| Patents for C07D 267 - Heterocyclic compounds containing rings of more than six members having one nitrogen atom and one oxygen atom as the only ring hetero atoms (2,022) |
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| 09/03/2008 | CN100415743C Derivatives of pyrimido [6.1-a] isoquinolin-4-one |
| 09/02/2008 | US7420051 Antitumor agents; microbiocides; antibiotics; forming a 1,4 bridge using a 1-labile, 10-hydroxy, 18-protected hydroxyl, di-6,8-en-5-one fused ring compound. After formation of the 1,4 brige, C-18 protection is removed before spiroamine introduction |
| 09/02/2008 | US7419974 Cyclohexyl(alkyl)propanolamines, preparation method and pharmaceutical compositions containing same |
| 09/02/2008 | US7419969 N-((hetero)arylalkyl)pyrimidonecarboxamides in which the ring is fused to a C4-7(hetero)cycloalkyl ring, which in turn has a spiro ring attached: e.g., N-[(4-fluorophenyl)methyl]-7',8'-dihydro-3'-hydroxy-8'-methyl-4'-oxo-spiro[cyclopentane-1,9'(6'H)-[4H]pyrazino[1,2-a]pyrimidine]-2'-carboxamide |
| 09/02/2008 | CA2273023C Aminoguanidines and alkoxyguanidines as protease inhibitors |
| 08/28/2008 | US20080207590 Inhibitors of Histone Deacetylase |
| 08/26/2008 | US7417040 hormone sensitive diseases such as prostate hypertrophia, benign prostatic hyperplasia, adenomas and neoplasies of the prostate, prostate cancer, hirsutism, and polycystic ovary syndrome; dibenz[b,f]azocine, dibenzo[b,f][1,4]thiazocine, dibenz[b,f][1,5]oxazocine derivatives; anticancer, antitumor agents |
| 08/21/2008 | US20080200671 Crystal form of asenapine maleate |
| 08/20/2008 | EP1957485A2 Substituted 4-amino-pyrrolotriazine derivatives useful for treating hyper-proliferative disorders and diseases associated with angiogenesis |
| 08/14/2008 | WO2008098138A1 Synthetic macrocyclic compounds for treating cancer |
| 08/14/2008 | US20080194672 Growth hormone secretagogue (ghrelin) receptor; gastrointestinal disorders; gastroesophageal reflux disease (GERD), gastric ulcers, Crohn's disease |
| 08/14/2008 | US20080194540 Desipramine, imipramine, trimipramine, amitriptyline, nortriptyline, doxepin, amoxapine, or maprotyline and chloroquine, promazine, quinine, biquinoline, phenothiazine or chlorpromazine; transfection or gene therapy |
| 08/13/2008 | EP1572672B1 Benzoxazocines and their use as monoamine-reuptake inhibitors |
| 08/12/2008 | US7411095 obtained using specific secondary amines are unexpectedly stable against water; reacting an aldehyde or ketone with an amine and treating the resulting reaction mixture with an acidic aqueous solution |
| 08/06/2008 | EP1951694A2 Salt forms |
| 08/06/2008 | EP1951693A2 Solid formulations |
| 08/05/2008 | US7407950 N-(heteroaryl)-1H-indole-2-carboxamide derivatives and their use as vanilloid TRPV1 receptor ligands |
| 07/30/2008 | EP1950206A1 Benzoxazocines and their use as monoamine-reuptake inhibitors |
| 07/17/2008 | US20080171692 Substituted amides |
| 07/16/2008 | EP1942901A2 Rifamycin analogs and uses thereof |
| 07/10/2008 | US20080167335 To obtain zotarolimus and other rapamycin products |
| 07/09/2008 | EP1276729B1 New neurokinin antagonists for use as medicaments |
| 07/03/2008 | US20080161555 Purification of Tacrolimus on Supports of Vegetable Origin |
| 07/03/2008 | US20080161554 Macrocyclic carbodiimides (MC-CDI) and their derivatives, syntheses and applications of the same |
| 07/02/2008 | EP1937677A1 Cb-1 modulating compounds and their use |
