| Patents for C07D 295 - Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms (34,005) |
|---|
| 03/18/2009 | EP2035401A2 Aryl- and heteroaryl-ethyl-acylguanidine derivatives, their preparation and their application in therapeutics |
| 03/18/2009 | EP2035369A1 Therapeutic compounds |
| 03/18/2009 | EP1805129B1 (biphenyl) carboxylic acids and derivatives thereof |
| 03/18/2009 | EP1689380A4 Method for treating adamts-5-associated disease |
| 03/18/2009 | CN101389617A Novel processes for the preparation of piperazinyl and diazapanyl benzamide derivatives |
| 03/18/2009 | CN101389616A Preparation of optically pure beta-amino acids having affinity for the alpha-2-delta protein |
| 03/18/2009 | CN100469764C Vitamin D derivatives |
| 03/17/2009 | US7504537 osteoarthritis or rheumatoid arthritis |
| 03/17/2009 | US7504528 Merocyanine derivatives for cosmetic use |
| 03/17/2009 | US7504520 8-({5-[4-(trifluoromethyl)phenyl]-1,3-oxazol-2-yl}amino)-3,4-dihydronaphthalen-2(1H) one; treating pain, bladder overactivity, and urinary incontinence |
| 03/17/2009 | US7504512 BCL-X1 protein inhibitors; anticarcinogenic agents |
| 03/17/2009 | US7504437 Acetylcholinesterase inhibitor; Alzheimer's diseases, Hubtington disease, antidepressants |
| 03/17/2009 | US7504436 Bioisosteres of actinonin |
| 03/17/2009 | US7504413 N-(4-(imidazo[1,2A]pyridin-YL)phenethyl)benzamide inhibitors of the mitotic kinesin CENP-E for treating certain cellular proliferation diseases |
| 03/17/2009 | US7504400 MTP inhibiting aryl piperydines or piperazines substituted with 5-membered heterocycles |
| 03/17/2009 | US7504399 Piperazine enamines as antiviral agents |
| 03/17/2009 | US7504393 Benzylamine analogues |
| 03/17/2009 | US7504378 Viricides; induction immunology response; compounds according to invention specifically inhibit NS3 protease and do not show significant inhibitory activity against other serine proteases such as human leukocyte elastase, porcine pancreatic elastase, bovine pancreatic chymotrypsin, or cysteine proteases |
| 03/17/2009 | CA2506016C 3-amino-piperidine derivatives and processes for their preparation |
| 03/17/2009 | CA2433684C Novel couplers for use in oxidative hair dyeing |
| 03/17/2009 | CA2412161C Thyroid receptor ligands, pharmaceutical compositions comprising them and their use in the treatment of disorders influenced by thyroid hormones |
| 03/12/2009 | WO2009033069A1 Simple pantoic acid ester neopentyl sulfonyl ester cyclization release prodrugs of acamprosate, compositions thereof, and methods of use |
| 03/12/2009 | WO2009033061A1 Masked carboxylate neopentyl sulfonyl ester cyclization release prodrugs of acamprosate, compositions thereof, and methods of use |
| 03/12/2009 | WO2009031202A1 Cinnamic acid derivatives and use thereof as ultraviolet absorber |
| 03/12/2009 | WO2008139492A3 A process for the preparation of highly pure ranolazine base |
| 03/12/2009 | US20090069432 Compounds, compositions and methods for the treatment of amyloid diseases and synucleinopathies such as alzheimer's disease, type 2 diabetes, and parkinson's disease |
| 03/12/2009 | US20090069344 Modulators of hcv replication |
| 03/12/2009 | US20090069310 Anti-inflammatory medicaments |
| 03/12/2009 | US20090069282 Alkyne compounds with mch antagonistic activity and medicaments comprising these compounds |
| 03/11/2009 | EP2033950A1 Substituted tetracycline compounds |
| 03/11/2009 | EP2033688A2 Oxalic acid derivatives and their use as physiological cooling agents |
| 03/11/2009 | EP2032535A1 Spirocyclic nitriles as protease inhibitors |
| 03/11/2009 | EP1940782B1 N-phenyl phenylacetamide non-nucleoside reverse transcriptase inhibitors |
