Patents
Patents for C07D 233 - Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings (34,408)
09/1999
09/30/1999CA2325472A1 Imidazolone anorectic agents: iii. heteroaryl derivatives
09/30/1999CA2322997A1 Novel cationic coupling agents, their use for oxidation dyeing of keratinous fibres, dyeing compositions and dyeing methods
09/30/1999CA2322992A1 Novel cationic compounds, their use as coupling agents for oxidation dyeing of keratinous fibres, dyeing compositions and dyeing methods
09/29/1999EP0945441A2 Process for the preparation of cyclic 4-oxoamidines
09/29/1999EP0945431A2 Process and intermediates for the preparation of phenylacetic derivatives
09/29/1999EP0944603A1 Process for making 2-amino-2-imidazoline, guanidine, and 2-amino-3,4,5,6-tetrahydropyrimidine derivatives
09/29/1999EP0944587A1 Metalloproteinase inhibitors
09/29/1999EP0944582A1 Ketobenzamides as calpain inhibitors
09/29/1999EP0944581A1 Process of preparing substituted acrylamides
09/29/1999EP0944387A1 Inhibitors of farnesyl-protein transferase
09/29/1999CN1230177A 'Beta'-sulfonyl hydroxamic acids as matrix metalloproteinases inhibitors
09/29/1999CN1230166A Illudin analogs useful as antitumor agents
09/29/1999CN1230110A Cell adhesion inhibitors
09/28/1999US5959113 Reacting a diketone derivative with an aldehyde derivative; administering to treat atherosclerosis, psoriasis, alopecia and tumors
09/28/1999US5958958 1,2,4-oxa diazolino and 1,24-oxa diazolidion heterocycles as useful nitric oxide synthase inhibitors
09/28/1999US5958954 2,2-dialkyl-4-aryl-substituted benzopyran and benzothiopyran derivatives
09/28/1999US5958839 Herbicidal compounds
09/27/1999CA2267080A1 Process for the preparation of cyclic 4-oxoamidines
09/23/1999WO1999047508A1 Benzenesulfonamide-derivatives and their use as medicaments
09/23/1999WO1999047504A1 Novel histidine derivatives preparation method and uses
09/23/1999WO1999047502A1 Cytotoxic metal chelators and methods for making and using same
09/23/1999CA2323783A1 Benzenesulfonamide-derivatives and their use as medicaments
09/23/1999CA2322742A1 Carboxylic acids and acylsulfonamides, compositions containing such compounds and methods of treatment
09/22/1999EP0943616A1 Substituted imidazole derivatives and their use as cytokine inhibitors
09/22/1999EP0663900B1 Metal-oxime chelates for use as radiopharmaceutical agents
09/22/1999CN1229082A Amine compound and its acid addition salt
09/22/1999CN1229080A Processes for preparing intermediate product used in method of diastereoselective syntheses of nucleosides
09/22/1999CN1229079A Processes for preparing intermediate product used in method of diastereoselective syntheses of nucleosides
09/22/1999CN1229078A Processes for preparing intermediate product used in method of diastereoselective syntheses of nucleosides
09/21/1999US5955617 Also for treatment of impaired glucose tolerance, obesity
09/21/1999CA2165137C Process for the manufacture of related intermediates including cistofur
09/16/1999WO1999046316A2 Enzyme inhibitors
09/16/1999WO1999046253A1 Heterocyclyl anthracyclinone derivatives
09/16/1999WO1999046246A1 Hetaryl-substituted benzyl phenyl ethers, method for the production thereof, and their use for combating harmful fungi and animal pests
09/16/1999WO1999046235A1 Fullerene derivatives
09/16/1999WO1999045914A1 Alkyl amine derivative and local anesthetic agent using the same
09/16/1999CA2323496A1 Enzyme inhibitors
09/16/1999CA2321832A1 Heterocyclyl anthracyclinone derivatives
09/15/1999EP0941080A2 Method of using cyclooxygenase-2 inhibitors as anti-angiogenic agents
09/15/1999EP0749421B1 Sulphonamide derivatives as aspartyl protease inhibitors
09/15/1999EP0741697B1 Amino acid derivatives and their use as phospholipase a2 inhibitors
09/15/1999CN1228771A 1,3-diheterocyclic metalloprotease inhibitors
09/15/1999CN1228765A New amidino derivatives and their use as thrombin inhibitors
09/15/1999CN1228414A New benzocyclobutane compounds, process for their preparation and pharmaceutical compositions containing them
09/14/1999US5952510 1,3-dihydro-1-(phenylalkenyl)-2H-imidazol-2-one derivatives having PDE IV and cytokine inhibiting activity
09/14/1999US5952507 Process for manufacture of chiral succinic acid derivatives
09/14/1999US5952497 N.sup.α -Bpoc amino acid pentafluorophenyl (Pfp) esters and 3,4-dihydro-4-oxo-1,2,3-benzotriazin-3-yl (ODhbt) esters
09/14/1999US5952381 Para-substituted phenylene derivatives
