Patents
Patents for C07D 295 - Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms (34,005)
05/2008
05/20/2008US7374749 Amino substituted hydroxyphenyl benzophenone derivatives
05/20/2008CA2395717C Fused imidazolium derivatives
05/20/2008CA2169695C Substituted benzenesulfonylureas and -thioureas, processes for their preparation, their use for the production of pharmaceutical preparations and medicaments containing them
05/15/2008US20080114169 Intermediates of active esters for peptide synthesis, labeling, analysis; purity
05/15/2008US20080114036 Novel Compounds, Their Preparations And Use
05/15/2008US20080114000 Suppressor of excess accumulation of intracellular sodium ions
05/15/2008US20080113989 For example, N-(1-Carbamoyl-1-oxo-3-phenylpropan-2-yl)-2-(E-2-(4-(1-pyrrolidinylmethyl)phenyl)ethen-1-yl)benzamide; calcium channel blockers; cardiovascular disorders; antiarthritic agents; inhibitors of enzymes, especially cysteine proteases such as calpain and cathepsins
05/15/2008US20080113975 Thiourea compounds
05/15/2008US20080113968 Substituted piperazines and diazepanes
05/15/2008DE19753655B4 α-Aminoacetophenonverbindungen, Massen, die diese Verbindungen enthalten und deren Verwendung als Photostarter α-Aminoacetophenonverbindungen, compositions containing these compounds and their use as photoinitiators
05/15/2008CA2672956A1 Calcium receptor modulating agents
05/14/2008EP1919883A1 N-oxides as prodrugs of piperazine&piperidine derivatives
05/14/2008EP1485365B1 Sulfonyl-derivatives as novel inhibitors of histone deacetylase
05/14/2008CN101180288A Aromatic substituted pentadienoic acid amide for combination with anti-infective drugs
05/14/2008CN101177420A Method for intermittent azeotropic rectifying separating N-ethylpiperazine-ethanolamine
05/14/2008CN101177419A Method for separating N-ethylpiperazine-ethanolamine azeotropic mixture by azeotropic rectifying intermittent operation
05/14/2008CN101177385A Aryl sulfonic acid amides and analogues as well as its purpose in curing neural degeneration disease
05/14/2008CN100387581C Process to produce oxazolidinones
05/13/2008US7371877 Glycerol ester derivative
05/13/2008US7371871 imidazole derivatives; Alzheimer's Disease, Down syndrome and Huntington's Disease; hypotensive agents, sleeping and eating disorders, anxiolytic agents, antidepressants, antiepileptic agents, drug abuse withdrawl
05/13/2008US7371855 Process for the synthesis of 5-(4-fluorophenyl)-1-[2-((2R,4R)-4-hydroxy-6-oxo-tetrahydro-pyran-2-yl)-ethyl]-2-isopropyl-4-phenyl-1H-pyrrole-3-carboxylic acid phenylamide
05/13/2008US7371766 Curcumin analogs with anti-tumor and anti-angiogenic properties
05/13/2008US7371765 Quinoline derivatives having VEGF inhibiting activity
05/13/2008US7371747 Cyanoalkylamino derivatives as protease inhibitors
05/13/2008US7371746 1,2,4-Thiadiazole compounds and pests controlling composition containing the same
05/13/2008CA2327854C Plant growth regulator compositions
05/08/2008WO2008053913A1 Sulfonylurea derivative capable of selectively inhibiting mmp-13
05/08/2008WO2008053023A1 Crosslinker for vulcanization, process for its preparation and rubber products
05/08/2008WO2008052658A1 Novel diphenylazetidinone substituted by piperazine-1-sulfonic acid having improved pharmacological properties
05/08/2008US20080108618 Compounds with activity on muscarinic receptors
05/08/2008US20080108601 anticancer agents; catalytic hydrogenation
05/08/2008US20080108595 Inhibitors of cathepsin s
05/08/2008US20080107599 Radiolabelled benzamide analogues, their synthesis and use in diagnostic imaging
05/08/2008CA2668094A1 Novel diphenylazetidinone substituted by piperazine-1-sulfonic acid and having improved pharmacological properties
