Patents
Patents for C07D 295 - Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms (34,005)
02/1995
02/16/1995WO1995004729A1 Amide derivatives as 5ht1d receptor antagonists
02/16/1995WO1995004715A1 Acylphenylglycine derivative and preventive and remedy for diseases caused by increased collagenase activity containing said compound as active ingredient
02/16/1995WO1995004713A1 2-aminoindans as selective dopamine d3 ligands
02/15/1995EP0638553A1 Carboxylic acid amides having a terminal carboxylic acid group as aggregation inhibiting drugs
02/15/1995EP0638548A1 Urea-subsituted benzoylguanidines, process for their preparation, their use as a medicament or diagnostic agent and a medicament containing them
02/15/1995EP0638073A1 1-piperazino-1,2-dihydroindene derivatives
02/15/1995CN1098713A Substituted ortho-ethenylphenylacetic acid derivatives
02/14/1995US5389680 Fluoroalkenyl compounds and their use as pest repellents
02/14/1995US5389645 Analgesics
02/14/1995US5389630 Diamine compound and brain protecting agent containing the same
02/14/1995US5389619 Fungicide, insecticide and miticide; phenylacetic acid derivatives
02/09/1995WO1995004051A1 Piperazine compounds used in therapy
02/09/1995WO1995004050A1 Novel 1,4-di(phenylalkyl)piperazine derivative
02/09/1995WO1995004049A1 PIPERAZINE DERIVATIVES AS α1A-ADRENERGIC RECEPTOR ANTAGONISTS
02/09/1995DE4325855A1 Novel benzoic acid derivatives, processes for their preparation and their use as medicaments
02/09/1995CA2168443A1 Piperazine derivatives as .alpha.1a-adrenergic receptor antagonists
02/09/1995CA2168264A1 Novel 1, 4-(diphenylalkyl)piperazine derivatives
02/08/1995EP0637774A1 1,1-Vinyl substituted nonlinear optical materials
02/08/1995EP0637318A1 Peptide derivatives corresponding to the carboxy terminal sequence of hirudin
02/08/1995EP0637304A1 1-piperazineacetic derivatives as fibrinogen receptor antagonists
02/08/1995EP0637303A1 N-aryloxy(thio)alkyl-azacycloalkanes useful as calcium channel antagonists
02/08/1995EP0637298A1 Substituted cyclohexene-1,2-bicarboxylic acid derivatives and raw materials for producing them
02/08/1995EP0637251A1 Radiopharmaceuticals for imaging the heart
02/08/1995EP0637242A1 Agents for treating substance abuse disorders
02/08/1995CN1098401A Process for preparing N-aliphatic substituted P-phenylenediamines
02/07/1995US5387594 Administering for topical and systemic treatment of
02/07/1995US5387593 Anxiolytic agents
02/06/1995CA2129374A1 Carbonamides, pharmaceutical compositions containing these compounds and processes for their preparation
02/03/1995CA2128991A1 Benzoylacetylene derivatives
02/02/1995WO1995003291A1 Novel substituted 1-propene derivatives, pharmaceutical compositions containing them and process for preparing same
02/02/1995WO1995003267A1 1,2-benzoquinones
02/02/1995CA2167504A1 1,2-benzoquinones
02/01/1995EP0636617A2 Process for the preparation of N-(2-hydromethyl)-piperazin
02/01/1995EP0636125A1 Basic derivatives of glutamic acid and aspartic acid as gastrin or cholecystokinin antagonists
02/01/1995EP0636026A1 Compounds useful for treating inflammatory diseases and inhibiting production of tumor necrosis factor
02/01/1995EP0636025A1 Compounds useful for treating allergic or inflammatory diseases
02/01/1995EP0556308B1 Oxysulfonyl urea acat inhibitors
01/1995
01/31/1995US5386041 Antibiotic
01/31/1995US5385942 Quinone derivatives and pharmacological use
01/31/1995US5385917 Carboxylic acid derivatives
01/31/1995US5385902 Bactericide, fungicide, viricide
01/31/1995US5385898 Hypertensive agents; cardiovascular disorders; renin inhibitors; glaucoma
01/31/1995US5385892 Ethylamino phenyl ethers having antifungal activity
01/26/1995WO1995002587A1 Substituted piperazinylcamphor derivatives as oxytocin antagonists
01/26/1995WO1995002567A1 Catalytic asymmetric reduction of trisubstituted olefins and enamines
01/26/1995CA2166974A1 Substituted amide derivatives of piperizinylcamphor sulfonyl and carbonyl oxytocin antagonists
01/25/1995EP0635485A1 Tetrahydrophthalamide derivative, intermediate for producing the same, production of both, and herbicide containing the same as active ingredient
01/25/1995EP0635018A1 4-(1H-2-METHYLIMIDAZO 4,5-c]PYRIDINYLMETHYL)PHENYLSULPHONAMIDE DERIVATIVES AS ANTAGONISTS OF PAF
01/25/1995EP0635008A1 Piperazides of substituted phenylalanine derivates as thrombin inhibitors
01/25/1995EP0635000A1 Novel phencyclidine derivatives and protein and polypeptide phencyclidine derivative conjugates and labels
