Patents
Patents for C07D 401 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom (107,979)
05/2006
05/31/2006CN1780621A Sulfonamide derivatives as gamma secretase inhibitors.
05/31/2006CN1780617A Imidazolin-2-ylaminophenyl amides as IP antagonists.
05/31/2006CN1778800A Chiral piperazine substrated quinolone carboxylic acid derivative, and preparation and use thereof
05/31/2006CN1257902C Method for producing cilostazol
05/31/2006CN1257901C Tetrahydroquinoline ketopiperidine compounds and their preparation and use
05/31/2006CN1257893C PPAR full activator of amino acids of aralkyl possessing excellent activity for lowering sugar and ester
05/31/2006CN1257892C New indole derivatives with 5-HT6 receptor affinity
05/31/2006CN1257891C Nitrogenous five-membered ring compounds
05/31/2006CN1257886C Dehydroamino acids compounds
05/30/2006USRE39113 Neuropathic pain; in humans, animals
05/30/2006US7053215 For therapy of inflammatory and immunoregulatory disorders and diseases, such as multiple sclerosis, rheumatoid arthritis and type I diabetes
05/30/2006US7053213 Therapeutic heterocycles
05/30/2006US7053113 Mannich base prodrugs of 3-(pyrrol-2-yl-methylidene)-2-indolinone derivatives
05/30/2006US7053112 Imidazolidinedione analogs useful as anticoagulants and antithrombotics
05/30/2006US7053110 Dietetics; osteoporosis; muscular disorders
05/30/2006US7053108 Indoline compounds
05/30/2006US7053107 Antiproliferative agents, angiogenesis inhibitors for treating cancer, eye disorders, diabetic retinopathy, neovascular glaucoma, rheumatoid arthritis, and psoriasis; N-Cyclopropyl-2-{3-[(E)-2-(4-methyl-pyridin-2-yl)-vinyl]-1H-indazol-6-ylamino}-benzamide
05/30/2006US7053105 Farnesyl transferase inhibiting quinoline and quinazoline derivatives as farnesyl transferase inhibitors
05/30/2006US7053095 A pyridyl-2yl-4-[1,2,3-triazole] derivatives therapeutic agent for treating cancer, glomerulonephritis, diabetic nephropathy, hepatic fibrosis, pulmonary fibrosis, hyperplasia, restenosis, skin disorders
05/30/2006US7053094 Increasing contractile force in cardiac muscle fiber by administering a N-[(3-yloxy)-phenyl]-arylamide derivatives; modulating at the cardiac sarcomere (cardiac beta myosin) for congestive heart failure
05/30/2006US7053091 Androgen sensitive diseases; prostate cancer; skin disorders; alopecia
05/30/2006US7053089 Such as 4-((methyl-pyrimidin-2-ylamino)-methyl)-piperidine-1-carboxylic acid benzyl ester; useful for pain relief; treating migraine, depression, anxiety, schizophrenia, Parkinson's disease, and stroke; N-methyl-D-aspartate (NMDA)
05/30/2006US7053088 Vanilloid receptor ligands and their use in treatments
05/30/2006US7053086 For cancer therapy
05/30/2006US7053085 EP4 receptor agonist, compositions and methods thereof
05/30/2006US7053084 Antagonist for preventing the deposits of amyloid protein, for treating neurodegenerative disease, Alzheimer's disease and Down's Syndrome; (2R,3S) N1-[1,3-dihydro-1-methyl-2-oxo-5-phenyl-2H-1,4-benzodiazepin-3-yl]-2-(2-methylpropyl)-3-allyl-butanediamide
05/30/2006US7053081 Cyclic malonamides as inhibitors of A-β protein production
05/30/2006US7053078 Serine protease inhibitors
05/30/2006US7053057 Caspase inhibitors and uses thereof
05/30/2006US7052673 Anticancer, antitumor agents; mixture of metal, drug, peptide and carriers
05/30/2006CA2398159C Sulphonylaminocarbonyltriazolinones having substitutents bonded via oxygen
