Patents
Patents for C07D 233 - Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings (34,408)
01/1999
01/12/1999US5859042 Alopecia, acne, diseases of the prostate glands
01/12/1999US5859041 Substituted imidazoles having cytokine inhibitory activity
01/12/1999US5859035 Arylheteroaryl inhibitors of farnesyl-protein transferase
01/12/1999US5859005 Inhibitors of thrombin and factor xa
01/12/1999US5859002 HIV protease inhibitors
01/12/1999US5858684 Contacting recombinant cell with test compound which is not verapamil or gallopamil, determining ability of compound to affect activities of inorganic ion receptor; determination of agonist and antagonist drugs
01/07/1999WO1999000654A2 Radiolabeled farnesyl-protein transferase inhibitors
01/07/1999WO1999000535A1 Method for preparing 2-aryl or 2-heterocyclyl chiral propionic acids and their esters
01/07/1999WO1999000361A1 Ace-inhibitor nitric salts
01/07/1999WO1999000359A1 Aromatic ring derivatives
01/07/1999WO1999000356A1 Substituted n-[(aminoiminomethyl or aminomethyl)phenyl]propyl amides
01/07/1999WO1999000121A1 Antithrombotic agents
01/07/1999EP0889036A1 HIV protease inhibitors
01/07/1999EP0889033A1 Alpha-substituted benzyl heterocyclic derivatives, intermediates for producing the same, and pesticides containing the same as active ingredient
01/07/1999EP0888317A1 Substituted 4-hydroxy-phenylalcanoic acid derivatives with agonist activity to ppar-gamma
01/07/1999EP0888309A1 Imidazole derivatives having affinity for alpha2 receptors activity
01/07/1999EP0888308A1 Process for preparing heterocyclic carbenes
01/07/1999EP0888292A1 TRICYCLIC COMPOUNDS HAVING ACTIVITY SPECIFIC FOR INTEGRINS, PARTICULARLY $g(a)v$g(b)3 INTEGRINS, METHOD FOR PREPARING SAME, INTERMEDIATES THEREFOR, USE OF SAID COMPOUNDS AS DRUGS, AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME
01/07/1999DE19829229A1 Hydrazinderivate Hydrazine
01/07/1999CA2294042A1 Antithrombotic agents
01/07/1999CA2292794A1 Ace-inhibitor nitric salts
01/07/1999CA2288786A1 Radiolabeled farnesyl-protein transferase inhibitors
01/05/1999US5856513 Methylating an n-alkylimidazoline with dimethyl carbonate and (b) reacting the resulting n-alkyl-n'-methylimidazolinium methyl carbonate with an organic acid, methanol solvent
01/05/1999US5856509 Hypotensive agents
01/05/1999US5856326 Inhibitors of farnesyl-protein transferase
01/05/1999US5856311 Derivatives of β-aminopropionic acid with a fungicidal activity
01/05/1999US5856273 Controlling weeds
01/05/1999CA2132017C Imidazolin derivatives and a method for producing the same and a therapeutic agent for maintaining blood pressure
12/1998
12/30/1998WO1998058934A1 Novel 2-(iminomethyl)amino-phenyl derivatives, preparation, application as medicines and compositions containing same
12/30/1998WO1998058902A1 INHIBITORS OF α4β1MEDIATED CELL ADHESION
12/30/1998EP0887346A2 Phenyl-and aminophenyl-alkylsulfonamide and urea derivatives, their preparation and their use as alpha1A/1L adrenoceptor agonists
12/30/1998EP0887340A1 Novel compounds and pharmaceutical use thereof
12/30/1998CN1203590A Substituted imidazoles having anti-cancer and cytokine inhibitory activity
12/30/1998CN1203228A Phenyl-and aminophenyl-alkylsulfonamide and urea derivatives
12/29/1998US5854289 Guanylhydrazones and their use to treat inflammatory conditions
12/29/1998US5854265 Biheteroaryl inhibitors of farnesyl-protein transferase
12/29/1998US5854251 Aminotetrazole derivatives useful as nitric oxide synthase inhibitors
12/29/1998US5854234 Amidino dervatives useful as nitric oxide synthase inhibitors
12/29/1998US5854232 Acyclic anc cyclic amides as neurotransmitter release enhancers
12/29/1998CA2036427C Acyl compounds
12/23/1998WO1998057972A1 Quaternary ammonium compounds as tachykinin antagonists
12/23/1998WO1998057632A1 ALPHA 1a ADRENERGIC RECEPTOR ANTAGONISTS
12/23/1998EP0885189A2 Method for the synthesis of poly-pyrrole and poly-imidazole carboxamides on a solid support
12/23/1998EP0885188A1 Hydroxyamidino derivatives useful as nitric oxide synthase inhibitors
12/23/1998EP0885186A1 Amino acid derivatives, pharmaceutical compositions containing these compounds and processes for preparing them
12/23/1998EP0720595B1 Method of resolution of two enantiomers by crystallization
12/23/1998CN1202882A New LH-RH antigonists with improved effectiveness
12/23/1998CA2430623A1 Phenyl-and aminophenyl-alkylsulfonamide and urea derivatives
12/23/1998CA2294591A1 Alpha 1a adrenergic receptor antagonists
12/22/1998US5852210 Cinnamic acid derivatives
12/22/1998US5852203 Hydroxy-functional polyhydantoin prepolymers and their use in coating compositions
