| Patents for C07D 401 - Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom (107,979) |
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| 12/04/2008 | US20080300239 Quinoline derivatives as pi3 kinase inhibitors |
| 12/04/2008 | US20080300237 Pharmaceutically Active Diazepanes |
| 12/04/2008 | US20080300236 Quinoline-derived amide modulators of vanilloid vr1 receptor |
| 12/04/2008 | US20080300234 N-(1-Methyl-1-phenyl-ethyl)-3-{[2-(2-oxo-2,3-dihydro-1H-indol-5-ylamino)-5-trifluoromethyl-pyrimidin-4-ylamino]-methyl}-benzenesulfonamide, useful in the treatment of breast cancer |
| 12/04/2008 | US20080300232 N-Piperidine Derivatives as Ccr3 Modulators |
| 12/04/2008 | US20080299639 adduct comprising a molecule binding with a kinase; antiinflammatory agents; modulating activation state of p38 kinase protein; switch control ligands to induce or restrict conformation |
| 12/04/2008 | DE102007025718A1 Pyridazinonderivate Pyridazinone derivatives |
| 12/04/2008 | CA2688599A1 Compounds with antiparasitic activity, applications thereof to the treatment of infectious diseases caused by apicomplexans |
| 12/04/2008 | CA2688518A1 Pyridazinone derivatives for use in the treatment of a disease which is influenced by inhibiton of met kinase |
| 12/04/2008 | CA2688517A1 Aryl ether pyridazinone derivatives for use in the treatment of tumours |
| 12/04/2008 | CA2688375A1 Spirocyclopropyl piperidine derivatives |
| 12/04/2008 | CA2688326A1 Tetrahydroisoquinolin-1-one derivative or salt thereof |
| 12/04/2008 | CA2688110A1 Azacyclylbenzamide derivatives as histamine-3 antagonists |
| 12/04/2008 | CA2687976A1 Therapeutic ((phenyl)imidazolyl)methylquinolinyl compounds |
| 12/04/2008 | CA2687973A1 ((bicylicheteroaryl) imidazolyl)methylheteroaryl compounds as adrenergic receptor agonists |
| 12/04/2008 | CA2687966A1 Thiazoles and pyrazoles useful as kinase inhibitors |
| 12/04/2008 | CA2687942A1 Therapeutic agent for cerebral infarction |
| 12/04/2008 | CA2687931A1 Ccr2 receptor antagonists and uses thereof |
| 12/04/2008 | CA2687821A1 Benzimidazolone chymase inhibitors |
| 12/04/2008 | CA2687625A1 3-(imidazolyl)-pyrazolo[3,4-b]pyridines |
| 12/04/2008 | CA2687365A1 4,4-disubstituted piperidine derivatives |
| 12/04/2008 | CA2687321A1 Pyridyl piperidine orexin receptor antagonists |
| 12/04/2008 | CA2687132A1 4' substituted compounds having 5-ht6 receptor affinity |
| 12/03/2008 | EP1997856A1 Optical recording medium and azo metal chelate compound |
| 12/03/2008 | EP1997823A1 Boronic ester and acid compounds, synthesis and uses |
| 12/03/2008 | EP1997818A2 Quinolinone derivatives and their use to treat pain |
| 12/03/2008 | EP1997811A2 Indazole, benzoxazole and pyrazolopyridine derivatives as P38 kinase inhibitors |
| 12/03/2008 | EP1997810A2 Indazole, benzoxazole and pyrazolopyridine derivatives for medical use |
| 12/03/2008 | EP1997809A2 Indazole, benzoxazole and pyrazolopyridine derivatives for medical use |
| 12/03/2008 | EP1997805A1 Compounds with antiparasitic activity, applications thereof to the treatment of infectious diseases caused by apicomplexans |
| 12/03/2008 | EP1997495A1 2-phenoxy- and 2-phenylsulfanyl-benzenesulfonamide derivatives with ccr3 antagonistic activity for the treatment of asthma and other inflammatory or immunological disorders |
| 12/03/2008 | EP1996585A2 Bicycloheteroaryl compounds as p2x7 modulators and uses thereof |
| 12/03/2008 | EP1996577A1 Heterocyclic substituted pyridine compounds with cxcr3 antagonist activity |
| 12/03/2008 | EP1996576A1 Ccr5 antagonists useful for treating hiv |
| 12/03/2008 | EP1996575A2 Crystal form of besipirdine chlorhydrate, process preparation and use thereof |
