Patents
Patents for C07D 401 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom (107,979)
04/2006
04/12/2006CN1759109A Substituted benzoylureidopyridyl-piperidine and -pyrrolidinecarboxylic acid derivatives, method for the production thereof and the use thereof
04/12/2006CN1759108A Biphenyl derivatives
04/12/2006CN1759101A Quinolinone / benzoxazinone derivatives and uses thereof
04/12/2006CN1759097A Chemical process for the preparation of intermediates to obtain N-formyl hydroxylamine compounds
04/12/2006CN1250540C Improved single-reactor synthesis of [2,8-di(trifluoromethyl)-4-quinolyl]-2-pyridyl methyl ketone and methylfluoro quine
04/12/2006CN1250539C Intermediate for preparing 1-[halogenarylradical] heterocyclic pesticide compound
04/12/2006CN1250533C Novel azoles having an insecticidal action
04/12/2006CN1250531C Novel compounds
04/12/2006CN1250218C Use of angiotensin II antagonists
04/12/2006CN1250192C 2, 5-diaminopyridine oxidation color display alkali for dyeing keratin fiber
04/12/2006CA2484473A1 1-[2-(4-benzyl-4-hydroxy-piperidin-1-yl)-ethyl]-3-(2-methyl-quinolin-4-yl)-urea salt
04/11/2006US7026498 Coordination catalyst containing ligand
04/11/2006US7026486 Process for production cilostazol
04/11/2006US7026485 inhibitors of HIV protease; N-heterocyclic moiety containing hydroxyethylamine compounds where the heterocyclic moiety may be octahydroisoquinoline
04/11/2006US7026482 Process for preparing imidazoquinolinamines
04/11/2006US7026479 Process for the production of quinazolines
04/11/2006US7026476 Intermediate arylamine compounds
04/11/2006US7026357 Diphenylurea compounds
04/11/2006US7026349 Sulfonamides
04/11/2006US7026346 Anticancer agents
04/11/2006US7026336 4-pyridinylimidazol-2-ylhydrocarbyl amine, (thio)urea, carbamic acid or sulfonamide derivatives, e.g., (2-(4-(4-Chloro-3-methoxy-phenyl)-5-pyridin-4-yl-1H-imidazol-2-yl)-2-methyl-propyl)-carbamic acid tert-butyl ester; Raf kinase inhibitors for the treatment of neurotraumatic diseases
04/11/2006US7026335 Melanocortin receptor ligands
04/11/2006US7026333 Retroviral protease inhibitors
04/11/2006US7026328 Heterocyclic compounds which inhibit leukocyte adhesion mediated by α4 integrins
04/11/2006US7026327 2-etherified 4-fluoroalkyl-6-(p-sulfonylphenyl)pyrimidines,e.g., 2-(4-fluorophenoxy)-4-[4-(methylsulfonyl)phenyl]-6](trifluoromethyl)pyrimidine; treatment of the pain, fever and inflammation of variety of conditions and diseases
04/11/2006US7026326 Substituted heterocyclic compounds and methods of use
04/11/2006US7026324 Amide containing a pyridinone or pyrazinone compound as serine protease enzyme inhibitors
04/11/2006US7026323 N-(naphth-2-ylaminocarbonylacetyl)- or N-(naphth-2-ylcarbonylamino- acetyl)- piperazine derivatives, e.g., 2-[((4-(ethoxycarbonyl)piperazin-1-yl)carbonylmethyl)carbonyl]aminonaphthalene; useful as antithrombotic agents
04/11/2006US7026314 Psychological disorders, antidepressants, anxiolytic agents, eating disorders; serotonin receptors antagonist
04/11/2006US7026312 Substituted piperidines, pharmaceutical compositions containing these compounds, their use and processes for the preparation thereof
04/11/2006US7026310 Heteroaryl derivatives and their use as medicaments
04/11/2006US7026270 malayamycin A and desmethylmalayamycin A prepared from a previously unknown strain of Streptomyces malaysiensis, used for combating or controlling phytopathogenic fungi
04/11/2006US7025978 Use of polysiloxanes containing quarternary amino groups as formulation auxiliary agents, and agents containing the same