12/22/1998US5852192 Cyclic urea derivatives, pharmaceutical compositions containing these compounds and processes for preparing them
12/22/1998US5852043 HIV protease inhibitors
12/22/1998US5852007 Cysteine and serine protease inhibitors containing D-amino acid at the P2 position, methods of making same, and methods of using same
12/22/1998CA1340284C Herbicidal substituted cyclic diones
12/17/1998WO1998056788A1 Imidazolyl-cyclic acetals
12/17/1998WO1998056779A1 4-sulfinyl benzamides as calcitonin gene-related peptide receptor antagonists
12/17/1998WO1998056769A1 Carbonyldiimidazoles, their ester derivatives and method for their production
12/17/1998WO1998056737A1 Bromination process
12/17/1998DE19724884A1 Carbonyldiimidazole, daraus abgeleitete Ester und Verfahren zu ihrer Herstellung Carbonyldiimidazoles, esters derived therefrom and methods for their preparation
12/17/1998CA2289020A1 Bromination process
12/16/1998EP0715618B1 Hydroxyethylamino sulphonamides useful as retroviral protease inhibitors
12/16/1998EP0673545B1 Process and apparatus for etching semiconductor wafers
12/16/1998EP0664791B1 Process for the preparation of oxime derivatives, certain intermediates and the use of the oxime derivatives as fungicides
12/16/1998CN1202103A Excitatory amino acid receptor antagonists
12/16/1998CN1201794A Process for preparation of (1S,4R)-or(1R,4S)-4-(2-amino-6-chloro-9H-purin-9-yl)-2-cyclopentene-1-methanol
12/15/1998US5849929 Process for the preparation of imidazoline nitroxyl
12/15/1998US5849923 Heterocyclic-substituted naphthalenyl retinobenzoic acid derivatives
12/15/1998US5849919 Fused benzeneoxyacetic acid derivatives which have PGI2 receptor anonist activity
12/15/1998US5849794 Guanylhydrazones and their use to treat inflammatory conditions
12/15/1998US5849777 Cell differentiation induction with mevalonate and mevalonolactone derivatives
12/15/1998US5849776 Medicaments based on metronidazole or on a synergic mixture of metronidazole and clindamycin
12/15/1998US5849775 Substituted benzoylguanidines process for their preparation, their use as a medicament or diagnostic, and pharmaceutical containing them
12/15/1998US5849767 Chloropyridylcarbonyl derivatives
12/15/1998US5849732 Phenol compound having antioxidative activity and the process for preparing the same
12/15/1998CA2163667C Imidazole lipoxygenase inhibitors
12/15/1998CA1340247C Choline salts of arylmethylenyl thiazolidinones and oxazolidinones
12/10/1998WO1998055476A1 2-{4-[4-(4,5-dichloro-2- methylimidazol-1-yl)butyl] -1-piperazinyl}-5-fluoropyrimidine, preparation and therapeutic use
12/10/1998WO1998055468A1 Oxazole compounds useful as pge2 agonists and antagonists
12/10/1998WO1998055463A1 Diphenyl-triazole derivatives and their use as anti-gestative, immuno-suppressant and anti-tumoral agents
12/10/1998WO1998055448A2 Fluoroalkene carboxylic acid derivatives, method for producing said derivatives, and insecticidal agents containing the same
12/10/1998WO1998055118A2 Use of nitrogen heterocyclic aromatic derivatives in the topical treatment of the epithelial tissues diseases
12/10/1998WO1998055112A1 Enhanced anti-cancer agent delivery to solid tumors by primer compounds
12/10/1998WO1998054966A1 A method of treating cancer
12/10/1998WO1998040374A3 Olefin polymerization catalysts containing group 8-10 transition metals, bidentate ligands, processes employing such catalysts and polymers obtained therefrom
12/10/1998CA2294547A1 Use of nitrogen heterocyclic aromatic derivatives in the topical treatment of the epithelial tissues diseases
12/10/1998CA2292746A1 2-{4-[4-(4,5-dichloro-2- methylimidazol-1-yl)butyl] -1-piperazinyl}-5-fluoropyrimidine, preparation and therapeutic use
12/10/1998CA2292699A1 Enhanced anti-cancer agent delivery to solid tumors by primer compounds
12/10/1998CA2292471A1 A method of treating cancer
12/10/1998CA2291441A1 Fluoroalkene carboxylic acid derivatives, method for producing said derivatives, and insecticidal agents containing the same
12/09/1998EP0882043A1 Halogen pyrimidines and its use thereof as parasite abatement means
12/09/1998EP0882024A1 Retroviral protease inhibiting compounds
12/09/1998EP0882023A1 Histamine h 3 receptor ligands
12/09/1998EP0882022A1 Aspartyl protease inhibitors
12/09/1998EP0632803B1 Arthropodicidal amides
12/09/1998CN1201454A Meta-guanidine, urea, thiourea or azacyclic amino benzoic acid derivatives as integrin antagonists
12/09/1998CN1041083C Preparation of beta-ketoesters compound useful for preparing quinolone antibiotics
12/09/1998CN1041053C Use of medicine of imidazole-1-yl chemical compound
12/08/1998US5847213 Process for production of tertiary amine compound
12/08/1998US5847201 N-protected/N-substituted-beta-amino hydroxy sulfonates