Patents
Patents for C07D 401 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom (107,979)
04/2006
04/27/2006WO2006043594A1 1,5-diheterocycle-1h-triazole derivative
04/27/2006WO2006043515A1 Pyrimidine-5-carboxylic acid derivative
04/27/2006WO2006043490A1 Pyrimidine derivative fused with nonaromatic ring
04/27/2006WO2006043064A1 Piperidines and related compounds for treatment of alzheimer's disease
04/27/2006WO2006042955A1 Pyridine derivatives and the preparation and the therapeutic use thereof
04/27/2006WO2006042638A1 3,6-substituted 5-arylamino-1h-pyidine-2-one derivatives and related compounds as poly(adp-ribose)polymerase (parp) inhibitors in the treatment of tissue damage or disease caused by necrosis or apoptosis
04/27/2006WO2006014290A3 Anti-inflammatory medicaments
04/27/2006WO2006012256A3 Fkbp binding composition and pharmaceutical use thereof
04/27/2006WO2006000371A3 Pyrimidine derivatives as 11beta-hsd1 inhibitors
04/27/2006WO2005101989A3 Piperidine derivatives as modulators of chemokine receptor ccr5
04/27/2006WO2005090320A3 Triazole derivatives and method of using the same to treat hiv infections
04/27/2006US20060089386 Novel process for substituted sulfoxides
04/27/2006US20060089383 Substituted piperidine compounds and methods of their use
04/27/2006US20060089380 Treating nervous system disorders such as mild cognitive impairment, Alzheimer's disease or dementia associated with Down syndrome; e.g. use of 5,7-dichloro-8-hydroxy-2-(2-pyridyl)-quinoline (PBT 1052)
04/27/2006US20060089379 Tetrahydropyranyl cyclopentyl tetrahydroisoquinoline modulators of chemokine receptor activity
04/27/2006US20060089371 Phenyl or heteroaryl amino alkane derivatives as ip receptor antagonist
04/27/2006US20060089369 pyrimidine and pyridine derivatives; diabetes, neurodegenerative disorders, obesity, atherosclerotic cardiovascular disease, hypertension, polycystic ovary syndrome, syndrome X, ischemia, traumatic brain injury, bipolar disorder, immunodeficiency, cancer
04/27/2006US20060089363 Antibacterial agents
04/27/2006US20060089354 ligands for receptor localization studies; for inhibiting binding of vanilloid ligand to a capsaicin receptor; Phosphoric acid dibenzyl ester 4-(4-tert-butyl-phenylamino)-7-(3-trifluoromethyl-pyridin-2-yl)-quinazolin-2-ylmethyl ester; to treat neuropathic pain, itch, urinary incontinence, cough, obesity
04/27/2006US20060089344 E.g., 2-(Methylamino)-2-oxoethyl 3-[1-(1-isoquinolyl)-4-piperidyl]propylcarbamate hydrochloride and 3{2-[1-(2-quinolyl)-4-piperidyl]-ethyl}-1,3-oxazolidine-2,4-dione; preventing or treating a pathology in which endogenous cannabinoids and/or any other substrate metabolized by the enzyme FA; analgesics
04/27/2006US20060089262 Substituted (thioxo)carbonylamino phenyl uraciles
04/27/2006CA2584504A1 Piperidines and related compounds for treatment of alzheimer's disease
04/27/2006CA2584422A1 1-(hetero)aryl-3-amino-pyrollidine derivatives for use as mglur3 receptor antagonists
04/27/2006CA2584328A1 Phosphodiesterase 4 inhibitors
04/27/2006CA2584262A1 Diphenyl substituted alkanes as flap inhiibitors
04/27/2006CA2583667A1 Sulfonamide peri-substituted bicyclics for occlusive artery disease
04/27/2006CA2583565A1 3,6-substituted 5-arylamino-1h-pyridine-2-one derivatives and related compounds as poly(adp-ribose)polymerase (parp) inhibitors in the treatment of tissue damage or disease causedby necrosis or apoptosis
04/27/2006CA2583534A1 Cgrp receptor antagonists
04/27/2006CA2583392A1 Imidazole derivatives as vanilloid receptor ligands
04/27/2006CA2583342A1 Spiropiperidine compounds useful as beta-secretase inhibitors for the treatment of alzhermer's disease
04/27/2006CA2583158A1 Triazoles and their use as bradykinin b1 receptor antagonists
04/27/2006CA2583153A1 1,5-diheterocycle-1h-triazole derivative
04/27/2006CA2582778A1 Pyridine derivatives and the preparation and the therapeutic use thereof
04/26/2006EP1650204A1 Process for producing 1,2,4-triazole compound and intermediate therefor
04/26/2006EP1650203A1 Process of preparation of benzimidazol-2-yl quinolinone derivatives
04/26/2006EP1650195A1 Method of inhibiting production of osteopontin
04/26/2006EP1650193A2 6-Phenylphenanthridines with PDE-IV inhibiting activity
04/26/2006EP1650192A1 Quinolone derivative or salt thereof
04/26/2006EP1649871A1 Retroviral protease inhibitor combinations
04/26/2006EP1648884A2 Pyrazolyl-indole derivatives active as kinase inhibitors, process for their preparation and pharmaceutical compositions comprising them
04/26/2006EP1648883A2 Lanthanide complexes preparation and uses thereof
04/26/2006EP1648882A1 3-fluoro-piperidines as nmda/nr2b antagonists
04/26/2006EP1648881A1 Substituted indole ligands for the orl-1 receptor
04/26/2006EP1648879A1 Heteroaryl-tetrahydropiperidyl compounds useful for treating or preventing pain
