Patents for C07D 231 - Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings (25,550) |
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06/25/2009 | WO2009078475A1 Process for production of pyrazolinone derivative |
06/25/2009 | WO2009078432A1 1-alkyl-4-amino-1h-pyrazole-3-carboxamide compound |
06/25/2009 | WO2009077954A1 Aminopyrazole derivatives |
06/25/2009 | WO2009077853A1 Process for the preparation of fipronil and analogues thereof |
06/25/2009 | WO2009077844A2 Inhibitors of biofilm formation of gram-positive and gram-negative bacteria |
06/25/2009 | WO2009077390A2 Azomethine direct dyes or reduced precursors of azomethine direct dyes obtained from 4,5 diaminopyrazole, and hair dyeing process using these dyes or precursors |
06/25/2009 | WO2009041705A3 5-membered heterocyclic compounds as proton pump inhibitors |
06/25/2009 | WO2009036235A3 Insecticidal carbamates exhibiting species-selective inhibition of acetylcholinesterase (ache) |
06/25/2009 | US20090163569 Process for the production of amides |
06/25/2009 | US20090163560 5-(3-(2-(4-(1-Hydroxyhexyl)phenyl)-3-oxopyrazolidin-1-yl)propyl)thiophene-2-carboxylic acid; bioisosteres; vision defects; glaucoma; hypotensive agents; ocular hypertension; kits |
06/25/2009 | US20090163546 Diacylglycerol acyltransferase inhibitors |
06/25/2009 | US20090163496 Antibacterial agents |
06/25/2009 | US20090163493 cell proliferation, such as cancer, inflammation, and angiogenesis; fungal infections; antimalaria; Heat hock protein 90 (HSP-90) inhibitor |
06/25/2009 | CA2709751A1 Process for the preparation of fipronil and analogues thereof |
06/25/2009 | CA2706836A1 Aminopyrazole derivatives |
06/24/2009 | EP1781614B1 Compounds which potentiate glutamate receptor and uses thereof in medicine |
06/24/2009 | CN100503577C Disubstituted pyrazolyl carboxanilides |
06/24/2009 | CN100503576C Substituted azole compounds, preparation and application thereof |
06/23/2009 | US7550624 For treating or inhibiting increased urinary urgency or urinary incontinence and/or pain |
06/23/2009 | US7550489 N-[3-(4-chlorophenyl)-2-(3-cyanophenyl)-1-methylpropyl]-2-(5-trifluoromethyl-2-pyridyloxy)-2-methylpropanamide and phentermine, metformin, or bupropion; obesity; antipsychotic agents; synergistic; cannabinoid receptor antagonists |
06/18/2009 | WO2009075080A1 Fluoroalkylsulfide derivative and pest control agent |
06/18/2009 | WO2009074782A1 Cannabinoid receptor modulators |
06/18/2009 | WO2009074590A1 N- (2 { [1-phenyl-1h-indaz0l-4-yl] amino} propyl) -sulfonamide derivatives as non-steroidal glucocorticoid receptor ligands for the treatment of inflammations |
06/18/2009 | WO2009010156A3 Substituted phenylpropoargyl compounds, methods for the production thereof, and use of same as herbicides and plant growth regulators |
06/18/2009 | WO2008072053A8 Substituted arylpyrazoles |
06/18/2009 | US20090156651 Heterocyclylethylbenzamide Derivatives |
06/18/2009 | US20090156616 Therapeutic agents |
06/18/2009 | US20090156592 Fungicidal Azocyclic Amides |
06/18/2009 | US20090155203 Thrombopoietin mimetics |
06/18/2009 | CA2708706A1 Cannabinoid receptor modulators |
06/17/2009 | EP2069311A1 Process for the preparation of fipronil, an insecticide, and related pyrazoles |
06/17/2009 | EP2069310A2 Sulfonylpyrazoline carboxamidine derivatives as 5-ht6 antagonists |
06/17/2009 | EP2069287A1 Insecticidal compounds |
06/17/2009 | EP1836166B1 Glucocorticoid mimetics, methods of making them, pharmaceutical compositions, and uses thereof |
06/17/2009 | EP1611088B1 Hydroxamates as therapeutic agents |
06/17/2009 | CN101460466A Thiazoles, imidazoles, and pyrazoles useful as inhibitors of protein kinases |