| 03/11/2009 | EP1485364B1 Aminocarbonyl-derivatives as novel inhibitors of histone deacetylase |
| 03/11/2009 | EP1485096B1 Methods for preventing or treating cardiac arrhythmia |
| 03/11/2009 | EP0976722B1 Benzamidine derivatives |
| 03/11/2009 | CN101381349A Dipfluzine addition salt and preparation method |
| 03/11/2009 | CN100467464C Long-chain aromatic piperazine modified duloxetine-like compound, and its preparation and use |
| 03/11/2009 | CN100467458C Indanyl-piperazine derivatives, process for their preparation and pharmaceutical compositions containing them |
| 03/11/2009 | CN100467449C Cyclic aminophenyl sulfamate derivative |
| 03/11/2009 | CN100467440C Quaternary bis-ammonium salt precursors and their uses as prodrugs having an antiparasitic activity |
| 03/10/2009 | US7501538 Erythropoietin receptor activators; inducing red blood cell production and maturation |
| 03/10/2009 | US7501519 reacting grignard reagents with chemical intermediate exo-1-(bi-cyclo[2.2.1]hept-5-en-2-yl)-3-piperidino-1-propanone, formed by conversion of exo-1-(bicyclo[2.2.1]hept-5-en-2-yl)-ethanone into an exo silyl enol ether, then reacting with N-methylenepiperidinium chloride |
| 03/10/2009 | US7501441 for treating uterine fibroid disease; [2-(4-hydroxyphenyl)-6-hydroxynaphthalen-1-yl][4-(2-(1-piperidinyl)ethoxy)phenyl]methane; therapy for post manupausal women |
| 03/10/2009 | US7501419 4-Squarylpiperazine derivatives as antiviral agents |
| 03/10/2009 | US7501417 Aminocarbonyl-derivatives as novel inhibitors of histone deacetylase |
| 03/10/2009 | US7501414 Substituted morpholine and thiomorpholine derivatives |
| 03/10/2009 | US7501408 2-(R)-Cyclohexylmethyl-N-[1-(S)-methyl-2-(4-trifluoromethoxy-phenylamino)-ethyl]-4-oxo-4-thiomorpholin-4-yl-butyramide; selective in presence of at least one other cathepsin isozyme; antiinflammatory agent: arthritis, atherosclerosis |
| 03/10/2009 | CA2394602C New modulators of dopamine neurotransmission |
| 03/05/2009 | WO2009028387A1 Therapeutic agent for cancer with resistance to protease inhibitor |
| 03/05/2009 | WO2009027510A1 Aldehydes containing hydroxyl groups |
| 03/05/2009 | WO2009027249A2 Method for producing amines from sugar alcohols |
| 03/05/2009 | WO2009027248A1 Method for producing amines from glycerin |
| 03/05/2009 | WO2008151957A9 Cyclohexyl derivatives |
| 03/05/2009 | WO2008148868A8 Piperidine/piperazine derivatives |
| 03/05/2009 | WO2008148849A8 Piperidine/piperazine derivatives |
| 03/05/2009 | US20090062530 Substituted arylalkanoic acid derivatives and use thereof |
| 03/05/2009 | US20090062340 Novel biaromatic compounds which activate ppary type receptors and cosmetic/pharmaceutical compositions comprised thereof |
| 03/05/2009 | US20090062287 thromboembolic and/or inflammatory disorders; 4-Aminomethyl-cyclohexanecarboxylic acid (1-biphenyl-3-yl-2-phenyl-ethyl)-amide; selective inhibitors of serine protease enzymes of the coagulation cascade and/or contact activation system; improved pharmacological properties, plasma kallikrein activity |
| 03/05/2009 | US20090062284 Thio-Substituted Biarylmethanesulfinyl Derivatives |
| 03/05/2009 | US20090062261 Nitrogen-containing heterocycle derivatives substituted with cyclic group |
| 03/04/2009 | EP2030968A2 Sulfur-containing compound, method of preparation and pharmaceutical uses thereof |
| 03/04/2009 | EP2030965A1 Aldehydes containing hydroxyl groups |
| 03/04/2009 | EP2029539A1 Piperidinyl, indolyl, pirinidyl, morpholinyl and benzimidazolyl urea derivatives as inhibitors of soluble epoxide hydrolase for the treatment of hypertension, inflammations and other diseases |