| 07/02/2008 | EP1496838A4 Substituted amides |
| 07/02/2008 | CN101209999A Macrocyclic carbodiimide and its derivatives, synthesis and application |
| 06/26/2008 | US20080154035 Coupling method between intramolecular carbon in unsaturated hydrocarbon compound using organo-indium compound as coupling agent |
| 06/26/2008 | US20080153801 Benzoxazepine compounds, their production and use |
| 06/25/2008 | EP1933845A2 Nitric oxide-releasing biodegradable polymers useful as medical devices and coatings therefore |
| 06/24/2008 | US7390797 Fused indazole compounds |
| 06/19/2008 | WO2008072745A1 Process for production of anthranilamide compound |
| 06/19/2008 | US20080146821 Internal 1,15-Lactones Of Fluprostenol And Related Prostaglandin F2a Analogs And Their Use In The Treatment Of Glaucoma And Intraocular Hypertension |
| 06/19/2008 | US20080146580 Anititumoral Ecteinascidin Derivatives |
| 06/19/2008 | US20080146542 Hydrazinocarbonyl-thieno[2,3-C]pyrazoles, Process for Preparing Them, Compositions Containing Them and Use Thereof |
| 06/19/2008 | US20080146536 2-Aminoimidazopyridines for treating neurodegenerative diseases |
| 06/18/2008 | CN101200472A Method for preparing 3-amido-4-imino rifamycin S |
| 06/17/2008 | US7388031 Reacting an epoxy compound with a aminocylcohexane-phenyl derivative; useful as anti-obesity, anti-diabetic, cicatrizing and tocolytic medicinal products |
| 06/12/2008 | US20080139811 Reacting an amino, hydroxy substituted amide with a heterocyclic substituted carboxylic acid to produce (2S,3S,5S)-2-(2,6-Dimethylphenoxyacetyl) amino-3-hydroxy-5-[2S-1-imidazolidin-2-onyl)-3-methyl-butanoyl] amino-1,6-diphenylhexane; inhibitors of HIV infection |
| 06/12/2008 | US20080139806 Triaminophosphine ligands for carbon-nitrogen and carbon-carbon bond formation |
| 06/12/2008 | US20080139577 Nitroheteroaryl-containing rifamycin derivatives |
| 06/12/2008 | US20080139530 7-Aryl 1,5-Dihydro-4,1-Benzoxazepin-2(3H)-One Derivatives And Their Use As Progesterone Receptor Modulators |
| 06/05/2008 | US20080132483 Administering (3R,5S)-N-propanesulfonyl-7-chloro-5-(2,3-dimethoxyphenyl)-1-(3-hydroxy-2,2-dimethylpropyl)-1,2,3,5-tetrahydro-4,1-benzoxazepine-3-acetamide; cerebral infarction |
| 06/05/2008 | US20080132482 3-(2(R)-Cyclopentylmethyl-3 (S)-hydroxyl-1-oxo-5-phenylpentyl)amino-1-methyl-5-(4-fluoro-phenyl)-2,3-dihydro-1H-1,4-benzodiazepin-2-one; neurological disorders related to beta -amyloid production, Alzheimer's disease, Down's Syndrome |
| 06/05/2008 | DE60129697T2 Kondensierte azepinderivate und ihre verwendung als antidiuretisches mittel Condensed azepine derivatives and their use as antidiuretic agent |
| 06/03/2008 | US7381743 Macrocycles for the treatment of cancer |
| 05/28/2008 | CN101189215A Benzoxazocines and their therapeutic use |
| 05/22/2008 | WO2008059948A1 Haloalkylsulfonanilide derivative or salt thereof, herbicide comprising the derivative as active ingredient, and use of the herbicide |
| 05/15/2008 | US20080113965 Skeletal muscle protecting agent |
| 05/15/2008 | US20080113964 7-Aryl 1,5-Dihydro-4,1-Benzoxazepin-2(3H)-One Derivatives and Their Use As Progesterone Receptor Modulators |
| 05/13/2008 | US7371853 Ring structuresC6.C6.C14N2O, C6.C6.C15N2O, C6.C6.C16N2O and C6.C6.C17N2O |
