Patents
Patents for C07D 241 - Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings (18,673)
09/2003
09/18/2003WO2003053368A3 Chalcone derivatives and their use to treat diseases
09/18/2003WO2002076925A3 Non-imidazole aryl alkylamines compounds as histamine h3 receptor antagonists, preparation and therapeutic uses
09/18/2003US20030176485 Calcium receptor active compounds
09/18/2003US20030176441 Inhibitsthe binding of eotaxin to the CCR-3 receptor and thereby provide a means of combating eosinophil induced diseases, such as asthma
09/18/2003US20030176440 For protecting skeletal muscles against damage resulting from trauma, protecting skeletal muscles subsequent to muscle or systemic diseases, therapy of shock conditions, preserving donor tissue and organs used in transplants
09/18/2003US20030176430 For therapy and prophylaxis of Tachykinin-mediated diseases
09/18/2003CA2479065A1 Aminoalcohol derivatives as beta-3 adrenergic receptor agonists
09/17/2003EP1344525A1 Aniline derivatives or salts thereof and cytokine production inhibitors containing the same
09/17/2003EP1343775A2 Piperazine derivatives
09/17/2003EP0984777B1 Arylsubstituted piperazines useful in the treatement of benign prostatic hyperlasia
09/17/2003EP0754682B9 Aminostilbazole derivative and medicine
09/17/2003CN1443170A Capsaicin receptor ligands
09/16/2003CA2167408C Process for making hiv protease inhibitors
09/16/2003CA2068089C Method and compositions for using non-ionic contrast agents to reduce the risk of clot formulation in diagnostic procedures
09/12/2003WO2003074495A1 Hppars activators
09/12/2003WO2003074476A1 Novel arylamidine derivative or salt thereof
09/11/2003US20030171461 Process for the synthesis of amine ethers from secondary amino oxides
09/11/2003US20030171352 Sulfonylaminocarboxylic acid N-arylamides as guanylate cyclase activators
09/11/2003US20030168970 Luminescent element material and luminescent element comprising the same
09/10/2003EP1341784A2 Process for making a thrombin inhibitor
09/10/2003EP1341764A1 Ortho-substituted nitrogen-containing bisaryl compounds used as potassium channel inhibitors
09/10/2003EP1341755A1 Carboxylic acid amide derivatives and their use in the treatment of thromboembolic diseases and tumours
09/10/2003EP1159237B1 Method of preparing surface-active alcohols and surface-active alcoholic ethers, products obtained by said method and their use
09/10/2003EP0998465B1 Polyhydroxyalkylpyrazine derivatives, preparation and medicines containing them
09/10/2003CN1441805A Antitumoral analogue of Et-743
09/10/2003CN1441789A Piperazinedione compounds
09/10/2003CN1441679A Compositions containing therapentically active components having enhanced solubility
09/10/2003CN1120878C Method for coal liquefaction
09/09/2003US6617317 Boronic ester and acid compositions
09/09/2003CA2138026C Novel 1,4-dihydroquinoxaline-2,3-diones and uses therefor as glycine receptor antagonists
09/09/2003CA2031480C Acetylenes disubstituted with a heteroaromatic group and a substituted phenyl group having retinoid like activity
09/04/2003WO2003072558A2 Arylsulfone derivatives
09/04/2003WO2003072537A2 Selective protein tyrosine phosphatatase inhibitors
09/04/2003WO2003072535A2 Substituted hydroxyethylamines
09/04/2003WO2003072056A2 Intranasal administration of mc4-r agonists
09/04/2003US20030166934 Using phase transfer catalyst
09/04/2003US20030166717 Substituted amide compound containing hydroxy and amino groups; useful for treating Alzheimer's disease and other similar diseases
09/04/2003US20030166690 Use of compounds for decreasing activity of hormone-sensitive
09/04/2003US20030166666 Diimino-piperazine derivatives for use as modulators of cell regulation
09/04/2003US20030166650 E.g., 3-(2-fluorophenyl)-N-(1-(3-morpholin-4-yl)phenyl)-propyl)acrylamide; disorders responsive to opening of KCNQ potassium channels; analgesics; migraine, bipolar disorders, anticonvulsants, antiepileptic, anxiolytic agents
09/04/2003US20030166644 Compounds and uses thereof for decreasing activity of hormone-sensitive lipase
09/04/2003US20030166637 Amines such as 9-(4-(4-(benzothiazol-2-yl)-piperazin-1-yl)-butyl)-9H-fluorene-9-carboxylic acid (2,2,2-trifluoroethyl) amide, used as microsomal triglyceride transfer protein antagonists, to prevent atherosclerosis or hyperlipemia
09/04/2003US20030166616 A tachykinin antagonist for used as antiinflammatory agent, antiallergic agent, analgesic, antiemetics, treating irritable colon syndrome, skin disorders
09/04/2003CA2477607A1 Substituted hydroxyethylamines
09/04/2003CA2476173A1 Arylsulfone derivatives
09/03/2003EP1341403A1 Luminescent element material and luminescent element comprising the same
09/03/2003EP1339701A1 Heteroaryl alkyl piperazine derivatives as fatty acid oxidation inhibitors
09/03/2003EP1339696A1 Benzyl(idene)-lactams and their use as 5ht1-receptor ligands
09/03/2003EP1339684A1 Mch antagonists and their use in the treatment of obesity
