Patents
Patents for C07D 263 - Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings (20,978)
07/2009
07/09/2009WO2009085637A1 Amorphous metaxalone and amorphous dispersions thereof
07/09/2009US20090176993 (N-{5-[(4-chlorophenyl)thio]pentyl}-N-[(1R)-1-(1-naphthyl)ethyl]amine); mimics/blocks effect of extracellular calcium in parathyroid cells, juxtaglomerular/proximal tubule kidney cells, parafollicular thyroid cells, bone osteoclasts, keratinocytes or placental trophoblasts; hyperparathyroidism
07/08/2009EP1836173A4 Anti-inflammatory medicaments
07/08/2009CN101479238A Amine derivative having npyy5 receptor antagonist activity
07/08/2009CN100510098C Optically active, heteroaromatic beta-hydroxy esters, processes for their preparation from beta-keto esters and processes for the preparation of these beta-keto esters
07/07/2009US7557214 Intermediate products for producing oxazolidinone-quinolone hybrids
07/07/2009CA2438324C Acylated 6,7,8,9-tetrahydro-5h-benzocycloheptenyl amines and their use as pharmaceutical
07/02/2009WO2009080788A2 Antibacterial agents
07/02/2009WO2009080446A1 2-methylthioethyl-substituted heyrrocycles as feed additives
07/02/2009WO2009061811A8 Substituted cyclopentanes having prostaglanding activity
07/02/2009WO2009012201A3 Process for the preparation of trifluoroalkyl-phenyl and heterocyclic sulfonamides
07/02/2009US20090170915 POLYMORPHIC FORMS OF (S)-1-cyanobutan-2-yl (S)-1-(3-(3-(3-methoxy-4-(oxazol-5-yl)phenyl)uriedo)phenyl)ethylcarbamate
07/02/2009US20090170908 Spiro compounds and pharmaceutical use thereof
07/02/2009US20090170883 3-arylphenyl sulfide derivative and insecticide and miticide
07/02/2009US20090170864 (S)-3-{5-[(1-Pyridin-2-yl-3-trifluoromethyl-1H-pyrazole-4-carbonyl)-amino]-pyridin-2-ylamino}-pyrrolidine-1-carboxylic acid ethyl ester; obesity, type II diabetes mellitus and metabolic syndrome
07/02/2009US20090170812 Transcription factor modulating compounds and methods of use thereof
07/02/2009CA2710170A1 2-methylthioethyl-substituted heterocycles as feed additives
07/01/2009EP2074089A2 Organic compounds
07/01/2009EP1599455B1 4-(3- (2-phenyl-oxazol-4-ylmethoxy)-cyclohexyloxy)-butane acid derivatives and related compounds as ppar modulators for treating diabetes of type 2 and atherosclerosis
07/01/2009CN100506805C Process for producing 5-substituted oxa zole compounds and 5-substituted imidazole compounds
07/01/2009CN100506788C Arylalkylcarbamate derivatives production and use thereof in therapy
07/01/2009CN100506776C NK1 antagonists
06/2009
06/30/2009US7554000 Reacting an arylhydrazine, hydrogen peroxide and an aryl compound using a catalytic metal of Group 5,6,7 or 8 or an oxide of a metal of Group 5,6,7 or 8 obtained by reacting the given metal with hydrogen peroxide; improved yield; quaternary amine as phase transfer agent; water solvent and by-product
06/30/2009US7553975 2-(((2-amino-1-oxo-3-mercapto-propyl)-amino)-methyl)-5-phenyl-thiazole-4-carbonyl-methionine; useful for treating restenosis or tissue proliferative diseases
06/30/2009US7553966 Glucocorticoid mimetics, methods of making them, pharmaceutical compositions, and uses thereof
06/30/2009US7553860 e.g.(S)-methyl 5-(((3-(4-(1-hydroxyhexyl)phenyl)-2-oxooxazolidin-4-yl)methoxy)methyl)thiophene-2-carboxylate; prostaglandin EP2 agonist; ocular hypotensive, antiinflammatory agent; glaucoma, inflammatory bowel disease and as presurgical adjuncts
06/25/2009WO2009079597A1 Piperazinyl derivatives useful as modulators of the neuropeptide y2 receptor
06/25/2009WO2009079593A1 Piperazinyl derivatives useful as modulators of the neuropeptide y2 receptor
06/25/2009WO2009078813A1 Method of forming oseltamivir and derivatives thereof
06/25/2009WO2009043027A3 Multi-armed forms of activated polyoxazoline and methods of synthesis thereof
06/25/2009WO2008152306A3 Novel peptidase substrates
