Patents for C07D 263 - Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings (20,978) |
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12/03/2009 | US20090298824 Organic compounds |
12/02/2009 | EP2125750A2 Cyclic urea and carbamate inhibitors of 11beta-hydroxysteroid dehydrogenase 1 |
12/02/2009 | EP2125711A1 2 -substituted- 3 -phenylpropionic acid derivatives and their use in the treatment of inflammatory bowel disease |
12/02/2009 | CN100564366C Derivatives of 1,3-diones having a herbicidal activity |
12/01/2009 | US7626035 Optically active, heteroaromatic β-hydroxy esters and processes for their preparation from β-keto esters and processes for the preparation of these β-keto esters |
12/01/2009 | US7626033 Compounds for the modulation of PPARγ activity |
12/01/2009 | US7625948 Ester that inhibits MTP in intestines as antilipemic agents for side effect reduction |
12/01/2009 | US7625933 PPAR gamma agonists or partial agonists; type II diabetes, including hyperglycemia, dyslipidemia, hyperlipidemia, hypercholesterolemia, hypertriglyceridemia, and obesity; compounds have a thiazolidinedione or an oxazolidinedione substituent |
12/01/2009 | US7625923 -4-[7-(hydroxy)-tetrahydro-pyrrolo[1,2-c]oxazol-3-ylideneamino]-2-chloro-3-methyl-benzonitrile; non-steroidal, non-toxic; side effect reduction; aging resistance; sarcopenia, osteoporosis and osteopenia, osteoporosis and osteopenia, cancer cachexia, eating disorders (e.g., anorexia) and chemotherapy |
12/01/2009 | US7625917 S-o-(phenylaminocarbonyl)phenyl-substituted, especially with a quaternary onium group; enhanced antiviral activity and better reactivity with zinc finger moieties, particularly, the zinc finger on HIV-1's NCp7 nucleocapsid protein |
12/01/2009 | US7625889 Substituted bis aryl and heteroaryl compounds as selective 5HT2A antagonists |
11/26/2009 | WO2009140932A2 Method of producing (3r,4s)-l-(4-fluorophenyl)-3-[(3s)-3-(4-fluorophenyl)- hydroxypropyl)]-4-(4-hydroxyphenyl)-2-azetidinone |
11/26/2009 | US20090291970 Substituted Aminoethers for the Treatment of Alzheimer's Disease |
11/26/2009 | US20090291923 Trioxane dimers having high anticancer and long-lasting antimalarial activities |
11/26/2009 | DE102008001932A1 Substiuierte Spiroisoxazoline Substiuierte Spiroisoxazoline |
11/25/2009 | EP2123665A2 Inhibitors of interleukin-1Beta converting enzyme |
11/25/2009 | EP2120576A2 Aminoazoline and urea derivatives for combating animal pests |
11/25/2009 | EP2120575A1 Sphingosine-1 -phosphate receptor agonist and antagonist compounds |
11/25/2009 | CN101585817A Method for the effective synthesis of optically active oxazoline-2-ketone derivative |
11/25/2009 | CN100562516C Beta-amyloid protein production/secretion inhibitors |
11/25/2009 | CN100562513C Benzamide derivative or salt thereof |
11/24/2009 | US7622490 Broadspecturm 2-amino-benzoxazole sulfonamide HIV protease inhibitors |
11/24/2009 | US7622479 For example, 2-(1,3-benzodioxol-5-yl)-6-phenyl-1H-imidazo[4,5-b]pyridinetyrosine; kinase-inhibiting activity; use in treatment of breast cancer, prostate cancer, lung cancer or pancreatic carcinoma |
11/24/2009 | CA2433197C Gyrase inhibitors and uses thereof |
11/24/2009 | CA2392050C Pharmaceutical formulations containing zolmitriptan |
11/24/2009 | CA2385882C Tyrosine derivatives |
11/19/2009 | WO2009139373A1 Amide compound |
11/19/2009 | US20090286988 chemical intermediates such as 2-(3-Methoxyphenyl)-4,5-dimethyloxazole 3-oxide, capable of being transformed to halomethyloxazoles smoothly with high yield and great purity |
11/19/2009 | US20090286985 Benzoxazole Derivative, and Light-Emitting Element, Light-Emitting Device, and Electronic Device Using the Same |
11/19/2009 | US20090286841 Certain chemical entities, compositions, and methods |
11/19/2009 | CA2724077A1 Amide compound |
11/18/2009 | EP2118078A2 New salt |
11/18/2009 | EP2117526A2 Inhibitors of diacylglycerol o-acyltransferase type 1 enzyme |
