Patents for C07D 267 - Heterocyclic compounds containing rings of more than six members having one nitrogen atom and one oxygen atom as the only ring hetero atoms (2,022) |
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08/12/2010 | US20100204203 Chemical Compounds 637: Pyridopyrimidinediones as PDE4 Inhibitors |
08/05/2010 | WO2010087430A1 N-acyl anthranilic acid derivative or salt thereof |
08/05/2010 | US20100197907 Phosphorus-containing compounds & uses thereof |
08/05/2010 | US20100197657 2-aryl or heteroaryl indole derivatives |
08/05/2010 | CA2750452A1 N-acyl anthranilic acid derivative or salt thereof |
08/03/2010 | US7767660 Macrocyclic indole compounds, e.g., (7R)-14-cyclohexyl-21,24-dimethyl-7,8-dihydro-6H-7,11-(epiminoethanoiminopropanothio iminomethano)indolo[1,2-e][1,5]benzoxazocin-15-one 17,17-dioxide; hepatitis C virus polymerase inhibitors |
07/29/2010 | US20100190766 Antibacterial agents |
07/22/2010 | WO2010082627A1 Process for producing 2-hydroxymethylmorpholine salt |
07/20/2010 | CA2431982C Novel benzazepines and related heterocyclic derivatives which are useful as orexin receptor antagonists |
07/13/2010 | CA2567776C Vasopressin v1a antagonists |
07/08/2010 | US20100173890 Compounds, Process for their Preparation, Intermediates, Pharmaceutical Compositions and their use in the Treatment of 5-HT6 Mediated Disorders such as Alzheimer's Disease, Cognitive Disorders, Cognitive Impairment Associated with Schizophrenia, Obesity and Parkinson's Disease |
07/08/2010 | US20100173823 Alpha2c adrenoreceptor agonists |
07/01/2010 | US20100168080 Novel compounds useful as cc chemokine receptor ligands |
06/24/2010 | US20100160627 (2,3-cis)-3-amino-2-phenyl-2,3-dihydro-1,5-benzoxazepin-4(5H)-one; for treatment of neurological disorders related to amyloid beta protein production such as Alzheimer's disease; inhibit gamma secretase and thereby inhibit the production of amyloid beta protein |
06/24/2010 | US20100160291 Tricyclic spiro-oxindole derivatives and their uses as therapeutic agents |
06/24/2010 | US20100160280 Aminopyridine and carboxypyridine compounds as phosphodiesterase 10 inhibitors |
06/17/2010 | US20100152440 NOVEL ANTI-ARRHYTHMIC AND HEART FAILURE DRUGS THAT TARGET THE LEAK IN THE RYANODINE RECEPTOR (RyR2) |
06/16/2010 | EP2196469A1 Conjugates with anti-inflammatory activity |
06/16/2010 | CN1989141B Bicyclic heterocycles as HIV integrase inhibitors |
06/10/2010 | WO2010065717A1 Morpholinone compounds as factor ixa inhibitors |
06/10/2010 | CA2745121A1 Morpholinone compounds as factor ixa inhibitors |
06/08/2010 | US7732434 9-Amino-14,30-dichloro-5-methyl-4,24-dioxa-3,8,10,16,19-pentaazatetracyclo-[23.2.2.212,15.02,6 ]hentriaconta-1(27),2,5,8,12,14,21,25,28,30-decaene-7,17-dione; inhibit the processing of amyloid precursor protein; Alzheimer's Disease (AD) and Down's Syndrome |
06/03/2010 | WO2010062565A1 Muscarinic agonists |
05/27/2010 | US20100129473 AMINO SUBSTITUTED DIARYL[a,d]CYCLOHEPTENE ANALOGS AS MUSCARINIC AGONISTS AND METHODS OF TREATMENT OF NEUROPSYCHIATRIC DISORDERS |
05/20/2010 | WO2010001407A8 Synthesis of 11-(4-[2-(2-hydroxyethoxy)ethyl]- piperazinyl)dibenzo[b,f][1,4]thiazepine and its fumarate salt |
05/18/2010 | US7718646 Cyclohexyl(alkyl)propanolamines, preparation method and pharmaceutical compositions containing same |
05/18/2010 | US7718645 4-[4-(4-Amino-5-oxo-7,8-dihydropyrimido[5,4-f][1,4]oxazepin-6(5H)-yl)phenyl]cycloalkylalkyl nitriles, carboxy acids or esters, amides, e.g., a -cyclohexylacetonitrile; diglyceride acyltransferase inhibitors for treating type II diabetes and obesity |
05/13/2010 | US20100120742 Rexinoid compound having alkoxy group |
05/13/2010 | US20100120716 Macrocyclic hepatitis c serine protease inhibitors and uses therefor |
05/12/2010 | CN1794997B 2,3,4,5-tetrahydrobenzo[f][1,4]oxazepine-5-carboxylic acid amide derivatives as gamma-secretase inhibitors for the treatment of alzheimer's disease |