06/25/2009WO2008098396A3 Oxazolidinones and their use as hypocholesterolemic agents
06/25/2009US20090163561 Amorphous metaxalone and amorphous dispersions thereof
06/25/2009US20090163549 Pharmaceutical Composition Comprising an Amide Derivative
06/25/2009US20090163496 Antibacterial agents
06/25/2009US20090163485 Heteroaryl derivatives as orexin receptor antagonists
06/25/2009US20090162474 2-methylthioethyl-substituted heterocycles as feed additives
06/25/2009DE102007062199A1 2-Methylthioethyl-substituierte Heterocyclen als Futtermitteladditive 2-methylthioethyl-substituted heterocycles as feed additives
06/25/2009DE102007061630A1 Preparing montelukast sodium, useful e.g. to antagonize leukotriene, comprises reacting sodium alkoxide compound with montelukast acid in organic solvent, where the montelukast acid is obtained by acidifying montelukast cyclohexylamine
06/24/2009EP2072505A2 A process for the preparation of oxazolidinone derivatives
06/24/2009EP1620093B1 Pesticidal (dihalopropenyl) phenylalkyl substituted benzoxazole and benzothiazole derivatives
06/24/2009CN101466688A Oxazole derivatives and their use in the treatment of diabetes and obesity
06/24/2009CN101466687A Activating agent for peroxisome proliferator activated receptor delta
06/24/2009CN100503600C Pesticidal heterocycles
06/24/2009CN100503568C Process for the preparation of perindopril, its analgous compounds and salts therof using 2,5 dioxo-oxazolidine intermediate compounds
06/23/2009USRE40795 Pesticides, drugs, fungicides; reacting p-toluenesulfony isocyanate with phosphorus oxychloride or phosgene in presence of phase transfer agent and base; final stable solution without irritating, nonexplosive
06/23/2009US7550511 amino alcohols; selective ribonucleic acid (RNA) binding agents; detecting the binding of small molecules to T-box antiterminator model mRNAs; screening for microbiocidal drug targets; use disinfecting; antiviral, anti-HIV; e.g. use of 1,2-dihydroxy-3-amino-4-phenylbutane
06/23/2009US7550489 N-[3-(4-chlorophenyl)-2-(3-cyanophenyl)-1-methylpropyl]-2-(5-trifluoromethyl-2-pyridyloxy)-2-methylpropanamide and phentermine, metformin, or bupropion; obesity; antipsychotic agents; synergistic; cannabinoid receptor antagonists
06/23/2009US7550448 Therapeutic compounds
06/18/2009WO2009075080A1 Fluoroalkylsulfide derivative and pest control agent
06/18/2009WO2009046841A3 Piperidine and piperazine derivatives for treating tumours
06/18/2009US20090156828 Novel Compounds and Methods for Forming Taxanes and Using the Same
06/18/2009US20090156807 Anti-tumor Compounds Derived From 1,4,5,8-tetrachloroanthraquinone
06/18/2009US20090156653 such as 2-amino-5-[4-(3-benzyloxyphenylthio)-2-chlorophenyl]-2-methylpentane-1-ol, used for treating autoimmune diseases, rheumatoid arthritis, psoriasis, dermatitis, asthma, hay fever or rejection of organ or bone morrow transplantation; side effect reduction
06/18/2009US20090156640 Nociceptin analogs
06/18/2009US20090156590 Vanilloid Receptor Ligands, Pharmaceutical Compositions Containing Them, Process for Making Them, and Use Thereof for Treating Pain and Other Conditions
06/18/2009US20090156588 such as 3-[4-(tert-Butyl-dimethyl-silanyloxy)-phenyl]-7-hydroxy-3,4-dihydro-benzo[e][1,3]oxazin-2-one, inhibitors macrophage migration inhibitory factor isomerase activity; treatment of vision defects, ischemia, inflammatory, autoimmune, bone, nervous system, cardiovascular and gastrointestinal disorders
06/18/2009US20090156556 Aminopropanol derivatives
06/17/2009EP1611088B1 Hydroxamates as therapeutic agents
06/17/2009EP1357115B1 Alkanoic acid derivatives, process for their production and use thereof
06/17/2009CN101460469A Chemical compounds
06/16/2009US7547790 Optically active 4,4-di-substituted oxazolidine derivative and method for producing same
