Patents
Patents for C07D 267 - Heterocyclic compounds containing rings of more than six members having one nitrogen atom and one oxygen atom as the only ring hetero atoms (2,022)
02/2004
02/25/2004EP1390034A1 N-substituted nonaryl-heterocyclo amidyl nmda/nr2b antagonists
02/25/2004CN1478084A Compounds useful in treatment of inflammatory diseases
02/25/2004CN1478074A Cyclohexyl (alkyl)-propanolamines, preparation method and pharmaceutical compositions containing same
02/19/2004WO2004014851A2 Tyrosine kinase inhibitors
02/19/2004US20040034018 2-amino-trihydroindole or tetrahydronapthalene-2-yl derivatives, useful for disease state associated with smooth muscle disorders, such as gastrointestinal and urogenital disorders
02/19/2004US20040033969 Such as penicillin G coupled to 2'deoxyazithromycin; drug delivery
02/19/2004DE10234697A1 Neue Verbindungen zur Stimulation des Nervenwachstums, zur Inhibition der Narbengewebsbildung und/oder Reduktion eines Sekundärschadens Novel compounds for stimulation of nerve growth, to inhibition of scar tissue formation and / or reduction of secondary damage
02/12/2004WO2004012649A2 Novel compounds for stimulation of nerve growth, for the inhibition of scar tissue formation and/or reduction of secondary damage
02/12/2004US20040029850 Central nervous system disorders; antidepressants; bipolar disorders; rhematic diseases
02/10/2004CA2108903C Substituted dibenzoxazepine compounds, pharmaceutical compositions and methods of use
02/04/2004CN1473053A High-density lipoprotein-cholesterol level elevating agent
01/2004
01/29/2004WO2004009530A1 Process for production of high-purity enamines
01/13/2004US6677332 Amide-substituted piperidine or azepine derivatives to treat drug abuse and tinnitus
01/02/2004EP1373188A1 Alanine 2,6-dialkoxyphenyl ester derivatives as hypnotics
01/01/2004US20040002539 Enzyme inhibitors; anticoagulants; blood collecting device
12/2003
12/31/2003WO2003068980A3 Method for extracting a macrolide from biomatter
12/24/2003WO2003105833A1 Formulation of nefopam and its use in the treatment of pain
12/24/2003WO2003105832A1 Use of nefopam for the treatment of nausea or emesis
12/24/2003CA2489315A1 Formulation of nefopam and its use in the treatment of pain
12/24/2003CA2489306A1 Use of nefopam for the treatment of nausea or emesis
12/23/2003US6667301 Therapy for muscular disorders, urogenital disorders, gastrointestinal disorders, respiratory system disorders
12/18/2003US20030232825 Benzoxazine derivatives and uses thereof
12/17/2003CN1462269A Fused azepine drivatives and their use as antidiuretic agents
12/16/2003US6664249 Bicyclic vasopressin agonists
12/11/2003WO2003101490A1 Drug composition containing calcium channel antagonist
11/2003
11/27/2003WO2003097618A1 Morpholinylmethylureas ccr-3 receptor antagonists
11/20/2003WO2003095434A1 Benzoxazine derivatives as 5-ht6 modulators and uses thereof
11/11/2003US6645980 Ligands for biological receptors such as opiate receptors or G-protein coupled receptors used for treating pain, drug dependence or tinnitus in mammals
11/11/2003US6645958 Benzocycloalkylenylamine derivatives as muscarinic receptor antagonists
11/04/2003US6642233 Strong affinity and high selectivity for the human NK1 receptors of substance P.
