Patents
Patents for C07D 295 - Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms (34,005)
04/1994
04/05/1994US5300501 Metalloproteinase inhibitors
04/05/1994US5300282 Agents for potentiating the effects of antitumor agents and combating multiple drug resistance
04/05/1994CA1328266C Process for the synthesis of a n,n-dialkyl-hydroxylamine
04/05/1994CA1328264C Spiro-substituted glutaramide diuretic agents
04/05/1994CA1328259C2 Alkylenediamine derivatives
03/1994
03/31/1994WO1994006784A1 1,2-disubstituted ethyl amides as inhibitors of acat
03/31/1994WO1994006768A1 Cyclic benzylamino, benzylamido and benzylimido derivatives as antipsychotic agents
03/31/1994WO1994006764A1 Preparation of beta-methyl carbapenem intermediates
03/31/1994WO1994006756A1 N-(acylaminomethyl)glutaryl amino acids and their use as dual inhibitors of neutral endopeptidase and angiotensin converting enzyme
03/31/1994WO1994006755A1 Alcohol derivative having renin-inhibiting activity and use thereof
03/31/1994DE4232505A1 Verfahren zur Reduktion von Carbonsäuren oder Carbonsäurederivaten sowie neue Verbindungen A process for the reduction of carboxylic acids or carboxylic acid derivatives and to novel compounds
03/31/1994CA2145206A1 1,2-disubstituted ethyl amides as inhibitors of acat
03/30/1994EP0589626A1 Preparation of beta-methyl carbapenem intermediates
03/30/1994EP0589484A1 1,2-Ethanediol derivative and salt thereof, process for producing the same, and cerebral function-improving agent comprising the same
03/30/1994EP0589445A1 Renin Inhibiting N-(2-Amino-2-oxoethyl)Butanediamide Derivatives
03/30/1994EP0589336A1 Benzoylguanidines, process for their preparation and their use as antiarrhythmic agents
03/30/1994EP0589322A1 5-Oxo-dibenzo[a,d]cyclohepta-1,4-dienes and their use as retroviral agents
03/30/1994EP0589039A1 Triphenylethylene derivative and pharmaceutical preparation containing the same
03/30/1994EP0589018A1 Amines as inhibitors of squalene synthase
03/29/1994US5298627 Anticholesterol, hypolipidemic agents, enzyme inhibitors
03/29/1994US5298514 Phenolic thioetheramides
03/29/1994US5298513 Serotonin antagonist
03/29/1994US5298505 Ethynyl alanine amino diol compounds having a piperazinyl-terminated group or a piperazinyl-alkylamino-terminated group for treatment of hypertension
03/29/1994US5298496 Inclusion complexes of 3-morpholino-sydnonimine or its salts or its tautomer isomer, process for the preparation thereof, and pharmaceutical compositions containing the same
03/29/1994CA2105100A1 Preparation of unsaturated amines
03/29/1994CA1328106C Anticholinergic compounds, pharmaceutical compositions and method of treatment
03/29/1994CA1328105C Derivatized alkanolamines as cardiovascular agents
03/26/1994CA2106892A1 5-oxo-dibenzo(a,d)cyclohepta-1,4-dienes
03/23/1994EP0588655A1 Amidinophenol derivatives
03/23/1994CN1084167A New process for the preparation of 3,3-diaryl acrylic acid amides
03/23/1994CN1084162A Octahydronaphthalene oxime derivatives for cholesterol biosynthesis inhibition, their preparation and use
03/22/1994US5296606 O-(3-amino-2-hydroxypropyl)-hydroximic acid halides and process for preparing the same
03/22/1994US5296596 Hexahydroazepine derivatives, a process for their preparation
03/22/1994US5296591 Trifluoromethylketone derivatives, processes for preparation thereof and use thereof
03/22/1994CA1327969C Substituted amine derivatives, their production and use
03/19/1994CA2106248A1 Preparation of beta-methyl carbapenem intermediates
03/17/1994WO1994005648A1 Diaryl piperazinoacetamide compounds as antimuscarinic agents
03/17/1994WO1994005639A1 Sulfonamide inhibitors of hiv-aspartyl protease
03/17/1994WO1994005628A1 Synthesis of 2-substituted quinazoline compounds (such as terazosin) and meobentine and bethanidine and intermediates therefor
03/17/1994WO1994005621A1 Process for the manufacture of cinnamic acid derivatives
03/17/1994CA2143744A1 Diaryl piperazinoacetamide compounds as antimuscarinic agents
03/16/1994EP0587221A1 Tertiary amino alcohol and method of producing the same
03/16/1994EP0587194A1 2-(Heterocycloalkoxy)-1-(subst.-phenyl)-ethanol derivatives as cerebral function improving agents
03/16/1994EP0587193A1 1,2-Ethanediol derivative and salt thereof, process for producing the same, and cerebral function-improving agent comprising the same
03/16/1994EP0586917A1 Substituted phenols, process for their preparation and their use in the treatment of all proliferation associated diseases
03/16/1994EP0445206B1 Hydroxamic acid based collagenase inhibitors
