Patents
Patents for C07D 241 - Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings (18,673)
05/2005
05/12/2005US20050101779 Antagonistic activity to alpha 4 integrin; antiinflammatory agents treating asthma, rheumatoid arthritis, inflammatory bowel diseases, lupus, diabetes; 1-[[(cyclohexyloxy)carbonyl]oxy]ethyl(2S)-2-[(2,6-dichlorobenzoyl)amino]-3-[4-[1-methyl-2,4-dioxo-1,4-tetrahydro-3-(2H)quinazolinyl]phenyl]Propionate
05/12/2005US20050101644 Benzylether amine compounds useful as CCR-5 antagonists
05/12/2005US20050100787 High density; stability; n-heterocyclic polymer or oligomer
05/12/2005CA2540843A1 Phenyl carboxamide and sulfonamide derivatives for use as 11-beta-hydroxysteroid dehydrogenase
05/11/2005EP1529530A1 Compounds affecting glucokinase
05/11/2005EP1529031A1 Acylated arylcycloalkylamines and their use as pharmaceuticals
05/11/2005EP1033362B1 Crystals of [s,s]-ethylenediamine-n,n'-disuccinic acid with high bulk density and method of obtaining the same
05/06/2005WO2005040137A1 Aminoalkyl-pyrazinones and -pyridones as thrombin inhibitors
05/05/2005US20050096468 Inhibitors of histone deacetylase
05/05/2005US20050096357 Antibiotics; therapy for infections which is caused by drug-resistant Streptococcus, or bacteria infections
05/05/2005US20050096337 for example (2-(3-methoxy-propyl)-4-{methyl-[2-methyl-6-(4-trifluoromethyl-phenyl)-pyridin-3-ylmethyl]-amino}-phenoxy)-acetic acid; Peroxisome Proliferator Activated Receptor (PPAR) activators; treating diabetes, dyslipidemia, cardiovascular disorders, polycystic ovary syndrome, proliferative disorders
05/05/2005US20050096312 Antiserotonine agents; antidepressants; eating disorders; anxiolytic agents; sleep disorders; gastrointestinal disorders; cardiovascular disorders; muscular disorders; endocrine system diseases; muscular disorders; psychological disorders
05/04/2005EP0886637B9 Inhibitors of microsomal triglyceride transfer protein and method
05/04/2005CN1612763A Composition and antiviral activity of substituted azaindoleoxoacetic piperazine derivatives
05/03/2005US6887905 Treatment of depression or generalized anxiety disorder
05/03/2005US6887875 2,5-diarypyrimidine compounds
05/03/2005US6887871 Use of phenylheteroakylamine derivatives
05/03/2005US6887865 N-heterocyclic derivatives as NOS inhibitors
05/03/2005US6887863 Such as (2RS,3R)-3-amino-4-cyclohexyl-2-hydroxy-N-phenoxybutanamide; methionine aminopeptidase type 2 inhibitors
05/03/2005CA2320388C Novel dihydroxyhexanoic acid derivatives
04/2005
04/28/2005WO2005037826A1 Substituted cyclic hydroxamates as inhibitors of matrix metalloproteinases
04/28/2005WO2005037809A1 Substituted aryl cycloalkanol derivatives and methods of their use
04/28/2005WO2005037807A1 Arylalkyl- and cycloalkylalkyl-piperazine derivatives and methods of their use
04/28/2005WO2005037803A1 Organic compounds
04/28/2005WO2005037793A1 Cyclopentene compounds
04/28/2005WO2005037786A1 Heterocyclyl compounds
04/28/2005WO2005037257A2 Novel alanyl-amino peptidase inhibitors for functionally influencing different cells and treating immunological, inflammatory, neuronal, and other diseases
04/28/2005WO2004014842A8 Acylated arylcycloalkylamines and their use as pharmaceuticals
04/28/2005US20050090669 Aminoalcohol derivatives as beta-3 adrenergic receptor agonists
04/28/2005US20050090630 Supported group 8-10 transition metal olefin polymerization catalysts
04/28/2005US20050090559 Heterocyclically-substituted pentanol derivatives, process for their production and their use as anti-inflammatory agents
