Patents
Patents for C07D 295 - Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms (34,005)
12/2011
12/21/2011EP2396300A1 New substituted tetrahydronapthalenes, method for the production thereof, and use thereof as drugs
12/21/2011EP2396295A1 Phenoxy acetic acid derivatives
12/21/2011EP2155736B1 Novel carbamoyloxy arylalkanoyl arylpiperazine compound, pharmaceutical compositions comprising the compound and method for treating pain, anxiety and depression by administering the compound
12/21/2011CN102285962A Phenoxy alkyl piperazine compounds, preparation method thereof and medicinal use thereof
12/21/2011CN101544629B 一种分离罗替戈汀、苯海索对映异构体的方法 An rotigotine, trihexyphenidyl enantiomer separation method
12/20/2011US8080656 Process for the preparation of aprepitant
12/20/2011US8080541 Carbocyclic GlyT-1 receptor antagonists
12/20/2011CA2492924C Novel piperazinone derivates for the treatment of 5-ht2a receptor-related disorders
12/20/2011CA2326777C Aminocyclohexyl ether compounds and uses thereof
12/15/2011WO2011154580A1 Novel cxcr4 inhibitors as anti-hiv agents
12/15/2011US20110306614 N-Hydroxylsulfonamide Derivatives as New Physiologically Useful Nitroxyl Donors
12/15/2011US20110306560 Boronic ester and acid compounds, synthesis and uses
12/15/2011US20110306133 Culture medium and method for inducing differentiation into adipocytes
12/14/2011EP2393794A1 Design, synthesis and evaluation of procaspase activating compounds as personalized anti-cancer drugs
12/14/2011EP2393776A1 Novel trifluoromethylsulfonamide gamma secretase inhibitor
12/14/2011EP1828160B1 Sulfonyl amino cyclic derivatives and use thereof as mmp inhibitors
12/14/2011CN102282129A 用于治疗癌症和免疫和自身免疫疾病的细胞程序死亡诱导药剂 Procedures for the treatment of cancer and cellular immune and autoimmune diseases inducing agent
12/14/2011CN102282128A 用于治疗癌症和免疫和自身免疫疾病的细胞程序死亡诱导药剂 Procedures for the treatment of cancer and cellular immune and autoimmune diseases inducing agent
12/14/2011CN102276557A 吡咯烷5-取代戊二烯酰胺类化合物的制备方法 The method for preparing 5-substituted pyrrolidine pentadienamide Compounds
12/14/2011CN102276556A 4-苄基哌连嗪乙亚胺酰(亚胺甲基苯)肼类化合物的制备方法 Preparation 4- benzylpiperazine even piperazine acetic acid imine (imine methylbenzene) hydrazines
12/14/2011CN102274736A Application of aluminum chloride in catalyzing amine and carbodiimide addition reaction
12/13/2011US8076342 Malonate salt of 4-((1R,3S)-6-chloro-3-phenylindan-1-yl)-1,2,2-trimethylpiperazine and uses of same
12/13/2011US8076326 N-phenyl- (piperazinyl or homopiperazinyl)-benzenesulfonamide or benzenesulfonyl-phenl-(piperazine or homopiperazine) compounds suitable for treating disorders that respond to modulation of the serotonin 5-HT6 receptor
12/13/2011CA2494628C Acylated arylcycloalkylamines and their use as pharmaceuticals
12/08/2011WO2011152658A2 Pharmaceutical composition comprising piperazine dithioctate and glimepiride
12/08/2011US20110301350 Process for preparing cycloalkyl-substituted piperazine compounds
12/08/2011US20110301200 Thyroid receptor ligands
12/08/2011US20110300567 Method for determining redox activity and screening compounds based on redox activity
12/08/2011US20110300218 Novel solid state forms of ranolazine salts
12/08/2011US20110300044 Corrosion inhibitors
12/08/2011CA2801074A1 Glycine transporter-1 inhibitors, methods of making them, and uses thereof