04/26/2006EP1648878A1 Piperidine compounds and pharmaceutical compositions containing them
04/26/2006EP1648877A1 Substituted pyridin-2-ylamine analogues
04/26/2006EP1648876A1 5-ht sb 2b /sb receptor antagonists
04/26/2006EP1648875A1 2-aminophenyl-4-phenylpyrimidines as kinase inhibitors
04/26/2006EP1648871A1 Piperidine or 8-aza-bicyclo 3.2.1 oct-3-yl derivatives useful as modulators of chemokine receptor activity
04/26/2006EP1648870A2 Sulfonic acid derivatives of polycyclic dyes used for analytical applications
04/26/2006EP1648867A1 Ppar active compounds
04/26/2006EP1648458A1 2-'4(phenylamino)-piperidin-1-yl]-n-phenyl-acetamine derivtives and related compounds as neuropeptide y5 (npy5) ligands for the treatement of obesity
04/26/2006EP1648448A1 Chemical compounds
04/26/2006EP1648447A1 Pyrazolines as par-1 antagonists for treatment of cardiovascular diseases
04/26/2006EP1648445A1 Indol-5-yl sulfonamide derivatives, their preparation and their use 5-ht-6 as modulators
04/26/2006EP1648443A1 1-sulfonylindole derivatives, their preparation and their use as 5-ht6 ligands
04/26/2006EP1648426A2 Benzimidazole derivatives and their use as protein kinases inhibitors
04/26/2006EP1379520B1 N-substituted nonaryl-heterocyclic nmda/nr2b antagonists
04/26/2006EP0915844B1 Process for preparing 3-pyrroline-2-carboxylic acid derivatives
04/26/2006CN1764668A Phosphonooxy quinazoline derivatives and their pharmaceutical use
04/26/2006CN1764659A Prostaglandin analogs as EP4 receptor antagonists
04/26/2006CN1764658A Preparation and use of 2-substituted-5-oxo-3- pyrazolidinecarboxylates
04/26/2006CN1764655A Aromatic sulfone hydroxamates and their use as protease inhibitors
04/26/2006CN1764651A Quinazoline derivatives as antitumor agents
04/26/2006CN1764650A 2, 3, 6-trisubstituted-4-pyrimidone derivatives
04/26/2006CN1764649A Benzyl-pyridazinons as reverse transcriptase inhibitors
04/26/2006CN1764648A hydroxamid acid derivatives as histone deacetylase (HDAC) inhibitors
04/26/2006CN1764641A Viral polymerase inhibitors
04/26/2006CN1764450A Crystalline N-formyl hydroxylamine compounds
04/26/2006CN1764380A N-phenyl- (4-pyridyl)- azinyl!amine derivatives as plant protection agents.
04/26/2006CN1762355A (imidazol-5-yl)methyl-2-quinolinone derivatives as inhibitors of smooth muscle cell proliferation
04/26/2006CN1253449C Indolylmaleimide derivatives as protein kinase C inibitors
04/26/2006CN1253442C Novel thiazine or pyrazine derivatives
04/26/2006CN1253441C Protease inhibitors
04/26/2006CN1253435C Aryl oxime-piperazines useful as CCR5 antagonists
04/25/2006US7034057 Controlling tumor necrosis factor; antiinflamamtory agents, autoimmune disease
04/25/2006US7034052 Anticancer agents; inflammatory bowel disorders; myelodysplastic syndrome
04/25/2006US7034049 3(5)-amino-pyrazole derivatives, process for their preparation and their use as antitumor agents
04/25/2006US7034047 Triazole derivative
04/25/2006US7034043 Cell adhesion inhibitors
04/25/2006US7034042 Corticotropin releasing factor receptor antagonist
04/25/2006US7034039 Fused heterocyclic compounds
04/25/2006US7034035 Having a high residual activity, greater activity at lower application rates, curative activity, and a broader spectrum of efficacy; heterocyclic aromatic amides having a hydroxy group adjacent to the amide functionality
04/25/2006US7034034 Substituted 2-cyclohexyl-4-phenyl-1H-imidazole derivatives
04/25/2006US7034033 Substituted quinazolinone compounds
04/25/2006US7034031 Modulators of TNF-α signaling
04/25/2006US7034029 1-aryl- or 1-alkylsulfonyl-heterocyclylbenzazoles as 5-hydroxytryptamine-6 ligands
04/25/2006US7034028 Treatment of inflammatory disorders
04/25/2006US7034022 Proteases, kinases enzyme inhibitors; cardiovascular disorders; central nervous system disorders; antiinflammatrory agents; bone disorders; infections
04/25/2006US7034019 Prodrugs of HIV replication inhibiting pyrimidines
04/25/2006US7034018 Substituted pyrrole mannich bases to combat pain and allergic reactions
04/20/2006WO2006042150A1 Diaminoalkane aspartic protease inhibitors
04/20/2006WO2006041888A2 Substituted aryl or heteroarylsulfonylbutanamides for use as anti-inflammatory agents
04/20/2006WO2006041635A2 Arylthiobenzylpiperidine derivatives
04/20/2006WO2006041405A1 Substituted amino-pyrimidones and uses thereof
04/20/2006WO2006040778A1 Process for preparations and purification of pantoprazole sesquihydrate
04/20/2006WO2006040728A1 1-[2-(4-benzyl-4-hydroxy-piperidin-1-yl)-ethyl]-3-(2-methyl-quinolin-4-yl)-urea as crystalline sulfate salt
04/20/2006WO2006040666A1 Substituted n-alkylpyrimidinones
04/20/2006WO2006040650A1 4-methoxyacridine-1-carboxamide derivatives and the phenazine and oxanthrene analogs as pde4-inhibitors for the treatment of asthma and chronic pulmonary disease (copd)
04/20/2006WO2006040646A1 Benzimidazole or indole amides as inhibitors of pin1