03/16/1994CN1083812A Benzimidazoles, pharmaceutical compositions containing these compounds and processes for preparing them
03/16/1994CN1083805A 7-(substituted)-9-|(substituted glycyl) amido¨-6-demethyl-6-deoxytetracyclines
03/16/1994CN1024004C Fungicides
03/15/1994US5294735 Semicarbazides and the use thereof for stabilizing polyamide fibre materials and the dyeings produced thereon
03/15/1994US5294720 1,4-diamino-2,3-dihydroxybutanes
03/15/1994US5294708 Guanidine derivatives
03/15/1994US5294643 Cinnamamide derivative
03/15/1994US5294624 Antiartheriosclerosis
03/15/1994US5294616 Fibrinogen receptor antagonists
03/15/1994US5294613 Method of treating endotoxic shock in mammals
03/15/1994CA1327795C Antidepressants which are aryloxy inadanamines
03/11/1994CA2105816A1 Substituted phenols, processes for their preparation and their use for the treatment of disorders caused by cell proliferation
03/09/1994EP0585682A2 Process for the preparation of 2,6-dimethylmorpholine from N-(2-hydroxypropyl)-2,6-dimethylmorpholine
03/09/1994EP0585500A1 Diaryl piperazineacetamides as antimuscarinic agents
03/09/1994EP0417210B1 Novel o-(3-amino-2-hydroxypropyl)-hydroximic acid halides and process for preparing the same
03/09/1994CN1083475A Chemical compounds
03/08/1994US5292897 Process for preparing halo acetals from enamines
03/08/1994US5292893 Catalytic asymmetric and non-asymmetric reduction of times and oximes using metal catalysts
03/08/1994US5292761 Piperidine, tetrahydropyridine and pyrrolidine compounds
03/08/1994US5292755 USPA benzolyguanidines
03/08/1994US5292726 N,N-diacylpiperazines
03/08/1994CA1327576C Phenoxyacetic acid amide derivatives and their use in the treatment of obesity and related conditions
03/03/1994WO1994004536A1 Ethynyl alanine amino diol compounds having a piperazinyl-terminated group or a piperazinyl-alkylamino-terminated group for treatment of hypertension
03/03/1994WO1994004523A1 Dioxacycloalkane compound with renin-inhibiting activity
03/03/1994WO1994004518A1 Morpholino/thiomorpholino-terminated alkylamino ethynyl alanine amino diol compounds as renin inhibitors
03/03/1994WO1994004495A1 Piperidinyl-terminated n-(dihydroxy alkyl)-ethynyl-alanine amides for treatment of hypertension
03/03/1994WO1994004492A1 Hydroxyethylamino sulfonamides useful as retroviral protease inhibitors
03/03/1994WO1994004172A1 Peptidyl activated ketone inhibitors containing natural and unnatural peptide sequences
03/03/1994CA2142883A1 Dioxacycloalkane compound having renin-inhibitory activity
03/03/1994CA2142839A1 Peptidyl activated ketone inhibitors containing natural and unnatural peptide sequences
03/03/1994CA2138521A1 Ethynyl alanine amino diol compounds having a piperazinyl-terminated group or a piperazinyl-alkylamino-terminated group for treatment of hypertension
03/03/1994CA2136842A1 Morpholino/thiomorpholino-terminated alkylamino ethynyl alanine amino diol compounds as renin inhibitors
03/02/1994EP0584903A1 Process for preparing aryl piperazinyl-heterocyclic compounds
03/02/1994EP0584191A1 Novel aromatic and polycyclic compounds and their use in human or veterinary medecine and in cosmetics.
03/02/1994CN1083062A 异羟肟酸衍生物 Hydroxamic acid derivatives
03/02/1994CN1083061A Process for preparation aryl piperazinyl-heterocyclic compounds
03/02/1994CN1083055A Pharmaceuticals
03/02/1994CN1083048A Heterocyclic compounds
03/02/1994CN1083047A Novel method of producing 7-(substituted)-9-|(substituted glycyl)-amido¨-6-demethyl-6-deoxytetra-cyclines
03/01/1994US5290951 Intermediates useful in preparing propenone oxime ethers
03/01/1994US5290932 Reaction of heterocyclic secondary amine with ketone
03/01/1994US5290793 Alzheimer's disease; induc nerve growth factor production
02/1994
02/23/1994EP0584046A1 Carbamic acid amide derivatives and their use as pesticides
02/23/1994EP0583605A1 Defined oligomeric liquid crystalline compounds with smectic liquid crystalline phases
02/22/1994US5288928 Asymmetrical hydrogenation
02/22/1994US5288910 In polar liquid medium
02/22/1994US5288757 Aminosulfonyl urea ACAT inhibitors and a method of lowering blood cholesterol levels therewith
02/22/1994CA1327200C Urea derivatives
02/22/1994CA1327197C Microbicidal agrochemical compositions
02/21/1994CA2104317A1 Carbamic acid derivatives
02/17/1994WO1994003436A1 Novel piprazine carboxamides
02/17/1994WO1994003424A1 Compound capable of intracerebral residence and use thereof
02/17/1994CA2141210A1 Novel piperazine carboxamides
02/17/1994CA2120248A1 Compounds which can be retained in brain