12/08/2011CA2800668A1 New forms of rifaximin and uses thereof
12/07/2011EP2391601A1 Sulfamoyl- phenyl-ureido benzamidine-derivatives as antimalarial agents
12/07/2011CN102271678A 2-酰胺基丙醇型葡糖神经酰胺合成酶抑制剂 2-acylaminopropanol type glucosyl ceramide synthase inhibitors
12/07/2011CN102267959A 一种瑞格列奈晶体、其制备方法及含有该晶体的固体口服制剂 One kind of repaglinide crystal, its preparation method and containing a solid oral formulations of the crystal
12/07/2011CN102267958A 芳族化合物的单硝化 Mononitration of aromatic compounds
12/07/2011CN102267924A 抗菌剂 Antibacterial agents
12/07/2011CN101787002B 1-芥子酰基-4-苄基哌嗪衍生物及其制备方法及抗自由基或抗炎活性应用 1- mustard-4-benzyl-piperazine derivatives and preparation method and application of anti-radical or anti-inflammatory activity
12/07/2011CN101747293B 萘哌地尔的制备方法 Naftopidil preparation
12/06/2011US8071787 Pyrrolidine compounds
12/06/2011US8071650 Vanilloid receptor modulators; analgesic, antiinflammatory and antiulcer effects; such as 1-(1H-indol-5-ylmethyl)-3-phenethylthiourea
12/06/2011US8071615 Carbonylamino-derivatives as novel inhibitors of histone deacetylase
12/06/2011US8071604 Thio-substituted arylmethanesulfinyl derivatives
12/06/2011US8071603 Heterocyclic derivatives and their use as stearoyl-CoA desaturase inhibitors
12/01/2011WO2011150347A2 Non-peptide bdnf neurotrophin mimetics
12/01/2011US20110294882 Novel derivatives of 3,3-diphenylpropylamines
12/01/2011US20110294822 Substituted Phenylpiperazinyl Aralkylalcohol Derivatives, Pharmaceutical Compositions Containing Such Derivatives and Uses Thereof
12/01/2011US20110294814 Compounds for treating proliferative disorders
12/01/2011US20110294793 Hydroxyphenyl sulfonamides as antiapoptotic bcl inhibitors
12/01/2011US20110294787 Substituted thiomorpholine derivatives
12/01/2011US20110294775 Novel compounds
12/01/2011US20110293703 Aminoalcohol lipidoids and uses thereof
11/2011
11/30/2011EP2389371A2 Bumetanide, furosemide, piretanide, azosemide, and torsemide analogs, compositions and methods of use
11/30/2011EP2389350A1 Methods for making valerenic acid derivatives and their use
11/30/2011EP2217583B1 Benzenesulfonanilide compounds suitable for treating disorders that respond to modulation of the serotonin 5-ht6 receptor
11/30/2011EP1633735B1 Derivatives of piperidinyl- and piperazinyl-alkyl carbamates, preparation methods thereof and application of same in therapeutics
11/30/2011CN102264710A 半胱氨酸蛋白酶抑制剂 Cystatin
11/30/2011CN102264693A 用作线粒体通透性转变抑制剂的丙烯酰胺衍生物 Is used as an inhibitor of mitochondrial permeability transition acrylamide derivative
11/30/2011CN102264692A 羰基化相应的叔胺来制备仲酰胺的方法 Carbonylation of the corresponding tertiary amine to prepare secondary amides
11/30/2011CN102260283A 杂环取代双齿胺基配体铝络合物及其制备方法和应用 Substituted heterocyclic amine bidentate ligand complexes of aluminum and its preparation method and application
11/30/2011CN102260225A 用于抑制肿瘤转移和肿瘤血管生长的苯基哌嗪类衍生物 For the inhibition of tumor metastasis and phenyl piperazine derivatives of tumor angiogenesis
11/30/2011CN102260188A 有机化合物 Organic compounds
11/30/2011CN102260187A 取代的氨甲酰基环己甲酸类化合物及其制法和用途 Carbamoyl substituted cyclohexyl carboxylic acid-based compound preparation and use
11/30/2011CN101768139B 哌嗪类衍生物及制备方法和用途 Piperazine derivatives and the preparation and use
11/29/2011US8067601 1-[2-(4-benzyl-4-hydroxy-piperidin-1 -yl )-ethyl]-3-(2-methyl-quinolin- 4-yl)- urea as crystalline sulfate salt