06/17/2009 | CN101456843A Synthetic method of 5-(4-chlorphenyl)-1-(2,4-dichlorobenzene)-4-methylpyrazole-3-carboxyl acid |
06/16/2009 | US7547725 Fluoro- and trifluoroalkyl-containing heterocyclic sulfonamide inhibitors of beta amyloid production and derivatives thereof |
06/16/2009 | US7547720 di-tert-butyl 4-{[1-(3,3-dimethyl-2-oxobutyl)-6-methoxy-1-H-indazole-3-yl]carbonyl}benzylphosphate; potassium channel blocker; eye neuroprotectant; hypotensive agent; glaucoma, elevated intraoccular pressure in the eye |
06/16/2009 | US7547719 Thrombopoietin mimetic; useful as an agonist of the TPO receptor, particularly in enhancing platelet production; treatment of thrombocytopenia |
06/16/2009 | US7547701 cathepsin S inhibitors; e.g. N-(1-cyanocyclopropyl)-3-phenylmethanesulfonyl-2-(2,2,2-trifluoro-1-phenylethylamino)-propionamide; autoimmune diseases such as rheumatoid arthritis or multiple sclerosis, pain, or atherosclerosis |
06/16/2009 | CA2447640C Substituted anilide derivative, intermediate thereof, agricultural and horticultural chemical and its usage |
06/11/2009 | WO2009071483A1 1- (indaz0l-5-yl) -ureas as diacylglycerol acyltransferase inhibitors |
06/11/2009 | WO2009051718A3 Calcium receptor modulating agents |
06/11/2009 | WO2008086962A3 Method for producing substituted pyrazolecarboxylic acid chlorides |
06/11/2009 | US20090149659 intermediates to manufacture of pharmaceutical 1-(aminoalkyl)indazoles (Yamanouchi Pharma, WO98/30548) which avoid undesired isomers and which are capable of producing large quantities of the desired compound |
06/11/2009 | US20090149524 N-(Phenylmethyl)-2-(1H-Pyrazol-4-yl) Acetamide Derivatives as P2X7 Antagonists for the Treatment of Pain, Inflammation and Neurodegeneration |
06/11/2009 | US20090149463 Therapeutic agents |
06/11/2009 | US20090149459 P38 inhibitors and methods of use thereof |
06/11/2009 | US20090149457 1H-Thieno[2,3-c]Pyrazole Compounds Useful as Kinase Inhibitors |
06/11/2009 | US20090149445 Tricyclic steroid hormone nuclear receptor modulators |
06/11/2009 | US20090149443 P38 inhibitors and methods of use thereof |
06/11/2009 | US20090149425 Malononitrile compound as pesticides |
06/10/2009 | EP2066641A1 Pyrazole derivatives as modulators of the 5-ht2a serotonin receptor useful for the treatment of disorders related thereto |
06/10/2009 | EP0976737B1 Pyrazole derivatives, process for preparing the same, intermediates, and pest control agent containing the same as active ingredient |
06/10/2009 | CN101454291A Sulphur containing pyrazole derivatives as selective cannabinoid CB1 receptor antagonists |
06/10/2009 | CN100497358C Iridium compound and organic electroluminescent device using the same |
06/10/2009 | CN100497326C Derivatives of 1-piperazine- and 1-homopiperazine-carboxylates, preparation method thereof and use of same in therapeutics |
06/10/2009 | CN100497302C Diarylurea derivatives and their use as chloride channel blockers |
06/09/2009 | US7544711 Cyclooxygenase inhibitors; musculoskeletal and cardiovascular disorders; antiinflammatory agents |
06/09/2009 | US7544707 Peroxisome Proliferator Activated Receptor (PPAR); 2-Methyl-4-[2-(4-trifluoromethylphenyl)-2H-indazol-7-ylmethylsulfanyl]phenoxyacetic Acid; diabetes, Metabolic and cardiovascular disorders, arthritis, demyelinating diseases |
06/04/2009 | WO2009069736A1 Nitrogenated compound |
06/04/2009 | WO2008059370A8 Substituted bicyclocarboxyamide compounds |
06/04/2009 | US20090143592 Glucagon Antagonists/Inverse Agonists |
06/04/2009 | US20090143579 Heterocyclic Inhibitors of MEK and Methods of Use Thereof |
06/04/2009 | US20090143455 Pyrazoles Useful in the Treatment of Inflammation |
