Patents for C07D 231 - Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings (25,550) |
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01/20/2010 | EP1654247B1 Alkynyl aryl carboxamides |
01/20/2010 | CN101628895A Preparation method of fipronil formed by oxidization of phenyl pyrazole derivatives |
01/20/2010 | CN100582096C Method for synthesizing pyrazoline derivatives capable of irradiating yellow green light |
01/20/2010 | CN100581543C Tetrahydronaphthalene derivatives, process for their production and their use as anti-inflammatory agents |
01/19/2010 | US7649104 producing 3-acyloxyacrylonitrile compound as an agricultural and horticultural pesticide; using the produced 3-oxopropionitrile compound as the intermediate |
01/19/2010 | US7649015 Saquinavir-like, a Lopinavir-like, a Ritonavir-like, a Indinavir-lik, a atazanavir-like, Nelfinavir-like.a Tipranavir-like, a Amprenavir-like, a KNI-like. a cyclic carbonyl-like phosphonate HIV protease inhibitors; drug designing |
01/19/2010 | US7649009 N-(trans-4-tert-butylcyclohexyl)-1-{4-[(1h-tetrazol-5-ylamino)carbonyl]benzyl }-3-(3,4,5-trifluoropbenyl)-1h-pyrazole-5-carboxamide; type 2 diabetes, hyperglycemia, diabetes or insulin resistance, Syndrome X, atherosclerosis |
01/19/2010 | US7649001 Fused benzene derivative and use |
01/19/2010 | US7648971 Thrombopoietin mimetics |
01/19/2010 | CA2143135C Process for sulfinylating heterocyclic compounds |
01/14/2010 | WO2009132453A8 Cyclylamine derivatives as calcium channel blockers |
01/14/2010 | WO2009000441A8 Processes for the preparation of pyrazoles |
01/14/2010 | US20100010123 Ultraviolet absorbent and polymer material containing the same |
01/14/2010 | US20100010063 Heterocyclocarboxamide derivatives |
01/14/2010 | US20100010061 Cb1 receptor modulators |
01/14/2010 | US20100010054 Therapeutic agent for amyotrophic lateral sclerosis |
01/14/2010 | US20100010045 PYRAZOLE-DERIVATIVES AS FACTOR Xa INHIBITORS |
01/14/2010 | US20100010038 Tricyclic compound and pharmaceutical use thereof |
01/13/2010 | EP2142511A2 Heterocyclyl-substituted-tetrahydro-naphthalen-amine derivatives, their preparation and use as medicaments |
01/13/2010 | EP1451160B1 Pyrazole-amides for use in the treatment of pain |
01/13/2010 | EP1144388B1 Acyl derivatives which treat vla-4 related disorders |
01/13/2010 | CN101627015A Fluorine-containing pyrazolecarbonitrile derivative and method for producing the same, and fluorine-containing pyrazolecarboxylic acid derivative obtained by using the fluorine-containing pyrazolecarb |
01/13/2010 | CN101624373A N-multisubstituted pyrazole amidine derivative and application thereof on insect pest and harmful mite prevention |
01/13/2010 | CN100579976C P38 inhibitors and methods of use thereof |
01/12/2010 | US7645885 (E)-Methyl 3-(1,2,3,4,8,8 alpha -hexahydro-8 alpha -methylspiro[1',3'-dithiolane-2',6(7H)naphthalen]-1-yl)acrylate; for treating or preventing diseases ( prostate cancer, benign prostatic hyperplasia, reproductive disorders, and male hypogonadism) associated with androgen binding to the androgen receptor |
01/12/2010 | US7645787 4'-((2-fluoro-4-methylphenyl)methyl)-1'-isopropyl-5'-methyl-1H-pyrazole-3'-O-(6-carbomethoxy)- beta -D-glucopyranoside; 4-[(3-fluoro-4-methoxyphenyl)methyl]-1-isopropyl-5-methyl-1H-pyrazole-3-O- beta -D-glucopyranoside; reducing reanal glucose reabsorption |
01/12/2010 | US7645786 Substituted arylpyrazoles |
01/12/2010 | US7645757 Derivatives of heteroaryl-alkylcarbamates, methods for their preparation and use thereof as fatty acid amido hydrolase enzyme inhibitors |
01/12/2010 | CA2442906C Reconstitutable parenteral composition containing a cox-2 inhibitor |