11/18/2009 | EP1789402B1 2-{-3-2-(phenyl)-oxazol-4-ylmethoxymethyl!-cyclohexylmethoxy };-propionic acid derivatives used as ppar ligandes (peroxisome proliferator-activated receptors) for the treatment of hyperlipidaemie and diabetes |
11/18/2009 | EP1660449B1 Aminopropanol derivatives |
11/18/2009 | EP1421071B1 Substituted piperazine and diazepane derivaives as histamine h3 receptor modulators |
11/17/2009 | US7619116 Intermediates for the synthesis of (R)-tamsulosin and of its pharmaceutically acceptable salts and process for their preparation |
11/17/2009 | US7618991 Diaryloxazole carboxamide derivatives for treating a disease selected from appetite disorder, metabolic disorder, gastrointestinal disorder, inflammatory phenomena, immune system disease, psychotic disorder, alcohol dependency and nicotine dependency |
11/17/2009 | US7618981 Imidazopyridinyl-benzamide anti-cancer agents |
11/17/2009 | CA2450801C Drugs that enhance synaptic responses mediated by ampa receptors |
11/17/2009 | CA2387464C Process for preparing n-carboxyanhydrides |
11/12/2009 | WO2009137340A1 Alpha2b and alpha2c agonists |
11/12/2009 | WO2009135526A1 Alpha-mercapto-amides |
11/12/2009 | WO2009063505A3 Process for preparation of (s) (n-[[3-[3-fluoro-4-(4-morpholinyl) hen l -2-oxo-5-oxazolidin l methyl]acetamide |
11/12/2009 | US20090281309 Method for producing 2-oxazoline analogue or 1,3-oxazine analogue |
11/12/2009 | US20090281279 Rigidized trimethine cyanine dyes |
11/12/2009 | US20090281155 Dimeric Small Molecule Potentiators of Apoptosis |
11/12/2009 | US20090281131 Diebenzofuran derivatives as inhibitors of pde-4 and pde-10 |
11/12/2009 | CA2723751A1 Alpha2b and alpha2c agonists |
11/12/2009 | CA2723550A1 Alpha-mercapto-amides |
11/11/2009 | EP2116535A1 Glucokinase-activating substance |
11/11/2009 | EP2116533A1 Glucokinase activator |
11/11/2009 | EP1874745B1 New 3-phenylpropionic acid derivatives and their use as ppar- gamma receptor ligands |
11/11/2009 | EP1477186B1 Antipruritics |
11/11/2009 | CN100558814C 树脂组合物 Resin composition |
11/11/2009 | CN100558712C Therapeutic molecules and methods-1 |
11/11/2009 | CN100558428C Calcitonin gene related peptide receptor antagonists |
11/11/2009 | CN100558356C Method of using benzenesulphoamides that are cyclooxygenase-2-inhibitors in the treatment and prevention of neoplasia |
11/05/2009 | WO2009132740A2 Reactive ionic liquids |
11/05/2009 | US20090275627 Alpha2b and alpha2c agonists |
11/05/2009 | US20090275598 Conformationally constrained 3-(4-hydroxy-phenyl)-substituted-propanoic acids useful for treating metabolic disorders |
11/05/2009 | US20090274637 Depigmenting or Brigthening Cosmetic Composition at Least One Oxazolin as an Active Ingredient |
11/05/2009 | US20090274632 Identification of human T2R receptors that respond to bitter compounds that elicit the bitter taste in compositions, and the use thereof in assays to identify compounds that inhibit (block) bitter taste in composition and use thereof |
11/04/2009 | EP2113031A1 Optically active, heteroaromatic beta-hydroxy esters, processes for their preparation from beta-keto esters and processes for the preparation of these beta-keto esters |
11/04/2009 | EP1651642B1 Pna monomer and precursor |
11/04/2009 | EP1473286B1 Process for producing biaryl compound |
11/04/2009 | EP1444739B1 Light emitting device and compounds for use therein |
11/04/2009 | EP1253152B1 Method of converting functional group through halogen-metal exchange reaction |
11/03/2009 | US7612210 Treating (4S or 4R)-4-benzyl-3-[(methoxyphenyl)acetyl]-1,3-oxazolidin-2-one with an aprotic amine base and titanium tetrachloride in chlorinated solvent under conditions which permit formation of corresponding anion, and mixing anion with titanium tetrachloride and cyclohexanone to permit aldol reaction |
11/03/2009 | US7612209 Pseudo proline dipeptides |
11/03/2009 | US7612105 3-arylphenyl sulfide derivative and insecticide and miticide |