09/14/1999US5952362 2-imidazoline, 2-oxazoline, 2-thiazoline, and 4-imidazole derivatives of methylphenyl, methoxyphenyl, and aminophenyl alkylsulfonamides and ureas and their use
09/14/1999US5952359 Thiazoles and their agricultural compositions
09/14/1999US5952356 Treating diabetes in a mammal with an active material and a glucosidase inhibitor
09/14/1999US5952343 HIV protease inhibitors
09/14/1999US5952316 2-amino-1,3-propanediol compound and immunosuppressant
09/14/1999US5952291 Controlling the alkalinity of the reaction of an alkylimidazoline or an open-ring derivative with a monohalo-acetic acid to a ph of 8.5-10; by-product inhibition
09/14/1999US5952283 Quaternary ammonium compounds as bleach activators and their preparation
09/10/1999WO1999045004A1 Nitrate salt of anti-ulcer medicine
09/10/1999WO1999044993A1 Acryronitrile-based compound, method for producing the same and pest controlling agent comprising the same
09/10/1999WO1999029670A3 Aminocarbonyltetralin and dihydronaphtalene derivates as thrombin inhibitors
09/10/1999CA2322493A1 Nitrate salt of anti-ulcer medicine
09/08/1999EP0940390A1 6- (Substituted-methyl) -3- cyclohexenyl formamide derivative, hair growth promoter and external composition for skin
09/08/1999EP0940386A1 Benzocyclobutan compounds, their process for preparation and pharmaceutical compositions containing them
09/08/1999EP0939629A1 Thiol sulfonamide metalloprotease inhibitors
09/08/1999EP0939628A1 Thiol sulfone metalloprotease inhibitors
09/08/1999EP0617009B1 Novel amino acid derivative
09/08/1999EP0592643B1 Pleuromutilin derivatives
09/08/1999CN1228080A Novel immunotherapeutic agents and their use in production of cytokine levels
09/08/1999CN1228078A Catalytic preparation process of N-acylglycine derivatives
09/08/1999CN1227842A Penems and their derivatives
09/02/1999WO1999043653A1 Synthesis of epothilones, intermediates thereto and analogues therof
09/02/1999WO1999024460A3 Dipeptide nitriles
09/01/1999CN1227551A N-sulfonylimidazoles used as fungicides
09/01/1999CN1227540A Hydroxamic and carboxylic acid derivatives having MMP and TNF inhibitory activity
09/01/1999CN1044911C Method for preparing prodrug
08/1999
08/31/1999US5945526 Energy transfer dyes with enhanced fluorescence
08/31/1999US5945413 Treating human immunodeficiency virus infections
08/31/1999US5945408 Hydroxyanidino derivatives useful as nitric oxide synthase inhibitors
08/31/1999CA2173328C Hiv protease inhibitors
08/31/1999CA2145835C Hydroxamic acid derivatives with tricyclic substitution
08/26/1999WO1999042455A1 Antiviral agents
08/26/1999WO1999042450A1 Solid phase synthesis of 1-aminohydantoins
08/26/1999WO1999042449A1 Novel compounds, hardening accelerator, resin composition, and electronic part device
08/26/1999WO1999042443A1 Sulfonylamino derivatives which inhibit matrix-degrading metalloproteinases
08/26/1999WO1999026909A3 Alpha-hydroxy, -amino and -fluoro derivatives of beta-sulphonyl hydroxamic acids as matrix metalloproteinases inhibitors
08/26/1999CA2321085A1 Solid phase synthesis of 1-aminohydantoins
08/25/1999EP0937076A1 Substituted oximes, hydrazones and olefins as neurokinin antagonists
08/25/1999EP0937042A1 Heteroaryl succinamides and their use as metalloproteinase inhibitors
08/25/1999EP0788485A4 Compacting halohydantoin and fatty amide and product therefrom
08/25/1999CN1226992A Ionic liquids as solvents
08/25/1999CN1226892A Compounds and compositions for treating diseases associated with tryptase activity
08/25/1999CN1226803A Diphenyl heterocycles as potassium channel modulators
08/24/1999US5942641 Fluorenone derivatives, process for preparing the same and central or peripheral nerve degeneration repair and protective agent
08/24/1999US5942632 Novel 4,5-bis(protected-amino), 2-(protected-carboxy)-1,3-dioxolane compounds that can be used to prepare hiv protease inhibitors by coupling to a solid support via an ester or an amide linkage
08/24/1999US5942627 Concentrated amphocarboxylpropionate surfactants produced from methyl acrylate and 2-alkyl imidazoline
08/24/1999US5942522 1-benzyl-3-ethoxycarbonyl-4-dimethylaminoethoxy-6-methyl-2-(1h) -quinolinone; antiviral against dna containing viruses, such as herpes group viruses
08/24/1999US5942493 LH-RH antagonists having improved action
08/19/1999WO1999041367A1 Heteroaromatic oligoamides as affinity ligands
08/19/1999WO1999041235A1 Farnesyl transferase inhibitors
08/19/1999WO1999040910A1 Anti-inflammatory agents
08/19/1999CA2320285A1 Anti-inflammatory agents
08/18/1999EP0935597A2 Dihydropyrones with improved antiviral activity