Patents
Patents for C07D 295 - Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms (34,005)
06/1995
06/14/1995EP0656885A1 Synthesis of 2-substituted quinazoline compounds (such as terazosin) and meobentine and bethanidine and intermediates therefor
06/14/1995EP0496836B1 Synthesis and use of amino acid fluorides as peptide coupling reagents
06/13/1995US5424319 Renin inhibitors
06/13/1995US5424309 Hypotensive agents
06/13/1995US5424307 Renin inhibitors
06/08/1995WO1995015319A1 Paramagnetic chelates for nuclear magnetic resonance diagnosis
06/08/1995WO1995015309A1 Dp-iv-serine protease inhibitors
06/08/1995CA2178066A1 Dp-iv-serine protease inhibitors
06/07/1995EP0656356A1 Dioxacycloalkane compound with renin-inhibiting activity
06/07/1995EP0655992A1 Fluorenone derivatives, process for preparing the same and central or peripheral nerve degeneration repair and protective agent
06/07/1995CN1028756C Pryidyl-and pyrimidyl derivatives
06/07/1995CN1028714C Pyrimidine derivatives their production and use
06/06/1995US5422367 Diphenylcyclopropyl analogs as antiestrogenic and antitumor agents
06/06/1995US5422349 Renin inhibitors
06/01/1995WO1995014688A1 Derivatives of 2,3,5,6-tetrafluorobenzoic acid and their use in combating pests
06/01/1995WO1995014651A1 Amphiphilic derivatives of piperazine
06/01/1995CA2176714A1 Amphiphilic derivatives of piperazine
05/1995
05/31/1995EP0655472A1 Microwave-polymerizable isocyanate/epoxy resins for heavy-duty applications
05/31/1995EP0655063A1 Ethynyl alanine amino diol compounds having a piperazinyl-terminated group or a piperazinyl-alkylamino-terminated group for treatment of hypertension
05/31/1995EP0655056A1 Piperidinyl-terminated n-(dihydroxy alkyl)-ethynyl-alanine amides for treatment of hypertension
05/31/1995CN1028638C Method for preparation of isoquinoline amides of sulphonic acids derivatives
05/30/1995US5420278 ω-(4-aryl or heteroarylpiperazine-1-yl)-2-aryl or aralkyl-propanoic or butanoic acids
05/30/1995US5420272 7-(substituted)-8-(substituted)-9-](substituted glycyl)amido]-6-demethyl-6-deoxytetracyclines
05/30/1995US5420165 Substituted hydrazones, amidrazones, crop protection
05/30/1995US5420164 Enzyme inhibitors
05/30/1995US5420158 Melatonin activity
05/30/1995US5420127 Morpholino-terminated non-peptidyl α-succinamidoacyl aminodiols as anti-hypertensive agents
05/30/1995US5419898 Antiallergic composition for ophthalmic or nasal use
05/26/1995WO1995014017A1 Non-peptide tachykinin receptor antagonists
05/26/1995CA2176735A1 Non-peptide tachykinin receptor antagonists
05/24/1995CN1028521C Therapeutic agents
05/23/1995US5418249 Renin inhibitors
05/23/1995US5417884 Defined oligomeric liquid-crystalline compounds having smectic liquid-crystalline phases
05/18/1995WO1995013264A1 Hydroxamic acid derivative and medicinal preparation containing the same
05/17/1995EP0652750A1 Use of alpha,omega-dicarboxylic acids as fibrinogen reducers
05/17/1995EP0510158B1 Improved anti-plaque compositions comprising a combination of morpholinoamino alcohol and metal salts
05/17/1995CN1102649A Piperidines and piperazines
05/17/1995CN1102640A Alpha, omega-diarylalkane derivatives, their preparation and their use in the treatment and prevention of circulatory diseases and psychosis
05/17/1995CN1028426C Process of preparing non-cyclic polyalkylenepolyamines employing group VB metal catalysts
05/16/1995US5416212 Anilide derivatives
05/16/1995US5416210 Polymers or monomers protecting and controlling microorganisms from fungi, bacteria, algae, viruses and yeasts on a variety of substrates
05/16/1995US5416193 Polymer with carbodiimide pendant groups
05/16/1995US5416111 Cyano-containing n-phenyl-amino-terminated non-peptidyl α-succinamidoacyl aminodiols as anti-hypertensive agents
05/16/1995US5416104 Oxazolidinyl-terminated non-peptidyl α-succinamidoacyl aminodiols as anti-hypertensive agents
05/16/1995US5416095 Tetrahydro-quinolinyl-terminated non-peptidyl α-succinamidoacyl aminodiols as anti-hypertensive agents
05/16/1995US5416092 3-azabicyclo[3.2.1]-oct-8-yl-terminated non-peptidyl α-succinamidoacyl aminodiols as anti-hypertensive agents
05/16/1995US5416085 3-oxa-8-azabicyclo[3.2.1]oct-8-yl terminated non-peptidyl α-succinamidoacyl aminodiols as anti-hypertensive agents
05/16/1995US5416084 Benzo-fused thiomorpholinyl-terminated alkylamino ethynyl alanine amino diol compounds for treatment of hypertension
05/16/1995US5416083 Benzodiazepinyl-terminated non-peptidyl α-succinamidoacyl aminodiols as anti-hypertensive agents
05/16/1995CA1335591C Ring-substituted 2-amino-1,2,3,4-tetrahydronaphthalenes
05/12/1995CA2135576A1 Microwave-polymerizable isocyanate/epoxy resins for heavy-duty applications