11/03/2009 | CA2384925C Process for the preparation of oxazole derivatives |
10/29/2009 | WO2009132119A2 Substituted oxazolidinones |
10/29/2009 | WO2009129953A1 2-(benzylsulfonyl)-oxazole derivatives, chiral 2- (benzylsulfinyl) -oxazole derivatives and 2-(benzylsulfanyl)-oxazole derivatives, methods for the production thereof, and use thereof as herbicides and plant growth regulators |
10/29/2009 | WO2009035951A3 Soluble epoxide hydrolase inhibitors |
10/29/2009 | US20090270469 Substituted oxazolidinones |
10/29/2009 | US20090270468 Preparation and use of aryl alkyl acid derivatives for the treatment of obesity |
10/29/2009 | US20090270365 such as N-(2,4-dimethyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)-2-(piperidin-1-ylmethyl)biphenyl-4-carboxamide, having vanilloid receptor 1 antagonistic activity, used as analgesics |
10/29/2009 | CA2722340A1 Small-molecule inhibitors of the androgen receptor |
10/29/2009 | CA2722214A1 2-(benzylsulfonyl)-oxazole derivatives, chiral 2- (benzylsulfinyl) -oxazole derivatives and 2-(benzylsulfanyl)-oxazole derivatives, methods for the production thereof, and use thereof as herbicides and plant growth regulators |
10/28/2009 | EP2112143A1 2-(benzylsulfonyl)-oxazol-derivatives, chiral 2-(benzylsulfinyl]-oxazol derivatives, 2-(benzylsulfanyl-oxazol) derivatives, process for their preparation, as well as their use as herbicide and plant growth regulators |
10/28/2009 | CN101565393A 3-(substituted bisulfonyl fluromethane)-1-propylene compound, synthetic method and applications thereof |
10/28/2009 | CN100554254C Oxazolidine compound for synthesizing taxone pharmaceutical side-chain and preparation method thereof |
10/27/2009 | US7608721 2-{4-[Ethyl-(thiazol-4-ylmethyl)-amino]-phenyl}-1,1,1,3,3,3-hexafluoro-propan-2-ol; liver-X-receptor modulators; anticholesterol agents; antiinflammatory agents; atherosclerosis; dyslipidemia; antidiabetic agents; alzheimer's disease; sepsis; skin disorders; cognition modulators |
10/27/2009 | US7608632 Sulfonamide inhibitors of aspartyl protease |
10/27/2009 | US7608631 1-(4-{3-[2,6-Dichloro-4-(3,3-dichloro-allyloxy)-phenoxy]-propoxy}-phenyl)-1H-pyrrole, for example; protecting soybean plants against pests such as caterpillars |
10/27/2009 | US7608619 [{4-[(4-benzyl-5-pyrrolidin-1-yl-oxazol-2-yl)-piperidin-1-yl-methyl]-cyclohexyl}-(4-fluorophenyl)-methyl]-dimethylamine; depression, urinary incontinence, diarrhoea, pruritus, alcohol and drug misuse, drug dependency, acute pain, neuropathic pain or chronic pain and anxiety |
10/27/2009 | US7608564 Herbicide; in crops such as wheat, rice, maize, soybeans and cotton they act against broad-leaved weeds and grass weeds without damaging the crop plants; compounds are based on 3-(5,5-disubstituted 2-isoxazolin-3-yl)benzoic acid, esters, thioesters and pyrazolyl ketones thereof |
10/27/2009 | CA2466724C Benzamide and heteroarylamide as p2x7 receptor antagonists |
10/27/2009 | CA2318976C Herbicidally active 3-hydroxy-4-aryl-5-oxopyrazoline derivatives |
10/22/2009 | WO2009129267A2 Small molecule inhibitors of the pleckstrin homology domain and methods for using same |
10/22/2009 | WO2009129097A1 Nitrated hydrocarbons, derivatives, and processes for their manufacture |
10/22/2009 | WO2009127338A1 Oxo-heterocyclic substituted carboxylic acid derivates and the use thereof |
10/22/2009 | US20090264487 Hemiasterlin analogs |
10/22/2009 | US20090264424 Vanilloid receptor ligands and their use in treatments |
10/22/2009 | US20090264405 Cetp Inhibitors |
10/22/2009 | CA2721371A1 Small molecule inhibitors of the pleckstrin homology domain and methods for using same |
10/22/2009 | CA2720646A1 Nitrated hydrocarbons, derivatives, and processes for their manufacture |
10/21/2009 | EP2109602A2 Tetracycline derivatives for the treatment of bacterial, viral and parasitic infections |
10/21/2009 | CN101560193A Alpha-polyhalide acetyl piperazinyl oxazolidone compound and antibacterium application thereof |