Patents for C07D 295 - Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms (34,005) |
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04/18/2012 | EP2440519A1 Alkanoylamino benzamide aniline hdac inihibitor compounds |
04/18/2012 | EP2225030B1 Method for producing an amine |
04/18/2012 | EP1409467B1 A n-acylsphingosine glucosyltransferase inhibitor |
04/18/2012 | CN102417489A 一种盐酸司他斯汀晶型f及其制备方法 One kind hydrochloride polymorph f setastine its preparation method |
04/17/2012 | US8158820 Compounds |
04/17/2012 | CA2569840C New disubstituted phenylpiperidines/piperazines as modulators of dopamine neurotransmission |
04/17/2012 | CA2427844C Naphthalene derivatives |
04/17/2012 | CA2371625C Polyamines and their use in therapy |
04/12/2012 | WO2012047907A1 Synthesis of c5-substituted tetracyclines, uses thereof, and intermediates thereto |
04/12/2012 | WO2012046771A1 Cycloalkane compound |
04/12/2012 | US20120088779 Heterocyclic sulfonamides |
04/12/2012 | US20120088769 Salts of arylsulfonamide ccr3 antagonists |
04/12/2012 | US20120088754 Sulfonyl-derivatives as novel inhibitors of histone deacetylase |
04/12/2012 | US20120088746 Amide derivatives as ion-channel ligands and pharmaceutical compositions and methods of using the same |
04/12/2012 | US20120088737 Novel acyl guanidine derivatives |
04/11/2012 | EP2439202A1 Inhibitor compounds of 11-beta-hydroxysteroid dehydrogenase type 1 |
04/11/2012 | EP2439201A1 Compounds with combined SERT, 5-HT3 and 5-HT1A activity |
04/11/2012 | EP2131845B1 5-(2,4-dihydroxy-5-isopropyl-phenyl)-4-(4-morpholin-4-ylmethyl-phenyl)-isoxazole-3-carboxylic acid ethylamide mesylate, hydrates and polymorphs thereof, and formulations comprising these forms |
04/11/2012 | EP1569893B1 Amino substituted hydroxyphenyl benzophenone derivatives |
04/11/2012 | EP1326840B1 Substituted heterocyclic compounds for treating multidrug resistance |
04/11/2012 | EP1261590B1 Piperidine- and piperazine substituted n-hydroxyformamides as inhibitors of metalloproteinases |
04/11/2012 | CN102414186A Abt-263的盐和其固体形式 Abt-263 salt and its solid form |
04/11/2012 | CN102408395A Novel piperazine and homopiperazine derivative and preparation method and use thereof |
04/11/2012 | CN102408286A 一种n,n-二取代磺酰胺类化合物的制备方法 One kind of n, n- disubstituted sulfonamide compounds prepared |
04/10/2012 | US8153843 Antibacterial agents |
04/10/2012 | US8153655 Compositions useful as inhibitors of voltage-gated sodium channels |
04/10/2012 | US8153637 Phenyl-alkyl piperazines having TNF-modulating activity, preparation method, and therapeutic use thereof |
04/10/2012 | US8153623 Compounds |
04/10/2012 | CA2687078C Novel solvate and crystalline forms of carbamoyl-cyclohexane derivatives |
04/10/2012 | CA2526540C Cyclicamino-phenyl sulfamate derivatives |
04/10/2012 | CA2486308C Hepatitis c virus inhibitors |
04/10/2012 | CA2414960C Epoxycarboxamide compound, azide compound, and amino alcohol compound, and process for preparing .alpha.keto amide compound using them |
04/05/2012 | WO2012043445A1 Cyclohexane derivative compound |
04/05/2012 | CA2812898A1 Cyclohexane derivative compound |
04/04/2012 | EP1960343B1 Indene derivatives, their preparation and use as medicaments |
04/04/2012 | EP1658277B1 Succinate and malonate salt of trans-4-(ir,3s)-6-chloro-3-phenylindan-1-yl)-1,2,2-trimethylpiperazine and the use as a medicament |
04/03/2012 | US8148422 Sulfonamides as TRPM8 modulators |
04/03/2012 | US8148414 Prodrugs of methyl hydrogen fumarate, pharmaceutical compositions thereof, and methods of use |
04/03/2012 | CA2505427C Bicyclic-substituted amines as histamine-3 receptor ligands |
03/29/2012 | WO2012038081A1 Substituted benzamide compounds |
03/29/2012 | US20120077977 Process for preparing (meth)acrylic esters of n,n-substituted amino alcohols |
03/29/2012 | US20120077677 Use of 4-phenylbutyric acid and/or salts thereof for enhancing stress tolerance in plants |
03/29/2012 | CA2811796A1 Substituted benzamide compounds |
03/28/2012 | EP2432769A1 N-PHENYL-(PIPERAZINYL OR HOMOPIPERAZINYL)-BENZENESULFONAMIDE OR BENZENESULFONYL-PHENYL-(PIPERAZINE OR HOMOPIPERAZINE) COMPOUNDS SUITABLE FOR TREATING DISORDERS THAT RESPOND TO MODULATION OF THE SEROTONIN 5-HT6 RECEPTOR& xA; |
03/28/2012 | EP1308438B9 3-substituted urea derivatives and medicinal use thereof |
03/28/2012 | CN102391209A Mesylate cinepazide crystal form II and preparation method thereof |
03/28/2012 | CN102389409A TRP-P8 active compounds and therapeutic treatment methods |
03/28/2012 | CN101928264B Apoptosis promoters |
03/28/2012 | CN101759665B Substituent phenylpiperazine aryl alkanol derivant and application thereof in preparing analgesics |
03/28/2012 | CN101084178B (benzyloxy-biphenyl) acetic acids and derivatives thereof |