05/11/2010 | US7713966 Heterobicyclic metalloprotease inhibitors |
05/06/2010 | US20100113770 O-substituted hydroxyaryl derivatives |
05/06/2010 | US20100113414 Thiazolyl-dihydro-indazoles |
05/05/2010 | CN101060847B Loxapine analogs and methods of use thereof |
05/04/2010 | US7709466 Pyridazinone derivatives, methods for their production and their use as pharmaceuticals |
04/29/2010 | US20100105657 Compounds, Process for their Preparation, Intermediates, Pharmaceutical Compositions and their use in the Treatment of 5-HT6 Mediated Disorders such as Alzheimer's Disease, Cognitive Disorders, Cognitive Impairment Associated with Schizophrenia, Obesity and Parkinson's Disease |
04/28/2010 | EP1363640B1 Nucleic acid derivatives |
04/28/2010 | CN1658855B O-substituted hydroxyaryl derivatives |
04/22/2010 | US20100099865 Heat shock protein 90 inhibitors |
04/08/2010 | US20100087418 Benzoxazepine derivatives and use thereof |
04/01/2010 | US20100081700 Hepatitis C Virus Inhibitors |
03/25/2010 | WO2010001407A3 Synthesis of ll-(4-[2-(2-hydroxyethoxy)ethyl]- piperazinyl)dibenzo[b,f][1,4]thiazepine and its fumarate salt |
03/25/2010 | US20100076046 Antiviral Indoles |
03/18/2010 | US20100069358 Use of 7-azaindoles in the inhibition of c-jun n-terminal kinase |
03/18/2010 | US20100069354 7-azaindole derivatives and their use in the inhibition of c-jun n-terminal kinase |
03/16/2010 | US7678784 4-amino-23,26-dichloro-13-oxa-3,5,18,21-tetraazatricyclo[20.2.2.29,12]octacosa-1(24),4,9,11,15,22,25,27-octaene-6,8,20-trione 8-(O-ethyloxime); beta -amyloid production blocking agent; neurodegenerative diseases, cognition activator; Alzheimer's disease, Down syndrome |
03/11/2010 | US20100063027 Amine Derivative Having NPY Y5 Receptor Antagonistic Activity |
03/09/2010 | US7674921 cloprostenol or latanoprost; topical use; highly crystalline structures that are easy to formulate into ophthalmic solutions; hydrolysis of these analogs releases only the active PGF2 alpha analog free acid, without the production of toxic and irritant small aliphatic alcohol coproducts |
02/25/2010 | WO2010021149A1 Spiro compound capable of inhibiting acid secretion |
02/18/2010 | WO2010018268A1 Novel (rs)-7- or 9-(1,2,3,5-tetrahydro-4,1-benzoxazepin-3-il)-7h or 9h-purines having antitumour activity |
02/18/2010 | US20100041637 1,3-Oxazepan-2-one and 1,3-diazepan-2-one inhibitors of 11ß-hydroxysteroid dehydrogenase 1 |
02/18/2010 | US20100041619 Lasonolide compounds as reagents for inducing premature chromosome condensation and methods for treating disorders |
02/16/2010 | CA2478183C Substituted amides |
02/09/2010 | US7659263 (E)-3-[4-({1-[(11-cyclohexyl-8-methoxy-4,5-dihydro-6-oxa-1-thia-3b-azabenzo[e]cyclopenta[a]azulene-2-carbonyl)amino]cyclobutanecarbonyl}amino)phenyl]acrylic acid; RNA-dependent RNA polymerase inhibitory activity; hepatitis C |
01/26/2010 | US7652003 Macrocyclic β-secretase inhibitors |
01/21/2010 | US20100016285 Heterocyclidene-n-(aryl) acetamide derivative |
01/21/2010 | US20100016284 Compounds and uses thereof - 151 |
01/21/2010 | US20100016283 Compounds and uses thereof - 150 |
01/21/2010 | US20100016272 Heteroarylacrylamides and their use as pharmaceuticals |
01/21/2010 | US20100016164 Haloalkylsulfonanilide derivatives or salt thereof, herbicide comprising the derivatives as active ingredient, and use of the herbicide |
01/19/2010 | US7649001 Fused benzene derivative and use |
01/07/2010 | US20100004222 Amide Derivatives as Ion-Channel Ligands and Pharmaceutical Compositions and Methods of Using the Same |
12/31/2009 | US20090325950 Benzoxazine derivatives and uses thereof |
12/30/2009 | EP2137157A1 Polymorphs of 7-[(3-chloro-6,11-dihydro-6-methyldibenzo[c,f][1,2]thiazepin-11-yl)amino]heptanoic acid s,s dioxide and methods of making and using the same |
12/30/2009 | EP1805202B1 Conjugates with anti-inflammatory activity |
12/24/2009 | US20090317328 Tricyclic oxazepines as in vivo imaging compounds |
12/22/2009 | CA2475383C Method for extracting a macrolide from biomatter |