06/04/2009 | US20090143454 Pyrazoline Derivatives and Their Use As Pesticides |
06/04/2009 | US20090143422 P38 inhibitors and methods of use thereof |
06/04/2009 | US20090143389 Heterocyclic inhibitors of mek and methods of use thereof |
06/04/2009 | US20090143380 2h- or 3h-benzo[e]indazol-1-yl carbamate derivatives, the preparation and therapeutic use thereof |
06/04/2009 | US20090143376 Fused Heterocyclic Compounds and Their Use as Sirtuin Modulators |
06/04/2009 | US20090143370 Non-nucleoside Reverse Transcriptase Inhibitors |
06/04/2009 | US20090143365 Derivatives of alkylpiperazine- and alkylhomopiperazine-carboxylates, preparation method thereof and use of same as fatty acid amido hydrolase enzyme inhibitors |
06/04/2009 | US20090143358 Inhibitors of ion channels |
06/03/2009 | EP2064177A2 Protease inhibitors |
06/03/2009 | EP1814860B1 Substituted 5-carboxyamide pyrazoles and [1,2,4]triazoles as antiviral agents |
06/03/2009 | EP1765788B1 3-aminoindazole derivatives and their use for the treatment of sgk-associated diseases |
06/03/2009 | EP1071668B1 5-aminoindeno[1,2-c]pyrazol-4-ones as anti-cancer and anti-proliferative agents |
06/03/2009 | CN101448792A Compounds which potentiate AMPA receptor and uses thereof in medicine |
06/03/2009 | CN101448791A FXR agonists |
06/03/2009 | CN101445501A Fused compounds that inhibit vanilloid receptor subtype 1 (VR1) receptor |
06/03/2009 | CN101445483A Method for preparing pesticide |
06/03/2009 | CN100494177C Bi-amido heterocyclic derivative with antitumour activity and its preparation method and use |
06/02/2009 | US7541378 tert-butyl 3-amino-1H-thieno[2,3-c]pyrazole-5-carboxylate; N-benzyl-3-[(4-fluorobenzoyl)amino]-1H-thieno[2,3-c]pyrazole-5-carboxamide; treats a disease caused associated with an altered (disregulated) protein kinase activity e.g cancer, cell proliferative disorders, Alzheimer's disease, viral infections |
06/02/2009 | US7541377 1-[2-(Aminomethyl)phenyl]-N-[2-methyl-6-[[(1-methylethyl)amino]carbonyl]phenyl]-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide; pesticides |
06/02/2009 | US7541376 3-(3-Fluoro-phenyl)-6-methoxy-1H-indazole-5-carboxylic acid(furan-2-ylmethyl)-amide; 3-Benzo[b]thiophen-2-yl-4-methoxy-1H-indazole-5-carboxylic acid[3-(2-oxo-pyrrolidin-1-yl)-propyl]-amide; Jun amino-terminal kinase (JNK) inhibitor; immunologic disease, inflammatory and neurodegenerative diseases |
06/02/2009 | US7541374 Malononitrile compounds and use thereof |
06/02/2009 | US7541370 1-aryl- or 1-alkylsulfonyl-heterocyclylbenzazoles as 5-hydroxytryptamine-6 ligands |
06/02/2009 | US7541358 1-aryl-or 1-alkylsulfonylbenzazole derivatives as 5-hydroxytryptamine-6 ligands |
06/02/2009 | CA2304425C Novel pyrazolone compound and ophthalmic plastic lens using the same |
05/28/2009 | WO2009067621A1 Biaryl pde4 inhibitors for treating pulmonary and cardiovascular disorders |
05/28/2009 | WO2009067600A2 Biaryl pde4 inhibitors for treating inflammation |
05/28/2009 | WO2008152138A3 Method for producing difluoromethyl-substituted pyrazole compounds |
05/28/2009 | WO2008152086A3 4,5-dihydro-(1h)-pyrazole derivatives as cannabinoid cb1 receptor modulators |
05/28/2009 | US20090137655 Non-Steroidal Ligands for the Glucocorticoid Receptor, Compositions and Uses Thereof |
05/28/2009 | US20090137611 Fungicide N-Cyclopropyl-Sulfonylamide Derivatives |
05/28/2009 | US20090137585 N-acylsulfonamide apoptosis promoters |
05/28/2009 | US20090137560 Imidazole compounds having pharmaceutical activity towards the sigma receptor |
05/28/2009 | US20090137524 Substituted arylpyrazoles |
05/28/2009 | US20090137420 Methods, compounds and compositions with genotype selective anticancer activity |