Patents
Patents for C07D 233 - Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings (34,408)
04/1999
04/28/1999EP0911018A1 Use of cationic copolymers of unsaturated acids and n-vinylimidazolium salts in hair cosmetic compositions
04/28/1999EP0910565A1 Amide derivatives as selective neuropeptide y receptor antagonists
04/28/1999EP0910564A1 D-amino acid derived inhibitors of cysteine and serine proteases
04/28/1999EP0910563A1 Integrin receptor antagonists
04/28/1999EP0910376A2 Use of clotrimazole and related compounds in the treatment of diarrhea
04/28/1999EP0618907B1 1-(arylalkyl-aminoalkyl)imidazole derivatives, processes of preparation and use as therapeutical agents
04/28/1999CN1215392A Histamine H3 receptor ligands
04/28/1999CN1215332A Use of subsitituted aryl imidazoles
04/22/1999WO1999019305A2 Substituted pyrimidine derivatives, their preparation and their use in the treatment of neurodegenerative or neurological disorders of the central nervous system
04/22/1999WO1999019301A1 Piperazine compounds and medicinal use thereof
04/22/1999WO1999019300A1 Prostaglandin agonists and their use to treat bone disorders
04/22/1999WO1999019296A1 Aminobutanoic acid derivatives
04/22/1999WO1999018781A1 Dipeptide apoptosis inhibitors and the use thereof
04/22/1999WO1999006361A3 N-hydroxyformamide derivatives as inhibitors of matrix metalloproteinases
04/22/1999WO1999005114A3 1h-4(5)-substituted imidazole derivatives, their preparation and their use as histamine h3 receptor ligands
04/22/1999WO1999002146A8 Amino acid derivatives
04/22/1999WO1998052548A3 Use of 1-ar(alk)yl-imidazolin-2-one for treating anxiety and stress conditions
04/22/1999CA2306811A1 Piperazine compounds and medicinal use thereof
04/22/1999CA2305255A1 Substituted pyrimidine derivatives, their preparation and their use in the treatment of neurodegenerative or neurological disorders of the central nervous system
04/21/1999EP0712397B1 Amide derivatives as 5ht1d receptor antagonists
04/21/1999EP0695184B1 Hiv protease inhibitors
04/21/1999CN1214682A Eprosartan dihydrate and process for its production and formulation
04/20/1999CA1340507C Azole-substituted cycloalkanol derivatives, a process for producing the same and a use of derivatives as an agricultural and horticultural fungicide
04/16/1999CA2248241A1 Use of cationic copolymers of unsaturated acids and n-vinylimidazolium salts in cosmetic hair formulations
04/15/1999WO1999018084A1 Method and reagents for n-alkylating ureides
04/15/1999WO1999018076A1 The preparation and use of ortho-sulfonamido bicyclic heteroaryl hydroxamic acids as matrix metalloproteinase and tace inhibitors
04/15/1999WO1999018075A1 Novel dihydronaphthalene compounds and process for producing the same
04/15/1999WO1999018074A1 Novel lactam metalloprotease inhibitors
04/15/1999WO1999017790A1 PEPTIDE-CONTAINING α-KETOAMIDE CYSTEINE AND SERINE PROTEASE INHIBITORS
04/15/1999WO1999017777A1 Inhibitors of prenyl-protein transferase
04/15/1999WO1998055118A3 Use of nitrogen heterocyclic aromatic derivatives in the topical treatment of the epithelial tissues diseases
04/15/1999CA2306746A1 Inhibitors of prenyl-protein transferase
04/15/1999CA2305679A1 Novel lactam metalloprotease inhibitors
04/15/1999CA2304116A1 Peptide-containing .alpha.-ketoamide cysteine and serine protease inhibitors
04/15/1999CA2303449A1 The preparation and use of ortho-sulfonamido bicyclic heteroaryl hydroxamic acids as matrix metalloproteinase and tace inhibitors
04/15/1999CA2298527A1 Novel dihydronaphthalene compounds and process for producing the same
04/14/1999EP0908445A1 Oxidation dyeing composition for keratin fibres containing an amino acid derivative as oxidation base and aminoacid derivatives
04/14/1999EP0907637A1 Phenylalamine derivatives as integrin inhibitors
04/14/1999EP0810991B1 1-aryl-2-acylamino-ethane compounds and their use as neurokinin especially neurokinin 1 antagonists
04/14/1999EP0513397B1 Benzohydroximoylazole derivative, production thereof and insecticide
04/14/1999CN1213663A Process for manufacture of chiral succinic acid derivatives of formula
04/14/1999CN1213535A Cosmetic skin lightening product for topical application
04/08/1999WO1999016754A1 Process for the preparation of imidazoline derivatives
04/08/1999WO1999016747A1 Sulfonyl derivatives
04/08/1999WO1999016746A1 Aminoalkylphenol derivatives and related compounds
04/08/1999WO1999016437A1 Use of an angiotensin ii receptor antagonist for the preparation of drugs to increase the survival rate of renal transplant patients
04/08/1999CA2304285A1 Sulfonyl derivatives
04/08/1999CA2302703A1 Process for the preparation of imidazoline nitroxyl
