484 Tyrosine kinase inhibitors; cancer, atherosclerosis, diabetic retinopathy, autoimmune diseases, inflammatory diseases
10/15/2002US6465482 Arylpiperazinyl-cyclohexyl indole derivatives for the treatment of depression
10/15/2002US6465478 Analgesics, antiinflammatories, diuretics, anesthetics, neuroprotective agents, antihypertensive or antianxiety agent, appetite control, hearing regulation
10/15/2002US6465476 Immuno-modulator exhibiting antimicrobial and anti-mycrobacterial activities, method for producing the same and pharmaceutical preparation
10/15/2002US6465471 Cinnamic acid derivatives
10/15/2002US6465467 Diseases related to the 5-ht2c receptor, especially eating, memory, mood, urinary and anxiety disorders, schizophrenia, pain, sexual dysfunctions
10/15/2002US6465459 Inhibit the enzyme, factor xa
10/15/2002US6465449 Heteroaromatic bicyclic derivatives useful as anticancer agents
10/15/2002US6465433 Boronic ester and acid compounds, synthesis and uses
10/15/2002CA2256438C Aromatic amidine derivatives useful as selective thrombin inhibitors
10/10/2002WO2002080161A2 Optical data carrier that contains a merocyanine dye as the light-absorbing compound in the information layer
10/10/2002WO2002079198A1 Pyridazinone aldose reductase inhibitors
10/10/2002WO2002079197A1 Inhibitors of c-jun n-terminal kinases (jnk) and other protein kinases
10/10/2002WO2002079195A1 Substituted 2-thio-3,5-dicyano-4-phenyl-6-aminopyridines with adenosine receptor-binding activity and their use as cardiovascular preparations
10/10/2002WO2002079194A1 Ccr5 antagonists useful for treating aids
10/10/2002WO2002079192A1 Novel tyrosine kinase inhibitors
10/10/2002WO2002079191A1 Viologen linked acridine based molecule and process for the preparation thereof
10/10/2002WO2002079190A1 3-substituted indoles as chemokine antagonists
10/10/2002WO2002079189A2 Spiroisoquinoline compounds, methods for their preparation and intermediates
10/10/2002WO2002079188A1 Pyrrolidine sulfonamides
10/10/2002WO2002079187A1 Methoxy-1,3,5-triazine derivatives as antiviral agents
10/10/2002WO2002079186A2 Aminopiperidine derivatives as modulators of chemokine receptor activity
10/10/2002WO2002079173A1 Benzotriazoles and their use as uv light stabilisers
10/10/2002WO2002079169A1 Cyano-substituted dihydropyrimidine compounds and their use to treat diseases
10/10/2002WO2002079168A1 Imidazolyl derivatives useful as histamine h3 receptor ligands
10/10/2002WO2002079165A1 Tetrahydroquinoline derivatives as stat6-modulators, preparation and use thereof
10/10/2002WO2002079163A1 Aminopyridine derivatives as estrogen receptor modulators
10/10/2002WO2002079157A1 Aryl oxime-piperazines useful as ccr5 antagonists
10/10/2002WO2002079156A1 Novel piperidine derivatives as modulators of chemokine receptor
10/10/2002WO2002079152A1 Cyclopropylindole derivatives as selective serotonin reuptake inhibitors
10/10/2002WO2002079151A1 3-substituted indoels or fused pyrroles as antagonists of the chemokine mcp-1 (ccr2b) receptor
10/10/2002WO2002079149A2 Novel cyano-substituted dihydropyrimidine compounds and their use to treat diseases
10/10/2002WO2002079146A2 Compounds useful as modulators of melanocortin receptors and pharmaceutical compositions comprising same
10/10/2002WO2002079145A1 BENZAMIDE INHIBITORS OF FACTOR Xa
10/10/2002WO2002078745A2 Use of mglur5 antagonists in the manufacture of a medicament in the treatment of autism, mental retardation, schizophrenia
10/10/2002WO2002078706A1 Farnesyl transferase inhibitors in combination with hmg coa reductase inhibitors for the inhibition for the treatment of cancer
10/10/2002WO2002078699A1 Compounds and methods
10/10/2002WO2002078697A1 Compounds and methods
10/10/2002WO2002078696A1 Compounds and methods
10/10/2002WO2002078693A2 N-(2-arylethyl)benzylamines as antagonists of the 5-ht6 receptor
10/10/2002WO2002078659A1 Dyeing composition for dyeing keratinous fibres comprising a cationic azo-dye
10/10/2002WO2002078641A2 Pyrrolidine sulfonamides
10/10/2002WO2002078639A2 A method of treating proliferative diseases using eg5 inhibitors
10/10/2002WO2002078628A2 Cyanamide, alkoxyamino, and urea derivatives of 1,3-benzodiazapines as hiv reverse transcriptase inhibitors
10/10/2002WO2002078626A2 Therapeutic combinations for cardiovascular and inflammatory indications
10/10/2002WO2002078625A2 Therapeutic combinations for cardiovascular and inflammatory indications
10/10/2002WO2002066440A8 Diaminopyrazole derivatives and their use for oxidation dyeing of keratinous fibres
10/10/2002WO2002062764A9 Fused heterocyclic compounds
10/10/2002WO2002062763A3 Inhibition of raf kinase using quinolyl isoquinolyl or pyridyl ureas
10/10/2002WO2002053516A3 N(phenylsulphonyl)glycine derivatives and their therapeutic use
10/10/2002WO2002050067A3 Pharmaceutical heterocyclic compounds
10/10/2002WO2002044173A3 Herbicidal heterocycles
10/10/2002WO2002006512A3 Method for detecting uracil biosynthesis inhibitors and their use as herbicides