10/2003
10/28/2003US6638931 Aminoguanidines and alkoxyguanidines as protease inhibitors
10/21/2003US6635661 Heterocyclic analgesic compounds and methods of use thereof
10/16/2003WO2002100347A3 Prodrugs of gaba analogs, compositions and uses thereof
10/07/2003US6630462 Delta agonist analgesics
10/01/2003EP1347967A1 Novel benzazepines and related heterocyclic derivatives which are useful as orexin receptor antagonists
10/01/2003CN1122670C Thiazolobenzoheterocycles, prepn method and medicines containing same
09/2003
09/30/2003US6627627 Aralkyl and aralkylidene heterocyclic lactams and imides
09/25/2003WO2003077847A2 Substituted amides
09/18/2003WO2003076424A1 Macrocyclic compounds useful as pharmaceuticals
09/18/2003US20030176668 C-nitroso compounds and use thereof
09/18/2003CA2478065A1 Macrocyclic compounds useful as pharmaceuticals
09/17/2003CN1121395C Compounds potentiating retinoid
09/10/2003EP1341753A1 Cyclohexyl(alkyl)-propanolamines, preparation method and pharmaceutical compositions containing same
09/10/2003CN1440971A Vitronectin receptor antagnist, its preparation and use
09/04/2003US20030166924 Method for extracting a macrolide from biomatter
09/03/2003EP1339696A1 Benzyl(idene)-lactams and their use as 5ht1-receptor ligands
09/02/2003US6613761 (3R,5S)-N- methanesulfonyl-7-chloro-5-(2,3-dimethoxyphenyl) -1-(3-hydroxy-2,2-dimethylpropyl)-2-oxo-1,2,3,5-tetrahydro-4, 1-benzoxazepine-3-acetamide, used as antilipemic agents and enzyme inhibitors
08/2003
08/28/2003WO2003070254A1 Antibiotic conjugates
08/28/2003US20030162964 Benzene-fused heterocycle derivatives and drugs containing the same as the active ingredient
08/28/2003CA2476448A1 Antibiotic conjugates
08/21/2003WO2003068980A2 Method for extracting a macrolide from biomatter
08/21/2003US20030158252 Especially trypsin-like serine proteases, such as chymotrypsin, trypsin, thrombin, plasmin and factor Xa.
08/20/2003CN1437587A Benzoxazepinones and their use as squalene synthase inhibitors
08/06/2003EP1332763A1 High-density lipoprotein-cholesterol level elevating agent
08/05/2003CA2075861C Dibenz[b,f][1,4]oxazepin-11(10h)-ones for multidrug resistance reversing agents
07/2003
07/30/2003EP1330425A2 C-nitroso compounds and use thereof
07/23/2003EP0929528B1 Aralkyl and aralkylidene heterocyclic lactams and imides
07/17/2003US20030135042 Atypical antipsychotic agents having low affinity for the D2 Receptor
07/16/2003CN1430610A Substituted 1-aminoalkyl-lactams compound and their use as muscarinic receptor antagonists
07/16/2003CN1430609A Substituted 1-aminoalkyl-lactams compound and their use as muscarinic receptor antagonists
07/09/2003EP1324992A1 Cyclized benzamide neurokinin antagonists for use in therapy
07/09/2003EP1324991A1 Compounds useful in the treatment of inflammatory diseases
07/02/2003EP1322314A2 Treatment of diabetes mellitus by inhibition of mitochondrial calcium/sodium antiporter
06/2003
06/26/2003US20030119811 Ion channel antagonists that are NMDA antagonists; treatment of migraine, depression, anxiety, schizophrenia, Parkinson's disease, or stroke.