| 03/04/2009 | EP2029521A1 Process for the preparation of an amine |
| 03/04/2009 | EP1948626B1 Process for the preparation of delmopinol and derivatives thereof |
| 03/04/2009 | EP1678102B1 Method and apparatus for the use of [11c] carbon monixi de in labeling synthesis by photo-initiated carbonylation |
| 03/04/2009 | EP1485370B1 Amino-derivatives as novel inhibitors of histone deacetylase |
| 03/04/2009 | EP1380306B1 Remedies for restless leg syndrome |
| 03/04/2009 | CN101379030A Sulfonamide derivatives to treat infection with hepatitis c virus |
| 03/04/2009 | CN101379027A Mutilin derivatives and their use as pharmaceutical |
| 03/04/2009 | CN101376648A Cinepazide maleate crystal form and preparation thereof |
| 03/04/2009 | CN101376637A High cubane diamide compound and use thereof |
| 03/03/2009 | US7498436 Substituted hydroxyethylamines |
| 03/03/2009 | US7498433 Process and intermediates for the preparation of olanzapine |
| 03/03/2009 | US7498421 Antibody specific for 4-methyl-3-vinylmaleimide derivatives; photolabile degradation product of bilirubin or biliverdin; antiinflammatory agents, infections,systemic inflammatory response syndrome |
| 03/03/2009 | US7498358 Human ADAM-10 inhibitors |
| 02/26/2009 | WO2009025914A2 Radiolabelled fluorobenzamide analogues, their synthesis and use in diagnostic imaging |
| 02/26/2009 | WO2009024550A1 N-benzyl, n' -arylcarbonylpiperazine derivatives as lxr modulators |
| 02/26/2009 | US20090054630 Compositions and methods for detecting and treating diseases and conditions related to chemokine receptors |
| 02/26/2009 | US20090054454 Benzofuranyl- and benzothienyl- piperazinyl quinolines and methods of their use |
| 02/26/2009 | US20090054448 Amino Acid Derivatives as Histone Deacetylase (HDAC) Inhibitors |
| 02/26/2009 | US20090054420 Bicyclic-substituted amines as histamine-3 receptor ligands |
| 02/26/2009 | DE102007039559A1 Piperazinpolyphosphat, Verfahren zu seiner Herstellung und seine Verwendung Piperazine, process for its preparation and its use |
| 02/26/2009 | CA2697256A1 Cyclopropyl amide derivatives |
| 02/26/2009 | CA2694604A1 N-benzyl, n' -arylcarbonylpiperazine derivatives as lxr modulators |
| 02/26/2009 | CA2689141A1 Radiolabelled fluorobenzamide analogues, their synthesis and use in diagnostic imaging |
| 02/25/2009 | EP2028226A1 Piperazin polyphosphate, method for its manufacture and application |
| 02/25/2009 | EP2027087A2 Intracellular kinase inhibitors |
| 02/25/2009 | CN101374826A Modulators of alpha7 nicotinic acetylcholine receptors and therapeutic uses thereof |
| 02/25/2009 | CN101374825A Cyclohexyl piperazinyl methanone derivatives and their use as histamine h3 receptor modulators |
| 02/25/2009 | CN101374811A Novel dual nk2/nk3-antagonists, pharmaceutical compositions comprising them and processes for their preparations |
| 02/25/2009 | CN101374810A Modulators of alpha7 nicotinic acetylcholine receptors and therapeutic uses thereof |
| 02/25/2009 | CN100463901C Alpha-ketoamide derivative, and production method and use thereof |
| 02/24/2009 | US7495022 α,β-unsaturated hydroxamic acid derivatives and their use as histone deacetylase inhibitors |
| 02/24/2009 | US7495012 Arylsulfonamides and uses related thereto |
| 02/24/2009 | US7494986 central nervous system disorders like Depression, anxiety, cognition enhancer, antiinflammatory agents; 4-((3,5-bis(trifluoromethyl)benzyloxy)methyl)-4-phenylazocane |
| 02/24/2009 | CA2417361C New phenyl- and phenylalkyl-substituted ethanolamines and ethylenediamines |
| 02/19/2009 | WO2009022633A1 Bicyclic acylguanidine derivative |
| 02/19/2009 | WO2009021946A1 Novel compounds |