04/28/2005US20050090503 5-HT receptor ligands and uses thereof
04/28/2005CA2549733A1 Fused-aryl and heteroaryl derivatives and methods of their use
04/28/2005CA2542723A1 Novel alanyl-amino peptidase inhibitors for functionally influencing different cells and treating immunological, inflammatory, neuronal, and other diseases
04/28/2005CA2541509A1 Substituted cyclic hydroxamates as inhibitors of matrix metalloproteinases
04/28/2005CA2540207A1 Substituted aryl cycloalkanol derivatives and methods of their use
04/28/2005CA2539763A1 Phenylpiperazine cycloalkanol derivatives and methods of their use
04/28/2005CA2539761A1 Arylalkyl- and cycloalkylalkyl-piperazine derivatives and methods of their use
04/27/2005EP1526131A1 Aminoalkyl-pyrazinones and -pyridones as thrombin inhibitors
04/27/2005EP1526127A2 Process for production of S,S-ethylenediamine-N,N'-disuccinic acid iron alkali salt
04/27/2005EP1525186A1 Inhibitors of hcv ns5b polymerase
04/27/2005EP1525183A1 Inhibitors of hcv ns5b polymerase
04/27/2005EP1025097B1 1-(2-naphthyl) and 1-(2-azanaphthyl)-4-(1-phenylmethyl)piperazines being dopamine d 4? receptor subtype ligands
04/27/2005EP0838453B1 Heterocyclic carboxylic acid derivatives and drugs containing the same
04/27/2005CN1610671A Quinoline compounds with 5-HT-antagonistic properties for therapy
04/27/2005CN1610669A Heteroaryl-substituted aminocyclohexane derivatives
04/27/2005CN1198839C Novel dipeptide amidines as thrombin inhibitors
04/27/2005CN1198806C Oxodiethylenediamine derivative and light stabilized composition
04/26/2005US6884821 Alkyloxypropanoic acid derivative containing sulfonamide or amide group are useful as insulin resistance agent
04/26/2005US6884808 Acids and salts such as 4-(4-(2-(2-(5,6,7,8-Tetrahydro-5,5,8, 8-tetramethylquinoxalyl))pyrrolyl))benzoic acid, used retinoic acid receptor agonists for the prophylaxis of cancer, skin disorders, asthma, alopecia or autoimmune diseases
04/26/2005US6884477 Electroluminescence device using liquid crystal compound
04/21/2005WO2005034857A2 Methods and compositions comprising diamines as new anti-tubercular therapeutics
04/21/2005WO2004062601A3 Antibacterial agents
04/21/2005US20050085667 N-biphenylmethyl aminocycloalkanecarboxamide derivatives
04/21/2005US20050085523 Imidazolyl and pyrazolyl ethyne compounds
04/21/2005US20050085509 KInase inhibitors; antiarthritic agents; autoimmune diseases; sepsis; cachexia; Alzheimer's disease; antihistamines; thrombosis; glomerulonephritis; inflammatory bowel disorders; crohn's disese; multiple sclerosis; antitumor agents; skin disorders
04/21/2005US20050085457 Therapeutic quinolone compounds with 5-ht-antagonistic properties
04/20/2005EP1349847B1 Oxybenzamides derivatives as factor xa inhibitors
04/20/2005CN1608054A Therapeutic quinolone compounds with 5-HT-antagonistic properties
04/20/2005CN1608052A Synthesis of enantiomerically pure amino-substituted fused bicyclic rings
04/20/2005CN1197863C Novel octahydro-2H-pyridino-[1, 2-a] pyrazine compound, its prepn. process and medicinal compound contg. them
04/20/2005CN1197856C Red fluorescence dyestuff and its synthesizing method and usage
04/19/2005US6881727 Sulfonated amino acid derivatives and metalloproteinase inhibitors containing the same
04/14/2005WO2005033119A1 Supramolecular compounds and their use as antitumour and antiviral agents
04/14/2005WO2005033105A2 Vanilloid receptor ligands and their use in treatments