05/07/2008EP1918278A1 Sulfonylamino derivatives which inhibit matrix-degrading metalloproteinases
05/07/2008EP1917254A2 Process of producing amorolfine
05/07/2008EP1436272B1 Biphenylcarboxylic amide derivatives as p38 kinase inhibitors
05/07/2008CN101175738A Apoptosis promoters
05/07/2008CN101175720A New haloalkylsulfone substituted compounds useful for treating obesity and diabetes
05/07/2008CN101172949A Catalytic esterification method for sulfonic group functionalization morpholine hyamine ion liquid
05/06/2008US7368605 Variously substituted derivatives of guanidine, and their use as medicines with anti-diabetes and/or anti-obesity activity
05/06/2008US7368479 Alpha-sulfonylamino-acetonitriles
05/06/2008US7368448 2-(arylalkoxy)-1-phenylethylamine derivatives as NK1 antagonist and serotonin reuptake inhibitors
05/06/2008CA2430601C Piperazine derivatives
05/02/2008WO2008051597A1 Process for the preparation of imatinib
05/02/2008WO2008050858A1 Amide compound, salt thereof, and biofilm remover using them
05/02/2008WO2008049806A1 Piperidine or piperazine substituted tetrahydro-naphthalene-1-carboxylic acid mtp inhibiting compounds
05/02/2008WO2008049605A1 Heterocyclyl pyridyl sulfonamide derivatives, their manufacture and use as pharmaceutical agents
05/02/2008CA2666885A1 Heterocyclyl pyridyl sulfonamide derivatives, their manufacture and use as pharmaceutical agents
05/02/2008CA2664141A1 Piperidine or piperazine substituted tetrahydro-naphthalene-1-carboxylic acid mtp inhibiting compounds
05/01/2008US20080103328 Synthetic and semisynthetic acanthoic acid derivatives; antiinflammatory, anticancer and antitumor agents
05/01/2008US20080103140 Cyclohexylamides as Dopamine D3, D2 and 5Ht1a Antagonists
05/01/2008US20080103135 Histamine H3 antagonists; do not contain imidazolyl moiety; such as 1-[4-(4-piperidin-1-ylmethyl-phenyl)-but-3-ynyl]-piperidine
05/01/2008US20080101989 Methods, Compositions and Kits Pertaining to Analyte Determination
04/2008
04/30/2008EP1915356A1 Therapeutic agents
04/30/2008EP1915355A1 Therapeutic agents
04/30/2008EP1915339A1 Beta-secretase inhibitors for use in the treatment of alzheimer's disease
04/30/2008CN101168532A Method for synthesizing N-methylpiperazine substituted anilin
04/29/2008US7365197 Method for the regioselective preparation of substituted benzo[g]quinoline-3-carbonitriles and benzo[g]quinazolines
04/29/2008US7365196 Sulphonamido-substituted bridged bicycloalkyl derivatives
04/29/2008US7365085 2-(3-{3-[[2-chloro-3-(trifluoromethyl)benzyl](2,2-dephenylethyl)amino]propoxy}phenyl)-ethanol; agonists of the nuclear receptors, LXR alpha and LXR beta used to increase ABCA1, ABCG1, and apolipoprotein E expression and inhibiting cholesterol absorption
04/29/2008US7365076 for the prevention and treatment of conditions ameliorated by monoamine reuptake including, inter alia, vasomotor symptoms (VMS), sexual dysfunction, gastrointestinal and genitourinary disorders, chronic fatigue syndrome, fibromylagia syndrome, nervous system disorders
04/29/2008US7365075 11-beta-hydroxysteroid dehydrogenase type 1 inhibitors; potentiation; diabetes and obesity; 2-(4-{4-[1-(6-chloro-pyridin-3-yl)cyclopropylmethyl]-2-(R)-methyl-piperazine-1-sulfonyl}phenyl)-1,1,1-trifluoro-propan-2-ol
04/29/2008US7365070 Such as N-{2-[2-(5-Bromo-2-methoxy-phenyl)-ethyl]-3-fluoro-benzoyl}-N'-butyl-guanidine; involuntary weight loss disorders
04/29/2008US7365068 Hepatitis C virus infections; -(3-cyclopropyl-4-(pentyloxy)phenyl)-3-nicotinoylthiourea;methyl 2-oxo-2-(5-((3-(4-(pentyloxy)-3-(trifluoromethyl)phenyl)thioureido)carbonyl)pyridin-2-ylamino)acetate
04/29/2008CA2343204C Arylsulfonanilide ureas