04/11/2006CA2274530C Process for producing 5-arylthio imidazole derivatives
04/11/2006CA2181570C Metalloproteinase inhibitors
04/11/2006CA2162382C Intercalators having affinity for dna and methods of use
04/06/2006WO2006037117A1 Substituted heterocyclic compounds and methods of use
04/06/2006WO2006037047A2 The r-isomer of 2-{2-[n-(2-indanyl)-n-phenylamino]ethyl}piperidine and other dermal anesthetic agents
04/06/2006WO2006036994A2 Modulators of crth2, cox-2 and faah
04/06/2006WO2006036981A2 Small molecule modulators of cytokine activity
04/06/2006WO2006036936A2 The s-isomer of 2-{2-[n-(2-indanyl)-n-phenylamino]ethyl}piperidine and other dermal anesthetic agents
04/06/2006WO2006036527A1 Substituted dipiperdine ccr2 antagonists
04/06/2006WO2006036507A1 4-(heteroaryl-methyl and substituted heteroaryl-methyl)-imidazole-2-thiones acting as alpha2 adrenergic agonists
04/06/2006WO2006036497A2 4-(condensed cyclicmethyl)-imidazole-2-thiones acting as alpha2 adrenergic agonists
04/06/2006WO2006036404A1 4-(substituted cycloalkylmethyl) imidazole-2-thones, 4-(substituted cycloalkenylmethyl) imidazole-2-thiones, 4-(substituted cyloalkylmethyl) imidazol-2-ones, 4-(substituted cycloalkenylmethyl) imidazol-2-ones and related compounds
04/06/2006WO2006036024A1 Proton pump inhibitors
04/06/2006WO2006036015A2 6- (pyridinyl) -4-pyrimidone derivates as tau protein kinase 1 inhibitors
04/06/2006WO2006035967A1 Pyridine derivatives and their use as medicaments for treating diseases related to mch receptor
04/06/2006WO2006035303A1 Muscarinic receptor antagonists
04/06/2006WO2006035280A1 3,4-dihydroisoquinoline compounds as muscrinic receptor antagonists for the treatment of respiratory, urinary and gastrointestinal diseases
04/06/2006WO2006035068A2 Hiv inhibiting 5-carbo- or heterocyclic substituted pyrimidines
04/06/2006WO2006035067A2 Hiv inhibiting 5-heterocyclyl pyrimidines
04/06/2006WO2006034833A1 Cyclic diarly ureas suitable as tyrosine kinase inhibitors
04/06/2006WO2006034769A1 Carbonyl compounds usable as coagulation factor xa inhibitors
04/06/2006WO2006023460A3 COMPOUNDS HAVING β2 ADRENERGIC RECEPTOR AGONIST AND MUSCARINIC RECEPTOR ANTAGONIST ACTIVITY
04/06/2006WO2005081687A3 Human hinge core mimetibodies, compositions, methods and uses
04/06/2006WO2005065195A3 Phenylamide and pyridylamide beta-secretase inhibitors for the treatment of alzheimer's disease
04/06/2006WO2005023796A8 New salts of omeprazole and esomeprazole i
04/06/2006US20060074247 Improving storage stability by reacting with hydrogen sulfate lithium- containing compound; aspartyl protease inhibitors
04/06/2006US20060074244 Pyridinyl substituted (1,2,3,)triazoles as inhibitors of the tgf-beta signalling pathway
04/06/2006US20060074243 Hydroxamic acid and amide compounds and their use as protease inhibitors
04/06/2006US20060074241 Enantioselective process
04/06/2006US20060074240 Process for the synthesis of derivatives of 2,3-dihydro-1,4-dioxino-[2,3-f] quinoline
04/06/2006US20060074237 Pyridines
04/06/2006US20060074123 Cyclic AMP-specific phosphodiesterase inhibitors
04/06/2006US20060074120 cyclopent[f]pyrazole derivatives; antiinflammatory agent; autoimmune diseases; side effect reduction, advantages over steroidal glucocorticoid ligands with respect to undesireable side-effects, efficacy, toxicity or metabolism
04/06/2006US20060074112 N-aryl (thio) anthranilic acid amide derivatives, their preparation and their use as VEGF receptor tyrosine kinase inhibitors
04/06/2006US20060074106 Treatment of inflammatory disorders