| 12/03/2008 | EP1996574A1 Quinoline and isoquinoline derivatives as phosphodiesterase 10 inhibitors |
| 12/03/2008 | EP1996562A1 Substituted 4-amino-quinazoline derivatives as regulators of metabotropic glutamate receptors and their use for producing drugs |
| 12/03/2008 | EP1996558A1 Heterobicyclic carboxamides as inhibitors for kinases |
| 12/03/2008 | EP1996555A1 Compounds which potentiate ampa receptor and uses thereof in medicine |
| 12/03/2008 | EP1996553A2 Tumor necrosis factor alpha inhibitors and their use in the treatment of human diseases |
| 12/03/2008 | EP1996550A2 Carboxyamine compounds and their use in the treatment of hdac dependent diseases |
| 12/03/2008 | EP1996548A1 Sigma receptor compounds |
| 12/03/2008 | EP1996546A2 Substituted gamma lactams as prostaglandin ep2 agonists |
| 12/03/2008 | EP1996545A1 Soluble epoxide hydrolase inhibitors and methods of using same |
| 12/03/2008 | EP1778633B1 Indoles useful in the treatment of inflammation |
| 12/03/2008 | EP1737463B1 Pyrimidines with tie2 (tek) activity |
| 12/03/2008 | EP1492785B1 2-hydroxy-3-heteroarylindole derivatives as gsk3 inhibitors |
| 12/03/2008 | EP1480954B1 Vanilloid receptor modulators |
| 12/03/2008 | EP1426371B1 Tetrazoyl oxime derivatives and agrochemicals containing the same as the active ingredient |
| 12/03/2008 | EP1423388B1 2-arylamino-pyrimidines for the treatment of gsk3-related disorders |
| 12/03/2008 | EP1377540B1 Inhibitors of integrin alpha-v-beta-6 |
| 12/03/2008 | EP1373218B9 Imidazolyl derivatives useful as histamine h3 receptor ligands |
| 12/03/2008 | EP1068202B1 1-(3-heteroarylpropyl- or -prop-2-enyl)-4-benzylpiperidines used as nmda receptor antagonists |
| 12/03/2008 | CN101316841A Arylmethylene urea derivative and use thereof |
| 12/03/2008 | CN101316840A 1,5-substituted indol-2-yl amide derivatives |
| 12/03/2008 | CN101316839A Acid addition salt of dihydropyridine derivative |
| 12/03/2008 | CN101316838A 1,1-dioxo-thiomorpholinyl indolyl methanone derivatives for use as h3 modulators |
| 12/03/2008 | CN101316837A Substituted pyrrolones as allosteric modulators of glucokinase |
| 12/03/2008 | CN101316836A Substituted dihydroisoindolones as allosteric modulators of glucokinase |
| 12/03/2008 | CN101316835A 5-substituted indole-2-carboxamide derivatives |
| 12/03/2008 | CN101316834A 1h-benzimidazole-4-carboxamides substituted with phenyl at the 2-position are potent PARP inhibitors |
| 12/03/2008 | CN101316823A 2,4,5-triphenyl imidazoline derivatives as inhibitors of the interaction between p53 and MDM2 proteins for use as anticancer agents |
| 12/03/2008 | CN101316587A 取代的吡唑化合物 Substituted pyrazole compounds |
| 12/03/2008 | CN101314595A Aromatic hydrocarbons connected multi-polyamine large-ring derivants, preparation method and medical use thereof |
| 12/03/2008 | CN100439359C Indolylmaleimide derivatives |
| 12/03/2008 | CN100439357C Benzo [b][1,4] dioxepine derivatives |
| 12/03/2008 | CN100439344C 4-anilino quinazoline derivatives as antiproliferative agents |
| 12/03/2008 | CN100439341C Indazole derivatives as CRF antagonists |
| 12/03/2008 | CN100439340C 3-cyanoquinolines, 3-cyano-1,6-naphthyridines, and 3-cyano-1,7-naphthyridines as protein kinase inhibitors |
| 12/03/2008 | CN100439339C 2-pyridone derivatives as netrophil elastase inhibitors and their use. |
| 12/03/2008 | CN100439337C Phenyl substituted piperidine compounds for use as PPAR activators |
| 12/03/2008 | CN100438872C Method of stabilizing lipid-rich plaque and method of preventing rupture thereof |
| 12/02/2008 | US7459580 Process for trans-4-amino-1-cyclohexanecarboxilic acid derivatives |
