Patents
Patents for C07D 241 - Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings (18,673)
02/2005
02/02/2005EP1501514A2 Protein kinase modulators and methods of use
02/02/2005EP1501513A2 Compositions and methods for combating lower urinary tract dysfunctions with delta opioid receptor agonists
02/02/2005EP1501508A1 Inhibitors of histone deacetylase
02/02/2005EP1286955B1 Aryl and heteroarylcyclopropyl oxime ethers and their use as fungicides
02/02/2005EP1184376B1 Novel heterocyclic carboxamide derivatives
02/02/2005CN1575283A Piperazine derivatives with CCRI receptor antagonist activity
02/02/2005CN1575275A Novel alpha-oxygenated or alpha-thiolated carboxylic acid penethylamide derivatives
02/02/2005CN1573599A Novel charge transport materials having heteroaromatic hydrazone groups
02/02/2005CN1187342C Substituted 1-aminoalkyl-lactams compound and their use as muscarinic receptor antagonists
02/02/2005CN1187341C N-hydroxy amidino compound and its preparation method
02/01/2005US6849739 N-heterocyclic derivatives as NOS inhibitors
02/01/2005US6849732 Metalloproteinase inhibitors, pharmaceutical compositions containing them and their pharmaceutical uses, and methods and intermediates useful for their preparation
02/01/2005US6849660 Antimicrobial biaryl compounds
02/01/2005US6849632 Heteroaryl alkyl piperazine derivatives
02/01/2005US6849630 Cyclized amino acid derivatives
01/2005
01/27/2005WO2004064972A3 Capture compounds, collections thereof and methods for analyzing the proteome and complex compositions
01/27/2005US20050020604 5-HT receptor ligands and uses thereof
01/27/2005US20050020601 Novel pyrazinones as CRF1 receptor antagonists
01/27/2005US20050020578 Oxidoreductase enzyme inhibitors such as (R)-1-[4-(2-methyl-4-phenyl-5,8-dihydro-6H-pyrido[3,4-d]pyrimidin-7-yl)-pyrimidin-2-yl-ethanol, used as antidiabetic agents
01/27/2005US20050020576 Opioid antagonist; analgesics; antiinflammatory agents; side effect reduction
01/27/2005US20050020450 Novel alpha-oxygenated or alpha-thiolated carboxylic acid penethylamide derivatives
01/26/2005EP1500653A1 Substituted arylpyrazines
01/26/2005EP1499599A1 Substituted pyrazine derivatives
01/26/2005EP1499578A2 Prime ring substituted thyroid receptor antagonists for the treatment of cardiac and metabolic disorders
01/26/2005EP1499319A1 Bicyclo 4.4.0 antiviral derivatives
01/26/2005EP0983267B1 Amidoaromatic ring sulfonamide hydroxamic acid compounds
01/26/2005CN1186332C New thryoid receptor ligands and process II
01/26/2005CN1186329C Process for catalytically synthesizing alkyl pyrazine compounds using granular solid super strong acid
01/25/2005US6846829 N-heterocyclic derivatives as NOS inhibitors
01/25/2005US6846825 Antibacterial agents
01/25/2005US6846815 Heterocyclic imines such as 2-anilino-6-quinoxalinol, used to suppress cell proliferation, differentiation, chemotaxis and/or activation; prophylaxis of restinosis; anticarcinogenic agents
01/20/2005WO2005005606A2 17-acetamido-4-azasteroid derivatives as androgen receptor modulators
01/20/2005WO2005005380A2 17-acetamido-4-azasteroid derivatives as androgen receptor modulators
01/20/2005WO2005005374A1 Aspartyl protease inhibitors
01/20/2005WO2005004802A2 N-alkyl phenylcarboxamide beta-secretase inhibitors for the treatment of alzheimer's disease
01/20/2005US20050014749 Piperazine derivatives and methods of use
01/20/2005US20050014740 E.g. 4-[2-(4-Methylphenoxy)- or 4-[2-(4-Methylphenylsulfanyl)-phenyl]-3,6-dihydro-2H-pyridine or piperazine or hydrochloride or oxalate; treating depression, anxiety, and obsessive compulsive disorders
01/20/2005US20050014724 Immunosuppressant compounds and compositions
01/20/2005CA2530182A1 17-acetamido-4-azasteroid derivatives as androgen receptor modulators
01/20/2005CA2530025A1 17-acetamido-4-azasteroid derivatives as androgen receptor modulators
01/20/2005CA2529994A1 N-alkyl phenylcarboxamide beta-secretase inhibitors for the treatment of alzheimer's disease
01/20/2005CA2529739A1 Aspartyl protease inhibitors
01/19/2005EP1498417A1 Heterocyclic amide derivatives
01/19/2005EP1498411A1 Diketohydrazine derivative compounds and drugs containing the compounds as the active ingredient
01/19/2005EP1497273A2 Hydroxamic acid derivatives
01/19/2005EP1497268A2 Nitric oxide donors, compositions and methods of use
01/19/2005EP1496906A1 Inhibitors of akt activity
01/19/2005EP1181271B1 Naphthalene ureas as glucose uptake enhancers
01/19/2005CN1568187A 2H-2, 3-dinitrogen phenodiazine-1-ketone and using method thereof
01/19/2005CN1568185A Compounds effecting glucokinase
01/19/2005CN1566096A Prostaglandin agonists and their use to treat bonedisorders
01/18/2005US6844404 Catalyst compositions for the polymerization of olefins
01/13/2005WO2005003102A1 Methods of preparation of dehydro-diketopiperazines in liquid phase or of solid supported phase
