Patents
Patents for C07D 241 - Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings (18,673)
03/2004
03/03/2004EP0929217B1 Sordarin derivatives
03/03/2004EP0853617B1 Novel 2,3-dioxo-1,2,3,4-tetrahydro-quinoyxalinyl derivatives
03/03/2004CN1479727A Piperazinylpyrazine compounds as agonist or antagonist of 5-hydroxytryptamine 5HT-2 receptor
03/03/2004CN1479715A Amide for inhibition of IL-8-induced chemiotaxis of neutrophil leucocytes
03/03/2004CN1140516C Quinoline and quinoxaline compounds which inhibits platelet-derived growth factor on/or p56lck tyrosine kinases
03/02/2004US6699893 Glucocorticoid receptor modulators
03/02/2004US6699891 Npyy5 antagonists
03/02/2004US6699890 Phosphodiesterase 4 inhibitors
03/02/2004US6699856 Pyrazinones, compositions containing such compounds and methods of use
02/2004
02/28/2004WO2004092177A1 Triazolopyrazines and methods of making and using the same
02/26/2004WO2004003599A3 Anisotropic films based on 1,8-naphthoylene-1',2'-benzimidazole sulfonates and lyotropic liquid crystal systems and methods for making
02/26/2004WO2003101444A8 Diarylurea compounds and derivatives as chk-1 inhibitors for the treatment of cancer
02/26/2004WO2002101003A3 Stereoselective preparation of cyclic l-amino acids
02/26/2004US20040039201 Functionalized compositions for improved immobilization
02/26/2004US20040038969 Substituted aminopyrimidines and aminopyridazines; analgesics particularly for migraines, neuropathic pain and associated hyperalgesia and allodynia; antiinflammatory agents; treating asthma, gastrointestinal disorders, etc.
02/26/2004US20040038858 Carboxamide derivatives and their use in the treatment of thromboembolic diseases and tumours
02/26/2004US20040037022 Aminoalcohol derivatives
02/25/2004EP1391952A2 Salts of pentacyclic or tetrapentaline derived anions, and their uses as ionic conductive materials
02/25/2004EP1391450A1 N-(heterocycle-methyl)alkylamine derivative, process for producing the same, and bactericide
02/25/2004EP1390361A2 Melanocortin receptor ligands
02/25/2004EP1390034A1 N-substituted nonaryl-heterocyclo amidyl nmda/nr2b antagonists
02/25/2004CN1478077A Benzamide compounds as APOB secretion inhibitors
02/25/2004CN1478076A MCH antagonists and their use in treatment of obesity
02/24/2004US6696434 Quinoline and quinoxaline compounds which inhibit platelet-derived growth factor and/or p56lck tyrosine kinases
02/24/2004CA2302727C Process for preparing cyclic thioamides
02/19/2004WO2004014892A1 Monocyclic derivatives as matrix metalloproteinase inhibitors
02/19/2004WO2004014876A1 Urea derivatives as kinase inhibitors
02/19/2004WO2004014875A1 Crystal forms of quinoxaline-2-carboxylic acid [4-carbamoyl-1-(3-fluorobenzyl)-2,7-dihydroxy-7-methyl-octyl]-amide
02/19/2004WO2004014871A1 Vanilloid receptor ligands and their use in treatments
02/19/2004WO2004014842A1 Acylated arylcycloalkylamines and their use as pharmaceuticals
02/19/2004US20040034225 Aryl-substituted n, n-heterocyclic compounds, method for their preparationand their use in therapeutics and diagnostics
02/19/2004US20040034104 2,2-Diphenylbutanamide derivatives and medicines containing the same
02/19/2004US20040034103 Cdc25 photophatase inhibitors
02/19/2004US20040034076 Such as methyl-3-azido-2-((4,6-dimethoxy-2-pyrimidinyl)oxy) 3,3-diphenylpropionate; for treatment of high blood pressure
02/19/2004US20040034048 Didepsipeptide-based endoparasiticides, new didepsipeptides and process for preparing the same
02/19/2004US20040034038 E.g., N-(2-(benzyl(2-hydroxyethyl)amino)-5-bromophenyl)-N'-(5-cyano-2- pyrazinyl)urea; anticarcinoma, -tumor, -proliferative and -metastatic agents; angiogenesis inhibition
02/19/2004US20040034034 Novel piperazine derivatives
02/19/2004US20040034027 E.g.N-(carbamimidoylphenyl)-N'-((1-(4-nitrophenyl)ethyl-2-phenyl -malonamide formate; reversible enzyme inhibitors of blood factor VIIa; a strong antithrombotic to treat thrombo-embolic diseases and restenoses; cardiovascular disorders
02/19/2004US20040034025 Having a high residual activity, greater activity at lower application rates, curative activity, and a broader spectrum of efficacy; heterocyclic aromatic amides having a hydroxy group adjacent to the amide functionality
02/19/2004US20040034018 2-amino-trihydroindole or tetrahydronapthalene-2-yl derivatives, useful for disease state associated with smooth muscle disorders, such as gastrointestinal and urogenital disorders
02/19/2004CA2494848A1 Urea derivatives as kinase inhibitors
02/19/2004CA2494776A1 Crystal forms of quinoxaline-2-carboxylic acid ¬4-carbamoyl-1-(3-fluorobenzyl)-2,7-dihydroxy-7-methyl-octyl|-amide
02/19/2004CA2494014A1 Monocyclic derivatives as matrix metalloproteinase inhibitors
02/18/2004EP1389611A1 20-hydroxyeicosatetraenoic acid production inhibitors
02/18/2004EP1389204A1 Novel sulfonamide derivatives, intermediate thereof, its preparation methods, and pharmaceutical composition comprising the same
