Patents
Patents for C07D 401 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom (107,979)
09/2004
09/28/2004US6797820 Succinate compounds, compositions and methods of use and preparation
09/28/2004US6797716 Imidazonaphthyridines
09/28/2004US6797713 1,4 substituted piperazines, 1,4 substituted piperidines, and 1-substituted,4-alkylidenyl piperidine compounds; dual acting molecules having both leukotriene inhibition properties
09/28/2004US6797710 Cardiovascular disorders; serine protease inhibitor; administering by mouth; bioavailability
09/28/2004US6797709 Sexual disorders
09/28/2004US6797708 Enzyme inhibitors such as 4-(2-(1-benzhydryl-2-(2-((benzyl-sulfonyl)amino)ethyl)-5-chloro-1h-indol-3 -yl)ethoxy) benzoic acid, used as analgesics or antiinflammatory agents
09/28/2004CA2461833A1 Process for the preparation of organic compounds containing a sulfinyl or sulfonyl group
09/28/2004CA2299013C Neuropeptide y antagonists
09/28/2004CA2224125C Pharmaceutical composition comprising a proteinase inhibitor and a monoglyceride
09/28/2004CA2128312C Use of n-(pyridinyl)-1h-indol-1-amines for the preparation of a medicament for the treatment of obsessive-compulsive disorders
09/23/2004WO2004081005A1 Melanin-concentrating hormone receptor antagonists and compositions and methods related thereto
09/23/2004WO2004081000A1 Quinazoline derivatives
09/23/2004WO2004080999A1 Pyrazole compounds useful in the treatment of inflammation
09/23/2004WO2004080998A1 Imidazol-4-yl-ethynyl-pyridine derivatives
09/23/2004WO2004080997A1 Process for the preparation of loratadine
09/23/2004WO2004080982A1 Pyrazine compounds as transforming growth factor (tgf) inhibitors
09/23/2004WO2004080981A1 Pyrimidin-2-one compounds and their use as dopamine d3 receptor ligands
09/23/2004WO2004080980A1 2, 4- di (phenylamino) pyrimidines useful in the treatment of neoplastic diseases, inflammatory and immune system disorders
09/23/2004WO2004080977A1 4-substituted-5-cyano-1h-pyrimidin-6-(thi)ones as gsk-3 inhibitors
09/23/2004WO2004080976A1 Phthalazinone derivatives
09/23/2004WO2004080975A1 Nitrogen-containing heterocycle derivative and organic electroluminescent element using the same
09/23/2004WO2004080973A1 Fused tri and tetra-cyclic pyrazole kinase inhibitors
09/23/2004WO2004080972A1 Pirazole modulators of atp-binding cassette transporters
09/23/2004WO2004080971A1 Tetrahydroquinoline derivatives useful as serine protease inhibitors
09/23/2004WO2004080970A1 Novel bicyclic aromatic compounds, the production and use thereof in the form of drugs
09/23/2004WO2004080969A1 Quinolinone / benzoxazinone derivatives and uses thereof
09/23/2004WO2004080968A1 6-substituted nicotinamide derivatives as opioid receptor antagonists
09/23/2004WO2004080964A1 Indole derivatives useful for the treatment of diseases
09/23/2004WO2004080961A2 Crystalline and amorphous solids of pantoprazole and processes for their preparation
09/23/2004WO2004080487A1 Preventive or remedy for teeth grinding
09/23/2004WO2004080480A1 Pharmaceutical preparations comprising acid-stabilised insulin
09/23/2004WO2004080463A1 Heterocyclic kinase inhibitors: methods of use and synthesis
09/23/2004WO2004080461A2 Stable pharmaceutical compositions of desloratadine
09/23/2004WO2004080423A2 7-amino- isoindolyl compounds amd their pharmaceutical uses
09/23/2004WO2004072027A3 Chemical derivatives binding very specifically with g-quadruplex dna structures and use thereof as a specific anti-cancer agent
09/23/2004WO2004052304A3 Antibacterial compounds having a (pyrrole carboxamide)-(benzamide)-(imidazole carboxamide) motif
09/23/2004WO2004050613A3 2-substituted-3-propenamide derivatives and methods of using the same
09/23/2004WO2004041258A3 Cyclic nucleotide phosphodiesterase inhibitors, preparation and uses
09/23/2004WO2004030637A3 Treatment of obesity and other disorders associated with excessive food intake
09/23/2004WO2003082268A3 Hemiasterlin derivatives and uses thereof in the treatment of cancer