04/29/2008CA2259203C Method for the synthesis of amines and amino acids with organoboron derivatives
04/29/2008CA2254833C Pharmaceutical for treatment of neurological and neuropsychiatric disorders
04/24/2008WO2007100506A3 Mass tags for quantitative analyses
04/24/2008US20080096936 Sulfur substituted sulfonylaminocarboxylic acid N-arylamides, their preparation, their use and pharmaceutical preparations comprising them
04/24/2008US20080096903 inhibitors of disease-related target, Heat Shock Protein 90 (HSP90); antiproliferative; 2-chloro-5'-sulfamoyladenosine analogs; derivatives of adenine and other purines; Sulfamic Acid 2-[6-amino-2-fluoro-8-(6-iodo-benzo[1,3]dioxol-5-ylmethyl)-purin-9-yl]-ethyl ester
04/24/2008US20080096889 Histone Deacetylases Inhibitors
04/24/2008US20080096876 Histamine receptor antagonists; 4-[3-(4-Piperidin-1-yl-but-1-ynyl)-benzyl]-thiomorpholine; antiallergens, antihistamines, antiepileptic agents; asthma, alzheimer's disease, narcolepsy, motion sickness, attention deficit disorder, schizophrenia
04/24/2008US20080096875 Hepatitis C virus infection; thiourea-substituted dibenzofuran, fluorene, or carbazole compounds
04/24/2008US20080096873 New compounds
04/24/2008US20080096869 Adamantyl acetamides as 11-beta hydroxysteroid dehydrogenase inhibitors
04/23/2008EP1912962A2 Crystalline non-solvated methanesulfonic acid salt of 1-(4-(2-piperidinylethoxy)phenoxy)-2-(3-hydroxyphenyl)-6-hydroxynaphthalene
04/23/2008EP1912961A2 Process of producing bepromoline
04/23/2008EP1912679A2 Amine-containing lipids and uses thereof
04/23/2008EP1303483B1 Novel thiourea derivatives and the pharmaceutical compositions containing the same
04/23/2008EP1007033B1 Lymphocyte function antigen-1 antagonists
04/23/2008CN100383116C Methoximinophenylacetic acid amides
04/22/2008US7361771 Process for the synthesis of 5-(4-fluorophenyl)-1-[2-((2R,4R)-4-hydroxy-6-oxo-tetrahydro-pyran-2-yl)-ethyl]-2-isopropyl-4-phenyl-1H-pyrrole-3-carboxylic acid phenylamide
04/22/2008US7361685 Compounds for use in the treatment of skin conditions
04/22/2008US7361662 Pyridopyrimidinone compounds, method for production thereof and medicaments comprising the same
04/22/2008US7361655 Pharmaceutically effective compounds
04/22/2008CA2388759C Substituted piperazine derivatives, the preparation thereof and their use as medicaments
04/22/2008CA2180816C 6-dimethylaminomethyl-1-phenyl-cyclohexane compounds as pharmaceutical active ingredients
04/17/2008WO2008045671A1 Matrix metalloprotease inhibitors
04/17/2008WO2008044033A1 Amide derivatives
04/17/2008WO2008043183A1 Cyclopropyl-piperazine compounds as calcium channel blockers
04/17/2008WO2007143745A3 Substituted phenyl acetic acids as dp-2 antagonists
04/17/2008US20080090839 Phenoxymethylalkyne inhibitors of lta4h for treating inflammation
04/17/2008US20080090822 Piperazine Derivatives As Glyt 1 Inhibitors
04/17/2008US20080090782 Inhibit DNA-dependent protein kinase; reduced side effects caused by radiation and chemotherapy drugs
04/17/2008US20080090779 2-Benzyloxy-5-(2-bromoacetyl)-N-[3,5-bis(trifluoromethyl)phenyl-benzamide; diseases caused by production of immunoglobulin E: inflammatory cytokine, histamine, leukotriene and degranulation from activated mast cell; pollinosis, bronchial asthma, atopic dermatitis, urticaria; endometriosis, hysteromyoma
04/17/2008CA2666275A1 Cyclopropyl-piperazine compounds as calcium channel blockers
04/16/2008EP1911762A1 Amino alcohols and their use as renin inhibitors
04/16/2008EP1911740A1 Potassium channel modulators
04/16/2008EP1911350A1 Amidine compound and herbicide
1 ... 64 65 66 67 68 69 70 71 72 73 74 75 76 77 78 79 80 81 82 83 84 ... 341