| 12/02/2008 | US7459566 1,2,4-oxadiazol-5-one-4-(benzimidazolylmethylamino)benzamidine compounds |
| 12/02/2008 | US7459562 Monocyclic heterocycles as kinase inhibitors |
| 12/02/2008 | US7459561 Containing pyridine, phenyl, thiazole and triazole rings, e.g., 1-[[N-methyl-N-3-[(methylamino)acetoxymethyl]pyridin-2-yl]carbamoyloxy]ethyl-1-[(2R,3R)-2-(2,4-difluorophenyl)-2-hydroxy-3-[4-(4-cyanophenyl)thiazol-2-yl ]butyl]-1H-[1,2,4]triazol-4-ium chloride; parenteral treatment of fungal diseases |
| 12/02/2008 | US7459556 Process for preparing substituted 8-azabicyclo[3.2.1]octan-3-ols |
| 12/02/2008 | US7459552 Reacting N-[2,4-bis(methylthio)-6-methylpyridin-3-yl]-2-[4-(2-hydroxyethyl)piperazin-1-yl]acetamide with 5-benzyloxy-2-mercaptobenzimidazole in presence of triphenylphosphine and diethyl azodicarboxylate; acyl-coenzyme A cholesterol acyltransferase (ACAT) inhibitor |
| 12/02/2008 | US7459480 Benzodioxepine derivatives |
| 12/02/2008 | US7459473 1-(phenylmethyl)sulfonyl-2-hydroxymethyl pyrrolidine for example; use treating neurological disorders including physically damaged nerves and neurodegenerative diseases; treating alopecia and promoting hair growth |
| 12/02/2008 | US7459470 For example, N-(Isoquinolin-3-yl)-2-(4-pyridylmethyl)aminobenzoic acid amide-N-oxide; use as pharmaceutical agents for treating diseases that are triggered by persistent angiogenesis, such as psoriasis, arthritis, hemangioma, angiofibroma, eye diseases, cirrhosis of the liver |
| 12/02/2008 | US7459466 Antiinflammatory agents; autoimmune diseases; anticancer agents |
| 12/02/2008 | US7459465 Isoquinoline compound and pharmaceutical use thereof |
| 12/02/2008 | US7459462 Water soluble groups on ring A; antitumor antibiotics; 1-Desoxy-5-C-[(8R)-4',9,9'-trihydroxy-6'-methoxy-1,1',3',5',8'-pentaoxo-1,1',2,3',5',6,7,8'-octahydrospiro[cyclopenta[g]isoquinoline-8,2'-cyclopenta[b]-naphthalene]-3-yl]pentitol; topoisomerase inhibitors; cyclodextrin inclusions; stereoisomers |
| 12/02/2008 | US7459460 Trisubstituted heteroaromatic compounds as calcium sensing receptor modulators |
| 12/02/2008 | US7459457 Polycyclic pyridines as potassium ion channel modulators |
| 12/02/2008 | US7459456 e.g. 3-(3-{2-[4-(2-methyl-5-quinolinyl)-1-piperazinyl]ethyl}phenyl)-1,3-oxazolidin-2-one; serotonin receptor antagonist and inverse agonists, agonists or partial agonists, serotonin reuptake inhibitor; antidepressant, anxiolytic agent |
| 12/02/2008 | US7459454 Aminopyrazine derivatives and compositions |
| 12/02/2008 | US7459453 Pyridazin-3(2H)-one derivatives as PDE4 inhibitors |
| 12/02/2008 | US7459452 Dihydroxypyrimidine carboxamide inhibitors of HIV integrase |
| 12/02/2008 | CA2461622C Substituted benzimidazole compounds and their use for the treatment of cancer |
| 12/02/2008 | CA2424600C Aliphatic nitrogenous five-membered ring compounds |
| 12/02/2008 | CA2361841C Mevinolin derivatives |
| 12/02/2008 | CA2344144C Pyridinium derivatives for the management of aging-related and diabetic vascular complications, process for their preparation and therapeutic uses thereof |
| 12/02/2008 | CA2305548C Prostaglandin agonists and their use to treat bone disorders |
| 12/02/2008 | CA2265672C Pyrazinones and triazinones and their derivatives thereof |
| 12/02/2008 | CA2186380C Novel carbamates and ureas as modifiers of multi-drug resistance |
| 11/27/2008 | WO2008144305A1 Diaryl-substituted tetrahydroisoquinolines as histamine h3 receptor and serotonin transporter modulators |
| 11/27/2008 | WO2008144299A1 5- (aminoazacyclyl) -3-sulfonyl-lh- indazoles as 5-hydroxytryptamine- 6 ligands for the treatment of cns disorders |
| 11/27/2008 | WO2008144266A1 Spiroindalones |