12/10/2009 | WO2009146772A1 New terpenes and macrocycles |
12/10/2009 | CA2726883A1 New terpenes and macrocycles |
12/02/2009 | EP2125750A2 Cyclic urea and carbamate inhibitors of 11beta-hydroxysteroid dehydrogenase 1 |
12/01/2009 | US7625887 e.g. 2-[3,5-trans-5-(3-aminophenyl)-7-chloro-1-neopentyl-2-oxo-1,2,3,5-tetrahydro-4,1-benzoxazepin-3-yl]-N-(2-fluorobenzyl)acetamide; G-protein-coupled receptor (TGR5) agonist; central nervous system diseases; antiinflammatory agent; learning enhancement; angina pectoris, arrhythmia, bronchial asthma |
11/25/2009 | EP2123644A1 Benzoxazepine derivatives and use thereof |
11/24/2009 | US7622461 Amino substituted diaryl[a,d]cycloheptene analogs as muscarinic agonists and methods of treatment of neuropsychiatric disorders |
11/18/2009 | EP2118079A1 Synthetic macrocyclic compounds for treating cancer |
11/12/2009 | WO2009071631A3 Dibenzoazepine and dibenzooxazepine trpa1 agonists |
11/10/2009 | US7615549 Substituted pyrrolidinones, their manufacture and their use as medicaments |
11/03/2009 | CA2449729C Prodrugs of gaba analogs, compositions and uses thereof |
10/22/2009 | US20090264404 Derivatives of 4-piperazin-1-yl-4-benzo[b]thiophene suitable for the treatment of cns disorders |
10/21/2009 | CN101563347A Vasopressin V1a antagonists |
10/15/2009 | US20090258901 Ligands for monoamine receptors and transporters, and methods of use thereof |
10/15/2009 | US20090258884 Substituted amides |
10/14/2009 | CN101558056A Process for production of anthranilamide compound |
10/13/2009 | US7601695 11-N-[4-(4-Pyridin-3-yl-imidazol-1-yl)-butyl]-6-O-methyl-5-O-(3-dimethylamino-2-hydroxy-propoxy)-3-oxo-erythronolide A, 11,12-carbamate; functionalized macrolides; antiviral, antiprotozoal, anticancer and antigastrointestinal |
10/06/2009 | US7598237 7-aryl 1,5-dihydro-4,1-benzoxazepin-2(3H)-one derivatives and their use as progesterone receptor modulators |
09/24/2009 | US20090239839 Receptor antagonist |
09/23/2009 | CN100543017C Novel keto-oxadiazole derivatives as cathepsin inhibitors |
09/22/2009 | US7592333 Loxapine analogs and methods of use thereof |
09/22/2009 | US7592331 2-(1-Amino-isoquinolin-6-ylamino)-4,11-diazatricyclo[14.2.2.1(6,10)]henicosa-1(19),6,8,10(21),16(20),17-hexaene-3,12-dione trifluoroacetic acid salt; serine protease inhibitors; arterial cardiovascular thromboembolic disorders; cerebral, kidney, pulmonary embolisms; acute coronary syndrome;prosthetics |
09/22/2009 | CA2360894C (1-phenacyl-3-phenyl-3-piperidylethyl) piperidine derivatives, method for the production thereof and pharmaceutical compositions containing the same |
09/08/2009 | US7585889 cloprostenol or latanoprost; topical use; highly crystalline structures that are easy to formulate into ophthalmic solutions; hydrolysis of these analogs does not have toxic and irritant small aliphatic alcohol coproducts; hypotensive agent for intraocular pressure |
09/03/2009 | WO2009107389A1 Tricyclic compound |
09/03/2009 | US20090221689 Macrocyclic Modulators of the Ghrelin Receptor |
09/03/2009 | US20090221551 Substituted fused[1,2] imidazo[4,5c] ring compounds and methods |
09/01/2009 | US7582752 Process for the resolution of nefopam |
09/01/2009 | US7582280 Conjugates of antioxidants with metal chelating ligands for use in diagnostic and therapeutic applications |
09/01/2009 | CA2417353C Single-step process for preparing 7,16-deoxy-2-aza-10-o-cladinosil-12-o-desosaminil-4,5-dihydroxi-6-ethyl-3,5,9,11,13,15-hexamethylbicycle (11.2.1)hexadeca-1(2)-en-8-one, and obtaining a new form of 9-deoxo-9a-methyl-9a-aza-9a-homoerythromycin a |
08/27/2009 | US20090215742 Amide resorcinol compounds |
08/25/2009 | US7579463 Crown ether derivatives |
08/20/2009 | US20090209593 Novel antibacterial agents |
08/18/2009 | US7576198 A hydroxy compound containing substituted orpyridine, pyrazine, pyrimidine, oxazole, thiadiazole, quinoline, isoquinoline etc. as anti HIV agent, for treating AIDS |