01/25/1995EP0634996A1 1,4 naphthoquinone derivtives with anti-protozoal and anti-parasitic activity
01/25/1995EP0634930A1 Compounds useful for treating allergic and inflammatory diseases
01/25/1995CN1097745A 取代的哌嗪 Substituted piperazine
01/25/1995CN1097744A Urea derivative containing heterocyclic ring
01/25/1995CN1097736A Novel antiarrhythmic agents I
01/24/1995US5384320 N-hydroxyurea derivatives which inhibit lipoxygenase
01/24/1995US5384319 Aminoalkylphenyl compounds
01/24/1995US5384108 Complexes of paramagnetic ions with hydrazide derivatives of polyaminocarboxylic acid chelate compounds
01/24/1995CA1334100C Benzocycloheptene compositions, process for their preparation thereof and pharmaceutical compositions holding same
01/24/1995CA1334093C Phosphorous acid salts, compositions holding same and their application as fireproofing agents
01/19/1995DE4323519A1 Process for the preparation of donor-substituted N-formylaminoaromatics and donor-substituted formanilides
01/18/1995EP0634448A1 Vulcanization accelerators
01/18/1995EP0634411A1 Process for the preparation of 8-(4'C4"-(pyrimidin-2'''-yl)-piperazin-1''-yl)-butyl)-8-aza-spiro(4,5)decan-7,9-dione and of its hydrochlorides of high purity
01/18/1995EP0634398A1 4-Phenylpiperidinyl-1/-piperazinyl-1-ethylsubstituted benzofusedheterocycles as antiarrhythmic agents
01/18/1995EP0634393A1 Polymerisable enamines
01/18/1995EP0633775A1 Compounds useful for treating inflammatory diseases and for inhibiting production of tumor necrosis factor
01/18/1995CN1097421A Adhesion receptor antagonists
01/18/1995CN1097413A Substituted ureas containing cyclic amines as chain extenders in polymeric systems
01/17/1995US5382661 Useful in treating spinal trauma, head injury, subarachnoid hemorrhage
01/17/1995US5382583 Piperazine derivatives
01/17/1995CA2128164A1 Process for the preparation of high purity buspiron and the hydrochloride thereof
01/12/1995WO1995001347A1 Novel cross-linking agents and use thereof
01/12/1995WO1995001326A1 Anti-atherosclerotic diaryl compounds
01/12/1995DE4322851A1 Telomers containing perfluorinated segments, and crosslinked resins prepared therefrom
01/12/1995DE4321843A1 Process for the preparation of nitrogen five-membered ring heterocycles
01/12/1995CA2166413A1 Anti-atherosclerotic diaryl compounds
01/11/1995EP0633260A1 2,3-Dihydro-1,4-benzodioxin-5-yl-piperazine derivatives having 5-HT1A-antagonistic activity
01/11/1995EP0633145A1 Thermal recording sheet
01/10/1995US5380941 From the phenylurea and an amine with the sulfur group
01/10/1995US5380888 7-(substituted)-9-[(substituted glycyl)amido]-6-demethyl-6-deoxytetracyclines
01/10/1995US5380855 Process for preparing N,N-substituted carbamoyl halides
01/10/1995US5380844 Nitrogen-containing perfluoroalkanoyl peroxide and method for production thereof
01/10/1995US5380841 Pyridinylpiperazinyl steroids
01/10/1995US5380840 Triazinylpiperazinyl steroids
01/10/1995US5380839 Phenylpiperazinyl steroids
01/10/1995US5380778 Fluorochemical aminoalcohols
01/10/1995US5380747 Treatment for atherosclerosis and other cardiovascular and inflammatory diseases
01/10/1995US5380733 Certain pyridyl-5-phenyl-1-cyclopropyl-dienamide pesticides
01/10/1995US5380726 Interleukin inhibitors
01/10/1995US5380725 Aryl- and heteroaryl piperazinyl carboxamides having central nervous system activity
01/10/1995US5380721 Aryl-fused and hetaryl-fused-2,4-diazepine and 2,4-diazocine antiarrhythmic agents
01/10/1995US5380629 Method of making and a photographic element containing bleach accelerator silver salts
01/10/1995CA1333905C Branched-chain alkyl esters of 2-[4-(2-piperidino-ethoxy) -benzoyl]-benzoic acid, processes for their preparation and their use as spasmolytic agents
01/09/1995WO1995001958A1 Difluoro statone analogs
01/05/1995WO1995000535A1 Optically pure calpain inhibitor compounds
01/05/1995WO1995000510A1 Processes and intermediates for the preparation of 5-[2-(4-(benzoisothiazol-3-yl)-piperazin-1-yl)ethyl]-6-chloro-1,3-dihydro-indol-2-one
01/05/1995WO1995000502A1 Novel intermediate for synthetic use and process for producing aminopiperazine derivative
01/05/1995WO1995000498A1 N,n-diacylpiperazines
01/05/1995WO1995000497A1 Inhibitors of farnesyl-protein transferase
01/05/1995WO1995000480A1 Novel intermediates for the preparation of antihistaminic 4-diphenylmethyl/diphenylmethoxy piperidine derivatives