11/29/2011US8067412 analogs of natural products radicicol and pochonins; (oxirane or cyclopropan) 2-benzoxacyclo(di)tetradecin derivatives; inhibition of kinase phosphorylation activity and heat shock proteins; anticarcinogenic, antiinflammatory agent; neurodegenerative diseases; antiallergen
11/29/2011CA2650248C Compounds and compositions as hedgehog pathway modulators
11/29/2011CA2453843C Substituted 4-aminocyclohexanol derivatives
11/24/2011US20110288104 Beta-3 receptor ligands and their use in therapy
11/24/2011US20110288101 Surgical compositions containing sigma-receptor agonists
11/24/2011US20110288094 1-aryl-1-hydroxy-2,3-diamino-propyl amines, 1-heteroaryl-1-hydroxy-2,3-diamino-propyl amines and related compounds having analgesic and/or immuno stimulant activity
11/24/2011US20110288068 Aza spiro alkane derivatives as inhibitors of metalloproteases
11/24/2011US20110288067 Pyrrolopyrazine Kinase Inhibitors
11/24/2011US20110288066 Phenoxy acetic acid derivatives
11/24/2011US20110288057 Salicylic acid derivatives being farnesyl pyrophosphate synthase activity inhibitors
11/23/2011EP2388258A1 Novel vanilloid receptor ligands and their use for producing medicaments
11/23/2011EP2388006A1 Urea derivatives as IL-8 receptor antagonists
11/23/2011EP2388003A2 Colchicine derivatives
11/23/2011EP2387560A2 Apoptosis-inducing agents for the treatment of cancer and immune and autoimmune diseases
11/23/2011EP2387559A1 Apoptosis-inducing agents for the treatment of cancer and immune and autoimmune diseases
11/23/2011EP1988902B1 Piperazine derivatives
11/23/2011CN1968921B Glucagon receptor antagonists, preparation and therapeutic uses
11/23/2011CN1907954B Water-soluble derivative of anesthetic 2,6-diisopropyl phenol and preparation method thereof
11/23/2011CN1535260B Perfluoroalkyl-substituted amines, acids, amino acids and thioether acids
11/23/2011CN102256955A Process for the preparation of piperazine derivatives
11/23/2011CN102256954A Process for the preparation of piperazine compounds and hydrochloride salts thereof
11/23/2011CN102256953A Piperazine salt and a process for the preparation thereof
11/23/2011CN102256929A Polymerizable photoinitiators and radiation curable compositions
11/23/2011CN102250045A Mycobacterium tuberculosis resisting compounds, and applications thereof
11/23/2011CN102250044A Piperazino photoinitiation sensitiser
11/23/2011CN102250043A Preparation method of N-(4-(2-ethylhexyloxy) phenyl)-1, 1-dioxothiomorpholino
11/23/2011CN102250042A Selective estrogen receptor modulators for the treatment of vasomotor symptoms
11/23/2011CN102250041A Pyrrolidine ionic compounds containing phenoxy substituents, and preparation method thereof
11/23/2011CN102250040A Method for preparing N-(3'-aryl allyl)pyrrole derivatives
11/23/2011CN102250039A Ionic liquid of N-methyl piperazine salt and preparation method thereof
11/23/2011CN101613246B Preparation method of N-substituted ethylene diamine derivative
11/22/2011US8063215 Cyclopropyl amide derivatives
11/22/2011US8063067 Hexenoic acid derivatives, processes for the preparation thereof, pharmaceutical compositions comprising them, and therapeutic applications thereof
11/22/2011US8063046 Benzamide derivative
11/22/2011CA2664720C Vitamin d derivatives
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