Patents for C07D 263 - Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings (20,978) |
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10/12/2010 | US7812041 such as 2-Morpholin-4-yl-thiazole-4-carboxylic acid (5,6-dimethyl-1H-benzoimidazol-2-yl)-amide, used for the treatment of dementia, amyotrophic lateral sclerosis, stroke, epilepsy, multiple sclerosis, myasthenia gravis, Huntington's, Alzheimer's, Parkinson's, Meniere's and Creutzfeld-Jacob Disease |
10/12/2010 | US7812040 Histamine-3 receptor antagonists |
10/07/2010 | WO2010114971A1 Compounds for treating disorders mediated by metabotropic glutamate receptor 5, and methods of use thereof |
10/07/2010 | WO2010113184A1 Kinetic resolution of (4s)-4-phenyl-3-[5(rs)-(4-fluorophenyl)-5-hydroxypentanoyl] -1,3 oxazolidin 2-one to (5s) isomer via lipase catalyzed enantioselective esterification of the (5r) isomer |
10/07/2010 | WO2010113182A1 Intermediates in the preparation of 1,4-diphenyl azetidinone |
10/07/2010 | WO2010112116A1 Heterocyclic compounds as autotaxin inhibitors |
10/07/2010 | WO2010112092A1 Compounds for treatment of duchenne musculary dystrophy |
10/07/2010 | WO2010112091A1 Compounds for treatment of duchenne muscular dystrophy |
10/07/2010 | US20100256923 Compounds for neutron radiation detectors and systems thereof |
10/07/2010 | US20100256385 Prostaglandin e receptor antagonists |
10/07/2010 | US20100256367 Pharmaceutical Composition For Preventing and Treating Metabolic Bone Diseases Containing Alpha-Arylmethoxyactylate Derivatives |
10/07/2010 | US20100256201 Cell differentiation inducer |
10/07/2010 | US20100256165 Large conductance calcium-activated k channel opener |
10/07/2010 | US20100256131 Carbonyl compounds |
10/07/2010 | US20100256130 Morpholinyl and pyrrolidinyl analogs |
10/07/2010 | US20100256114 Amido Compounds And Their Use As Pharmaceuticals |
10/07/2010 | CA2757722A1 Enzymatic process for the preparation of (s)-5-(4-fluoro-phenyl)-5-hydroxy- 1morpholin-4-yl-pentan-1-one, an intermediate of ezetimibe and further conversion to ezetimibe |
10/07/2010 | CA2757413A1 Heterocyclic compounds as autotaxin inhibitors |
10/07/2010 | CA2756989A1 Compounds for treating disorders mediated by metabotropic glutamate receptor 5, and methods of use thereof |
10/06/2010 | EP2234990A1 Bifeprunox derivatives |
10/06/2010 | CN1942186B Pyrrolidine compounds |
10/06/2010 | CN101855213A Therapeutic compounds |
10/06/2010 | CN101855212A Heterocyclyl substituted fused carbocyles useful in the treatment of conditions such as glaucoma and pain |
10/06/2010 | CN101851235A Heterocyclic compound and light-emitting element, light-emitting device, lighting device, and electronic device using the same |
10/06/2010 | CN101851214A Method for synthesizing polyarylation substituted oxazolidine |
10/06/2010 | CN101851173A Inhibitors of histone deacetylase |
10/06/2010 | CN101849953A Inflammatory cytokine release inhibitor |
10/06/2010 | CN101323589B Preparation of novel compound and montelukast sodium |
10/05/2010 | US7807842 Synthesis of tetracyclines and analogues thereof |
10/05/2010 | US7807841 Spiro-containing compounds and compositions as modulators of steroid hormone nuclear receptors |
10/05/2010 | US7807701 Dibenzylamine compounds and pharmaceutical use thereof |
10/05/2010 | US7807700 Inhibitors of 11-β-hydroxy steroid dehydrogenase type 1 |
10/05/2010 | US7807697 Disorders related to memory and cognition processes, neurological processes, cardiovascular function, and body weight; benzoxazole, benzimidazole, and indole compounds substituted with pyrrole, azepane, piperidine or azetidine e.g. 4-{2-[2-(2-methyl-pyrrolidin-1-yl)-ethyl]-benzooxazol-5-yl}-benzonitrile |
10/05/2010 | US7807692 peroxisome proliferator activated receptor agonists useful in the treatment and control of hyperglycemia that is symptomatic of non-insulin dependent diabetes, as well as dyslipidemia, hyperlipidemia, hypercholesterolemia, hypertriglyceridemia and obesity that are often associated with type II diabetes |