| 04/22/2008 | US7361666 Ligands for cellular receptors, including opiate receptors; side effect reduction; base structure is a saturated nitrogen-containing ring substituted with a tertiary amide that is N-substituted with an arylalkyl group |
| 04/22/2008 | US7361648 1-(4-{ethyl-[2-(4-methanesulfonylphenyl)-1-methylethyl]amino}butyl)-4-methanesulfonyl-[1,4]diazepan-2-one; repiratory system disorders: asthma and chronic obstructive pulmonary disease; nervous system, muscular,urogenital, gastrointestinal disorders; antiallergens; side effect reduction |
| 04/17/2008 | US20080091008 Methods of manufacturing crystalline forms of rapamycin analogs |
| 04/17/2008 | US20080090805 Cb-1 modulating compounds and their use |
| 04/17/2008 | US20080090804 (cis)-8-fluorodibenzo[b,f]pyrido[1,2-d]oxazepine-1-amine derivatives; contraception, hormone replacement therapy (HRT) or gynaecological disorders, adjuvant therapy in cancer |
| 04/16/2008 | EP1910321A1 New compounds, process for their preparation, intermediates, pharmaceutical compositions and their use in the treatment of 5-ht6 mediated disorders such as alzheimer's disease, cognitive disorders, cognitive impairment associated with schizophrenia, obesity and parkinson's disease |
| 04/15/2008 | US7358275 cloprostenol or latanoprost; topical use; highly crystalline structures that are easy to formulate into ophthalmic solutions; The hydrolysis of these analogs releases only the active PGF2 alpha analog free acid, without the production of toxic and irritant small aliphatic alcohol coproducts |
| 04/09/2008 | CN101160280A Compounds and uses thereof |
| 04/08/2008 | US7355042 Sleep disorders; side effect reduction |
| 04/08/2008 | US7354914 1-[3-Methyl-1-(5-methyl-6-oxo-benzo[b]-1,4-oxazepin-7-ylcarbamoyl)-butyl]-cyclohexanecarboxylic acid amide; inhibit processing of amyloid precursor protein (production of A beta -peptide); neurological disorders related to beta -amyloid production: Alzheimer's disease, Down's Syndrome |
| 04/08/2008 | CA2187541C Benzoxazepine derivatives, salts thereof, and drugs containing the same |
| 04/01/2008 | US7351824 Intermediates for oxazolidinone antibacterials; N-[3-Chloro-2-(R)-hydroxypropyl]-3-fluoro-4-morpholinyl aniline |
| 04/01/2008 | CA2298974C Thiazolobenzoheterocycles, preparation and medicines containing same |
| 03/27/2008 | US20080076918 Quinoxaline compounds |
| 03/27/2008 | US20080076812 Lyophilized powder includes an antioxidant, a buffer and a bulking agent; storage stability; improved stability upon reconstitution; treating endothelin-mediated disorders such as hypertension |
| 03/27/2008 | US20080076752 substituted structure of 3-amino-2-(2,5-difluorophenyl)-2,3-dihydro-1,5-benzothiazepin-4(5H)-one; 6-amino-7-phenyl-1,4-thiazepan-5-one; -amino-2-phenyl-2,3-dihydro-1,5-benzoxazepin-4(5H)-one for treating neurological disorders such as Alzheimer's; inhibit the production of amyloid beta protein |
| 03/26/2008 | EP1902714A1 Prodrugs of gaba analogs, compositions and uses thereof |
| 03/26/2008 | EP1902041A1 New compounds, process for their preparation, intermediates, pharmaceutical compositions and their use in the treatment of 5-ht6 mediated disorders such as alzheimer s desease, cognitive disorders, cognitive impairment associated with schizophrenia, obesity and parkinson's disease |
| 03/20/2008 | US20080070978 cloprostenol or latanoprost; topical use; highly crystalline structures that are easy to formulate into ophthalmic solutions; hydrolysis of these analogs does not have toxic and irritant small aliphatic alcohol coproducts; hypotensive agent for intraocular pressure |