06/16/2009US7547711 Heterocyclic inhibitors of kinases
06/11/2009WO2009073713A1 Oximyl macrocyclic derivatives
06/11/2009WO2008152305A3 Novel nitroreductase enzymatic substrates
06/11/2009WO2007083320A3 Conversion of aromatic diazonium salt to aryl hydrazine
06/11/2009US20090149657 Process for the synthesis of intermediates of chloramphenicol or its analogues
06/11/2009US20090149520 Oxazolidinones containing oxindoles as antibacterial agents
06/11/2009US20090149519 Phenylamino-benzoxazole substituted carboxylic acids, method for their production and use thereof as medicaments
06/11/2009US20090149445 Tricyclic steroid hormone nuclear receptor modulators
06/11/2009US20090149425 Malononitrile compound as pesticides
06/10/2009EP2066647A1 Benzoxazoles and oxazolopyridines being useful as janus kinases inhibitors
06/10/2009EP2066632A1 Benzophenone derivatives useful for inhibiting formation of microtubule
06/10/2009CN101454299A Ureide derivative and use thereof for medical purposes
06/10/2009CN100497323C New heterocyclic oxime compounds, preparing process and medical composition thereof
06/09/2009US7544809 Peroxisome proliferator activated receptor agonists
06/09/2009US7544687 (2S)-3-{4-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)-ethoxy]-phenyl}-2-(4-m-tolyl-piperazin-1-yl)-propionic acid; hyperglycemia, dyslipidemia, type II diabetes mellitus; (2S)-2-[4-(4-nitro-benzenesulfonyl)-piperazin-1-yl]-3-{4-[2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)-ethoxy]-phenyl}-propionic acid;
06/04/2009US20090143353 Antifungal bicyclic hetero ring compounds
06/03/2009EP2064195A2 Crystal forms of 2-(3-fluoro-4-hydroxyphenyl)-7-vinyl-1,3-benzoxazol-5-ol and pharmaceutical formulations thereof
06/03/2009EP1786790B1 Oxazole derivatives as histamine h3 receptor agents, preparation and therapeutic uses
06/03/2009CN101445490A Method for preparing optically pure L-goitrin and D-goitrin by adopting liquid chromatogram and chiral separation analytical method
06/02/2009US7541474 Catalyzed process of making C-5-substituted heterocyclic inhibitors of 11β-hydroxy steroid dehydrogenase type 1
06/02/2009US7541472 3-Aryl-3-hydroxy-2-methylenepropionic acid esters as fungicides
06/02/2009US7541356 Compounds for use in weight loss and appetite suppression in humans
05/2009
05/28/2009WO2009067663A1 Alkynes and methods of reacting alkynes with 1,3-dipole-functional compounds
05/28/2009WO2009067618A1 Substituted benzoazole pde4 inhibitors for treating pulmonary and cardiovascular disorders
05/28/2009WO2009067604A1 Substituted benzoazole pde4 inhibitors for treating inflammatory, cardiovascular and cns disorders
05/28/2009WO2009066060A2 4-substituted-6-isopropyl-benzene-1,3-diol compounds and their use
05/28/2009WO2009049180A3 Heteroaryl amides useful as inhibitors of voltage-gated sodium channels
05/28/2009WO2009032294A3 Processes for the preparation of a linezolid intermediate, linezolid hydroxide
05/28/2009US20090137817 Spatially-defined macrocyclic compounds useful for drug discovery
05/28/2009US20090137611 Fungicide N-Cyclopropyl-Sulfonylamide Derivatives
05/28/2009US20090137596 G-protein inhibitor
05/28/2009US20090137585 N-acylsulfonamide apoptosis promoters
05/28/2009US20090137548 1,3-Oxazolidin-2-One Derivatives Useful as Cetp Inhibitors
05/28/2009US20090137453 Composition comprising at least one oxazoline to inhibit migration of langerhans cells, and uses thereof
05/28/2009US20090137420 Methods, compounds and compositions with genotype selective anticancer activity
05/28/2009US20090136448 Antiviral 2-Carboxy-Thiophene Compounds
05/28/2009CA2722591A1 Substituted benzoazole pde4 inhibitors for treating pulmonary and cardiovascular disorders
05/28/2009CA2722586A1 Substituted benzoazole pde4 inhibitors for treating inflammatory, cardiovascular and cns disorders
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