05/30/2006CA2321380C 6-azauracil derivatives as thyroid receptor ligands
05/30/2006CA2195243C Triazole compounds and the use thereof
05/30/2006CA2141692C Prodrugs of imidazole carboxylic acids as angiotensin ii receptor antagonists
05/26/2006WO2006055760A1 Triazole compounds that modulate hsp90 activity
05/26/2006WO2006055463A2 2-amino-3-functionalized tetralin derivatives and related glycogen phosphorylase inhibitors
05/26/2006WO2006055462A1 2-amino-4-functionalized tetralin derivatives and related glycogen phosphorylase inhibitors
05/26/2006WO2006055187A1 Sulfonyl-substituted bicyclic compounds as modulators of ppar
05/26/2006WO2006054912A1 Aryl(hetaryl)-3-aminomethyl-quinilone-2 derivatives in the form of no-synthetase i and cyclooxygenase-2 nhibitors, methods for the production thereof and compositions based thereon
05/26/2006WO2006054700A1 Optical filter
05/26/2006WO2006054623A1 Novel pyridonecarboxylic acid derivatives or salts thereof
05/26/2006WO2006054560A1 Aromatic amide derivatives, medicinal compositions containing the same, medical uses of both
05/26/2006WO2006054314A1 Polymorphic forms of imatinib mesylate
05/26/2006WO2006054143A1 Polymorphs of {5-[3-(4,6-difluoro-1h-benzoimidazol-2-yl)-1h-indazol-5-yl]-4-methyl-pyridin-3-ylmethyl}-ethyl-amine
05/26/2006WO2006053643A1 N-heterocyclyl phthalic acid diamides as insecticides
05/26/2006WO2006053429A1 Process for the manufacture of 3-hydroxy-n-alkyl-1-cycloalkyl-6-alkyl-4-oxo-1,4-dihydropyridine-2-carboxamide and its related analogues
05/26/2006WO2006026760A3 1-amino imidazo-containing compounds and methods
05/26/2006WO2006026703A8 Chemical compounds
05/26/2006WO2006010079A3 Process for preparing naratriptan hydrochloride
05/26/2006WO2005123080A3 Nitrogen-containing heterocyclyl substituted imidazoquinolines and imidazonaphthyridines
05/26/2006WO2005108358A3 Pyrrolidine derivatives useful as bace inhibitors
05/26/2006CA2588768A1 Aromatic amide derivatives, medicinal compositions containing the same, medical uses of both
05/26/2006CA2588766A1 Heterocycle substituted carboxylic acids
05/26/2006CA2588513A1 3-phenyl-pyrazole derivatives as modulators of the 5-ht2a serotonin receptor useful for the treatment of disorders related thereto
05/26/2006CA2588034A1 Pyridonecarboxylic acid derivatives or salts thereof
05/26/2006CA2587482A1 N-heterocyclyl phthalic acid diamides as insecticides
05/26/2006CA2586612A1 Triazole compounds that modulate hsp90 activity
05/26/2006CA2585378A1 Anthranilamide insecticides
05/26/2006CA2585172A1 Sulfonyl-substituted bicyclic compounds as modulators of ppar
05/25/2006US20060111573 Resolution of mefloquine with o,o-di-p-aroyltartaric acid
05/25/2006US20060111567 Nonpeptide substituted spirobenzoazepines as vasopressin antagonists
05/25/2006US20060111425 To treat diseases of respiratory, urinary and gastrointestinal systems; highly selective; significant potency; (2R,2S)(1 alpha ,5 alpha ,6 alpha )-N-{-[4-(1,3-dioxo-1,3-dihydro-isoindol-2-yl)-butyl]-3-azabicyclo[3.1.0]hex-6-yl-methyl}-2-hydroxy-2-cyclopentyl-2-phenylacetamide
05/25/2006US20060111424 Treating nuclear hormone receptor-associated conditions such as cancer and immune disorders; (3a alpha ,4 alpha ,7 alpha ,7a alpha )-2-(3-Chloro-4-hydroxyphenyl)hexahydro-4,7-methano-1H-isoindole-1,3(2H)-dione
05/25/2006US20060111419 Novel fused indazole compounds
05/25/2006US20060111403 Cyano anthranilamide insecticides
05/25/2006US20060111400 Piperidinetriol derivatives as inhibitors of glycosylceramidsynthase