09/23/2004US20040186295 G protein-coupled receptors activators such as 2-[2-(3-chlorophenyl)-2H-tetrazol-5-yl]pyridine, used as analgesics, anxiolytic, antidepressants, and for prophylaxis of psychological disorders
09/23/2004US20040186292 Indole, azaindole and related heterocyclic 4-alkenyl piperidine amides
09/23/2004US20040186290 transferase enzyme modulators such as 2-(6-Chloropyridin-3-yl)-3-cyclopentyl-N-thiazol-2-ylpropionamide, used for prophylaxis of hyperglycemia and diabetes
09/23/2004US20040186288 3,5-Diamino-1,2,4-triazoles as kinase inhibitors
09/23/2004US20040186159 used to treat glaucomatous optic neuropathy and/or lower and control intraocular pressure (IOP) associated with normal-tension glaucoma, ocular hypertension, and/or glaucoma in warm blooded animals, including man
09/23/2004US20040186154 treating or preventing a hypercholesterolemia-related or an inflammation-related condition ; apical sodium co-dependent bile acid transport inhibitor and an amount of a cyclooxygenase-2 (COX-2) selective inhibitor or its prodrug; kits
09/23/2004US20040186153 Pharmaceutical use of N-carbamoylazole derivatives
09/23/2004US20040186148 E.g., 1-(pyrid-2-yl-so2-),2-((4-(isopropylphenyl)-so2-),5-(isopropoxy)benzene; antiinflammatory agents; immunomodulatory activity rheumatoid arthritis, asthma, allergy, psoriasis, Crohn's disease, systemic lupus erythematosus, multiple sclerosis, diabetes, cancer, glaucoma, osteoporosis, renal ischemia
09/23/2004US20040186146 E.g., R-N-2-[4-(pyrrolidin-1'-yl)methylphenyl]propionyl-methanesulfonamide; inhibition of chemotaxis of neutrophils induced by interleukin-8; antiinflammatory agents; psoriasis, ulcerative cholitis, glomerular nephritis, acute respiratory insufficiency, idiopathic fibrosis, and rheumatoid arthritis
09/23/2004US20040186145 Sulfur substituted sulfonylaminocarboxylic acid N-arylamides, their preparation, their use and pharmaceutical preparations comprising them
09/23/2004US20040186141 Arthropodicidal anthranilamides
09/23/2004US20040186140 Cyclic derivatives as modulators of chemokine receptor activity
09/23/2004US20040186139 Process for preparation of crystalline form-1 of pantoprazole sodium sesquihydrate
09/23/2004US20040186135 Substituted piperidine compounds
09/23/2004US20040186134 Inhibitors of Factor Xa are useful as anticoagulants in the treatment of cardiovascular disorders associated with thromboses; e.g., 1,1-dimethylethyl 1-[1-(-2-(-3-[2-(5-Chloro-thiophen-2-yl)-ethenesulfonylamino]-2-oxo-piperidin-1-yl)-acetyl)-pyrrolidin-2- yl-methyl]-pyrrolidin-3-yl}-methyl-carbamate
09/23/2004US20040186133 preferably antagonists used in the therapeutic and/or preventive treatment of disfunctions of the heart, kidney, respiratory system, central nervous system
09/23/2004US20040186132 Steroid receptor modulator compounds and methods
09/23/2004US20040186129 2-Aroylimidazole compounds for treating cancer
09/23/2004US20040186125 E.g , 3-cyclohexyl-2-furan-3-yl-1Hindole-5-carboxylic acid; hepatitis C viricides that target RNA dependent RNA polymerases (Ns5B) in mammals, an enzyme essential to viral replication; used in conjunction with an mmunomodulatory agent, such as beta -, delta - gamma -, and omega -interferon
09/23/2004US20040186123 such as 2[(Benzyloxy)methyl]-8-methyl-2,3-dihydro[1,4]dioxino[2,3-f]quinoline; serotonin receptor antagonists for treatment of depression, obsessive compulsive disorders, panic disorder, generalized anxiety disorder, social anxiety disorders, sexual dysfunction, and eating disorders
09/23/2004US20040186119 glycogen synthase kinase (GSK-3) inhibitors; for treatment of diabetes and alzheimer's disease
09/23/2004US20040186118 Chk-, Pdk- and Akt-inhibitory pyrimidines, their production and use as pharmaceutical agents
09/23/2004US20040186116 such as 2-(7-acetylamino-1-furano-2-ylmethyl-2,4-dioxo-1,4-dihydro-2H-quinazolin-3-yl)-succinic acid; for treatment of autoimmune diseases, proliferative diseases, angiogenic disorders, and/or cancers; catheters, prosthetics
09/23/2004US20040186114 Cytokine inhibitors