01/07/2010 | WO2010003025A1 Bicyclic heterocycles as mek kinase inhibitors |
01/07/2010 | WO2010001869A1 Tetra-substituted benzene compound and use thereof |
01/07/2010 | WO2010000372A2 New drug for inhibiting aggregation of proteins involved in diseases linked to protein aggregation and/or neurodegenerative diseases |
01/07/2010 | US20100004307 Process for the Sulfinylation of a Pyrazole Derivative |
01/07/2010 | US20100004280 Substituted imidazoles as bombesin receptor subtype-3 modulators |
01/07/2010 | US20100004271 Heterocyclic compounds as aganist for the thyroid receptor |
01/07/2010 | US20100004207 Inhibitors of cyclin-dependent kinases, compositions and uses related thereto |
01/07/2010 | US20100004129 Herbicidally active 4-(3-alkylsulfinylbenzoyl)pyrazoles |
01/07/2010 | CA2727250A1 Bicyclic heterocycles as mek kinase inhibitors |
01/07/2010 | CA2726999A1 New drugs for inhibiting aggregation of proteins involved in diseases linked to protein aggregation and/or neurodegenerative diseases |
01/06/2010 | EP2141150A1 Bicyclic compound and pharmaceutical use thereof |
01/06/2010 | EP2140864A2 Use of GAL3 receptor antagonists for the treatment of depression and / or anxiety and compounds useful in such methods |
01/06/2010 | EP2140862A2 Use of GAL 3 receptor antagonists for the treatment of depression and /or anxiety and compounds useful in such methods |
01/06/2010 | EP2139862A1 Cosmetic preparations designed to reduce unsightly cellulite |
01/06/2010 | EP2139489A2 Mineralocorticoid receptor modulators |
01/06/2010 | EP2139328A2 Hexahydro-cycloheptapyrazole cannabinoid modulators |
01/06/2010 | EP1005361B1 USE OF FVIIa OR FVIIai FOR THE TREATMENT OF ENDOTHELIAL DYSFUNKTION AND FOR THE INHIBITION OF ANGIOGENESIS RESPECTIVELY |
01/06/2010 | CN101622233A Tricyclic compound and pharmaceutical use thereof |
01/06/2010 | CN100577648C 2H- or 3H-benzo[e]indazol-1-yle carbamate derivatives, the preparation and therapeutic use thereof |
01/06/2010 | CN100577163C Compounds effecting glucokinase |
01/05/2010 | US7642360 Composition for dyeing keratinous fibers comprising at least one diamino-N,N-dihydropyrazolone derivative |
01/05/2010 | US7642359 Pyrazolyl-substituted heterocycles and their use as phytosanitary products |
01/05/2010 | US7642358 Antidiabetic agents; modulate insulin drug resistance |
01/05/2010 | US7642276 N-[4-methyl-3-(3-piperidin-4-yl-1,2-benzisoxazol-6-yl)phenyl]-2-pyrrolidin-1-ylisonicotinamide; rheumatoid arthritis |
12/31/2009 | US20090326242 Process for preparing 3-dihalomethyl-pyrazole-4-carboxylic acid derivatives |
12/31/2009 | US20090326241 PROCESS FOR PREPARING SUBSTITUTED 5-AMINO-PYRAZOLO-[4,3-e]-1,2,4-TRIAZOLO[1,5-c]PYRIMIDINES |
12/31/2009 | US20090326240 Iron-Copper Co-Catalyzed Process for Carbon-Carbon or Carbon-Heteroatom Bonding |
12/31/2009 | US20090325974 1,5-diphenylpyrazoles ii as hsp90 inhibitors |
12/31/2009 | US20090325962 Tyrosine derivative |
12/31/2009 | US20090324625 Heterocyclic Aromatic Compounds Useful As Growth Hormone Secretagogues |
12/31/2009 | US20090324569 Biaryl pde4 inhibitors for treating inflammatory, cardiovascular and cns disorders |
12/30/2009 | WO2009158369A1 Synthesis and use of heterocyclic antibacterial agents |
12/30/2009 | WO2009157196A1 Amide compound |
12/30/2009 | WO2009156090A2 Insecticidal sulfur-derivatized 1-azinylpyrazoles |
12/30/2009 | WO2008157680A3 Methods and compositions for modulating p300/cbp activity |
12/30/2009 | WO2008151719A8 3-cyclopropyl-4-(3-thiobenzoyl)pyrazoles and their use as herbicides |
12/30/2009 | EP2138483A1 Oxidative color-developing compounds, salts thereof, process for production of the same, reagent compositions and test tools made by using the same |
