Patents
Patents for C07D 295 - Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms (34,005)
12/2008
12/18/2008WO2008153573A1 4-phenylpiperazine derivatives with functionalized linkers as dopamine d3 receptor selective ligands and methods of use
12/18/2008WO2008153159A1 Amine compound and pharmaceutical use thereof
12/18/2008WO2008152650A1 Process for preparation of substantially optically pure levorotatory and dextrorotatory enantiomers of cetirizine using novel intermediates
12/18/2008WO2008152090A1 Novel compound
12/18/2008WO2008152089A1 Novel compounds
12/18/2008WO2008151969A1 Piperazine and [1,4] diazepan derivatives as nk antagonists
12/18/2008WO2008151957A1 Cyclohexyl derivatives
12/18/2008WO2008151702A1 Substituted 2- [2- (phenyl) ethylamino] alkaneamide derivatives and their use as sodium and/or calcium channel modulators
12/18/2008WO2008130332B1 Subsituted sulphonamides, process for their preparation, pharmaceutical composition comprising thereof and their use
12/18/2008WO2008130321A3 Novel n-tetrahydronaphtalene or 5-heterocyclyl-chromane or 8-heterocyclyl-tetrahydronaphtalene derivatives for the treatment of pain
12/18/2008WO2008130319A3 Novel n-tetrahydronaphtalene or n-chromane carboxamide derivatives for the treatment of pain
12/18/2008WO2008113756A3 Compounds having aryl-sulphonamidic structure useful as metalloproteases inhibitors
12/18/2008WO2008087654A3 PIPERIDINES AS INHIBITORS OF 11β-HYDROXYSTEROID DEHYDROGENASE TYPE 1
12/18/2008WO2008064054A3 Compounds which modulate the cb2 receptor
12/18/2008US20080312237 Amide derivatives as ion-channel ligands and pharmaceutical compositions and methods of using the same
12/18/2008US20080311113 Method for treating adamts-5-associated disease
12/18/2008CA2691987A1 Antibacterial agents
12/18/2008CA2690913A1 Ire-1alpha inhibitors
12/18/2008CA2690789A1 4-phenylpiperazine derivatives with functionalized linkers as dopamine d3 receptor selective ligands and methods of use
12/18/2008CA2690686A1 Amine compound and pharmaceutical use thereof
12/18/2008CA2690299A1 Piperazine and [1,4] diazepan derivatives as nk antagonists
12/18/2008CA2689561A1 Substituted 2- [2- (phenyl) ethylamino] alkaneamide derivatives and their use as sodium and/or calcium channel modulators
12/18/2008CA2688585A1 Cyclohexyl derivatives
12/17/2008EP2001847A2 Soluble adenylate cyclase inhibitors
12/17/2008EP2001838A2 Selective hydroxamate based mmp inhibitors
12/17/2008EP2001831A2 Compounds which inhibit the glycine transporter and uses thereof
12/17/2008EP1919883B1 N-oxides as prodrugs of piperazine&piperidine derivatives
12/17/2008EP1917254B1 Process of producing amorolfine
12/17/2008EP1423106B1 Arylsulfonyl derivatives with 5-ht 6 receptor affinity
12/17/2008CN101326171A Novel dual peptidase inhibitors as prodrugs for the therapy of inflammatory and other disorders
12/17/2008CN101323590A Novel synthetic method of aripiprazole and intermediate thereof
12/16/2008US7465733 trans-1-{2-[(3,5-dibromobenzyl)oxy]-2,3-dihydro-1H-inden-1-yl}piperazine; serotonin reuptake inhibitor and/or neurokinin NK1 antagonist; antidepressant, anxiolytic agent; cognition activator; psychological disorders; obesity, gastrointestinal disorders
12/11/2008WO2008150486A2 2-acylaminopropoanol-type glucosylceramide synthase inhibitors
12/11/2008WO2008148868A1 Piperidine/piperazine derivatives