02/18/2004EP1389194A2 Inhibitors of bace
02/18/2004EP1389111A1 COMPOSITION FOR INHIBITING HIV ACTIVITY EXTRACTED FROM i PAECILOMYCES SP. /i (TOCHU-KASO) J300
02/17/2004US6693123 (4-(3-pyridylaminomethylene)-2-phenylbenzoyl)-n -methylmethionine, methyl ester for example; restenosis, hyperplasia
02/17/2004US6693112 Compounds for enhancing chemotherapy
02/12/2004WO2004013084A1 Sphingosinoids and external preparations for skin containing the same
02/12/2004WO2003049702A3 Vanilloid receptor ligands and their use in treatments
02/12/2004US20040029928 Tumor necrosis factor alpha-converting enzyme inhibitor; rheumatic diseases; antiarthritic agents; infections; autoimmune diseases; antidiabetic agents
02/12/2004US20040029889 Bone disorders; antiarrhythmia agents; cardiovascular disorders
02/12/2004US20040029881 Herbicides, and chemical intermediates thereof
02/12/2004US20040029814 Cathepins inhibitor; antiinflammatory agents; antiarthritic agents
02/12/2004US20040029720 Supported group 8-10 transition metal olefin polymerization catalysts
02/11/2004EP1388535A1 Acylated arylcycloalkylamines and their use as pharmaceuticals
02/11/2004CN1474689A CDC25 phosphatase inhibitors
02/11/2004CN1473818A Process for catalytically synthesizing alkyl pyrazine compounds using granular solid super strong acid
02/11/2004CN1137886C Novel 2,3-dioxo-1,2,3,4-tetrahydro-quinoyxalinyl derivatives
02/10/2004US6689886 Treatment of inflammation and other immune disorders
02/05/2004US20040024180 By heating suitable dipeptides in organic solvent whilst removing water by distillation; use as chiral catalysts, e.g. for the production of chiral cyanohydrines
02/05/2004US20040024059 Novel pleuromutilin derivatives
02/05/2004US20040023999 Glucocorticoid mimetics, methods of making them, pharmaceutical compositions, and uses thereof
02/05/2004US20040023986 Treating epilepsy, neuropathic pain, and tissue damage form ischemic events; antihypoxic agents
02/05/2004US20040023060 Structure including at least three planar moieties, which are linearly configured such that one planar moiety is located between two neighboring planar moieties and shares an atom with each of the moieties
02/05/2004US20040022856 Carriers for drug delivery
02/04/2004EP1385818A2 Biurethane derivatives
02/04/2004EP0813525B9 Benzamidine derivatives their preparation and their use as anti-coagulants
02/04/2004CN1473158A Radiopharmaceuticals for diagnosing alzheimer's disease
02/04/2004CN1137101C Ammoxidation process of preparing 2-cyano pyrazine
02/03/2004US6686356 Pyridoquinoxaline antivirals
01/2004
01/29/2004WO2004009586A1 Novel piperazinyl-pyrazinone derivatives for the treatment of 5-ht2a receptor-related disorders
01/29/2004WO2004009552A1 Phosphodiesterase 4 inhibitors, including n-substituted aniline and diphenylamine analogs
01/29/2004WO2004009017A2 Modulators of the glucocorticoid receptor and method
01/29/2004WO2003053971A8 Pyridoquinoxaline antivirals
01/29/2004US20040019217 Dihydoxyhexanoic acid derivatives, their intermediates, and methods of making
01/29/2004US20040019056 Anititumoral analogs of et-743
01/29/2004DE10232525A1 Neue Anthracen-Derivate und deren Verwendung als Arzneimittel Novel anthracene derivatives and their use as medicaments
01/29/2004CA2492907A1 Phosphodiesterase 4 inhibitors, including n-substituted aniline and diphenylamine analogs
01/28/2004EP1384716A1 Preparation of ethenylpyrazines
01/28/2004CN1471534A 桥(连)哌嗪衍生物 Bridge (even) piperazine derivatives
01/28/2004CN1136201C Pharmacologucally active enantiomers and method for their preparation
01/28/2004CN1136200C Pharmacollogically active enantiomers and method for their preparation
01/28/2004CN1136193C Imide derivatives ar Salts thereof
01/27/2004US6683211 Fungicides for crops
01/27/2004US6683184 Piperazine derivatives and process for the preparation thereof
01/27/2004US6683074 Cyclic amine derivatives-CCR-3 receptor antagonists
01/27/2004CA2214720C Arylsulfonylamino hydroxamic acid derivatives
01/22/2004WO2004007472A1 Ccr4 antagonist and medicinal use thereof
01/22/2004WO2004007470A1 Novel anthracene derivatives and the use thereof as a medicament
01/22/2004US20040014968 Such as 2-(3-chloro-phenyl)-3-cyclopentyl-N-thiazol-2-yl-propionamide which increases insulin secretion in treatment of type II diabetes
01/22/2004US20040014796 Antiinflammatory agents; rheumatic diseases; antitumor agents
01/22/2004US20040014774 Aryl and heteroaryl quinazoline compounds which inhibit CSF-1R receptor tyrosine kinase
01/22/2004US20040014767 Central nervous system diosrders; antidepressants, anxiolytic agents, anxiolytic agents
01/22/2004US20040014765 Chk-1 inhibitors
01/22/2004US20040014745 Amide compounds
01/22/2004US20040014744 Anticancer, antitumor agents
01/21/2004EP1381590A1 3,4-di-substituted cyclobutene-1,2-diones as cxc-chemokine receptor ligands
01/21/2004EP1305028A4 Antimicrobial biaryl compounds