05/11/1995WO1995012603A1 Matrix metalloprotease inhibitors________________________________
05/11/1995WO1995012394A1 Use of nitric oxide releasing compounds as protective agents in ischemia reperfusion injury
05/11/1995CA2175667A1 Matrix metalloprotease inhibitors________________________________
05/11/1995CA2175467A1 Use of nitric oxide releasing compounds as protective agents in ischemia reperfusion injury
05/10/1995EP0652208A1 Phenylalkan(en)oic acids with leukotriene B4 antagonistic activity
05/10/1995EP0652003A1 Methods for inhibiting smooth muscle cell proliferation and restinosis
05/10/1995EP0651738A1 Natural amino acid derivatives as metalloproteinase inhibitors
05/10/1995EP0651737A1 O-benzyl oxime ether derivatives and their use as pesticides
05/10/1995EP0651735A1 Pharmacologically active alpha-(tertiary-aminomethyl)-phenylmethanol derivatives
05/09/1995US5414087 Preparation of N-alkylpiperazines
05/09/1995US5414086 Preparation of 4-methylpyrimidines
05/09/1995US5414083 Dialkylating a urea in the presence of solid base and phase-transfer catalyst
05/09/1995US5414012 Indalyl-terminated non-peptidyl α-succinamidoacyl aminodiols as anti-hypertensive agents
05/09/1995US5413998 Benzo-fused thiazopinyl-terminated alkylamino ethynyl alanine amino diol compounds for treatment of hypertension
05/09/1995US5413997 Triphenylmethane derivatives
05/03/1995EP0650964A1 1 2H-1-benzopyran-2-one-8-yl -piperazine derivatives
05/03/1995EP0650958A1 Hydrazones of indane-triones and their application in therapy
05/03/1995EP0650595A1 Universal standard reagents, method of preparing same and use thereof
05/03/1995EP0650372A1 Compounds for cancer imaging and therapy
05/03/1995CA2134630A1 1-[2h-1-benzopyran-2-one-8-yl]-piperazine derivatives
05/02/1995US5411989 Nitric acid esters of cyclohexanol derivatives
05/02/1995US5411987 Fungicidal substituted amino acid amides
05/02/1995US5411975 Thiazolidinyl terminated alkylamino ethynyl alanine amino diol compounds for treatment of hypertension
05/02/1995US5411972 Arylamide derivatives for treating hyperlipemia
05/02/1995US5411962 Benzomorpholinyl-terminated non-peptidyl α-succinamidoacyl aminodiols as anti-hypertensive agents
05/02/1995US5411961 Benzo-fused morpholinyl terminated alkylamino ethynyl alanine amino diol compounds for treatment of hypertension
05/02/1995US5411959 1,4-Thiomorpholino-terminated alkylamino ethynyl alanine amino diol compounds for treatment of hypertension
05/02/1995US5411958 Benzothiomorpholinyl-terminated non-peptidyl α-succinamidoacyl aminodiols as anti-hypertensive agents
05/02/1995US5411957 3-azabicyclo[3.2.1]-nonanyl-terminated non-piptidyl alpha-succinamidoacyl aminodiols as anti-hypertensive agents
05/02/1995US5411954 Benzo-fused oxazopinyl-terminated alkylamino ethynyl alanine amino diol compounds for treatment of hypertension
05/02/1995US5411953 Oxazopinyl terminated alkylamino ethynyl alanine amino diol compounds for treatment of hypertension
05/02/1995US5411950 Benzo-fused oxazocinyl terminated alkylamino ethynyl alanine amino diol compounds for treatment of hypertension
05/02/1995US5411933 Bromopropargyl quarternary ammonium compounds having antimicrobial activity
05/02/1995CA1335447C Preparation of linear polyethylenepolyamines by reacting monoethanolamine with ethylenediamine in the presence of a phosphorus/titania/zirconia catalyst
04/1995
04/27/1995WO1995011240A1 Amine derivatives as calcium channel antagonists
04/27/1995WO1995011239A1 Novel phenoxyalkylpiperazine derivative
04/27/1995WO1995011238A1 Heterocyclic amines for treating ischaemic strokes
04/27/1995WO1995011228A1 2,3-diaminopropionic acid derivative
04/27/1995CA2174516A1 2,3-diaminopropionic acid derivative
04/26/1995EP0649835A1 Halopropiolamide compound, production and use thereof
04/26/1995EP0649420A1 New process for the preparation of 3,3-diaryl acrylic acid amides.
04/26/1995EP0649419A1 N-cycloalkylpiperazine derivatives, methods of obtaining them and pharmaceutical compositions containing them
04/26/1995EP0649414A1 Opioid diarylmethylpiperazines and piperidines
04/26/1995EP0649407A1 Dimeric piperidine, tetrahydropyridine and piperazine derivatives
04/25/1995US5409945 Benzyo-fused thiazolidinyl terminated alkylamino ethylnyl alanine amino diol compounds for treatment of hypertension
04/25/1995US5409931 1,3-substituted cycloalkenes and cycloalkanes as central nervous system agents
04/25/1995US5409925 Oxazobicyclo terminated alkylamino ethynyl alanine amino diol compounds for treatment of hypertension
04/25/1995US5409924 Benzo-fused oxazobicyclo terminated alkylamino ethynyl alanine amino diol compounds for treatment of hypertension
04/25/1995US5409922 Renin inhibitors