12/11/2008WO2008148856A1 N- ( (3, 5-dichlorophenyl) methyl) -2- u-methyl-1-piperazinyl) -2- ( 1-naphtalenyl) ethan amide as ghrelin receptor modulator
12/11/2008WO2008148853A1 N-phenyl hydrazides as modulators of the ghrelin receptor
12/11/2008WO2008148851A1 Piperidine/piperazine derivatives
12/11/2008WO2008148849A2 Piperidine/piperazine derivatives
12/11/2008WO2008024892A3 Cyclic 11-beta hydroxysteroid dehydrogenase type i inhibitors
12/11/2008US20080306273 Process for the Preparation of 1-Aminopiperidine Derivatives
12/11/2008US20080306260 Method for Producing Aryl Amines, Aryl Ethers and Aryl Thioethers
12/11/2008US20080306258 Cyclopropane compounds and pharmaceutical use thereof
12/11/2008US20080306087 1-(10,11-Dihydro-5H-dibenzo[a,d]cyclohepten-5-yl)-4-(2-nitro-phenylmethanesulfonyl)-piperazine; acylation or sulfonamidation of the piperazine ring; psychological disorders, Parkinson's, Alzheimer's, Huntington's Diseases; antidepressants, entiepileptics
12/11/2008US20080306085 Non-imidazole aryloxyalkylamines
12/11/2008US20080306068 Suppression cytokines, tumor necrosis factor
12/11/2008US20080305528 Isolation of nucleic acids
12/11/2008US20080305082 1,4-Bis-N-Oxide-5,8- Dihydroxyanthracenedione Compounds and the Use Thereof
12/11/2008CA2690004A1 Tri-aryl compounds and compositions comprising the same
12/11/2008CA2687918A1 Piperidine/piperazine derivatives
12/11/2008CA2687754A1 Piperidine/piperazine derivatives
12/11/2008CA2687243A1 Piperidine/piperazine derivatives
12/10/2008EP2000462A2 Non-imidazole alkylamines as histamine H3-receptor ligands and their therapeutic applications
12/10/2008EP1999121A1 Novel tetralins as 5-ht6 modulators
12/10/2008EP1999099A1 Process for preparing an amine
12/10/2008EP1999098A2 Compounds that modulate ppar activity, their preparation and use
12/10/2008EP1841752B1 3,4-dihydro-2-naphthamide derivatives and their therapeutic applications
12/10/2008EP1391199B1 Carboxylic acid derivatives and drugs containing the same as the active ingredient
12/10/2008CN101321741A Process for selective synthesis of enantiomers of substituted 1-(2-amino-1-phenyl-ethyl)-cyclohexanols
12/10/2008CN101321730A Cyclopropyl amines as modulators of the histamine H3 receptor
12/10/2008CN101318943A Substituted diethylenediamine compounds, preparation method, uses and medicament composition containing the compounds
12/10/2008CN101318909A Benzoyl fluoride benzene salicylamide compounds, preparation and application thereof
12/10/2008CN100441556C Triphenylalkene derivatives and their use as selective estrogen receptor modulators
12/09/2008US7462746 Amino polyols and amino sugars
12/09/2008US7462718 Process for the production of high-purity rac-1-{4-[2-hydroxy-3-(5-quinolyloxy)propyl]-piperazin-1-yl}-2,2-diphenylethan-1-one fumarate and high-purity rac-1-{4-[2-hydroxy-3-(5-quinolyloxy)propyl]piperazin-1-yl}-2,2-diphenylethan-1-one fumarate
12/09/2008US7462630 Diarylalkene derivatives and novel diarylalkane derivatives
12/09/2008US7462617 Substituted acylpiperazine derivatives
12/09/2008CA2379061C Antibacterial agents
12/09/2008CA2217855C Tetralines
12/05/2008WO2005115146A1 Piperazin derivatives and their use in controlling pests
12/04/2008WO2008148057A2 Cationic lipids compositions and methods for enhancing immune responses to vaccines
12/04/2008US20080300271 Novel compounds and a novel process for their preparation
12/04/2008US20080300258 Anhydrous ciprofloxacin hydrochloride