03/28/2012 | CA2715907A1 Group 5 metal complexes useful for amine functionalization and synthetic process for manufacture thereof |
03/27/2012 | US8143463 Process for the preparation of delmopinol and derivatives thereof |
03/27/2012 | US8143201 Morpholine derivatives as ashless TBN sources and lubricating oil compositions containing same |
03/27/2012 | CA2676456C Tosylate salt of a therapeutic compound and pharmaceutical compositions thereof |
03/27/2012 | CA2552304C Labeling reagents, labeled analytes, including mixtures thereof, and fragment ions derived therefrom and methods for the analysis thereof |
03/22/2012 | US20120071651 Processes for Preparing 1,2-Substituted Cyclopropyl Derivatives |
03/22/2012 | US20120071461 Substituted Benzamide Compounds |
03/22/2012 | US20120071457 Metallo-beta-lactamase inhibitors |
03/22/2012 | US20120071429 Novel antibacterial agents |
03/21/2012 | EP2430008A2 Stable forms of n-(2,6-dimethyl-4-morpholin-4-yl-phenyl)-3,3-dimethyl-butyramide |
03/21/2012 | EP1954678B1 Novel nk1 and nk2 antagonists |
03/21/2012 | EP1928818B1 Pesticide benzyloxy- and phenetyl-substituted phenyl-amidine derivatives |
03/21/2012 | EP1926706B1 Pesticide bi-phenyl-amidine derivatives |
03/21/2012 | EP1233961B9 Method for producing 5-(1-piperazinyl)-benzofuran-2-carboxamide by transition metal-catalyzed amination |
03/21/2012 | CN1984895B Synthesis and uses of synephrine derivatives |
03/21/2012 | CN101591310B Method for preparing cinepazide maleate |
03/21/2012 | CN101538253B Method for preparing repaglinide intermediate |
03/21/2012 | CN101466694B Aryl- and heteroaryl-ethyl-acylguanidine derivatives, their preparation and their application in therapeutics |
03/21/2012 | CN101302205B Preparation of piperazine acidamide compound |
03/21/2012 | CN101298427B Diaryl urea compound and use thereof |
03/21/2012 | CN101007803B Piperazinyl-, piperidinyl- and morpholinyl-derivatives as novel inhibitors of histone deacetylase |
03/20/2012 | US8138353 Synthesis of UDP-glucose: N-acylsphingosine glucosyltransferase inhibitors |
03/20/2012 | CA2504410C Bifunctional phenyliso(thio)cyanates; method and intermediate products for the production thereof |
03/15/2012 | US20120065404 Process for Preparing Ethyl (s)-2-Ethoxy-4-[N-[1-(2-Piperidinophenyl)-3-Methyl-1-Butyl]Aminocarbonyl Methyl]Benzoate and Use Thereof for the Preparation of Repaglinide |
03/15/2012 | US20120065398 Method for producing 3-amidinophenylalanine derivatives |
03/15/2012 | US20120065358 Biodegradable poly(beta-amino esters) and uses thereof |
03/15/2012 | US20120065206 Compounds for treating proliferative disorders |
03/15/2012 | US20120065114 Amine reaction compounds comprising one or more active ingredient |
03/14/2012 | EP2427444A1 Inhibitors of the renal outer medullary potassium channel |
03/14/2012 | EP2427425A2 Tetracycline compounds |
03/14/2012 | EP1948627B1 Novel dual peptidase inhibitors as prodrugs for the therapy of inflammatory and other disorders |
03/14/2012 | CN101712658B 1-butyl-2-hydroxy aralkyl piperazine derivative and application as antidepressant |
03/13/2012 | USRE43244 Phenylethylamines and condensed rings variants as prodrugs of catecholamines, and their use |
03/13/2012 | US8134005 Preparation and use of magnesium amides |
03/13/2012 | US8133905 Biphenyl compounds useful as muscarinic receptor antagonists |
03/08/2012 | WO2012029942A1 Cyclic amide derivative |
03/08/2012 | WO2012028629A1 2 - (benzyloxy) benzamides as lrrk2 kinase inhibitors |
03/08/2012 | US20120059007 Pharmacologically-active vanilloid carbamates |
03/08/2012 | US20120058945 Neuroprotective iron chelators and pharmaceutical compositions comprising them |
03/08/2012 | CA2809112A1 Cyclic amide derivative |
03/07/2012 | EP2426154A1 Photosensitive composition, pattern forming method using the photosensitive composition and compound for use in the photosensitive composition |
03/07/2012 | EP2425840A1 Triazine derivatives and their therapeutical applications |
03/07/2012 | EP2424849A1 Salt of abt-263 and solid-state forms thereof |
03/07/2012 | EP2424844A1 Benzenesulfonanilide compounds suitable for treating disorders that respond to modulation of the serotonin 5-ht6 receptor |
03/07/2012 | EP2424840A1 Cxcr3 receptor antagonists |
03/07/2012 | CN102367241A Preparation method of ranolazine |
03/07/2012 | CN102367216A Preparation method of diselenoaminoformate derivatives |
03/07/2012 | CN101774983B Manufacture method of cinepazide maleate compound |
03/07/2012 | CN101698649B Short-acting hypnotizing and calming compound used for anesthetization |
03/06/2012 | US8129407 Hemiasterlin derivatives and uses thereof in the treatment of cancer |