04/14/2005WO2005033088A1 Quinoxaline compounds
04/14/2005WO2005016286A8 Pyrazine modulators of cannabinoid receptors
04/14/2005US20050080267 Synthesis of enantiomerically pure amino-substituted fused bicyclic rings
04/14/2005US20050080263 Method for producing ss-heteroaryl-alpha-alanine compounds using 2-amino-2-(heteroarylmethyl) carboxylic acid compounds
04/14/2005US20050080121 for example, 4S-[(naphthalene-2-carbonyl)-amino]-5-(2-oxo-pyrrolidin-3S-yl)-pent-2-enoic acid ethyl ester; treatment of viral infections caused by human rhinoviruses, human polioviruses, human coxsackieviruses, human echoviruses, among others
04/14/2005US20050080119 Diaminopropionic acid derivatives
04/14/2005US20050080106 Such as 2-[3,5-Di(2-chlorobenzyloxy)benzoyl)amino]-thiazole; for treatment of diabetes
04/14/2005US20050080092 Such as N-(6-aminohexyl)-N'-(3,5-diamino-6-chloropyrazine-2-carbonyl)guanidine Dihydrochloride; for hydration of mucosal surfaces, treating chronic bronchitis, cystic fibrosis, sinusitis, vaginal dryness, dry eye, esophogitis, emphysema, and pneumonia
04/14/2005US20050080091 Capped pyrazinoylguanidine sodium channel blockers
04/14/2005US20050080073 Sulfonylaminocarboxiylic acid N-arylamides as guanylate cyclase activators
04/14/2005DE10343098A1 Tetrahydrochinoxaline und ihre Verwendung Tetrahydroquinoxalines and their use
04/14/2005CA2540640A1 Vanilloid receptor ligands and their use in treatments
04/14/2005CA2540638A1 Quinoxaline compounds
04/13/2005EP1521748A1 Novel anthracene derivatives and the use thereof as a medicament
04/13/2005CN1606548A Aryloxyphenyl and arylsulfanylphenyl piperazine derivatives
04/13/2005CN1606443A Substituted diketopiperazines as oxytocin antagonists
04/13/2005CN1196681C (+)-Norcisapride useful for 5-HT3 and 5-HT4 mediated disorbers
04/13/2005CN1196680C Modulators of dopamine neurotransmission
04/12/2005US6878743 Controlling apoptosis; central nervous system disorders
04/12/2005US6878732 5,7-diazaspiro(3.4)octane and -octene derivatives; treating diseases including emesis, depression, anxiety and cough
04/12/2005US6878712 E.g., (R)-((2S,5R)-2-methyl-5-methyl-4-(4-carboxyphenyl-sulphonyl)-1-(3,3,3 -trifluoro-2-hydroxy-2-methylpropionyl)-piperazine); antidiabetic agents
04/12/2005US6878704 Heterocyclic mutilin esters and their use as antibacterials
04/12/2005US6878700 Cell adhesion-inhibiting antiinflammatory and immune-suppressive compounds
04/12/2005CA2203936C Boronic ester and acid compounds, synthesis and uses
04/12/2005CA2081836C Aromatic amidine derivatives and salts thereof
04/07/2005WO2005030794A2 Hemiasterlin derivatives and uses thereof
04/07/2005WO2004014871A8 Vanilloid receptor ligands and their use in treatments
04/07/2005US20050075390 HIV protease inhibitors
04/07/2005US20050074668 Perfluorinated amide salts and their uses as ionic conducting materials
04/07/2005CA2539823A1 Hemiasterlin derivatives and uses thereof
04/07/2005CA2539444A1 Hexa- and octahydro-pyrido[1,2-a]pyrazine derivatives with nk1 antagonistic activity
04/06/2005EP1520452A2 Electronic devices made with electron transport and/or anti-quenching layers
04/06/2005EP1520308A2 Polymeric charge transport compositions and electronic devices made with such compositions
04/06/2005EP1520305A2 Charge transport compositions and electronic devices made with such compositions
04/06/2005EP1519935A2 Charge transport compositions comprising fluorinated phenanthroline derivatives
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