01/13/2005WO2005003101A2 Pyrazine and pyridine derivatives as rho kinase inhibitors
01/13/2005WO2005003098A1 Heterocyclically substituted pentanol derivatives, method for the production thereof, and use thereof as anti-inflammatory agents
01/13/2005US20050010031 2-(S)-{3-(S)-allyl-4-[2-(R)-amino-3-(4-fluorophenyl)propionyl]-2-oxo-piperazin-1-yl}-N-methyl-3-naphthalen-2-yl-propionamide for example; various diseases and disorders including controlling appetite and treating diabetes
01/13/2005US20050009844 Inhibitors of p38
01/13/2005US20050009786 Immunosuppressant compounds and compositions
01/13/2005CA2531060A1 Heterocyclically-substitued pentanol derivatives, process for their production and their use as anti-inflammatory agents
01/13/2005CA2530389A1 Pyrazine and pyridine derivatives as rho kinase inhibitors
01/12/2005EP1496060A1 Antitumoral analogs of ET-743
01/12/2005EP1496057A1 Novel crystal of quinoxalinedione derivative anhydride
01/12/2005EP1495002A1 Benzamide derivatives useful as histone deacetylase inhibitors
01/12/2005EP1495000A1 Alpha, omega-dicarboximide derivatives as useful uro-selective a1a adrenoceptor blockers
01/12/2005EP1494997A1 Substituted aryl amides
01/12/2005EP1494676A1 Fused quinoxaline derivatives as inhibitors of akt activity
01/12/2005EP1494674A1 Carboximide derivatives as useful uro-selective alpha-1a adrenoceptor blockers
01/12/2005EP1494672A1 Aminocarbonyl substituted pyridines, pyridazines, pyrimidines, pyrazines and triazines having antiangiogenic activity
01/12/2005EP0991628B1 QUINOLINE AND QUINOXALINE COMPOUNDS WHICH INHIBIT PLATELET-DERIVED GROWTH FACTOR AND/OR P56lck TYROSINE KINASES
01/12/2005CN1184209C Chuanxiong alkoxide derivative and its preparation and medicinal composition containing it and use thereof
01/11/2005US6841676 Stereospecific catalysts for polymerization of addition polymerizable monomers
01/11/2005US6841674 N-heterocyclic derivatives as NOS inhibitors
01/11/2005US6841673 Enzyme inhibitors; antiinflammatory agents; rheumatic diseases; antidiabetic agents
01/06/2005US20050004230 Retroviral protease inhibitors
01/06/2005US20050004212 Antitumor/cancer activity; topoisomerase I inhibitors
01/06/2005US20050004211 Inhibiting topoisomerase I; blocking S or G2/M phase of tumor and/or cancer cells
01/06/2005US20050004140 Such as n-(4-fluorobenzyl)-6-(4-methyl-1H-imidazol-1-yl)pyrazin-2-amine; protein kinase associated disease states
01/06/2005US20050004133 Inhibiting ligand gated ion channel vanilloid receptor (VR1); pain relievers; such as 6-(3,4-dichloro-phenyl)-N-(2-oxo-2,3-dihydro-1H-benzoimidazol-5-yl)-nicotinamide
01/06/2005US20050004130 New metabotropic glutamate receptor compounds
01/05/2005EP1493733A2 Fungicidal heterocyclic aromatic amides, their compositions and methods of use
01/05/2005EP1492792A2 3-heteroaryl-3,5-dihydro-4-oxo-4h-pyridazino 4,5-b]indole-1-acetamide derivatives, preparation and use thereof in medicaments
01/05/2005EP1492757A1 (2-((2-alkoxy)-phenyl)-cyclopent-1-enyl) aromatic carbo- and heterocyclic carboxylic acid and derivatives
01/05/2005EP1492534A1 Carbamic acid compounds comprising a piperazine linkage as hdac inhibitors
01/05/2005CN1561336A Phenyl-piperazine derivatives as serotonin reuptake inhibitors
01/05/2005CN1183120C Method for producing high melting point crystals of phenoxypropionic acid derivative
01/05/2005CN1183119C Arylpiperzines as metalloproteinase inhibiting agents (MMP) and their use
01/05/2005CN1183113C Tri-aryl acid derivatives as PPAR receptor ligands
01/04/2005US6838483 Sulfonated amino acid derivatives and metalloproteinase inhibitors containing the same
12/2004
12/30/2004US20040266782 Cyclic amine derivatives-CCR-3 receptor antagonists
12/30/2004US20040266774 Amide compounds
12/29/2004WO2004113311A1 Amorphous und crystal forms of (5-chloro-2-{2-
12/29/2004WO2004078714A3 Processes for preparing imidazoquinoxalinones, heterocyclic-substituted imidazopyrazinones, imidazouinoxalines and heterocyclic-substituted imidazopyrazines
12/29/2004WO2004002940A8 Inhibitors of hcv ns5b polymerase
12/29/2004EP1491190A1 Decomposition inhibitor for extracellular matrix of cartilage
12/29/2004EP1490346A2 Stereoselective alkylation of chiral 2-methyl-4-protected piperazines
12/29/2004EP1490066A1 Use of ranolazine for the preparation of a medicament for the treatment of arrhythmias
12/29/2004EP1490062A1 Glucocorticoid mimetics, methods of making them, pharmaceutical compositions, and uses thereof
12/29/2004EP0994834A4 Ligated platinum group metal catalyst complex and improved process for catalytically converting alkanes to esters and derivatives thereof
12/29/2004CA2529949A1 Antiviral compounds and methods
12/28/2004US6835495 Pentacyclic anion salts or tetrazapentalene derivatives and their uses as ionic conducting materials
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