12/04/2008US20080299639 adduct comprising a molecule binding with a kinase; antiinflammatory agents; modulating activation state of p38 kinase protein; switch control ligands to induce or restrict conformation
12/04/2008DE102008020361A1 Preparing 2,5-dimethylphenylthioacetomorpholide comprises reacting 2,5-dimethylacetophenone with sulfur and morpholine in a liquid reaction system
12/04/2008CA2688346A1 Compositions and methods for enhancing immune responses to vaccines
12/03/2008EP1997823A1 Boronic ester and acid compounds, synthesis and uses
12/03/2008EP1997804A1 Mmp-13-selective inhibitor
12/03/2008EP1997495A1 2-phenoxy- and 2-phenylsulfanyl-benzenesulfonamide derivatives with ccr3 antagonistic activity for the treatment of asthma and other inflammatory or immunological disorders
12/03/2008EP1997489A1 Adamantylglycine derivatives as inhibitors of dipeptidyl peptidase IV for the treatment of diabetes
12/03/2008EP1996550A2 Carboxyamine compounds and their use in the treatment of hdac dependent diseases
12/03/2008EP1996545A1 Soluble epoxide hydrolase inhibitors and methods of using same
12/03/2008EP1353638A4 Novel couplers for use in oxidative hair dyeing
12/03/2008EP1353637A4 Novel couplers for use in oxidative hair dyeing
12/03/2008CN101316811A Puleganic amides as insect repellants
12/03/2008CN100439336C Methods for producing cyclic benzamidine derivatives
12/03/2008CN100439332C Novel thiourea derivatives and the pharmaceutical compositions containing thd same
12/03/2008CN100439329C 5-amidino-2-hydroxybenzenesulfonamide derivatives, pharmaceutical compositions containing the same and intermediates for their preparation
12/02/2008US7459580 Process for trans-4-amino-1-cyclohexanecarboxilic acid derivatives
12/02/2008US7459558 Enzyme inhibitor on NO-synthase enzymes; treating STROKE, NEURODEGENERATIVE DISEASES, preventing ISCHEMIC OR HEMORRAGIC CARDIAC OR CEREBRAL INFARCTIONS; inhibiting lipidic peroxidation
12/02/2008US7459552 Reacting N-[2,4-bis(methylthio)-6-methylpyridin-3-yl]-2-[4-(2-hydroxyethyl)piperazin-1-yl]acetamide with 5-benzyloxy-2-mercaptobenzimidazole in presence of triphenylphosphine and diethyl azodicarboxylate; acyl-coenzyme A cholesterol acyltransferase (ACAT) inhibitor
12/02/2008US7459472 Aryl and heteroaryl compounds, compositions, and methods of use
12/02/2008US7459106 a mixture of chromogens having a two-photon or multi-photon absorptiion, and photoacid generators, that can be patterned by photochemistry
12/02/2008CA2306371C Use of flunarizine for the topical treatment of glaucoma
11/2008
11/27/2008WO2008142461A1 Metabolites of (thio)carbamoyl-cyclohexane derivatives
11/27/2008WO2007136790A3 Intracellular kinase inhibitors
11/27/2008WO2005025498A3 Substituted acetanilides and benzamides for the treatment of asthma and pulmonary inflammation
11/27/2008US20080293940 Amide Derivative and Medicine
11/27/2008US20080293727 Amine hydroxyalkyl sulfonamides as enzyme inhibitors; for example, N-1-(3-((3-acetylamino-4-fluoro-benzenesulfonyl)-benzyl-amino)-(1S,2 syn)-1-benzyl-2-hydroxy-propyl)-2-((quinoline-2-carbonyl)-amino)-succinamide; may be used as anti-viral agents against the HIV-1 and HIV-2 viruses
11/27/2008US20080293722 Ion Channel Modulators
11/27/2008US20080293712 Benzo[C][2,7]Naphtyridine Derivatives, Methods of Making Thereof and Methods of Use Thereof
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