| 03/20/2008 | US20080070950 Amorphous rapamycin 42-ester with 3-hydroxy-2-(hydroxymethyl)-2- methylpropionic acid and its pharmaceutical compositions |
| 03/19/2008 | CN101146785A Novel anti-arrythmic and heart failure drugs that target the leak in the ryanodine receptor (RYR2) |
| 03/12/2008 | CN101142197A N-hydroxyamides omega-substituted with tricyclic groups as histone deacetylase inhibitors, their preparation and use in pharmaceutical formulations |
| 03/06/2008 | US20080058310 High-density lipoprotein-cholesterol level elevating agent |
| 02/21/2008 | US20080045497 Substituted aniline derivatives |
| 02/12/2008 | US7329746 Ring structures C6.C6.C13N and C6.C6.C12NO |
| 02/12/2008 | US7329652 Janus Kinase JAK2 and JAK3; 4-chloro-6-(3,5-dimethylpiperazin-1-yl)pyrimidine; chemotherapeutic, antiproliferative, antiinflammatory, immunomodulatory agent; allergies, asthma, autoimmune diseases, transplant rejection, rheumatoid arthritis, multiple sclerosis |
| 02/07/2008 | US20080031951 Compositions and methods for the inhibition of phospholipase A2 |
| 01/31/2008 | WO2008012524A1 Substituted aniline derivatives |
| 01/31/2008 | US20080027211 Enantiopure Heterocyclic Compound Useful for the Preparation of Peptides Which Can Be Potentially Used as Medicaments |
| 01/31/2008 | US20080027038 N-Acylated lipophilic amino acid derivatives |
| 01/31/2008 | CA2658913A1 Substituted aniline derivatives |
| 01/30/2008 | CN101115730A 新分子探针 New molecular probes |
| 01/29/2008 | US7323455 1,2,3,5-Tetrahydro-4,1-benzoxazepine derivatives: 4-methyl-5-(5-methyl-2-oxo-5-phenyl-1,2,3,5-tetrahydro-4,1-benzoxazepin-7-yl)thiophene-2-carbonitrile; contraceptives; hormone replacement therapy |
| 01/24/2008 | WO2007132255A3 Racemisation of enantiomers of nefopam and analogues |
| 01/23/2008 | EP1880215A2 Compositions and methods for detection of sirolimus |
| 01/23/2008 | EP1879863A1 Amide resorcinol compounds |
| 01/22/2008 | US7320973 5,11-Dihydrodiaryl[b,e][1,4,]oxazepine derivatives for gastrointestinal disorder treatment; irritable bowel syndrome |
| 01/17/2008 | US20080015213 Macrocyclic Aminopyridyl Beta-Secretase Inhibitors For The Treatment Of Alzheimer's Disease |
| 01/10/2008 | WO2007135295A3 Derivatives of 2-alkoxy-3,4,5-trihydroxy-alkyl amides, preparation and use thereof, and compositions containing the same |
| 01/10/2008 | WO2007050425A3 Lxr modulators |
| 01/10/2008 | US20080009619 Process for the preparation of asenapine and intermediate products used in said process |
| 12/27/2007 | US20070299051 Tricyclic Guanidine Derivatives as Sodium-Proton Exchange Inhibitors |
| 12/27/2007 | US20070299019 Macrolides and methods for producing same |
| 12/20/2007 | US20070293472 Novel 14 and 15 Membered Ring Compounds |
| 12/20/2007 | US20070293470 Carboxamide Spirolactam Cgrp Receptor Antagonists |
| 12/19/2007 | EP1347967B1 Novel benzazepines and related heterocyclic derivatives which are useful as orexin receptor antagonists |
| 12/19/2007 | CN101090908A Conjugates with anti-inflammatory activity |
| 12/13/2007 | US20070287697 Cgrp Receptor Antagonists |
| 12/13/2007 | US20070287696 ligands for Calcitonin gene related peptide; azepinone ligands; migranes; N-[5-(2,3-Difluorophenyl)-1-(2-methoxyethyl)-2-oxopiperidin-3-yl]-4-(2-oxo-2,3-dihydro-1H-imidazo[4,5-b]pyridin-1-yl)piperidine-1-carboxamide |