10/05/2010 | US7807669 Peroxisome proliferator-activated receptor type gamma (PPAR- gamma) modulators such as (S)-3-{3'-[(benzoylmethylamino)methyl]biphenyl-4-yl}-2-(1-methyl-3-oxo-3-phenylpropenylamino)propionic acid, suited for use in dermatology, immunology, cardiovascular diseases and/or hyperlipemia |
09/30/2010 | WO2010111303A2 Imaging agents for detecting neurological disorders |
09/30/2010 | WO2010108903A1 2,3-diaryl- or heteroaryl-substituted 1,1,1-trifluoro-2-hydroxypropyl compounds |
09/30/2010 | WO2009157019A3 Process for preparing ezetimibe using novel allyl intermediates |
09/30/2010 | US20100249428 Process for the preparation of propionic acid derivatives |
09/30/2010 | US20100249349 Novel Polymers |
09/30/2010 | US20100249124 2,3-diaryl- or heteroaryl-substituted 1,1,1-trifluoro-2-hydroxypropyl compounds |
09/30/2010 | US20100249123 Novel benzamide derivatives as modulators of the follicle stimulating hormone |
09/30/2010 | US20100248313 Novel optically active, heteroaromatic beta-hydroxy esters and processes for their preparation from beta-keto esters and processes for the preparation of these beta-keto esters |
09/30/2010 | CA2756137A1 Imaging agents for detecting neurological disorders |
09/30/2010 | CA2754176A1 2,3-diaryl- or heteroaryl-substituted 1,1,1-trifluoro-2-hydroxypropyl compounds |
09/29/2010 | CN101845025A Preparation method of 3-alpha,beta-unsaturated acyl-1,3-oxazolidine-2-ketone |
09/28/2010 | US7803954 Mandelic acid derivatives and their use as thrombin inhibitors |
09/28/2010 | US7803950 Method for the production of diarylcycloalkyl derivatives |
09/28/2010 | US7803797 Substituted arylcyclopentenes as therapeutic agents |
09/28/2010 | CA2429267C Cyclohexyl(alkyl)-propanolamines, preparation method and pharmaceutical compositions containing same |
09/28/2010 | CA2383524C Thiazolyl alkynyl compounds and methods of use thereof |
09/23/2010 | WO2010108067A1 Alpha-(n-benzenesulfonamido)cycloalkyl derivatives |
09/23/2010 | US20100240721 desoxyepothilone A and B; Fludelone; anticarcinogenic agents; drug resistance; water solubility for formulability; industrial scale; cytotoxic or growth inhibitory effects on CAG myeloma cells lines; ability to polymerize tubulin; minimum toxicity; stabilizing microtubules |
09/23/2010 | US20100240708 Alpha-(N-Benzenesulfonamido)Cycloalkyl Derivatives |
09/23/2010 | US20100240659 Nitrogen-containing heterocyclic derivative having 11ss-hydroxysteroid dehydrogenase type i inhibitory activity |
09/23/2010 | US20100240657 Chemical compounds |
09/23/2010 | US20100239551 Compounds and compositions as channel activating protease inhibitors |
09/22/2010 | EP1853565B1 Menthane carboxamide derivatives having cooling properties |
09/21/2010 | US7799927 optical recording media with said organic dye as recording layer; high density Disk-Recordable (HD DVD-R) |
09/21/2010 | US7799828 selective estrogen receptor modulators such as 4-[(4-Hydroxyphenyl)(3,3,5,5-tetramethylcyclohexylidene)methyl]benzoic acid, used for the treatment of osteoporosis, obesity, breast cancer, depression, vaginal dryness, rheumatoid arthritis, vasomotor symptoms and urogenital or vulvar vaginal atrophy |
09/21/2010 | CA2590575C 3-phenylpropionic acid derivatives and their use as ppar- gamma receptor ligands |
09/21/2010 | CA2411111C Thiazolyl, oxazolyl and pyrazolyl-substituted heterocycles and their use as pesticides and herbicides |
09/21/2010 | CA2401502C Carboxylic acid derivatives as ip antagonists |
09/16/2010 | WO2010103281A1 Cyclic carbamate compounds useful in energy-curable compositions |
09/16/2010 | WO2010062490A3 Method for making carbamates, ureas and isocyanates |
09/16/2010 | US20100234591 Biaryl heterocyclic compounds and methods of making and using the same |
09/16/2010 | US20100234365 Compounds and compositions as inhibitors of cannabinoid receptor 1 activity |