04/06/2006US20060074105 Substituted quinoline and quinazoline inhibitors of quinone reductase 2
04/06/2006US20060074092 Cysteine protease inhibitors with 2-cyano-4-amino-pyrimidine structure and cathepsin K inhibitory activity for the treatment of inflammations and other diseases
04/06/2006US20060074085 Bcl-XL inhibitors; N-{[4-({(1R)-5-(dimethylamino)-1-[(phenylthio)methyl]pentyl}amino)-3-nitrophenyl]sulfonyl}-4-(4-fluorophenyl)piperidine-1-carboxamide; useful for promoting apoptosis; Anticancer agents; autoimmune diseases; antiinflammatory agents
04/06/2006US20060074075 including cystic fibrosis transmembrane conductance regulator ("CFTR"), used for treating genetic disorders; respiratory system disorders
04/06/2006US20060074072 2-[3-(4-chlorophenyl)ureido] N-[4-(2-oxo-2H-pyridin-1-yl)phenyl]-4-methanesulfonylbutyramide; prophylaxis and/or therapy of thromboembolic diseases and for the treatment of tumors
04/06/2006US20060074069 e.g. (2R-trans) [4-(4-azetidin-3-yl-piperazin-1-yl)-2-benzyl-piperidin-1-yl]-(3,5-bis-trifluoromethyl-phenyl)-methanone;tachykinins, substance P inhibitor; antidepressant, anxiolytic, antiinflammatory agent, cognition activator; neurodegenerative diseases; addiction, sleep, eating disorders
04/06/2006US20060074068 Chemical compounds with dual activity, processes for their preparation and pharmaceutical compositions
04/06/2006US20060073472 Anti-inflammatory and protein kinase inhibitor compositions and related methods for downregulation of detrimental cellular responses and inhibition of cell death
04/06/2006DE102004047272A1 Inhibitoren der löslichen Adenylatzyklase Inhibitors of soluble adenylate cyclase
04/06/2006DE102004044829A1 5-Heterocyclylpyrimidine 5-Heterocyclylpyrimidine
04/06/2006CA2582777A1 Proton pump inhibitors
04/06/2006CA2582225A1 Substituted dipiperdine ccr2 antagonists
04/06/2006CA2581828A1 4-(heteroaryl-methyl and substituted heteroaryl-methyl)-imidazole-2-thiones acting as alpha2 adrenergic agonists
04/06/2006CA2581823A1 4-(condensed cyclicmethyl)-imidazole-2-thiones acting as alpha2 adrenergic agonists
04/06/2006CA2581732A1 Carbonyl compounds usable as coagulation factor xa inhibitors
04/06/2006CA2581179A1 6-(pyridinyl)-4 pyrimidone derivatives as tau protein kinase 1 inhibitors
04/06/2006CA2580838A1 Substituted heterocyclic compounds and methods of use
04/06/2006CA2579240A1 Small molecule modulators of cytokine activity
04/06/2006CA2577467A1 Hiv inhibiting 5-heterocyclyl pyrimidines
04/06/2006CA2577185A1 Cyclic diarly ureas suitable as tyrosine kinase inhibitors
04/06/2006CA2573976A1 Hiv inhibiting 5-carbo- or heterocyclic substituted pyrimidines
04/05/2006EP1642899A1 2,4-bis(trifluoroethoxy)pyridine compound and medicine containing the same
04/05/2006EP1641780A1 Processes for the preparation of 1- [(benzoimidazole-1yl) quinolin-8-yl] piperidin-4-ylamine derivatives
04/05/2006EP1641779A1 2-substitued 5, 6-diaryl-pyrazine derivatives as cb1 modulator.
04/05/2006EP1641778A1 Process for preparing intermediates useful to prepare certain antibacterial n-formyl hydroxylamines
04/05/2006EP1641777A1 Indole derivatives with apoptosis-inducing effect
04/05/2006EP1641776A1 Novel piperidine derivatives
04/05/2006EP1641775A1 2-pyridine alkyne derivatives useful for treating pain
04/05/2006EP1641765A1 Aryl-heteroaromatic products, compositions containing same and use thereof
04/05/2006EP1641764A1 5-membered heterocycle-based p38 kinase inhibitors
04/05/2006EP1641763A2 4-cyanopyrazole-3-carboxamide derivatives preparation and therapeutic application thereof
04/05/2006EP1641762A2 Cck-1 receptor modulators