06/18/2003EP1318988A2 Ligands for monoamine receptors and transporters, and methods of use thereof (neurotransmission)
06/12/2003US20030109524 Benzocycloalkylenylamine derivatives as muscarinic receptor antagonists
06/05/2003US20030105102 Oxo-substituted compounds, process of making, and compositions and methods for inhibiting PARP activity
05/2003
05/30/2003WO2003043618A2 Amino diols useful in the treatment of alzheimer's disease
05/30/2003CA2467476A1 Amino diols useful in the treatment of alzheimer's disease
05/29/2003US20030100755 For example (2S, 3S, 5S)-2-(2,6-dimethylphenoxyacetyl)amino-3-hydroxy-5-(2S-(1-tetrahydro-pyrimid-2-onyl)-3-methyl butanoyl)amino-1,6-diphenylhexane; HIV therapy
05/13/2003US6562963 Coupling using organosilicon compound
05/13/2003US6562813 Aralkyl and aralkylidene heterocyclic lactams and imides
05/01/2003US20030083382 Orally administered dosage forms of GABA analog prodrugs having reduced toxicity
04/2003
04/24/2003US20030078251 Triglyceride and cholesterol lowering activity and treats hyperlipidemia
04/23/2003EP1304326A1 Single-step process for preparing 7,16-deoxy-2-aza-10-o-cladinosil-12-o-desosaminil-4,5-dihydroxi-6-ethyl-3,5,9,11,13,15-hexamethylbicycle (11.2.1)hexadeca-1(2)-en-8-ona and obtaining a new form of 9-desoxo-9a-methyl-9a-aza-9a-homoerythromycin a
04/10/2003US20030069418 Ligands for cellular receptors, including opiate receptors; side effect reduction; base structure is a saturated nitrogen-containing ring substituted with a tertiary amide that is N-substituted with an arylalkyl group
04/09/2003EP0674623B1 Bicyclic fibrinogen antagonists
03/2003
03/27/2003WO2003024941A1 Naphthalene compounds and use thereof as drugs
03/26/2003EP1294698A1 Fused azepine derivatives and their use as antidiuretic agents
03/26/2003CN1103775C Vitronectin receptor antagonists, their preparation and use
03/25/2003US6538116 For therapy of inflammatory or painful disorder
03/19/2003EP1292585A1 Benzoxazepinones and their use as squalene synthase inhibitors
03/13/2003US20030050309 A gelatinase inhibitor for modulating the activity of a dopamine, serotonin, or norepinephrine receptor or transporter
03/12/2003EP1289965A1 Substituted 1-aminoalkyl-lactams and their use as muscarinic receptor antagonists
03/12/2003EP1289964A1 Substituted 1-aminoalkyl-lactams and their use as muscarinic receptor antagonists
03/04/2003US6528504 Compounds such as (R)-5,11-dihydro-5-(1-(4-methoxyphenethyl)-piperidine-2-ylmethyl) -dibenzo(b,e)(1,4) oxazepine are useful for treating or preventing abnormal motor functions of gastrointestinal tracts, e.g., irritable bowel syndrome.
03/04/2003US6528492 Azithromycin by treating erythromycin A with O-mesitylene sulfonyl hydroxylamine in the presence of sodium bicarbonate to produce 9-deoxo-6-deoxy-6,9-epoxy-9,9a- didehydro-9a-aza-homoerythromycin A intermediate, the 6,9-iminoether
02/2003
02/27/2003WO2003016245A1 Chromatographic separation of enantiomers of protected amino acids via smb-method
02/13/2003US20030032635 Heterocyclic esters and amides
02/11/2003US6518310 Non-peptidic; inhibits trypsin-like protease, thrombin and embolus formation; anticoagulant
02/06/2003US20030027807 Vitronectin receptor antagonists, their preparation and their use
01/2003
01/27/2003WO2002010144A1 Single-step process for preparing 7,16-deoxy-2-aza-10-o-cladinosil-12-o-desosaminil-4,5-dihydroxi-6-ethyl-3,5,9,11,13,15-hexamethylbicycle (11.2.1)hexadeca-1(2)-en-8-ona and obtaining a new form of 9-desoxo-9a-methyl-9a-aza-9a-homoerythromycin a
01/22/2003EP1276729A1 New neurokinin antagonists for use as medicaments
01/14/2003US6506744 Benzazepinone-derivatives
01/14/2003CA2141494C Mediators suitable for the electrochemical regeneration of nadh, nadph or analogs thereof
01/09/2003WO2003002147A1 Preventives/remedies for organ functional disorders and organ dysfunction
01/09/2003CA2451163A1 Agent for preventing or treating organ functional disorders and order dysfunction
01/07/2003US6503898 Administering 4,7-dibenzyl-5,6-dihydroxy-N,N*-di(m-aminobenzyl)--1,3-diazepin-2-one or salt to treat human immunodeficiency virus infection
01/03/2003WO2003000670A1 A11-piperazinyldibenzo (b, f) (1, 4) oxazepines and thiazepines as atypical antipsychotic agents having low affinity for the d2 receptor
01/03/2003WO2002060870A3 Delta agonist analgesics
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