05/25/2006US20060111392 Substituted biaryl-carboxylate derivatives
05/25/2006US20060111389 Therapeutic acridone and acridine compounds
05/25/2006US20060111377 Heterocyclic derivatives
05/25/2006US20060111375 Compound having tgfß inhibitory activity and medicinal composition containing the same
05/25/2006US20060111371 Protein tyrosine kinase inhibitors
05/25/2006US20060111364 Reversible inhibitors of cysteine proteases S, K, F, L and B; N-[2-(Benzylamino)pyrimidin-4-yl]-N-(cyanomethyl)-L-phenylalaninamide
05/25/2006US20060111357 Quinoline compounds for use in mch receptor related disorders
05/25/2006US20060111323 Use of polysiloxanes having quaternary ammonium groups as formulation auxiliaries, and compositions comprising them
05/25/2006US20060111322 Indazole compounds, pharmaceutical compositions, and methods for mediating or inhibiting cell proliferation
05/25/2006US20060111303 N-[(1S)-3-{(2Z)-2-[(4R)-3,4-dimethyl-1,3-thiazolidin-2-ylidene]hydrazino}-2,3-dioxo-1-(tetrahydro-2H-pyran-4-yl)propyl]cycloheptanecarboxamide; cysteine protease inhibitors; for the treatment of inflammatory, immune, ischemic, respiratory,circulatory, neuronal, blood, hepatic and metabolic diseases
05/25/2006US20060110638 Electrochromic compounds
05/24/2006EP1659129A1 Coordination metal compound, material for organic electroluminescence device, material for luminescent coating formation and organic electroluminescence device
05/24/2006EP1659120A1 3-substituted quinoline-4-carboxamide derivatives as NK-3 and NK-2 receptor antagonists
05/24/2006EP1659111A2 Piperidine derivatives useful as ccr5 antagonists
05/24/2006EP1658847A2 Indane derivatives as dermal anesthetic agents
05/24/2006EP1658503A1 Chemiluminescent compounds
05/24/2006EP1658284A1 3,5 disubstituted indazole compounds, pharmaceutical compositions, and methods for mediating or inhibiting cell proliferation
05/24/2006EP1658283A2 Substituted pyrrole derivatives and their use as hmg-co inhibitors
05/24/2006EP1658280A1 Quinazoline derivatives as angiogenesis inhibitors
05/24/2006EP1658270A1 Novel 6-phenylphenantridines
05/24/2006EP1658269A1 Fused compounds that inhibit vanilloid receptor subtype 1 (vr1) receptor
05/24/2006EP1575935B1 Process for the preparation of sulphinyl derivatives by oxidation of the corresponding sulfides
05/24/2006EP1506185B1 Compounds and their use as inhibitors of 5-ht
05/24/2006EP1487452B1 Use of 4-(4-methylpiperazin-1-ylmethyl)-n 4-methyl-3-(4-pyridin-3-yl) pyrimidin-2-ylamino) phenyl -benzamide for treating seminomas
05/24/2006EP1355900B1 Heterocyclylalkylindole or -azaindole compounds as 5-hydroxytryptamine-6 ligands
05/24/2006EP1320529B1 Quinoline derivatives as antibacterials
05/24/2006EP1254904B1 Novel piperidine compounds and drugs containing the same
05/24/2006EP1226129B1 Methods and compositions utilizing quinazolinones
05/24/2006EP1212298B1 Isolation of natural l-beta-3-indolylalanine and enrichment of natural aliphatic amino acid mixtures with natural l-beta-3-indolylalanine
05/24/2006DE102004055582A1 N-Heterocyclyl-phthalsäurediamide N-heterocyclyl-Phthalamides
05/24/2006CN1777600A 4-, 6- o 7-hydroxyindoles having n-oxide groups and the use thereof as therapeutic agents
05/24/2006CN1777599A 5-hydroxyindoles with n-oxide groups and use thereof as a phosphodiesterase 4 inhibitor
05/24/2006CN1777598A Polymorphs of s-omeprazole.
05/24/2006CN1777597A Indazole having analgesic activity