09/23/2004US20040186113 Heterocyclic amines for the treatment of conditions associated with gsk-3
09/23/2004US20040186111 Therapeutic agents useful for treating pain
09/23/2004US20040186110 Nitrogenous heterocylic compounds
09/23/2004US20040186102 such as {4-Chloro-3-[2-(3,4-dihydro-1H-isoquinolin-2-yl)ethoxy]phenyl}-(2-methylquinolin-4-yl)amine for treatment of cardiovascular disorders, kidney disorders, pain and inflammation
09/23/2004US20040186099 Novel heterocyclic compounds, their preparation, pharmaceutical compositions containing them and their use in medicine
09/23/2004US20040186098 Method for preventing and treating hearing loss using sensorineurotrophic compounds
09/23/2004US20040186097 such as N-phenyl-3-[[4-(phenylmethyl)-1-piperidinyl]methyl]-1-piperidinecarboxamide for prevention of asthma and allergies
09/23/2004US20040186092 Tertiary carbocyclic amides such as 1-(3-Piperazin-1-yl-benzyl)-3,4-dihydro-1H-quinolin-2-one, used as serotonin receptor antagonists for prophylaxis of nervous system disorders and gastrointestinal disorders
09/23/2004US20040186091 Triazole compounds useful in therapy
09/23/2004US20040186088 Mercapto-cycloalkyl or heterocyclyl ring-sulfonyl-aryl or heteroaryl derivatives; preventing the cleavage Of tumor necrosis factor- alpha from cell membranes in mammal; treating autoimmune diseases, inflammation, inflammatory bowel disease, Crohn's disease, asthma, sepsis and septic shock
09/23/2004US20040186080 Beta 2-adrenergic receptor agonists
09/23/2004US20040186078 Substituted N'-(arylcarbonyl)-benzhydrazides, N'-(arylcarbonyl)-benzylidene-hydrazides and analogs as activators of caspases and inducers of apoptosis and the use thereof
09/23/2004US20040185352 Photothermographic element comprising improved base precursors and methods for their use
09/23/2004US20040185299 Tertiary diamines containing heterocyclic groups and their use in organic electroluminescent devices
09/23/2004DE10311065A1 New 1-(cyclic amino-alkyl)-pyrimidin-2(1H)-one derivatives, are selective dopamine D3 receptor ligands useful for treating CNS disorders, especially schizophrenia or depression
09/23/2004DE10310278A1 New N-(benzazinyl)-(hetero)aralkylamine derivatives, are inhibitors of factor Xa and/or related serine proteases, useful e.g. as antithrombotic agents and intermediates
09/23/2004CA2518999A1 Crystalline and amorphous solids of pantoprazole and processes for their preparation
09/23/2004CA2518584A1 7-amino- isoindolyl compounds and their pharmaceutical uses
09/23/2004CA2518403A1 Quinolinone/benzoxazinone derivatives and uses thereof
09/23/2004CA2518398A1 Heterocyclic kinase inhibitors: methods of use and synthesis
09/23/2004CA2518194A1 6-substituted nicotinamide derivatives as opioid receptor antagonists
09/23/2004CA2517885A1 Fused tri and tetra-cyclic pyrazole kinase inhibitors
09/23/2004CA2517720A1 Pyrazine compounds as transforming growth factor (tgf) inhibitors
09/23/2004CA2517569A1 Indole derivatives useful for the treatment of diseases
09/22/2004EP1460073A1 Substituted piperidine and piperazine derivatives as melanocortin-4 receptor modulators
09/22/2004EP1460070A1 Substituted piperidine and piperazine derivatives as melanocortin-4 receptor modulators
09/22/2004EP1460069A1 Substituted cyclohexyl and piperidinyl derivatives as melanocortin-4 receptor modulators
09/22/2004EP1460066A1 Piperazine compounds
09/22/2004EP1460065A1 Processes for production of cyclic diamine compounds or salts thereof
09/22/2004EP1460064A1 Indole-2-carboxamide derivatives useful as beta-2 agonists
09/22/2004EP1460062A1 Nitrogenous cyclic ketone derivative, process for producing the same, and use
09/22/2004EP1458718A1 Quinolinones as prostaglandin receptor ligands
09/22/2004EP1458714A1 3,4-dihydro-1h-isoquinoloin-2-yl-derivatives
09/22/2004EP1458713A1 Indolinone derivatives useful as protein kinase inhibitors
09/22/2004EP1458712A2 Novel compounds
09/22/2004EP1458710A1 Heteroaryl substituted pyrrole modulators of metabotropic glutamate receptor-5