09/03/2003EP1339673A1 Malonamide and malonamic ester derivatives with antithrombotic activity, their preparation and their use
09/03/2003EP1070065B1 Azabicyclic 5ht1 receptor ligands
09/03/2003CN1440414A Synthesis of cuttlefish compound
09/03/2003CN1440383A PPARγ调制剂 PPARγ modulators
09/03/2003CN1440281A Medicine for reducing intraocular pressure
09/03/2003CN1439638A Preparation of tetrahydrobenzothiogenin oxidate containing antimer richfully
09/02/2003US6613769 Tryptase inhibitors
09/02/2003US6613743 Sulfonamide inhibitors of aspartyl protease
09/02/2003US6613345 Conjugates of sodium channel blockers and methods of using the same
08/2003
08/28/2003WO2003070709A1 Novel phenylalanine derivative
08/28/2003WO2003070184A2 Sodium channel blockers
08/28/2003WO2003070182A2 Sodium channel blockers
08/28/2003US20030162799 Squaric acid derivatives
08/28/2003US20030162789 4-alkylpiperazine substituted phenol derivative or 4-alkylamide substituted phenols for treating neurodegerative diseases such as aging, cancer, diabetes, ischemic stroke, Parkinson's disease, dementia and Huntinton's disease
08/28/2003US20030162786 Use of cysteine derivatives for the preparation of a medicament intended to treat pathologies which result from the formation of the heterotrimeric G protein
08/28/2003US20030162776 Substituted 5-membered polycyclic compounds useful for selective inhibition of the coagulation cascade
08/28/2003CA2476837A1 Sodium channel blockers
08/27/2003EP1338592A1 Novel 2-phenylpiperazine derivatives
08/27/2003EP1337518A1 Piperazinylpyrazines compounds as antagonists of serotonin 5-ht2 receptor
08/27/2003EP1337251A1 Monocyclic or bicyclic carbocycles and heterocycles as factor xa inhibitors
08/27/2003EP1337218A2 Substituted felbamate derived compounds
08/27/2003EP1185540B1 Ruthenium dimeric complexes suitable as antimetastatic and antineoplastic agents
08/27/2003EP0906906B1 Process for preparing optically active 2-piperazinecarboxylic acid derivatives
08/27/2003CN1119346C Benzothiadiaxoles and derivatives
08/27/2003CN1119336C Novel compounds with analgesic effect
08/26/2003US6610854 Reacting (Z)-5-Fluoro-2-methyl-(4-pyridylidene)-3-(N-benzyl) indenylacetamide with hydrochloric acid to produce (Z)-5-fluoro-2-methyl-(4-pyridylidene)-3-(N-benzyl)indenylacetamide hydrochloride
08/26/2003US6610846 Heteroaromatic glucokinase activators
08/26/2003US6610284 Preparation for prevention and healing of inflammation affections
08/21/2003WO2003069703A1 Electrode-active materials, electrodes made by using the same, and cells equipped with the electrodes
08/21/2003WO2003069397A2 Controlled diffusion coefficient electrochromic materials for use in electrochromic mediums and associated electrochromic devices
08/21/2003WO2003068759A1 Piperazine derivatives as anti-inflammatory agents
08/21/2003WO2003018549A3 Bicyclic compounds as inhibitors of chemokine binding to us28
08/21/2003WO2002020463A3 Fxr modulators
08/21/2003WO2002002512A3 Compounds to treat alzheimer's disease
08/21/2003US20030158411 Methods for preparing 5- and 6-benzyl-functionalized quinoxalines
08/21/2003US20030158205 N-benzyl-substituted, e.g., (2S)-1-(p-chlorophenoxy)methyl)-carbonyl-2-methyl-4-(p -fluorobenzyl)piperazine; inhibit the activity of the chemokines, MIP-1 alpha and RANTES
08/21/2003US20030158202 Substituted fused ring sulfonamides containing, e.g., naphthalene, isoquinoline, quinoline, benzofuran or benzothiophene rings; treatment of conditions relating to obesity, type II diabetes and CNS disorders
08/21/2003US20030158186 Compositions and methods for treating heart failure
08/21/2003US20030158185 Novel use of phenylheteroakylamine derivatives
08/21/2003CA2464451A1 Controlled diffusion coefficient electrochromic materials for use in electrochromic mediums and associated electrochromic devices
08/20/2003EP1336608A1 Dibenzosberanyl piperazine derivatives and drug-resistance overcoming agents containing the derivatives
08/20/2003EP1335907A1 Piperazinylpyrazine compounds as agonist or antagonist of serotonin 5ht-2 receptor
08/20/2003EP1282608B1 Production of 2-ethyl-3-methyl-1,4-diazine
08/20/2003EP1150944B1 N2-phenylamidine derivatives
08/20/2003CN1118456C 1,2-dihydro-2-oxoquinoline derivatives
08/19/2003US6608195 Process for the preparation of 2-(4-alkyl-1-piperazinyl)-benzaldehyde and -benzylidenyl compounds
08/19/2003US6608067 Inhibitors of serine proteases, particularly HCV NS3 protease
08/19/2003US6608063 For example: (2-(3-amino-4-nitrophenyl)amino)ethyl)(6-(2,4-dichlorophenyl-5-nitropyrazin -2-yl)-amine; antidiabetic, -carcingenic and ischemic agents; nervous and cardiovascular system disorders; immunotherapy; obesity; syndromes
08/19/2003US6608060 Treating inflammatory diseases, destructive bone disorders, reperfusion/ischemia in stroke, myocardial ischemia, renal ischemia, cardiac hypertrophy, rheumatoid arthritis, inflammatory bowel disease, or Crohn's disease
08/19/2003US6607741 Conjugates of sodium channel blockers and methods of using the same
08/14/2003WO2003066604A2 Novel aryl- and heteroarylpiperazines