12/30/2009 | EP2137178A2 Novel vanilloid receptor ligands and the use thereof for the production of pharmaceuticals |
12/30/2009 | EP2137160A1 4-(4-trifluoromethyl-3-thiobenzoyl)pyrazoles, and use thereof as herbicides |
12/30/2009 | EP2137159A1 4-(3-aminobenzoyl)-1-ethylpyrazole and the use thereof as herbicides |
12/30/2009 | CN101616897A Heterocyclyl-substituted-ehylamino-phenyl derivatives, their preparation and use as medicaments |
12/30/2009 | CN101613318A Dihalo-propylene compound and preparation method and application thereof |
12/30/2009 | CN100575341C Tetrahydro-indolone derivative and tetrahydro-indazolone derivatives and their use |
12/30/2009 | CA2729227A1 2-heterocyclylaminoalkyl-(p-quinone) derivatives for treatment of oxidative stress diseases |
12/30/2009 | CA2728210A1 Synthesis and use of heterocyclic antibacterial agents |
12/29/2009 | US7638514 Agriculture |
12/29/2009 | CA2370250C Di-aryl acid derivatives as ppar receptor ligands |
12/24/2009 | US20090318703 Carboxylic acid derivatives and pharmaceutical agent comprising the same as active ingredient |
12/24/2009 | US20090318495 Ethenyl carboxamide derivatives useful as microbiocides |
12/23/2009 | WO2009155399A1 1-substituted-3-(naphthalen-1-ylsulfonyl)-5-(piperazin-1-yl)-1h-indazole compounds as 5-hydroxytryptamine-6 ligands |
12/23/2009 | WO2009155362A1 Small molecule hematopoietic growth factor mimetic compounds and their uses |
12/23/2009 | WO2009154557A1 Benzoxazinone derivatives acting as beta2-adrenoreceptor agonist for the treatment of respiratory disorders |
12/23/2009 | WO2009153804A1 Process for preparing form i of rimonabant |
12/23/2009 | WO2009153592A1 Pyrazole compounds 436 |
12/23/2009 | WO2009153180A1 Heteroaromatic monoamides as orexinin receptor antagonists |
12/23/2009 | WO2009117626A3 Methods for making central nervous system agents that are trpv1 antagonists |
12/23/2009 | EP2134175A1 Inhibitors of akt activity |
12/23/2009 | EP1534390B1 3'- (2z)- 1-(3,4-dimethylphenyl)-1,5-dihydro-3-methyl-5-oxo-4h-pyrazol-4-ylidene hydrazino -2'-hydroxy- 1,1'-biphenyl -3-carboxylic acid bis-(monoethanolamine) |
12/23/2009 | EP1523475B1 Heterocyclically substituted benzoylureas, method for their production and their use as medicaments |
12/23/2009 | CN101611015A Indazolyl ester and amide derivatives for the treatment of glucocorticoid receptor mediated disorders |
12/23/2009 | CN101611014A Acylaminopyrazoles as FGFR inhibitors |
12/23/2009 | CN101611013A Pyrazole derivatives as modulators of the 5-HT2A serotonin receptor useful for the treatment of disorders related thereto |
12/23/2009 | CN101607957A Intermediate for preparing 3-halo-4,5-dihydro-1h-pyrazoles |
12/23/2009 | CN101607941A Fluoride-containing pyrazole compound as well as preparation and application thereof |
12/23/2009 | CN101607940A Fluorine Anthranilamide compound for killing arthropod |
12/23/2009 | CN100572361C Process for the preparation of phenyl pyrazole compounds |
12/23/2009 | CA2728063A1 Pyrazole compounds 436 |
12/23/2009 | CA2726746A1 Benzoxazinone derivatives acting as beta2-adrenoreceptor agonist for the treatment of respiratory disorders |
12/23/2009 | CA2726703A1 Heteroaromatic monoamides as orexinin receptor antagonists |
12/22/2009 | US7635695 4-Amino-2-(4-methyl-thiophen-2-yl)thieno[3,2-c]pyridine-7-carboxylic acid amide; 4-amino-2-cyclopent-1-enyl-thieno[3,2-c]pyridine-7-carboxylic acid amide; for therapy and prophylaxis of disease or condition associated with inflammation, a metabolic disorder, infection, cancer or an immune disease |
12/22/2009 | US7635684 Pyrazole derivatives, medicinal composition containing the same, medicinal use thereof, and intermediate for production thereof |