09/16/2010 | US20100234364 Ccr2 inhibitors and methods of use thereof |
09/16/2010 | DE102009012445A1 New substituted bisoxazoline ligands, useful as chiral catalyst in asymmetric organic synthesis, preferably nitroaldol reaction |
09/16/2010 | CA2754712A1 Cyclic carbamate compounds useful in energy-curable compositions |
09/15/2010 | EP2227453A2 Heteroaryl amides useful as inhibitors of voltage-gated sodium channels |
09/15/2010 | EP1836150B1 Hydroxyphenol derivatives, processes for the preparation thereof, pharmaceutical compositions comprising them, and therapeutic uses thereof |
09/15/2010 | CN101835762A 2-aminooxazole derivatives as TRPV1 antagonists useful for treating pain |
09/15/2010 | CN101835745A Process for production of disulfonic acid compound, asymmetric mannich catalyst, process for production of beta-aminocarbonyl derivative, and novel disulfonate salt |
09/15/2010 | CN101830894A Benzo[d]oxazole compounds and preparation method thereof |
09/15/2010 | CN101830860A Copper ion hapten penicillenic acid mercaptan copper salt and preparation method thereof |
09/15/2010 | CN101830855A Substituted nitrogen-containing benzoheterocycle compounds and preparation method and application thereof |
09/14/2010 | US7795291 Glycine, N-[[3-[[2-(4-chlorophenyl)-5-methyl-4-oxazolyl]methoxy]phenyl]methyl]-N-(methoxycarbonyl)-, used for treating atherosclerosis, dyslipidemia, diabetes, non-insulin dependent diabetes, hyperglycemia, hyperinsulinemia and obesity |
09/14/2010 | US7795251 such as 3-[4-(tert-Butyl-dimethyl-silanyloxy)-phenyl]-7-hydroxy-3,4-dihydro-benzo[e][1,3]oxazin-2-one, inhibitors macrophage migration inhibitory factor isomerase activity; treatment of vision defects, ischemia, inflammatory, autoimmune, bone, nervous system, cardiovascular and gastrointestinal disorders |
09/14/2010 | CA2584311C Synthesis of amino acid, n-carboxyanhydrides |
09/10/2010 | WO2010101247A1 Cyclohexane derivative having npy y5 receptor antagonism |
09/09/2010 | US20100227902 Bis-aryl sulfonamides |
09/09/2010 | US20100227901 Compounds for the treatment of metabolic disorders |
09/09/2010 | US20100226882 Linked diimidazole antivirals |
09/08/2010 | EP2225216A1 Substituted benzoazole pde4 inhibitors for treating pulmonary and cardiovascular disorders |
09/08/2010 | EP2225215A1 Substituted benzoazole pde4 inhibitors for treating inflammatory, cardiovascular and cns disorders |
09/08/2010 | EP2019822B1 A new process for the synthesis of 2-aminoxazole compounds |
09/08/2010 | EP1382336B1 Use of the abc expression promotor pioglitazone for the treatment of arteriosclerosis obliterans |
09/07/2010 | US7790903 Process for production of optically active PPAR-activating compound and intermediate of the same |
09/07/2010 | US7790726 chemokine receptor antagonists such as 6-Chloro-3-{2-[4-(4-chloro-3-methoxy-phenyl)-4-hydroxy-piperidin-1-yl]-2-oxo-ethyl}-3H-benzooxazol-2-one, having in vivo antiinflammatory activity |
09/07/2010 | CA2179935C Novel dipeptide compound or pharmaceutically acceptable salt thereof and medical use thereof |
09/02/2010 | US20100222580 Process For The Preparation Of Onium Alkylsulfates Having A Low Halide Content |
09/02/2010 | US20100222326 New Heterocyclic Derivatives Useful For The Treatment of CNS Disorders |
09/02/2010 | US20100221764 Novel nitroreductase enzymatic substrates |
09/01/2010 | EP2224013A1 Methods for the determination of telomerase activity using click chemistry |
09/01/2010 | EP2222654A1 2-methylthioethyl-substituted heyrrocycles as feed additives |
09/01/2010 | EP1555261B1 Valerolactone compounds and perfume composition |
09/01/2010 | EP1379508B1 N-(aryl)-2-arylethenesulfonamides and therapeutic uses thereof |
09/01/2010 | CN101821238A Compounds which inhibit BETA-SECRETASE activity and methods of use thereof |
09/01/2010 | CN101817799A Cyanoacrylate compound and application thereof in pesticide and medicine |