04/07/1999EP0906927A1 Epoxy resin curing agents
04/07/1999EP0906917A2 Method for chemical synthesis of oligonucleotides
04/07/1999EP0906905A1 Process for the preparation of cyclic ureas
04/07/1999EP0906311A1 N-sulfonylimidazoles used as fungicides
04/07/1999EP0906307A1 Substituted imidazoles having cytokine inhibitory activity
04/07/1999EP0906296A1 Process for the preparation of chiral keto-heterocycles of basic amino acids
04/07/1999EP0906091A1 Amidinohydrazones as protease inhibitors
04/07/1999EP0854716A4 Androgenic directed compositions
04/07/1999EP0620821B1 Antiviral compositions and method for their use
04/06/1999US5892114 Hetero-linked phenylglycinolamides
04/06/1999US5892052 Process for making retroviral protease inhibiting compounds
04/06/1999US5891912 Endopeptidase 24.11 inhibitors
04/06/1999US5891909 Amidinohydrazones as protease inhibitors
04/06/1999US5891881 Propane 1,2,3-substituted with one of each: ether or sulfide group; hydroxy group; and aminoheterocyclic group; wound healing promoter for mammals
04/03/1999CA2247580A1 Process for preparing chiral succinic acid derivatives
04/01/1999WO1999015507A1 Hydrazono-benzazulene derivatives, pharmaceutical compositions and intermediates
04/01/1999WO1999015506A1 Tricyclic compounds, preparation method and said method intermediates, application as medicines and pharmaceutical compositions containing same
04/01/1999WO1999015493A1 9,10-dihydro-9,10-ethanoanthracene derivatives as phospholipase inhibitors
04/01/1999WO1999015490A1 C3a receptor ligands
04/01/1999WO1999015481A1 Asymmetric hydrogenation
04/01/1999WO1999003826A3 Metalloproteinase inhibitors
04/01/1999DE19743016A1 New 5-tetrahydroxybutyl-2,4-imidazolidine-dione compounds
04/01/1999DE19742844A1 New substituted imidazolidine-2,4-diones useful in preparation of enzyme inhibitors, especially protease inhibitors
04/01/1999CA2304879A1 New tetracycles, process for their production and pharmaceutical preparations containing these compounds
04/01/1999CA2303883A1 C3a receptor ligands
03/1999
03/31/1999EP0905139A2 5 ring heterocyles, process for preparation, use as inhibitors of leukocyte adhesion and pharmaceutical preparations comprising them
03/31/1999EP0904274A1 Farnesyl transferase inhibitors
03/31/1999EP0904262A1 Conformationally restricted aromatic inhibitors of microsomal triglyceride transfer protein and method
03/31/1999EP0904076A1 Inhibitors of farnesyl-protein transferase
03/31/1999CN1212685A Azole compounds endowed with antimycotic activity for human and veterinary use
03/30/1999US5889163 Method for producing azo dye compounds
03/30/1999US5889130 Monomeric and polymeric cyclic amine and N-halamine compounds
03/30/1999US5889059 Phenylacetic acid derivatives, preparation thereof and intermediates therefor, and compositions containing them
03/30/1999US5889038 Methods and products for treating diarrhea and scours: use of clotrimazole and related aromatic compounds
03/30/1999US5889037 Prevention, therapy tissue damage from lipid peroxidation
03/30/1999US5889014 Heterocyclic compounds for inhibiting phosphodiesterase IV
03/25/1999WO1999014200A1 Imidazoline compounds
03/25/1999WO1999001427A3 Novel nitric oxide-releasing amidine- and enamine-derived diazeniumdiolates, compositions and uses thereof and method of making same
03/25/1999WO1999001103A3 Peptide derivatives or pharmaceutically acceptable salts thereof, method for producing the same, use of said derivatives and pharmaceutical composition
03/25/1999WO1999000654A3 Radiolabeled farnesyl-protein transferase inhibitors
03/25/1999DE19742014A1 Use of new and known tetracyclene compounds as phospholipase inhibitors
03/25/1999DE19741636A1 New 1-benzyl-imidazole and known tetrazole derivatives
03/25/1999CA2303385A1 Imidazoline compounds
03/24/1999EP0903353A1 Imidazolidine derivates, their preparation and use, and pharmaceutical compositions containing them
03/24/1999EP0903337A1 Process for the preparation of 1-alkoxycarbonyl-3-phenylpropyl derivatives
03/23/1999US5886190 Reacting glycerol-1,3-ditosylate-2-o-acetylate with 2-nitroimidazole to form chemical intermediate 1-(2'-nitro-1'-imidazolyl)-2-o-acetyl-3-o-tosylpropanol in presence of dimethylformamide and cesium carbonate
03/23/1999US5886177 Phosphate linked oligomers
03/23/1999US5886175 Tetracycline antibiotics
03/23/1999US5886036 Treating hiv infections
03/23/1999US5885990 Fibrinolysis promoting action; thrombolysis action
03/23/1999US5885985 Antiinflammatory agents
03/23/1999CA2247735A1 Novel 5-membered ring heterocycles, their preparation, their use and pharmaceutical preparations comprising them